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List of works by Angela Casini

A gold coordination compound as a chemical probe to unravel aquaporin-7 function

scientific article published on 28 May 2014

A golden future in medicinal inorganic chemistry: the promise of anticancer gold organometallic compounds

scientific article published on March 2014

A multi-technique approach to predicting the molecular structure of cuprizone in the gas phase and in the crystalline state

A new target for gold(I) compounds: Glutathione-S-transferase inhibition by auranofin

scientific article published on 24 August 2012

Activity of Rat Cytosolic Thioredoxin Reductase Is Strongly Decreased bytrans-[Bis(2-amino-5- methylthiazole)tetrachlororuthenate(III)]: First Report of Relevant Thioredoxin Reductase Inhibition for a Ruthenium Compound

scientific article published on 02 November 2007

Adjusting the DNA Interaction and Anticancer Activity of Pt(II) N-Heterocyclic Carbene Complexes by Steric Shielding of the Trans Leaving Group

scientific article published on 16 July 2015

An Organogold Compound as Potential Antimicrobial Agent against Drug-Resistant Bacteria: Initial Mechanistic Insights

scientific article published on 23 July 2021

Anticancer activity of new organo-ruthenium, rhodium and iridium complexes containing the 2-(pyridine-2-yl)thiazole N,N-chelating ligand

scholarly article by Michaël Gras et al published April 2010 in Journal of Organometallic Chemistry

Anticancer therapeutics that target selenoenzymes: synthesis, characterization, in vitro cytotoxicity, and thioredoxin reductase inhibition of a series of gold(I) complexes containing hydrophilic phosphine ligands

scientific article

Antimalarial properties of green tea.

scientific article published on 11 December 2006

Antiproliferative Activity of Gold(I) Alkyne Complexes Containing Water-Soluble Phosphane Ligands

Application of mass spectrometric techniques to delineate the modes-of-action of anticancer metallodrugs ⬇️

scientific article published on July 21, 2013

Aquaporin inhibition by gold(III) compounds: new insights

scientific article published on 7 May 2013

Aquaporins in cancer development: opportunities for bioinorganic chemistry to contribute novel chemical probes and therapeutic agents

scientific article

BODIPY-phosphane as a versatile tool for easy access to new metal-based theranostics.

scientific article

Bio-based and bio-inspired adhesives from animals and plants for biomedical applications

scientific article published on 13 January 2022

Bioconjugation of Supramolecular Metallacages to Integrin Ligands for Targeted Delivery of Cisplatin

scientific article published on 13 November 2018

Bioconjugation strategies to couple supramolecular exo-functionalized palladium cages to peptides for biomedical applications

scientific article published on 12 January 2017

Biophysical characterisation of adducts formed between anticancer metallodrugs and selected proteins: new insights from X-ray diffraction and mass spectrometry studies

scientific article published on 08 January 2008

Caffeine-based gold(I) N-heterocyclic carbenes as possible anticancer agents: synthesis and biological properties

scientific article published on 5 February 2014

Carbon-Phosphorus Coupling from C^N Cyclometalated AuIII Complexes

scientific article published on 06 March 2020

Carbonic Anhydrase Inhibitors: Synthesis and Inhibition of Cytosolic/Membrane-Associated Carbonic Anhydrase Isozymes I, II, and IX with Sulfonamides Incorporating Hydrazino Moieties

scientific article published on 01 March 2005

Carbonic Anhydrase Inhibitors: Water-Soluble 4-Sulfamoylphenylthioureas as Topical Intraocular Pressure-Lowering Agents with Long-Lasting Effects

scientific article published on 01 December 2000

Carbonic anhydrase activators. The selective serotonin reuptake inhibitors fluoxetine, sertraline and citalopram are strong activators of isozymes I and II.

scientific article published in August 2003

Carbonic anhydrase inhibitors

scientific article (publication date: March 2003)

Carbonic anhydrase inhibitors with strong topical antiglaucoma properties incorporating a 4-(2-aminopyrimidin-4-yl-amino)-benzenesulfonamide scaffold

scientific article published in February 2002

Carbonic anhydrase inhibitors. Inhibition of cytosolic isozyme XIII with aromatic and heterocyclic sulfonamides: a novel target for the drug design.

