(E,E)-10-(1,3-Dihydro-4,6-dihydroxy-7-methyl-3-oxoisobenzofuran-5-yl)4,8-dimethyldeca-4,8-dienoic acid: total synthesis and role in mycophenolic acid biosynthesis

1,4-addition to α,β-unsaturated carbonyl compounds bearing a γ-stereocenter: A molecular mechanics model for steric interactions in the transition state

article

1-t-Butylthio-1-t-butyldimethylsilyloxyethylene

1-t-Butylthio-1-t-butyldimethylsilyloxypropene

1-t-Butylthio-1-t-butyldimethylsilyloxypropene

1-tert-Butylthio-1-tert-butyldimethylsilyloxyethylene

2,3-Dihydroxybenzoate pathway in Pseudomonas putida. 1H n.m.r. study on the ring-cleavage site

scientific article published on February 1981

2-Benzoylamino-2-deoxy-2-hydroxymethyl-D-hexono-1,4-lactones: synthesis from D-fructose and utilization in the total synthesis of thermozymocidin (myriocin)

article

6-Farnesyl-5,7-dihydroxy-4-methylphthalide oxidation mechanism in mycophenolic acid biosynthesis

article

A Catalytic and Enantioselective Desymmetrization of meso Cyclic Allylic Bisdiethylphosphates with Organozinc Reagents

A Catalytic and Enantioselective Desymmetrization of meso Cyclic Allylic Bisdiethylphosphates with Organozinc Reagents

scholarly article by Umberto Piarulli et al published 13 January 2003 in Angewandte Chemie International Edition

A Formal Total Synthesis of Eleutherobin (IV) Using the Ring-Closing Metathesis (RCM) Reaction of a Densely Functionalized Diene as the Key Step: Investigation of the Unusual Kinetically Controlled RCM Stereochemistry

A Formal Total Synthesis of Eleutherobin Through an Unprecedented Kinetically Controlled Ring-Closing Metathesis Reaction of a Densely Functionalized Diene

A Formal Total Synthesis of Eleutherobin Through an Unprecedented Kinetically Controlled Ring-Closing-Metathesis Reaction of a Densely Functionalized Diene

scholarly article by Damiano Castoldi et al published 14 January 2005 in Angewandte Chemie International Edition

A Highly Stereoselective Total Synthesis of (+)-9-epi-Dictyostatin

A Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts

scholarly article by Marc Renom-Carrasco et al published 12 July 2016 in Advanced Synthesis & Catalysis

A Modular Approach to a New Class of Monodentate Chiral Phosphorus Ligands and Their Application in Enantioselective Copper-Catalysed Conjugate Additions of Diethylzinc to Cyclohexenone

article

A Practical Synthesis of the C1-C9 Fragment of Dictyostatin

A carbonylative cross-coupling strategy to the total synthesis of the sarcodictyins: preliminary studies and synthesis of a cyclization precursor

A computational study of the 1,4-addition of lithium enolates to conjugated carbonyl compounds

A computational study of the 1,4-addition of lithium enolates to conjugated carbonyl compounds

A dimeric bicyclic RGD ligand displays enhanced integrin binding affinity and strong biological effects on U-373 MG glioblastoma cells

scientific article published on 26 September 2019

A formal total synthesis of eleutherobin using the ring-closing metathesis (RCM) reaction of a densely functionalized diene as the key step: investigation of the unusual kinetically controlled RCM stereochemistry.

scientific article published in December 2005

A highly enantio- and diastereoselective aldol reaction for α-heterosubstituted thioacetates

A highly stereoselective synthesis of the C10–C23 fragment of (–)-dictyostatin

scientific article published on 01 November 2007

A library approach to the development of BenzaPhos: highly efficient chiral supramolecular ligands for asymmetric hydrogenation

scientific article

A new method for the solution and solid phase synthesis of chiral β-sulfonopeptides under mild conditions

article

A practical approach to the resolution of racemic N-benzyl alpha-amino acids by liquid-liquid extraction with a lipophilic chiral salen-cobalt(III) complex

scientific article published in April 2006

A straightforward total synthesis of (-)-chaetominine.

