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List of works by Timothy J. Ritchie

1-(2-Nitrophenyl)thiosemicarbazides: a novel class of potent, orally active non-peptide antagonist for the bradykinin B(2) receptor

scientific article

Analysis of the calculated physicochemical properties of respiratory drugs: can we design for inhaled drugs yet?

scientific article published on 01 April 2009

Antihyperalgesic activity of a novel nonpeptide bradykinin B1 receptor antagonist in transgenic mice expressing the human B1 receptor

scientific article

Chemoinformatics: manipulating chemical information to facilitate decision-making in drug discovery.

scientific article

Heterocyclic replacements for benzene: Maximising ADME benefits by considering individual ring isomers

scientific article

How drug-like are 'ugly' drugs: do drug-likeness metrics predict ADME behaviour in humans?

scientific article published on 21 January 2014

Nonpeptide bradykinin B2 receptor antagonists: conversion of rodent-selective bradyzide analogues into potent, orally-active human bradykinin B2 receptor antagonists

scientific article

Physicochemical descriptors of aromatic character and their use in drug discovery

scientific article published on 03 June 2014

Potent and orally bioavailable non-peptide antagonists at the human bradykinin B(1) receptor based on a 2-alkylamino-5-sulfamoylbenzamide core

scientific article published in September 2004

Should medicinal chemists do molecular modelling?

scientific article published on 16 January 2012

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

scientific article

The graphical representation of ADME-related molecule properties for medicinal chemists

scientific article

The impact of aromatic ring count on compound developability--are too many aromatic rings a liability in drug design?

scientific article published on September 2009

The impact of aromatic ring count on compound developability: further insights by examining carbo- and hetero-aromatic and -aliphatic ring types

scientific article published on December 2010