scientific article

Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors

scientific article published in May 2003

Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides

scientific article published in December 2004

Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.

scientific article

Carbonic anhydrase inhibitors: 4-sulfamoyl-benzenecarboxamides and 4-chloro-3-sulfamoyl-benzenecarboxamides with strong topical antiglaucoma properties

scientific article

Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX.

scientific article published in January 2004

Carbonic anhydrase inhibitors: Inhibition of the tumor-associated isozymes IX and XII with polyfluorinated aromatic/heterocyclic sulfonamides

scientific article published in June 2005

Carbonic anhydrase inhibitors: N-(p-sulfamoylphenyl)-alpha-D-glycopyranosylamines as topically acting antiglaucoma agents in hypertensive rabbits

scientific article published in January 2004

Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV.

scientific article

Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.

scientific article

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase

scientific article published in January 2004

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one?

scientific article published in August 2003

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a topically acting antiglaucoma sulfonamide

scientific article published in May 2004

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride

scientific article published in January 2004

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the perfluorobenzoyl analogue of methazolamide. Implications for the drug design of fluorinated inhibitors

scientific article published in August 2003

Carbonic anhydrase inhibitors: aliphatic N-phosphorylated sulfamates--a novel zinc-anchoring group leading to nanomolar inhibitors

scientific article published in June 2004

Carbonic anhydrase inhibitors: design of thioureido sulfonamides with potent isozyme II and XII inhibitory properties and intraocular pressure lowering activity in a rabbit model of glaucoma

scientific article published in September 2005

Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives

scientific article

Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates

scientific article

Carbonic anhydrase inhibitors: sulfonamides incorporating furan-, thiophene- and pyrrole-carboxamido groups possess strong topical intraocular pressure lowering properties as aqueous suspensions

scientific article published on 01 August 2000

Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity

scientific article

Carbonic anhydrase inhibitors: the first on-resin screening of a 4-sulfamoylphenylthiourea library

scientific article

Carbonic anhydrase inhibitors: the first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX.

scientific article published in February 2004

Carbonic anhydrase inhibitors: topically acting antiglaucoma sulfonamides incorporating esters and amides of 3- and 4-carboxybenzolamide

scientific article published in September 2003

Cellular transport mechanisms of cytotoxic metallodrugs: an overview beyond cisplatin.

scientific article published on 29 September 2014

Characterization of CA XIII, a novel member of the carbonic anhydrase isozyme family

scientific journal article

Characterization of Hydrophilic Gold(I) N-Heterocyclic Carbene (NHC) Complexes as Potent TrxR Inhibitors Using Biochemical and Mass Spectrometric Approaches

scientific article published on 2 November 2017

Chemistry, antiproliferative properties, tumor selectivity, and molecular mechanisms of novel gold(III) compounds for cancer treatment: a systematic study

scientific article

Clioquinol decreases amyloid-beta burden and reduces working memory impairment in a transgenic mouse model of Alzheimer's disease

scientific article

Conjugation of organoruthenium(II) 3-(1H-benzimidazol-2-yl)pyrazolo[3,4-b]pyridines and indolo[3,2-d]benzazepines to recombinant human serum albumin: a strategy to enhance cytotoxicity in cancer cells

scientific article published on 23 November 2011

Correlation between the Stereochemistry and Bioactivity in Octahedral Rhodium Prolinato Complexes

scientific article published on 7 August 2015

Cyclodextrin complexes of sulfonamide carbonic anhydrase inhibitors as long-lasting topically acting antiglaucoma agents

scientific article

Cyclometalated Au III Complexes for Cysteine Arylation in Zinc Finger Protein Domains: towards Controlled Reductive Elimination

scientific article published on 09 May 2019

Cytotoxic Profile and Peculiar Reactivity with Biomolecules of a Novel "Rule-Breaker" Iodidoplatinum(II) Complex

scientific article published on 21 July 2010

Cytotoxic gold compounds: synthesis, biological characterization and investigation of their inhibition properties of the zinc finger protein PARP-1.