scientific article published in August 2009

A trifunctional steroid-based scaffold for combinatorial chemistry

article

Acceleration of hemiacetal cleavage through hydrogen bonding: a new synthetic catalyst with balanced conformational flexibility and preorganization

Acetogenin synthesis. Organocopper reagents, anions of 1,3-dithians and of protected cyanohydrins as intermediates in ketide side-chain synthesis

Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source

scholarly article by Marc Renom-Carrasco et al published 6 July 2015 in Advanced Synthesis & Catalysis

Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts

scientific article published on 03 June 2016

Asymmetric Synthesis with Enol Ethers

Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process

Asymmetric synthesis of functionalized α -amino-β-hydroxy acids via chiral norephedrine-derived oxazolidines

Asymmetric synthesis of trans- β -lactams through TiCl4-mediated addition to imines

article

Auxiliary structure and asymmetric induction in the “Mukaiyama-aldol” reactions of chiral silyl ketene acetals

Bicyclic carbohydrate-derived scaffolds for combinatorial libraries

scientific article

Bifunctional 2,5-Diketopiperazines as Efficient Organocatalysts for the Enantioselective Conjugate Addition of Aldehydes to Nitroolefins

article

Bifunctional 2,5-Diketopiperazines as Rigid Three-Dimensional Scaffolds in Receptors and Peptidomimetics

article

Biosynthesis of ascochitine and synthesis of its biogenetic precursors

article published in 1980

Biosynthesis of ascochitine: incorporation studies with advanced precursors

Biosynthesis of austdiol and synthesis of a deuterium labelled biogenetic precursor

Biosynthesis of citrinin

Biosynthesis of citrinin and synthesis of its biogenetic precursors

Biosynthesis of cochlioquinones

Biosynthesis of cochlioquinones

Biosynthesis of mycophenolic acid. Oxidation of 6-farnesyl-5,7-dihydroxy-4-methylphthalide in a cell-free preparation from Penicillium brevicompactum

article published in 1978

Biosynthetic origin and revised structure of ascochitine, a phytotoxic fungal metabolite. Incorporation of [1-13C]- and [1,2-13C2]-acetates and [Me-13C]methionine

Boron aldol reaction of α-halosubstitued thioacetates with silyl imines: A highly enantio- and diastereoselective synthesis of aziridines

CONFORMATIONAL CONTROL IN NATURAL PRODUCTS SYNTHESIS

Chelation controlled aldol additions of the enolsilane derived from tert-butyl thioacetate : a stereosetective approach to 1β-methylthienamycin

article

Chelation-controlled enantioselective synthesis of key intermediates for the preparation of carbapenem antibiotics PS-5 and 1.beta.-methyl-PS-5

ChemInform Abstract: A Carbonylative Cross-Coupling Strategy to the Total Synthesis of the Sarcodictyins: Preliminary Studies and Synthesis of a Cyclization Precursor

ChemInform Abstract: A Highly Stereoselective Synthesis of the C10—C23 Fragment of (-)-Dictyostatin

ChemInform Abstract: Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source

ChemInform Abstract: Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs′ Metathesis Catalysts: On the Way to a Tandem Process

ChemInform Abstract: Bifunctional 2,5-Diketopiperazines as Efficient Organocatalysts for the Enantioselective Conjugate Addition of Aldehydes to Nitroolefins

article

ChemInform Abstract: Bifunctional 2,5-Diketopiperazines as Rigid Three-Dimensional Scaffolds in Receptors and Peptidomimetics

ChemInform Abstract: Chiral (Cyclopentadienone)iron Complexes for the Catalytic Asymmetric Hydrogenation of Ketones

ChemInform Abstract: Combination of a Binaphthol-Derived Phosphite and a C1-Symmetric Phosphinamine Generates Heteroleptic Catalysts in Rh- and Pd-Mediated Reactions

