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List of works by Alex M Szpilman

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species

scientific article published on 16 August 2018

A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides

scientific article published on June 2003

Azido-Enolonium Species in C-C and C-N Bond-Forming Coupling Reactions

scientific article published on 09 January 2020

Cross-coupling of dissimilar ketone enolates via enolonium species to afford non-symmetrical 1,4-diketones.

scientific article

Design concept for α-hydrogen-substituted nitroxides

scientific article published on 06 February 2015

Enolonium Species-Umpoled Enolates

scientific article published on 27 January 2017

First α-deuterium nitroxides; synthesis and EPR study

scientific article published on 01 August 2019

Indium(III) Catalyzed Reactions of Vinyl Azides and Indoles

scientific article published on 24 April 2020

Iron(II)-induced degradation of antimalarial beta-sulfonyl endoperoxides: evidence for the generation of potentially cytotoxic carbocations

scientific article

Mechanism of the Copper/TEMPO-Catalyzed Aerobic Oxidation of Alcohols

scientific article

Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy.

scientific article published on 27 January 2016

Organocatalytic oxidation of aldehydes to mixed anhydrides.

scientific article published on 11 September 2012

Oxidative asymmetric umpolung alkylation of Evans' β-ketoimides using dialkylzinc nucleophiles

scientific article published on 01 March 2015

Oxidative umpolung α-alkylation of ketones

scientific article published on 06 January 2015

Probing the Biology of Natural Products: Molecular Editing by Diverted Total Synthesis

scientific article published on December 10, 2010

Sunlight assisted direct amide formation via a charge-transfer complex.

scientific article published on 25 August 2017

Synthesis and biological evaluation of amphotericin B derivatives

scientific article published on 16 June 2010

Synthesis and biological studies of 35-deoxy amphotericin B methyl ester

scientific article published in January 2008

Synthesis and biophysical studies on 35-deoxy amphotericin B methyl ester.

scientific article published in July 2009

Synthesis and stability of cyclic α-hydrogen nitroxides

scientific article published on 01 November 2015

Synthesis of 35-deoxy amphotericin B methyl ester: a strategy for molecular editing

scientific article published in January 2008

Total syntheses of Yingzhaosu A and of its C(14)-epimer including the first evaluation of their antimalarial and cytotoxic activities

scientific article

Transition-Metal-Free Intermolecular α-Arylation of Ketones via Enolonium Species.

scientific article published on 15 November 2017

Visible-Spectrum Solar-Light-Mediated Benzylic C-H Oxygenation Using 9,10-Dibromoanthracene As an Initiator

scientific article published on 25 November 2020

α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species

scientific article published on 15 January 2018

β-Glycosidation of Sterically Hindered Alcohols

scientific article published on 01 March 2009