scientific article published on 31 January 2012

Cytotoxic gold(I) N-heterocyclic carbene complexes with phosphane ligands as potent enzyme inhibitors

scientific article published on 26 March 2014

DNA as a possible target for antitumor ruthenium(III) complexes

scientific article

DOTAP/DOPE and DC-Chol/DOPE lipoplexes for gene delivery studied by circular dichroism and other biophysical techniques

article

Design Strategies and Medicinal Applications of Metal-Peptidic Bioconjugates

scientific article published on 03 April 2020

Designing of novel carbonic anhydrase inhibitors and activators.

scientific article

Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation

scientific article

Development of bimetallic titanocene-ruthenium-arene complexes as anticancer agents: relationships between structural and biological properties.

scientific article published on October 2010

ESI mass spectrometry and X-ray diffraction studies of adducts between anticancer platinum drugs and hen egg white lysozyme

scientific article

ESI–MS Characterisation of Protein Adducts of Anticancer Ruthenium(II)-Arene PTA (RAPTA) Complexes

scientific article published on 01 May 2007

Effects of two representative antitumor ruthenium(III) complexes on thermal denaturation profiles of DNA

scholarly article by L. Messori et al published May 2000 in Inorganica Chimica Acta

Emerging protein targets for anticancer metallodrugs: inhibition of thioredoxin reductase and cathepsin B by antitumor ruthenium(II)-arene compounds

scientific article published on 4 October 2008

Emerging protein targets for metal-based pharmaceutical agents: An update

article published in 2013

Evaluation of New Palladium Cages as Potential Delivery Systems for the Anticancer Drug Cisplatin

scientific article published on 12 January 2016

Ex vivo toxicological evaluation of experimental anticancer gold(i) complexes with lansoprazole-type ligands

scientific article published on 20 September 2019

Excellent correlation between cathepsin B inhibition and cytotoxicity for a series of palladacycles

scientific article

Exploiting soft and hard X-ray absorption spectroscopy to characterize metallodrug/protein interactions: the binding of [trans-RuCl4(Im)(dimethylsulfoxide)][ImH] (Im = imidazole) to bovine serum albumin

scientific article published on 23 August 2008

Exploring Metallodrug–Protein Interactions by ESI Mass Spectrometry: The Reaction of Anticancer Platinum Drugs with Horse Heart Cytochrome c

scholarly article by Angela Casini et al published 10 April 2006 in ChemMedChem

Exploring metallodrug-protein interactions by mass spectrometry: comparisons between platinum coordination complexes and an organometallic ruthenium compound

scientific article published on 14 March 2009

Exploring the gating mechanisms of aquaporin-3: new clues for the design of inhibitors?

scientific article published on 10 March 2016

Exploring the mechanisms of metalbased pharmacological agents via an integrated approach ⬇️

scientific article published on December 29, 2011

Exploring the potential of gold(III) cyclometallated compounds as cytotoxic agents: variations on the C^N theme.

scientific article published on 10 June 2015

Fluorescent silver(I) and gold(I)-N-heterocyclic carbene complexes with cytotoxic properties: mechanistic insights

scientific article published on August 2013

Formation of Supramolecular Structures between DNA and Starburst Dendrimers Studied by EPR, CD, UV, and Melting Profiles

Frontiers in radionuclide imaging and therapy, a chemical journey from naturally radioactive elements to targeted theranostic agents.

scientific article published on 23 October 2017

Functional inhibition of aquaporin-3 with a gold-based compound induces blockage of cell proliferation

scientific article published on November 2014

Gold Organometallics with Biological Properties

Gold compounds as anticancer agents: chemistry, cellular pharmacology, and preclinical studies

scientific article published on May 2010

Gold compounds as aquaporin inhibitors: new opportunities for therapy and imaging

Gold compounds for catalysis and metal-mediated transformations in biological systems

scientific article published on 18 February 2020

Gold finger formation studied by high-resolution mass spectrometry and in silico methods

scientific article published on 01 January 2015

Gold(I) N-heterocyclic carbene complexes with an “activable” ester moiety: Possible biological applications

Gold(I) NHC-based homo- and heterobimetallic complexes: synthesis, characterization and evaluation as potential anticancer agents

scientific article published on 23 July 2015

Gold(I) carbene complexes causing thioredoxin 1 and thioredoxin 2 oxidation as potential anticancer agents

scientific article published on 4 June 2012

Gold(III) Pyridine-Benzimidazole Complexes as Aquaglyceroporin Inhibitors and Antiproliferative Agents

article published in 2018

Gold(III) compounds as anticancer agents: relevance of gold-protein interactions for their mechanism of action

scientific article published on 28 November 2007

Gold(i) compounds with lansoprazole-type ligands: synthesis, characterization and anticancer properties in vitro