ChemInform Abstract: Computer-Assisted Design and Synthetic Applications of Chiral Enol Borinates: Novel, Highly Enantioselective Aldol Reagents

ChemInform Abstract: Conformational Preferences of Peptides Containing Reverse-Turn Mimetic Bicyclic Lactams: Inverse γ-Turns versus Type-II′ β-Turns - Insights into β-Hairpin Stability

ChemInform Abstract: Discovery of a New Efficient Chiral Ligand for Copper-Catalyzed Enantioselective Michael Additions by High-Throughput Screening of a Parallel Library

ChemInform Abstract: Discovery of a New Efficient Chiral Ligand for Copper-Catalyzed Enantioselective Michael Additions by High-Throughput Screening of a Parallel Library

ChemInform Abstract: Effect of Ligands and Additives on the Palladium-Promoted Carbonylative Coupling of Vinyl Stannanes and Electron-Poor Enol Triflates

ChemInform Abstract: Enantioselective Rh-Catalyzed Addition of Arylboronic Acids to N-Tosylarylimines

article

ChemInform Abstract: Enantioselective Synthesis of 1-Vinyltetrahydroisoquinolines Through Palladium-Catalyzed Intramolecular Allylic Amidation with Chiral PhthalaPhos Ligands

ChemInform Abstract: Natural Products with Taxol-like Antitumor Activity

ChemInform Abstract: Optimization of New Chiral Ligands for the Copper-Catalyzed Enantioselective Conjugate Addition of Et2Zn to Nitroolefins by High-Throughput Screening of a Parallel Library

article

ChemInform Abstract: Synthesis of (R)-BINOL-Derived (Cyclopentadienone)Iron Complexes and Their Application in the Catalytic Asymmetric Hydrogenation of Ketones

ChemInform Abstract: Synthesis of a 4-Vinyltetrahydrocarbazole by Palladium-Catalyzed Asymmetric Allylic Alkylation of Indole-Containing Allylic Carbonates

ChemInform Abstract: Synthetic Studies on Sarcodictyins and Eleutherobin: Synthesis of Fully Functionalized Cyclization Precursors

ChemInform Abstract: Ureas: New Efficient Lewis Base Catalysts for the Allylation of Aldehydes

Chiral (Cyclopentadienone)iron Complexes for the Catalytic Asymmetric Hydrogenation of Ketones

article published in 2015

Chiral (salen)Co(III)(N-benzyl-l-serine)-derived phosphites: monodentate P-ligands for enantioselective catalytic applications

Chiral Formyl-Group Equivalents: Conjugate Addition to α,β-Unsaturated Ketones

article

Chiral acyl anion and enolonium ion equivalents. Asymmetric synthesis of α-methoxy-aldehydes

Chiral acyl anion equivalents: asymmetric synthesis of 11-deoxy-ent-prostaglandin intermediates

Chiral acyl anion equivalents: asymmetric synthesis of α-methoxytolualdehyde

Chiral α-sulphinyl hydrazones as effective reagents for stereoselective aldol-type condensation

Combination of a binaphthol-derived phosphite and a C1-symmetric phosphinamine generates heteroleptic catalysts in Rh- and Pd-mediated reactions

scientific article published on 21 May 2009

Combinations of Acidic and Basic Monodentate Binaphtholic Phosphites as Supramolecular Bidentate Ligands for Enantioselective Rh-Catalyzed Hydrogenations

Combinatorial Libraries of Chiral Ligands for Enantioselective Catalysis

Combinatorial Libraries of Chiral Ligands for Enantioselective Catalysis

scientific article published on 01 August 2003

Combinatorial Libraries: Studies in Molecular Recognition and the Quest for New Catalysts

article published in 1997

Computational studies on the aldol-type addition of boron enolates to imines: An ab-initio approach

article

Computer-Assisted Design and Synthetic Applications of Chiral Enol Borinates: Novel, Highly Enantioselective Aldol Reagents

article published in 1998

Computer-Assisted Design of Chiral Boron Enolates: A Novel, Highly Enantioselective Aldol Reaction for Thioacetates and Thiopropionates

scholarly article by Cesare Gennari et al published November 1993 in Angewandte Chemie International Edition

