List of works - Prashant Murumkar

3D-quantitative structure-activity relationship studies on benzothiadiazepine hydroxamates as inhibitors of tumor necrosis factor-alpha converting enzyme

scientific article published on 14 February 2008

A comprehensive patents review on cannabinoid 1 receptor antagonists as antiobesity agents

scientific article published on 10 July 2015

Advances in studies on collagenase inhibitors

scientific article published on January 2012

Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists--a perspective

scientific article

Current perspective of TACE inhibitors: a review.

scientific article published on 03 December 2008

Design of selective TACE inhibitors using molecular docking studies: Synthesis and preliminary evaluation of anti-inflammatory and TACE inhibitory activity

scientific article published on 01 January 2015

Design, synthesis and evaluation of 4,7-disubstituted 8-methoxyquinazoline derivatives as potential cytotoxic agents targeting β-catenin/TCF4 signaling pathway

scientific article published on 21 March 2022

Developing steroidal aromatase inhibitors-an effective armament to win the battle against breast cancer

scientific article published on 03 October 2015

Development of highly predictive 3D-QSAR CoMSIA models for anthraquinone and acridone derivatives as telomerase inhibitors targeting G-quadruplex DNA telomere

scientific article published on July 15, 2010

Development of predictive 3D-QSAR CoMFA and CoMSIA models for beta-aminohydroxamic acid-derived tumor necrosis factor-alpha converting enzyme inhibitors.

scientific article published in January 2009

Development of predictive pharmacophore model for in silico screening, and 3D QSAR CoMFA and CoMSIA studies for lead optimization, for designing of potent tumor necrosis factor alpha converting enzyme inhibitors.

scientific article

Discovery of anti-malarial agents through application of in silico studies

scientific article published on January 2015

Exploring structural requirements for peripherally acting 1,5-diaryl pyrazole-containing cannabinoid 1 receptor antagonists for the treatment of obesity

scientific article

Novel TACE inhibitors in drug discovery: a review of patented compounds

scientific article published on January 2010

Novel methods and strategies in the discovery of TACE inhibitors

scientific article published on 12 December 2012

One-pot synthesis, biological evaluation, and docking study of new chromeno-annulated thiopyrano[2,3-c]pyrazoles

scientific article

Prospective therapeutic agents for obesity: molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonists

scientific article published on 05 April 2014

Structural investigations of acridine derivatives by CoMFA and CoMSIA reveal novel insight into their structures toward DNA G-quadruplex mediated telomerase inhibition and offer a highly predictive 3D-model for substituted acridines.

scientific article published in May 2009

Studies on novel 2-imidazolidinones and tetrahydropyrimidin-2(1H)-ones as potential TACE inhibitors: design, synthesis, molecular modeling, and preliminary biological evaluation

scientific article published on 8 April 2009

Synthesis and biological evaluation of some novel pyrido[1,2-a]pyrimidin-4-ones as antimalarial agents

scientific article published on 13 April 2014

Synthesis, preliminary biological evaluation and molecular modeling of some new heterocyclic inhibitors of TACE

scientific article published on 21 September 2011

Unequivocal role of pyrazine ring in medicinally important compounds: a review

scientific article published on October 2013

List of works by Prashant Murumkar

3D-quantitative structure-activity relationship studies on benzothiadiazepine hydroxamates as inhibitors of tumor necrosis factor-alpha converting enzyme

A comprehensive patents review on cannabinoid 1 receptor antagonists as antiobesity agents

Advances in studies on collagenase inhibitors

Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists--a perspective

Current perspective of TACE inhibitors: a review.

Design of selective TACE inhibitors using molecular docking studies: Synthesis and preliminary evaluation of anti-inflammatory and TACE inhibitory activity

Design, synthesis and evaluation of 4,7-disubstituted 8-methoxyquinazoline derivatives as potential cytotoxic agents targeting β-catenin/TCF4 signaling pathway

Developing steroidal aromatase inhibitors-an effective armament to win the battle against breast cancer

Development of highly predictive 3D-QSAR CoMSIA models for anthraquinone and acridone derivatives as telomerase inhibitors targeting G-quadruplex DNA telomere

Development of predictive 3D-QSAR CoMFA and CoMSIA models for beta-aminohydroxamic acid-derived tumor necrosis factor-alpha converting enzyme inhibitors.

Development of predictive pharmacophore model for in silico screening, and 3D QSAR CoMFA and CoMSIA studies for lead optimization, for designing of potent tumor necrosis factor alpha converting enzyme inhibitors.

Discovery of anti-malarial agents through application of in silico studies

Exploring structural requirements for peripherally acting 1,5-diaryl pyrazole-containing cannabinoid 1 receptor antagonists for the treatment of obesity

Novel TACE inhibitors in drug discovery: a review of patented compounds

Novel methods and strategies in the discovery of TACE inhibitors

One-pot synthesis, biological evaluation, and docking study of new chromeno-annulated thiopyrano[2,3-c]pyrazoles

Prospective therapeutic agents for obesity: molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonists

Structural investigations of acridine derivatives by CoMFA and CoMSIA reveal novel insight into their structures toward DNA G-quadruplex mediated telomerase inhibition and offer a highly predictive 3D-model for substituted acridines.

Studies on novel 2-imidazolidinones and tetrahydropyrimidin-2(1H)-ones as potential TACE inhibitors: design, synthesis, molecular modeling, and preliminary biological evaluation

Synthesis and biological evaluation of some novel pyrido[1,2-a]pyrimidin-4-ones as antimalarial agents

Synthesis, preliminary biological evaluation and molecular modeling of some new heterocyclic inhibitors of TACE

Unequivocal role of pyrazine ring in medicinally important compounds: a review