Hypoxia activates the capacity of tumor-associated carbonic anhydrase IX to acidify extracellular pH.

scientific article

Identifying and validating the presence of Guanine-Quadruplexes (G4) within the blood fluke parasite Schistosoma mansoni

scientific article published on 18 February 2021

Improved synthesis of N-benzylaminoferrocene-based prodrugs and evaluation of their toxicity and antileukemic activity

scientific article published on 9 February 2015

Influence of the π-coordinated arene on the anticancer activity of ruthenium(II) carbohydrate organometallic complexes

scientific article

Inhibition Mechanism of Urease by Au(III) Compounds Unveiled by X-ray Diffraction Analysis

Insights into the Mechanisms of Aquaporin-3 Inhibition by Gold(III) Complexes: the Importance of Non-Coordinative Adduct Formation

scientific article published on 15 January 2019

Insights into the Selectivity Mechanisms of Grapevine NIP Aquaporins

scientific article published on 13 September 2020

Insights into the molecular mechanisms of protein platination from a case study: the reaction of anticancer platinum(II) iminoethers with horse heart cytochrome c.

scientific article published on 9 October 2007

Insights into the strong in-vitro anticancer effects for bis(triphenylphosphane)iminium compounds having perchlorate, tetrafluoridoborate and bis(chlorido)argentate anions

scientific article published on 5 September 2015

Interactions of anticancer Pt compounds with proteins: an overlooked topic in medicinal inorganic chemistry?

scholarly article by Angela Casini & Jan Reedijk published 2012 in Chemical Science

Interactions of two cytotoxic organotin(IV) compounds with calf thymus DNA.

scientific article

Light-stable bis(norharmane)silver(I) compounds: synthesis, characterization and antiproliferative effects in cancer cells

scientific article

Luminescent iminophosphorane gold, palladium and platinum complexes as potential anticancer agents.

scientific article published on 07 March 2014

Mass Spectrometry Uncovers Molecular Reactivities of Coordination and Organometallic Gold(III) Drug Candidates in Competitive Experiments That Correlate with Their Biological Effects

scientific article published on 11 February 2016

Mass spectrometric analysis of ubiquitin–platinum interactions of leading anticancer drugs: MALDI versus ESI

article

Mechanistic studies on two dinuclear organogold(III) compounds showing appreciable antiproliferative properties and a high redox stability

scientific article

Metal-Based Inhibition of Poly(ADP-ribose) Polymerase − The Guardian Angel of DNA ⬇️

scientific article published on March 3, 2011

Molecular Basis of Aquaporin-7 Permeability Regulation by pH

scientific article published on 10 November 2018

Molecular Mechanisms and Proposed Targets for Selected Anticancer Gold Compounds ⬇️

scientific article published on January 1, 2011

Multinuclear cytotoxic metallodrugs: physicochemical characterization and biological properties of novel heteronuclear gold-titanium complexes

scientific article

Nanoformulations of a potent copper-based aquaporin inhibitor with cytotoxic effect against cancer cells

scientific article published on 7 July 2016

New Copper(II)/Cyclic Tetrapeptide System That Easily Oxidizes to Copper(III) under Atmospheric Oxygen

scientific article published on 03 November 2007

New Gold(I) Organometallic Compounds with Biological Activity in Cancer Cells

New Luminescent Polynuclear Metal Complexes with Anticancer Properties: Toward Structure-Activity Relationships

scientific article published on 11 February 2016

New Variations on the Theme of Gold(III) C∧N∧N Cyclometalated Complexes as Anticancer Agents: Synthesis and Biological Characterization

scientific article published on 20 November 2018

New heteronuclear gold(I)-platinum(II) complexes with cytotoxic properties: are two metals better than one?