Computer-assisted design of chiral boron enolates: The role of ate complexes in determining aldol stereoselectivity

Computerunterstütztes Design von chiralen Borenolaten: Eine neue, hoch enantioselektive Aldolreaktion für Thioacetate und Thiopropionate

Computerunterstütztes Design von chiralen Borenolaten: eine neue, hoch enantioselektive Aldolreaktion für Thioacetate und Thiopropionate

Conformational Preferences of Peptides Containing Reverse-Turn Mimetic Bicyclic Lactams: Inverse γ-Turns versus Type-II′ β-Turns – Insights into β-Hairpin Stability

article published in 1999

Conformational Studies of Chiral Vinylogous Sulfonamidopeptides

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

scientific article published on 07 June 2019

Copper Phosphoramidite-Catalyzed Enantioselective Desymmetrization of meso-Cyclic Allylic Bisdiethyl Phosphates

Copper Phosphoramidite-Catalyzed Enantioselective Desymmetrization ofmeso-Cyclic Allylic Bisdiethyl Phosphates

scientific article published in 2003

Copper catalysed 1,4-addition of organozinc reagents to α,β-unsaturated carbonyl compounds: a mechanistic investigation

article

Copper-Catalysed, Enantioselective Desymmetrisation ofmeso Cyclic Allylic Bis(diethyl phosphates) with Organozinc Reagents

Copper-Catalyzed, Enantioselective Desymmetrization of meso Cyclic Allylic Bis(diethyl phosphates) with Organozinc Reagents

Cyclative cleavage via solid-phase supported stabilized sulfur ylides: synthesis of macrocyclic lactones

Cyclic RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands

Cyclic RGD-peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands.

scientific article published in November 2009

Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists.

scientific article

Cyclic isoDGR peptidomimetics as low-nanomolar αvβ3 integrin ligands.

scientific article published on 19 February 2013

Detection of one symmetrical precursor during the biosynthesis of the fungal metabolite austdiol using [1,2-13C2]acetate and [Me-13C]methionine

article

Determination of the binding epitope of RGD-peptidomimetics to αvβ3 and α(IIb)β3 integrin-rich intact cells by NMR and computational studies.

scientific article published on June 2013

Developing a force field for the transition state of the aldol reaction of enolborinates: Evaluation of the use of fixed point charges

Diastereofacial selectivity in the aldol reactions of chiral α-methyl aldehydes: a computer modelling approach

Direct synthesis of Z-unsaturated esters. A useful modification of the horner-emmons olefination

Discovery of a New Efficient Chiral Ligand for Copper-Catalyzed Enantioselective Michael Additions by High-Throughput Screening of a Parallel Library

article

Discovery of a new efficient chiral ligand for copper-catalyzed enantioselective Michael additions by high-throughput screening of a parallel library.

scientific article

Effect of Ligands and Additives on the Palladium-Promoted Carbonylative Coupling of Vinyl Stannanes and Electron-Poor Enol Triflates

article

Effects of Allylic and Homoallylic Substituents on the Ring Closing Metathesis Reaction Used to Synthesise Simplified Eleuthesides

Effects of allylic and homoallylic substituents on the ring closing metathesis reaction used to synthesise simplified eleuthesides

Efficient resolution of racemic N-benzyl beta3-amino acids by iterative liquid-liquid extraction with a chiral (salen)cobalt(III) complex as enantioselective selector.

scientific article

Enantioselective Conjugate Addition of Phenylboronic Acid to Enones Catalyzed by a Chiral Tropos/Atropos Rhodium Complex at the Coalescence Temperature

article

Enantioselective Cyanosilylation of Aldehydes Catalyzed by a Diastereomeric Mixture of Atropisomeric Thioureas

