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List of works by Khondaker M. Rahman

A novel small-molecule inhibitor of IL-6 signalling.

scientific article

An overview of bacterial efflux pumps and computational approaches to study efflux pump inhibitors.

scientific article published on 29 January 2016

Antibiotic resistance breakers: current approaches and future directions

scientific article published on 01 September 2019

Antimicrobial molecules in the lung: formulation challenges and future directions for innovation

scientific article published on 23 February 2018

Antistaphylococcal activity of DNA-interactive pyrrolobenzodiazepine (PBD) dimers and PBD-biaryl conjugates.

scientific article

Author Correction: Mapping the Dynamic Functions and Structural Features of AcrB Efflux Pump Transporter Using Accelerated Molecular Dynamics Simulations

scientific article published on 28 November 2019

Author Correction: The Aurora B specificity switch is required to protect from non-disjunction at the metaphase/anaphase transition

scientific article published on 03 June 2020

Biaryl polyamides as a new class of DNA quadruplex-binding ligands.

scientific article

C8-Linked Pyrrolobenzodiazepine Monomers with Inverted Building Blocks Show Selective Activity against Multidrug Resistant Gram-Positive Bacteria

scientific article published on 20 December 2017

Computational Study Reveals the Molecular Mechanism of the Interaction between the Efflux Inhibitor PAβN and the AdeB Transporter from Acinetobacter baumannii.

scientific article published on 28 June 2017

Computational studies support the role of the C7-sibirosamine sugar of the pyrrolobenzodiazepine (PBD) sibiromycin in transcription factor inhibition

scientific article published on 11 August 2014

Covalent Bonding of Pyrrolobenzodiazepines (PBDs) to Terminal Guanine Residues within Duplex and Hairpin DNA Fragments

scientific article

Crispenes F and G, cis-Clerodane Furanoditerpenoids from Tinospora crispa, Inhibit STAT3 Dimerization

scientific article

Current Advances in Developing Inhibitors of Bacterial Multidrug Efflux Pumps

scientific article

Cytotoxic Naphthoquinone and Azaanthraquinone Derivatives from an Endophytic Fusarium solani

scientific article

Cytotoxicity and antibacterial activity of extractives from Wedelia calendulacea.

scientific article

DNA Sequence Preference and Adduct Orientation of Pyrrolo[2,1-c][1,4]benzodiazepine Antitumor Agents

scientific article

Diverse signalling of the platelet P2Y1 receptor leads to a dichotomy in platelet function

scientific article published on 11 March 2018

Effect of base sequence on the DNA cross-linking properties of pyrrolobenzodiazepine (PBD) dimers

scientific article published on 21 March 2011

Effect of hairpin loop structure on reactivity, sequence preference and adduct orientation of a DNA-interactive pyrrolo[2,1-c][1,4]benzodiazepine (PBD) antitumour agent

scientific article published on April 2015

Effect of microwave irradiation on covalent ligand-DNA interactions

scientific article

Effectiveness of Efflux Pump Inhibitors as Biofilm Disruptors and Resistance Breakers in Gram-Negative (ESKAPEE) Bacteria

scientific article published on 19 November 2019

Effects of Systematic Shortening of Noncovalent C8 Side Chain on the Cytotoxicity and NF-κB Inhibitory Capacity of Pyrrolobenzodiazepines (PBDs)

scientific article published on 13 February 2019

Evaluating the level of nitroreductase activity in clinical Klebsiella pneumoniae isolates to support strategies for nitro drug and prodrug development

scientific article published on 06 August 2019

Fluoxetine and thioridazine inhibit efflux and attenuate crystalline biofilm formation by Proteus mirabilis

scientific article published on 22 September 2017

From Anthramycin to Pyrrolobenzodiazepine (PBD)-Containing Antibody-Drug Conjugates (ADCs).

scientific article

Fusaproliferin, a Fungal Mycotoxin, Shows Cytotoxicity against Pancreatic Cancer Cell Lines