scientific article published on 12 August 2014

New uses for old drugs. Auranofin, a clinically established antiarthritic metallodrug, exhibits potent antimalarial effects in vitro: Mechanistic and pharmacological implications

scientific article published on 21 February 2008

Next-Generation Anticancer Metallodrugs ⬇️

scientific article published on January 1, 2012

Nitrate as a probe of cytochrome c surface: crystallographic identification of crucial "hot spots" for protein-protein recognition

scientific article published on 11 March 2014

Nonconventionaltrans-Platinum Complexes Functionalized with RDG Peptides: Chemical and Cytototoxicity Studies

On the Mechanism of Gold/NHC Compounds Binding to DNA G-Quadruplexes: Combined Metadynamics and Biophysical Methods

On the binding modes of metal NHC complexes with DNA secondary structures: implications for therapy and imaging

scientific article published on 27 June 2017

On the toxicity and transport mechanisms of cisplatin in kidney tissues in comparison to a gold-based cytotoxic agent.

scientific article published on 6 November 2017

Organometallic Antitumour Agents with Alternative Modes of Action

Organometallic ruthenium(II) arene compounds with antiangiogenic activity

scientific article published on 16 May 2011

Organometallic ruthenium-based antitumor compounds with novel modes of action

Outstanding plasmodicidal properties within a small panel of metallic compounds: Hints for the development of new metal-based antimalarials

scientific article published on 17 October 2008

Peculiar mechanistic and structural features of the carboplatin-cytochrome c system revealed by ESI-MS analysis

scientific article

Potent in vitro antiproliferative properties for a triplatinum cluster toward triple negative breast cancer cells

scientific article published on 27 June 2016

Potential anticancer heterometallic Fe-Au and Fe-Pd agents: initial mechanistic insights

scientific article published on 02 July 2013

Potential pathogenic role of beta-amyloid(1-42)-aluminum complex in Alzheimer's disease

scientific article published on 22 October 2007

Protease inhibitors of the sulfonamide type: anticancer, antiinflammatory, and antiviral agents

scientific article

Proteins as possible targets for cytotoxic trans-platinum(II) complexes with aliphatic amine ligands: Further exceptions to the DNA paradigm

scientific article published on August 2010

Rationalization of the inhibition activity of structurally related organometallic compounds against the drug target cathepsin B by DFT.

scientific article published on 14 May 2010

Re(VII) and Tc(VII) trioxo complexes stabilized by tridentate ligands and their potential use as radiopharmaceuticals

Reactivity and biological properties of a series of cytotoxic PtI2(amine)2 complexes, either cis or trans configured

scientific article

Reactivity of Cys4 Zinc Finger Domains with Gold(III) Complexes: Insights into the Formation of “Gold Fingers”

scientific article published on 03 April 2015

Reactivity of an antimetastatic organometallic ruthenium compound with metallothionein-2: relevance to the mechanism of action

scientific article published on 11 August 2009

Reactivity of anticancer metallodrugs with serum proteins: new insights from size exclusion chromatography-ICP-MS and ESI-MS

scientific article

Ruthenium anticancer drugs and proteins: a study of the interactions of the ruthenium(III) complex imidazolium trans-[tetrachloro(dimethyl sulfoxide)(imidazole)ruthenate(III)] with hen egg white lysozyme and horse heart cytochrome c

scholarly article by Angela Casini et al published 7 August 2007 in Journal of Biological Inorganic Chemistry

Ruthenium(II) arene complexes with oligocationic triarylphosphine ligands: Synthesis, DNA interactions and in vitro properties

Selective targeting of PARP-1 zinc finger recognition domains with Au(iii) organometallics

scientific article published on 2 January 2018

Self-Assembled Palladium and Platinum Coordination Cages: Photophysical Studies and Anticancer Activity

Self-assembled M2L4 coordination cages: Synthesis and potential applications

Self-assembly of highly luminescent heteronuclear coordination cages

scientific article published in August 2016

Solution behaviour and biomolecular interactions of two cytotoxic trans-platinum(II) complexes bearing aliphatic amine ligands

scientific article

Stability of an organometallic ruthenium-ubiquitin adduct in the presence of glutathione: relevance to antitumour activity

scientific article published on 23 August 2008

Structural and solution chemistry, antiproliferative effects, and DNA and protein binding properties of a series of dinuclear gold(III) compounds with bipyridyl ligands

scientific article published on September 2006

Structural characterization, solution studies, and DFT calculations on a series of binuclear gold(III) oxo complexes: relationships to biological properties