Enantioselective Rh-Catalyzed Addition of Arylboronic Acids to N-Tosylarylimines

article

Enantioselective Synthesis of (-)-(R)-5-Hydroxy-1-(4-hydroxy-3-methoxyphenyl)-3-decanone [(-)-(R)-[6]-Gingerol]

Enantioselective binding of dipeptides using acyclic receptors

article published in 2001

Enantioselective conjugate addition of phenylboronic acid to enones catalysed by a chiral tropos/atropos rhodium complex at the coalescence temperature

scientific article published on 21 September 2005

Enantioselective cyanosilylation of aldehydes catalysed by a diastereomeric mixture of atropisomeric thioureas

Enantioselective synthesis of 1-vinyltetrahydroisoquinolines through palladium-catalysed intramolecular allylic amidation with chiral PhthalaPhos ligands

scholarly article by Luca Pignataro et al published May 2014 in Tetrahedron: Asymmetry

Enantioselective synthesis of anti-.alpha.-methyl-.beta.-hydroxy esters through titanium tetrachloride-mediated aldol condensation

scholarly article by Cesare Gennari et al published October 1985 in Journal of the American Chemical Society

Entdeckung eines effizienten chiralen Liganden für die Cu-katalysierte enantioselektive Michael-Addition durch High-Throughput-Screening einer Parallelbibliothek

article

Ethylene Chloroboronate

Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols

article

Fast Cyclization of a Proline-Derived Self-Immolative Spacer Improves the Efficacy of Carbamate Prodrugs

scientific article published on 22 January 2020

Festphasensynthese von vinylogen Sulfonylpeptiden

Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αV β3

High diastereoface selection in an ester enolate addition to .alpha.-alkoxy aldehydes: stereoselective synthesis of .alpha.-methylene-.beta.-hydroxy-.gamma.-alkoxy esters

article

High diastereoselectivity in lewis acid mediated aldol condensations using thioester silyl ketene acetals

Highly Stereoselective Total Synthesis of (+)-9-epi-Dictyostatin and (-)-12,13-Bis-epi-dictyostatin

Highly enantio- and diastereoselective boron aldol reactions of α-heterosubstituted thioacetates with aldehydes and silyl imines

Highly enantioselective Rh-catalyzed hydrogenations with heterocombinations of pentafluorobenzyl- and methoxybenzyl-derived binaphthyl phosphites

Hydrogen-Bonding Donor/Acceptor Scales inβ-Sulfonamidopeptides

Improved enantioselective synthesis of anti α-methyl-β-hydroxyesters through TiCl4-PPh3 mediated aldol condensation

Improving C=N Bond Reductions with (Cyclopentadienone)iron Complexes: Scope and Limitations

Innovative Linker Strategies for Tumor-Targeted Drug Conjugates

scientific article published on 20 September 2019

Inside Cover: Cyclic RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands (Chem. Eur. J. 20/2012)

Inside Cover: Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols (ChemCatChem 22/2016)

scholarly article by Piotr Gajewski et al published 22 November 2016 in ChemCatChem

Insights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live-Cell NMR And Computational Studies

scientific article

Investigating the Interaction of Cyclic RGD Peptidomimetics with αVβ₆ Integrin by Biochemical and Molecular Docking Studies

scientific article published on 21 September 2017

Investigation of a New Family of Chiral Ligands for Enantioselective Catalysis via Parallel Synthesis and High-Throughput Screening

Ketenetert-Butyldimethylsilyl Methyl Acetal

Ketenetert-Butyldimethylsilyl Methyl Acetal

Lewis acid mediated aldol condensations using thioester silyl ketene acetals

Lewis acid promoted aldol additions of α-thiosilylketeneacetals to α-alkoxy aldehydes: diastereoselective synthesis of -α-methylene-β-hydroxy-∂-alkoxy esters

article

Mechanistic insights from ab initio calculations on a nitrogen analogue of the boron-mediated aldol reaction

Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake

scientific article published on 30 March 2020

Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αV β3.

scientific article published on 17 August 2017

Natural Products with Taxol-like Antitumor Activity — Synthetic Approaches to the Sarcodictyins and Eleutherobin

Natural products with taxol-like anti-tumor activity: Synthetic approaches to eleutherobin and dictyostatin

article published in 2007

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

scientific article published on 27 December 2018

Novel reverse-turn mimics inhibit farnesyl transferase

scientific article published on 01 March 1999

Optimization of New Chiral Ligands for the Copper-Catalysed Enantioselective Conjugate Addition of Et2Zn to Nitroolefins by High-Throughput Screening of a Parallel Library

article

Origins of stereoselectivity in chiral boron enolate aldol reactions: A computational study using transition state modellings

Origins of stereoselectivity in the addition of allyl- and crotylboronates to aldehydes : the development and application of a force field model of the transition state

article

Origins of stereoselectivity in the addition of allyl- and crotylboronates to aldehydes: The development and application of a force field model of the transition state

article

Origins of stereoselectivity in the addition of chiral allyl- and crotylboranes to aldehydes: the development and application of a force field model of the transition state

article

Origins of π-face selectivity in the aldol reactions of chiral E-enol borinates: a computational study using transition state modelling

Peptide bond formation using an enzyme mimicking approach

Peptide bond formation using an enzyme mimicking approach

PhthalaPhos: Chiral Supramolecular Ligands for Enantioselective Rhodium-Catalyzed Hydrogenation Reactions

scientific article published on 01 September 2010

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

scientific article published on 29 March 2019

Rationally Designed Bicyclic Lactams Control Different Turn Motifs and Folding Patterns in Hexapeptide Mimics

Rationally designed chiral enol borinates: Powerful reagents for the stereoselective synthesis of natural products

Reagent Control in the Aldol Addition Reaction of Chiral Boron Enolates with Chiral .alpha.-Amino Aldehydes. Total Synthesis of (3S,4S)-Statine

article

Reagent control in the aldol addition reaction of chiral boron enolates with chiral aldehydes

article

Reagent control in the aldol addition reaction of chiral boron enolates with chiral aldehydes. Total synthesis of (3S,4S)-Statine

article

Resolution of RacemicN-Benzyl α-Amino Acids by Liquid-Liquid Extraction: A Practical Method Using a Lipophilic Chiral Cobalt(III) Salen Complex and Mechanistic Studies

scholarly article by Pawel Dzygiel et al published March 2008 in European Journal of Organic Chemistry

Rh-Catalyzed Asymmetric Hydrogenation of Prochiral Olefins with a Dynamic Library of Chiral TROPOS Phosphorus Ligands

Rh-catalysed asymmetric hydrogenations with a dynamic library of chiral tropos phosphorus-ligands

Rh-catalyzed asymmetric hydrogenation of prochiral olefins with a dynamic library of chiral TROPOS phosphorus ligands

scientific article

Rh-catalyzed enantioselective conjugate addition of arylboronic acids with a dynamic library of chiral tropos phosphorus ligands

scientific article

Rhodium-Catalyzed Asymmetric Reactions with a Dynamic Library of Chiral Tropos Phosphorus Ligands

scholarly article by Cesare Gennari et al published 25 July 2006 in ChemInform

Rhodium-catalyzed asymmetric hydrogenation of olefins with PhthalaPhos, a new class of chiral supramolecular ligands

scientific article

Rhodium-catalyzed asymmetric reactions with a dynamic library of chiral tropos phosphorus ligands

scholarly article by Cesare Gennari et al published 1 January 2006 in Pure and Applied Chemistry

Riding the Wave of Monodentate Ligand Revival: From the A/B Concept to Noncovalent Interactions

scientific article published on 18 July 2016

Selective O-acylation of unprotected N-benzylserine methyl ester and O,N-acyl transfer in the formation of cyclo[Asp-Ser] diketopiperazines

article

Semisynthese von Taxol: eine hochenantio- und -diastereoselektive Synthese der Seitenkette und eine neue Methode zur Esterbildung an C13 unter Verwendung von Thioestern

Semisynthesis of Taxol: A Highly Enantio- and Diastereoselective Synthesis of the Side Chain and a New Method for Ester Formation at C13 Using Thioesters

Solid-Phase Synthesis of Peptides Containing Reverse-Turn Mimetic Bicyclic Lactams

Solid-Phase Synthesis of Vinylogous Sulfonyl Peptides

Stereocontrolled synthesis of polyketide libraries: Boron-mediated aldol reactions with aldehydes on solid support

article

Stereoselective aldol additions to α-alkoxy aldehydes using thioester silyl ketene acetals,

article

Stereoselective aldol condensations via alkenyloxy dialkoxyboranes : mechanistic and stereochemical details

Stereoselective aldol condensations via alkenyloxy dialkoxyboranes: synthetic applications using thioesters

Stereoselective aldol condensations via enolboronates

Stereoselective aldol reactions of γ-thiobutyrolactone: The benzaldehyde anomaly

Stereoselective aldol reactions using ticl4 as stereochemical template

Stereoselective radical-mediated cyclization of norephdrine derived α-iodoamides: synthesis of enantiopure pyrrolidines and trandition state modelling1

Stereoselective radical-mediated cyclization of norephedrine derived o-bromobenzamides: Enantioselective synthesis of 4-substituted 1,2,3,4-tetrahydroisoquinolines

article published in 1993

Stereoselective radical-mediated cyclization of norephedrine derived α-iodoamides: Experiments and TS-modelling

Stereoselective synthesis of α-methylene-β-hydroxy-γ-alkoxy esters from α-alkoxy aldehydes

Stereoselectivity in (Z)-Vinylmetal Additions to the Dictyostatin C1-C9 β-Silyloxy Aldehyde

article

Stereoselectivity of intramolecular nitrile oxide cycloadditions to Z and E chiral alkenes

Stereospecific Synthesis of Chiral α-Sulfinylhydrazones

Supramolecular ligand-ligand and ligand-substrate interactions for highly selective transition metal catalysis.

scientific article

Synthese von Sulfonamid-Pseudopeptiden: neue chirale synthetische Oligomere

article

Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αV β3 -Integrin Ligands for Tumor Targeting

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin αV β3

scientific article published on 22 March 2019

Synthesis and Screening of New Chiral Ligands for the Copper-Catalysed Enantioselective Allylic Substitution

scholarly article by Sandrine Ongeri et al published October 2002 in Helvetica Chimica Acta

Synthesis and Screening of New Chiral Ligands for the Copper-Catalyzed Enantioselective Allylic Substitution

Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine-glycine-aspartate (RGD) peptidomimetic-paclitaxel conjugates targeting integrin αVβ3.

scientific article

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting.

scientific article

Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers

scientific article

Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting α(v)β(3)/α(v)β(5) integrins and IAP proteins.

scientific article published on 16 April 2014

Synthesis and conformational studies of peptidomimetics containing a new bifunctional diketopiperazine scaffold acting as a beta-hairpin inducer.

scientific article published on 13 December 2007

Synthesis of (R)-BINOL-Derived (Cyclopentadienone)iron Complexes and Their Application in the Catalytic Asymmetric Hydrogenation of Ketones

Synthesis of Chiral Vinylogous Sulfonamidopeptides (vs-Peptides)

Synthesis of Combinatorial Libraries of Vinylogous Sulfonamidopeptides (vs-Peptides)

Synthesis of Sulfonamido-Pseudopeptides: New Chiral Unnatural Oligomers

scholarly article by Cesare Gennari et al published 2 November 1994 in Angewandte Chemie International Edition

Synthesis of [Bis(hexamethylene)cyclopentadienone]iron Tricarbonyl and its Application to the Catalytic Reduction of C=O Bonds

scholarly article by Sofia Vailati Facchini et al published 28 March 2017 in ChemCatChem

Synthesis of a 4-Vinyltetrahydrocarbazole by Palladium-Catalyzed Asymmetric Allylic Alkylation of Indole-Containing Allylic Carbonates

article

Synthesis of a simplified sarcodictyin analogue which retains microtubule stabilising properties

article

Synthesis of novel simplified eleutheside analogues with potent microtubule-stabilizing activity, using ring-closing metathesis as the key-step

Synthesis of novel simplified sarcodictyin/eleutherobin analogs with potent microtubule-stabilizing activity, using ring closing metathesis as the key-step

article

Synthesis of novel, simplified, C-7 substituted eleutheside analogues with potent microtubule-stabilizing activity

article published in 2005

Synthesis of tertiary acyloins using acyl anions formed from 1,3-dithians. Total synthesis of (±)-(2E)-1,7-dihydroxy-3,7,11-trimethyl-dodeca-2,10-dien-6-one

Synthesis of the C15–C23 fragment of dictyostatin using a highly stereoselective Carreira alkynylation

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors

scientific article

Synthesis, Conformational Studies and Binding Properties of Acyclic Receptors for N-Protected Amino Acids and Dipeptides

article

Synthetic Receptors Based on Vinylogous Sulfonyl Peptides

Synthetic opportunities offered by anti .alpha.-methylene-.beta.-hydroxy-.gamma.-alkoxy esters: stereoselective reactions at the double bond

Synthetic studies on sarcodictyins and eleutherobin: Synthesis of fully functionalized cyclization precursors

Synthetic studies on the sarcodictyins: synthesis of fully functionalized cyclization precursors

Synthetische Rezeptoren aus vinylogen Sulfonylpeptiden

Taxol Semisynthesis: A Highly Enantio- and Diastereoselective Synthesis of the Side Chain and a New Method for Ester Formation at C-13 Using Thioesters

The Importance of Detail: How Differences in Ligand Structures Determine Distinct Functional Responses in Integrin α v β 3

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The Italian Chemical Society Is 100 Years Old (Eur. J. Org. Chem. 18/2009)

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The Italian Chemical Society Is 100 Years Old (Eur. J. Org. Chem. 19/2009)

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The rational design and systematic analysis of asymmetric aldol reactions using enol borinates: Applications of transition state computer modelling

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The rational design of highly stereoselective boron enolates using transition-state computer modeling: a novel, asymmetric anti aldol reaction for ketones

Theoretical studies of stereoselective aldol condensations

TiCl4-mediated reactions of silyl ketene acetals derived from n-methylephedrine esters:asymmetric synthesis ofβ-lactams

Titanium chloride-mediated reactions of the silyl ketene acetals derived from N-methylephedrine esters: an asymmetric variant of the Mukaiyama reaction

scholarly article by Cesare Gennari et al published June 1987 in Journal of Organic Chemistry

Titanium tetrachloride-mediated enantioselective synthesis of trans β-lactones

scholarly article by Silvia Cardani et al published July 1992 in Tetrahedron

Total Synthesis of (+)-7,11-Helianane and (+)-5-Chloro-7,11-helianane through Stereoselective Aromatic Claisen Rearrangement

Total Synthesis of (+)-7,11-Helianane and (+)-5-Chloro-7,11-helianane through Stereoselective Aromatic Claisen Rearrangement

Total synthesis of (+)-thermozymocidin (myriocin) from D-fructose

Transition-state modeling of the aldol reaction of boron enolates: a force field approach

scholarly article by Anna Bernardi et al published May 1990 in Journal of Organic Chemistry

Tumor Targeting with an isoDGR-Drug Conjugate

scientific article published on 27 April 2017

Ureas: New efficient Lewis base catalysts for the allylation of aldehydes

Use of the Trost Ligand in the Ruthenium-Catalyzed Asymmetric Hydrogenation of Ketones

scholarly article by Mattia Cettolin et al published 27 June 2017 in ChemCatChem

αvβ3 Integrin-Targeted Peptide/Peptidomimetic-Drug Conjugates: In-Depth Analysis of the Linker Technology

scientific article published on July 2015

β-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate

scientific article published on 01 May 2019