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List of works by Jay H. Kalin

A novel role for histone deacetylase 6 in the regulation of the tolerogenic STAT3/IL-10 pathway in APCs.

scientific article

A selective phenelzine analogue inhibitor of histone demethylase LSD1.

scientific article published on 7 April 2014

An Fc domain protein-small molecule conjugate as an enhanced immunomodulator

scientific article

An Fc-Small Molecule Conjugate for Targeted Inhibition of the Adenosine 2A Receptor.

scientific article

An optimized RAD51 inhibitor that disrupts homologous recombination without requiring Michael acceptor reactivity.

scientific article

Bicyclic-Capped Histone Deacetylase 6 Inhibitors with Improved Activity in a Model of Axonal Charcot-Marie-Tooth Disease

scientific article published on 24 November 2015

Chiral Mercaptoacetamides Display Enantioselective Inhibition of Histone Deacetylase 6 and Exhibit Neuroprotection in Cortical Neuron Models of Oxidative Stress

scientific article published on 10 January 2012

Creating zinc monkey wrenches in the treatment of epigenetic disorders.

scientific article published on 21 June 2009

Development and Therapeutic Implications of Selective Histone Deacetylase 6 Inhibitors ⬇️

scientific article published on May 15, 2013

Exploration of the labeling of [11C]tubastatin A at the hydroxamic acid site with [11C]carbon monoxide.

scientific article

Histone deacetylase 6 inhibition improves memory and reduces total tau levels in a mouse model of tau deposition.

scientific article

Inhibiting the coregulator CoREST impairs Foxp3+ Treg function and promotes antitumor immunity

scientific article published on 01 April 2020

Investigation into the use of histone deacetylase inhibitor MS-275 as a topical agent for the prevention and treatment of cutaneous squamous cell carcinoma in an SKH-1 hairless mouse model

scientific article published on 13 March 2019

Lysine-14 acetylation of histone H3 in chromatin confers resistance to the deacetylase and demethylase activities of an epigenetic silencing complex.

scientific article published on 5 June 2018

Lysine-Specific Demethylase 1 Mediates AKT Activity and Promotes Epithelial-to-Mesenchymal Transition in PIK3CA-Mutant Colorectal Cancer

scientific article published on 08 November 2019

Rational design and simple chemistry yield a superior, neuroprotective HDAC6 inhibitor, tubastatin A

scientific article

Second-generation histone deacetylase 6 inhibitors enhance the immunosuppressive effects of Foxp3+ T-regulatory cells

scientific article published on 5 January 2012

Site-Specific Protein Labeling with N-Hydroxysuccinimide-Esters and the Analysis of Ubiquitin Ligase Mechanisms

scientific article published on 23 July 2018

Synthesis and antitubercular activity of quaternized promazine and promethazine derivatives

scientific article published on 02 December 2006

Targeting the CoREST complex with dual histone deacetylase and demethylase inhibitors

scientific article published on 4 January 2018

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