scientific article

Structural investigation of cisplatin-protein interactions: selective platination of His19 in a cuprozinc superoxide dismutase

scientific article published in February 2006

Structure and biological activities of metal complexes of flumequine

scholarly article in RSC Advances, vol. 6 no. 23, 2016

Structure, solution chemistry, antiproliferative actions and protein binding properties of non-conventional platinum(II) compounds with sulfur and phosphorus donors

scientific article published on 6 January 2011

Sulfonamide derivatives with protease inhibitory action as anticancer, anti-inflammatory and antiviral agents

article published in 2002

Sulfonamides and sulfonylated derivatives as anticancer agents

scientific article

Supramolecular exo-functionalized palladium cages: fluorescent properties and biological activity

Synthesis, characterisation and biological properties of gold(III) compounds with modified bipyridine and bipyridylamine ligands

scientific article

Synthesis, molecular structure and solution chemistry of the iridium(III) complex imidazolium [trans(bisimidazole)tetrachloro iridate(III)] (IRIM)

scholarly article by P Mura et al published January 2001 in Inorganica Chimica Acta

Targeted imaging of integrins in cancer tissues using photocleavable Ru(ii) polypyridine complexes as mass-tags

scientific article published on 29 April 2020

Targeting aquaporin function: potent inhibition of aquaglyceroporin-3 by a gold-based compound

scientific article

The Promise of Self-Assembled 3D Supramolecular Coordination Complexes for Biomedical Applications

scientific article published on 27 November 2017

The formation of oxytocin dimers is suppressed by the zinc-aspartate-oxytocin complex

scientific article

The influence of auranofin, a clinically established antiarthritic gold drug, on bone metabolism: analysis of its effects on human multipotent adipose-derived stem cells, taken as a model

scientific article published in August 2008

The inhibition of glycerol permeation through aquaglyceroporin-3 induced by mercury(II): A molecular dynamics study

scientific article

The mechanism of aquaporin inhibition by gold compounds elucidated by biophysical and computational methods

scientific article

The molecular mechanisms of antimetastatic ruthenium compounds explored through DIGE proteomics

scientific article

The reaction of artemisinins with hemoglobin: a unified picture

scientific article published on 10 January 2006

The x-ray structure of the adduct between NAMI-A and carbonic anhydrase provides insights into the reactivity of this metallodrug with proteins

scientific article

Thiolato gold(I) complexes containing water-soluble phosphane ligands: a characterization of their chemical and biological properties.

scientific article

Thioredoxin reductase, an emerging target for anticancer metallodrugs. Enzyme inhibition by cytotoxic gold(iii) compounds studied with combined mass spectrometry and biochemical assays

Thioredoxin reductase: A target for gold compounds acting as potential anticancer drugs

Toward anticancer gold-based compounds targeting PARP-1: a new case study

scholarly article in RSC Advances, vol. 6 no. 82, 2016

Trace copper(II) or zinc(II) ions drastically modify the aggregation behavior of amyloid-beta1-42: an AFM study

scientific article

Trans-cis-cis-[RuCl2(DMSO)2(2-amino-5-methyl-thiazole)2], (PMRu52), a novel ruthenium(II) compound acting as a strong inhibitor of cathepsin B.

scientific article published on 9 October 2009

Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: new pharmacological opportunities due to related binding site recognition

scientific article

Unravelling the chemical nature of copper cuprizone

scientific article published on 11 April 2007

Unveiling the Mechanisms of Aquaglyceroporin-3 Water and Glycerol Permeation by Metadynamics

scientific article published on 03 June 2019

X-ray absorption spectroscopy studies of the adducts formed between cytotoxic gold compounds and two major serum proteins

scientific article published on 24 December 2010

[Au2(phen(2Me))2(μ-O)2](PF6)2, a Novel Dinuclear Gold(III) Complex Showing Excellent Antiproliferative Properties

scientific article published on 2 July 2010

fac-{Ru(CO)3}2+-core complexes and design of metal-based drugs. synthesis, structure, and reactivity of Ru-thiazole derivative with serum proteins and absorption-release studies with acryloyl and silica hydrogels as carriers in physiological media

scientific article published in January 2007

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