GC-targeted C8-linked pyrrolobenzodiazepine-biaryl conjugates with femtomolar in vitro cytotoxicity and in vivo antitumor activity in mouse models

scientific article published on 21 March 2013

Identification of novel telomeric G-quadruplex-targeting chemical scaffolds through screening of three NCI libraries

scientific article published on February 16, 2012

In Silico and in Vitro Screening for P-Glycoprotein Interaction with Tenofovir, Darunavir, and Dapivirine: An Antiretroviral Drug Combination for Topical Prevention of Colorectal HIV Transmission

scientific article published on 25 June 2017

Investigation of the protein alkylation sites of the STAT3:STAT3 inhibitor Stattic by mass spectrometry

scientific article published on 29 May 2013

Mapping the Dynamic Functions and Structural Features of AcrB Efflux Pump Transporter Using Accelerated Molecular Dynamics Simulations

scientific article published on 11 July 2018

Methylene-linked bis-phenylbenzimidazoles - a new scaffold to target telomeric DNA/RNA hybrid duplex

scientific article published on 2 March 2018

Noncytotoxic Pyrrolobenzodiazepine-Ciprofloxacin Conjugate with Activity against Mycobacterium tuberculosis

scientific article published on 03 December 2019

Novel 1-(2-aryl-2-adamantyl)piperazine derivatives with antiproliferative activity.

scientific article

Novel pyridyl nitrofuranyl isoxazolines show antibacterial activity against multiple drug resistant Staphylococcus species.

scientific article

Novel pyrrolobenzodiazepine benzofused hybrid molecules inhibit NF-κB activity and synergise with bortezomib and ibrutinib in hematological cancers

scientific article published on 07 May 2020

Observation of a dynamic equilibrium between DNA hairpin and duplex forms of covalent adducts of a minor groove binding agent.

scientific article

Observation of a single-stranded DNA/pyrrolobenzodiazepine adduct.

scientific article

Observation of the reversibility of a covalent pyrrolobenzodiazepine (PBD) DNA adduct by HPLC/MS and CD spectroscopy

scientific article published on 21 January 2011

Preliminary Cytotoxicity Screening of Some Medicinal Plants of Bangladesh

article

Pyrrolobenzodiazepines (PBDs) do not bind to DNA G-quadruplexes

scientific article

Recent advances in targeting the telomeric G-quadruplex DNA sequence with small molecules as a strategy for anticancer therapies

scientific article published on 21 July 2016

Role of bacterial efflux pumps in biofilm formation

scientific article published on 28 February 2018

Schiff bases of sulphonamides as a new class of antifungal agent against multidrug-resistant Candida auris

scientific article published on 01 August 2021

Sequence-selective binding of C8-conjugated pyrrolobenzodiazepines (PBDs) to DNA.

scientific article published in September 2017

SmvA is an important efflux pump for cationic biocides in Klebsiella pneumoniae and other Enterobacteriaceae

scientific article published in Scientific Reports

Stereochenols A and B, two quinones from Stereospermum chelonoides

scientific article published on 06 October 2006

Synthesis, pharmacological evaluation and docking studies of progesterone and testosterone derivatives as anticancer agents

scientific article published on 18 May 2018

The Aurora B specificity switch is required to protect from non-disjunction at the metaphase/anaphase transition

scientific article published on 13 March 2020

The minor groove-binding agent ELB-21 forms multiple interstrand and intrastrand covalent cross-links with duplex DNA and displays potent bactericidal activity against methicillin-resistant Staphylococcus aureus

scientific article

The prenylated dioxopiperazine alkaloid Cristatin A has selective telomeric DNA G-quadruplex stabilising properties

scientific article

The pyrrolobenzodiazepine dimer SJG-136 forms sequence-dependent intrastrand DNA cross-links and monoalkylated adducts in addition to interstrand cross-links.

scientific article

The use of molecular dynamics simulations to evaluate the DNA sequence-selectivity of G-A cross-linking PBD-duocarmycin dimers

scientific article published on 12 October 2016

Topical delivery of anthramycin I. Influence of neat solvents

scientific article

Topical delivery of anthramycin II. Influence of binary and ternary solvent systems

scientific article published on 07 May 2018

Topical therapies for skin cancer and actinic keratosis

scientific article published on 16 June 2015

Towards identifying the mode of action of drugs using live-cell FTIR spectroscopy

scientific article published on 01 April 2019

Triaryl Benzimidazoles as a New Class of Antibacterial Agents against Resistant Pathogenic Microorganisms.

scientific article published on 26 June 2017