List of works - Daniele Castagnolo

A facile and regioselective multicomponent synthesis of chiral aryl-1,2-mercaptoamines in water followed by monoamine oxidase (MAO-N) enzymatic resolution

scientific article published on 04 October 2019

A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides

A mild and chemoselective CALB biocatalysed synthesis of sulfoxides exploiting the dual role of AcOEt as solvent and reagent

scientific article published on 12 November 2020

A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes

Antimicrobial drugs bearing guanidine moieties: A review

scientific article published in 2021

Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethylocta-2,6-dienyl)ethane-1,2-diamine (SQ109) Pyrrole Hybrid Derivatives: Discovery of Potent Antitu

scientific article published on 23 February 2016

Design, Synthesis and Discovery of N,N'-Carbazoyl-aryl-urea Inhibitors of Zika NS5 Methyltransferase and Virus Replication

scientific article published on 07 January 2020

Guanylated Diamines, Triamines, and Polyamines: Chemistry and Biological Properties ⬇️

scientific article published on 09 June 2011

Microwave-Assisted Domino Reactions of Propargylamines with Isothiocyanates: Selective Synthesis of 2-Aminothiazoles and 2-Amino-4-methylenethiazolines

Monoamine Oxidase (MAO-N) Whole Cell Biocatalyzed Aromatization of 1,2,5,6-Tetrahydropyridines into Pyridines

Novel Macrocyclic Amidinoureas: Potent Non-Azole Antifungals Active against Wild-Type and Resistant Candida Species

scientific article

Photo-biocatalytic one-pot cascades for the enantioselective synthesis of 1,3-mercaptoalkanol volatile sulfur compounds

scientific article published on 13 March 2018

Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents

scientific article published on 12 September 2015

Synthesis and Biological Evaluation of Amidinourea and Triazine Congeners as Inhibitors of MDA-MB-231 Human Breast Cancer Cell Proliferation.

scientific article published on 11 January 2017

Synthesis and Reactivity of Propargylamines in Organic Chemistry.

scientific article published on 22 November 2017

Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis