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List of works by Thomas Rades

"This body does not want free medicines": South African consumer perceptions of drug quality

scientific article published on 2 September 2009

A New Approach to Dissolution Testing by UV Imaging and Finite Element Simulations ⬇️

scientific article published on January 11, 2013

A Promising New Method to Estimate Drug-Polymer Solubility at Room Temperature

article

A case study of real-time monitoring of solid-state phase transformations in acoustically levitated particles using near infrared and Raman spectroscopy

scientific article

A comparison of pseudo-ternary diagrams of aqueous mixtures of Quil A, cholesterol and phospholipid prepared by lipid-film hydration and dialysis

scientific article

A method for the incorporation of ovalbumin into immune stimulating complexes prepared by the hydration method

scientific article published in July 2002

A non-destructive method for quality control of the pellet distribution within a MUPS tablet by terahertz pulsed imaging

scientific article published on 19 October 2017

A novel image analysis methodology for online monitoring of nucleation and crystal growth during solid state phase transformations

scientific article published on 04 May 2012

A platform for preparing homogeneous proteinaceous sub-visible particles with distinct morphologies.

scientific article published on 21 March 2018

A slow cooling rate of indomethacin melt spatially confined in microcontainers increases the physical stability of the amorphous drug without influencing its biorelevant dissolution behaviour

article published in 2014

A theoretical and spectroscopic study of co-amorphous naproxen and indomethacin

scientific article

A theoretical and spectroscopic study of γ-crystalline and amorphous indometacin

scientific article published on 01 February 2007

Activation of the NLRP3 inflammasome is not a feature of all particulate vaccine adjuvants

scientific article published on 01 April 2014

Adsorption of bovine serum albumin (BSA) onto lecithin studied by attenuated total reflectance Fourier transform infrared (ATR-FTIR) spectroscopy.

scientific article

Advanced characterisation techniques

scientific article published on 21 March 2011

Aerosol OT Microemulsions as Carriers for Transdermal Delivery of Hydrophobic and Hydrophilic Local Anesthetics

scientific article published on 01 June 2008

Amino Acids as Co-amorphous Excipients for Simvastatin and Glibenclamide: Physical Properties and Stability

scientific article published on 04 June 2014

Amino acids as co-amorphous stabilizers for poorly water soluble drugs--Part 1: preparation, stability and dissolution enhancement

scientific article published on 26 March 2013

Amino acids as co-amorphous stabilizers for poorly water-soluble drugs--Part 2: molecular interactions.

scientific article published on 6 April 2013

Amino acids as stabilizers for spray-dried simvastatin powder for inhalation

scientific article published on 31 October 2019

Amorphization within the tablet: Using microwave irradiation to form a glass solution in situ

scientific article published on 20 January 2017

Amorphous is not always better—A dissolution study on solid state forms of carbamazepine

An oral delivery system for indomethicin engineered from cationic lipid emulsions and silica nanoparticles

scientific article published on 14 January 2010

An overview of recent studies on the analysis of pharmaceutical polymorphs

scientific article published on 22 December 2010

Analysis of 3D Prints by X-ray Computed Microtomography and Terahertz Pulsed Imaging

scientific article

Analysis of Quil A–phospholipid mixtures using drift spectroscopy

scientific article published on 06 May 2007

Analysis of coating structures and interfaces in solid oral dosage forms by three dimensional terahertz pulsed imaging

scientific article

Analysis of lecithin-cholesterol mixtures using Raman spectroscopy

scientific article published on 15 February 2006

Analysis of matrix dosage forms during dissolution testing using raman microscopy

scientific article published on 10 May 2011

Analysis of sustained-release tablet film coats using terahertz pulsed imaging

article

Anhydrate to hydrate solid-state transformations of carbamazepine and nitrofurantoin in biorelevant media studied in situ using time-resolved synchrotron X-ray diffraction

scientific article published on 13 January 2016

Anti-ageing effects of Sonchus oleraceus L. (pūhā) leaf extracts on H₂O₂-induced cell senescence.

scientific article

Application of a Salt Coformer in a Co-Amorphous Drug System Dramatically Enhances the Glass Transition Temperature: A Case Study of the Ternary System Carbamazepine, Citric Acid, and l-Arginine

scientific article published on 9 April 2018

Application of an online post-column derivatization HPLC-DPPH assay to detect compounds responsible for antioxidant activity in Sonchus oleraceus L. leaf extracts.

scientific article published on 25 September 2012

Application of spray-drying and electrospraying/electospinning for poorly water-soluble drugs: a particle engineering approach

scientific article published on January 2014

Application of terahertz pulsed imaging to analyse film coating characteristics of sustained-release coated pellets

scientific article published on 27 May 2013

Applications of terahertz pulsed imaging to sustained-release tablet film coating quality assessment and dissolution performance

scientific article published on 12 January 2008

Applying thermodynamic and kinetic parameters to predict the physical stability of two differently prepared amorphous forms of simvastatin.

scientific article

Are phytosomes a superior nanodelivery system for the antioxidant rutin?

Aspartame as a co-former in co-amorphous systems

Assessment of crystalline disorder in cryo-milled samples of indomethacin using atomic pair-wise distribution functions.

scientific article

Atomic pairwise distribution function analysis of the amorphous phase prepared by different manufacturing routes.

scientific article published on 31 January 2012

Bicontinuous cubic liquid crystals as sustained delivery systems for peptides and proteins.

scientific article published on October 2010

Biorelevant characterisation of amorphous furosemide salt exhibits conversion to a furosemide hydrate during dissolution

scientific article published on 16 September 2013

Cage-like complexes formed by DOTAP, Quil-A and cholesterol

scientific article

Cationic cage-like complexes formed by DC-cholesterol, Quil-A, and phospholipid

scientific article published in August 2005

Characterisation of bicontinuous cubic liquid crystalline systems of phytantriol and water using cryo field emission scanning electron microscopy (cryo FESEM).

scientific article published on 20 September 2006

Characterisation of colloidal drug delivery systems from the naked eye to Cryo-FESEM.

scientific article

Characterisation of indomethacin and nifedipine using variable-temperature solid-state NMR.

scientific article published in November 2005

Characterisation of pore structures of pharmaceutical tablets: A review.

scientific article published on 13 January 2018

Characterisation of quaternary polymethacrylate films containing tartaric acid, metoprolol free base or metoprolol tartrate.

scientific article published on 3 August 2009

Characterising glass transition temperatures and glass dynamics in mesoporous silica-based amorphous drugs

scientific article published on 01 September 2019

Characterising lipid lipolysis and its implication in lipid-based formulation development

scientific article

Characterization and in vitro permeation study of microemulsions and liquid crystalline systems containing the anticholinesterase alkaloidal extract from Tabernaemontana divaricata

scientific article published on 13 May 2013

Characterization of Amorphous and Co-Amorphous Simvastatin Formulations Prepared by Spray Drying.

scientific article

Characterization of Temperature-Induced Phase Transitions in Five Polymorphic Forms of Sulfathiazole by Terahertz Pulsed Spectroscopy and Differential Scanning Calorimetry

article

Characterization of chitosan–magnesium aluminum silicate nanocomposite films for buccal delivery of nicotine

scientific article published on 05 January 2013

Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with hydrophilic amorphous polymers

scientific article

Characterization of the Hydrodynamics in a Miniaturized Dissolution Apparatus

scientific article published on 9 December 2017

Characterization of the bulk properties of pharmaceutical solids using nonlinear optics--a review

scientific article

Characterizing colloidal structures of pseudoternary phase diagrams formed by oil/water/amphiphile systems

scientific article published in January 2001

Characterizing the conversion kinetics of carbamazepine polymorphs to the dihydrate in aqueous suspension using Raman spectroscopy.

scientific article

Characterizing the freezing behavior of liposomes as a tool to understand the cryopreservation procedures

scientific article published on 24 August 2007

Chemical imaging and solid state analysis at compact surfaces using UV imaging

scientific article published on 31 October 2014

Chitosan hydrogels containing liposomes and cubosomes as particulate sustained release vaccine delivery systems

scientific article published on 22 December 2011

Chitosan-magnesium aluminum silicate composite dispersions: characterization of rheology, flocculate size and zeta potential

scientific article published on 5 October 2007

Chitosan-magnesium aluminum silicate nanocomposite films: physicochemical characterization and drug permeability

scientific article published on 14 April 2010

Co-amorphous simvastatin and glipizide combinations show improved physical stability without evidence of intermolecular interactions

article

Co-former selection for co-amorphous drug-amino acid formulations

scientific article published on 19 December 2018

Coamorphous drug systems: enhanced physical stability and dissolution rate of indomethacin and naproxen.

scientific article published on 15 August 2011

Combining diagnostic methods for antimicrobial susceptibility testing - A comparative approach

scientific article published on 14 November 2017

Comparative Study of Different Methods for the Prediction of Drug-Polymer Solubility

scientific article published on 27 July 2015

Comparative effects of intraduodenal infusions of lauric and oleic acids on antropyloroduodenal motility, plasma cholecystokinin and peptide YY, appetite, and energy intake in healthy men

scientific article published on 01 May 2008

Comparative study of liposomes, transfersomes, ethosomes and cubosomes for transcutaneous immunisation: characterisation and in vitro skin penetration ⬇️

scientific article published on May 9, 2012

Comparison of bulk and microfluidics methods for the formulation of poly-lactic-co-glycolic acid (PLGA) nanoparticles modified with cell-penetrating peptides of different architectures

scientific article published on 13 August 2019

Comparison of chitosan nanoparticles and chitosan hydrogels for vaccine delivery

scientific article published on 01 December 2008

Comparison of induction methods for supersaturation: pH shift versus solvent shift

scientific article published on 20 November 2019

Comparison of lipases for in vitro models of gastric digestion: lipolysis using two infant formulas as model substrates

scientific article

Comparison of the Structure and Properties of Liposomes Prepared from Milk Fat Globule Membrane and Soy Phospholipids

scientific article published on 01 May 2006

Comparison of two DSC-based methods to predict drug-polymer solubility

scientific article published on 6 February 2018

Comparison of two different PEGylation strategies for the liposomal adjuvant CAF09: Towards induction of CTL responses upon subcutaneous vaccine administration

article

Correction: Formation of drug nanocrystals under nanoconfinement afforded by liposomes

scholarly article in RSC Advances, vol. 6 no. 15, 2016

Correlating thermodynamic and kinetic parameters with amorphous stability

scientific article published on 23 April 2009

Corrigendum to "Formulation and characterization of self-nanoemulsifying drug delivery systems containing monoacyl phosphatidylcholine" [Int. J. Pharm. 502 (1-2) (2016) 151-160]

scholarly article published in International Journal of Pharmaceutics

Cryo-responses of two types of large unilamellar vesicles in the presence of non-permeable or permeable cryoprotecting agents

scientific article

Crystal Morphology Modification by the Addition of Tailor-Made Stereocontrolled Poly(N-isopropyl acrylamide)

article

Crystalline adduct of moxifloxacin with trans-cinnamic acid to reduce the aqueous solubility and dissolution rate for improved residence time in the lungs

scientific article published on 17 June 2019

Cubosomes containing the adjuvants imiquimod and monophosphoryl lipid A stimulate robust cellular and humoral immune responses

scientific article published on 8 November 2012

Current advances and future trends in characterizing poorly water-soluble drugs using spectroscopic, imaging and data analytical techniques.

scientific article

Deeper insight into the drug release mechanisms in Eudragit RL-based delivery systems.

scientific article published on 25 January 2010

Design of Inhalable Solid Dosage Forms of Budesonide and Theophylline for Pulmonary Combination Therapy

scientific article published on 07 March 2019

Determination of Stable Co-Amorphous Drug-Drug Ratios from the Eutectic Behavior of Crystalline Physical Mixtures

scientific article published on 24 November 2019

Determination of methylphenidate in Calliphorid larvae by liquid-liquid extraction and liquid chromatography mass spectrometry--forensic entomotoxicology using an in vivo rat brain model.

scientific article published on 26 June 2012

Determination of moisture content in relation to thermal behaviour and plasticization of Eudragit RLPO.

scientific article published on 20 October 2011

Determination of polymorphic forms of ranitidine-HCl by DRIFTS and XRPD.

scientific article published in July 2001

Determination of the Optimal Molar Ratio in Amino Acid-Based Coamorphous Systems

scientific article published on 09 March 2020

Determining Thermal Conductivity of Small Molecule Amorphous Drugs with Modulated Differential Scanning Calorimetry and Vacuum Molding Sample Preparation

scientific article published on 10 December 2019

Development and characterisation of modified poloxamer 407 thermoresponsive depot systems containing cubosomes

article

Development of a Video-Microscopic Tool To Evaluate the Precipitation Kinetics of Poorly Water Soluble Drugs: A Case Study with Tadalafil and HPMC.

scientific article

Development of a high-throughput in vitro intestinal lipolysis model for rapid screening of lipid-based drug delivery systems

Development of a novel magnetic resonance imaging contrast agent for pressure measurements using lipid-coated microbubbles.

scientific article published in December 2009

Development of a screening method for co-amorphous formulations of drugs and amino acids.

scientific article published on 13 August 2016

Differential scanning calorimetry predicts the critical quality attributes of amorphous glibenclamide

scientific article published on 18 August 2015

Dipeptides as co-formers in co-amorphous systems

scientific article published on 20 November 2018

Direct Comparison of Standard Transmission Electron Microscopy and Cryogenic-TEM in Imaging Nanocrystals Inside Liposomes

scientific article published on 27 February 2019

Direct Measurement of Amorphous Solubility

scientific article published on 14 May 2019

Direct Measurement of Lateral Molecular Diffusivity on the Surface of Supersaturated Amorphous Solid Dispersions by Atomic Force Microscopy

scientific article published on 01 April 2020

Direct detection of dissolution of 14 C-labeled compounds into an oil phase by the fat scintillation proximity method

scientific article published on 01 March 2000

Distribution of binder in granules produced by means of twin screw granulation.

scientific article published on 19 December 2013

Dose-related effects of lauric acid on antropyloroduodenal motility, gastrointestinal hormone release, appetite, and energy intake in healthy men.

scientific article published on 16 June 2005

Drug hydrate systems and dehydration processes studied by terahertz pulsed spectroscopy

scientific article published on 21 October 2006

Drug nanocrystallisation within liposomes

scientific article published on 02 September 2018

Drug quality in South Africa: perceptions of key players involved in medicines distribution

scientific article published on January 2009

Dry Hybrid Lipid−Silica Microcapsules Engineered from Submicron Lipid Droplets and Nanoparticles as a Novel Delivery System for Poorly Soluble Drugs

scientific article published on 01 May 2009

Effect of amorphous phase separation and crystallization on the in vitro and in vivo performance of an amorphous solid dispersion

scientific article published on 03 July 2018

Effect of composition of simulated intestinal media on the solubility of poorly soluble compounds investigated by design of experiments

scientific article published on 3 October 2017

Effect of different preparation methods on the dissolution behaviour of amorphous indomethacin

scientific article published on 14 October 2011

Effect of incorporation of the adjuvant Quil A on structure and immune stimulatory capacity of liposomes

scientific article published on 01 October 2004

Effect of milling conditions on the solid-state conversion of ranitidine hydrochloride form 1

scientific article published on 22 July 2006

Effect of polymer type and drug dose on the in vitro and in vivo behavior of amorphous solid dispersions

scientific article

Effects of alcohols and diols on the phase behaviour of quaternary systems

scientific article published on 10 March 2000

Effects of film coating thickness and drug layer uniformity on in vitro drug release from sustained-release coated pellets: a case study using terahertz pulsed imaging

scientific article published on 27 August 2009

Effects of formulation variables on characteristics of poly (ethylcyanoacrylate) nanocapsules prepared from w/o microemulsions

scientific article published in March 2002

Effects of intraduodenal fatty acids on appetite, antropyloroduodenal motility, and plasma CCK and GLP-1 in humans vary with their chain length

scientific article

Effects of lauric acid on upper gut motility, plasma cholecystokinin and peptide YY, and energy intake are load, but not concentration, dependent in humans

Effects of meal consistency and ingested fluid volume on the intragastric distribution of a drug model in humans--a magnetic resonance imaging study.

scientific article

Efflux Inhibitor Bicalutamide Increases Oral Bioavailability of the Poorly Soluble Efflux Substrate Docetaxel in Co-Amorphous Anti-Cancer Combination Therapy

scientific article published on 11 January 2019

Elucidating Pathway and Anesthetic Mechanism of Action of Clove Oil Nanoformulations in Fish

scientific article published on 22 April 2022

Elucidating the Molecular Interactions Occurring during Drug Precipitation of Weak Bases from Lipid-Based Formulations: A Case Study with Cinnarizine and a Long Chain Self-Nanoemulsifying Drug Delivery System

scientific article published on 22 September 2015

Emerging trends in the stabilization of amorphous drugs.

scientific article published on 28 April 2012

Enhanced dissolution rate and synchronized release of drugs in binary systems through formulation: Amorphous naproxen-cimetidine mixtures prepared by mechanical activation

scientific article

Enhancing Stability and Tooth Bleaching Activity of Carbamide Peroxide by Electrospun Nanofibrous Film

scientific article published on 11 November 2020

Evaluating the effect of coating equipment on tablet film quality using terahertz pulsed imaging

scientific article published on 4 April 2013

Evaluation of Drug–Polymer Solubility Curves Through Formal Statistical Analysis: Comparison of Preparation Techniques

scientific article published on 31 October 2014

Exploring the fate of liposomes in the intestine by dynamic in vitro lipolysis

Factors affecting incorporation of drug into solid solution with HPMCP during solvent change co-precipitation

scientific article published in October 2002

Factors influencing the entrapment of hydrophilic compounds in nanocapsules prepared by interfacial polymerisation of water-in-oil microemulsions

scientific article published in May 2002

Fat digestion modulates gastrointestinal sensations induced by gastric distention and duodenal lipid in humans

scientific article

Formation Mechanism of Coamorphous Drug-Amino Acid Mixtures.

scientific article published on 23 June 2015

Formation and physical stability of the amorphous phase of ranitidine hydrochloride polymorphs prepared by cryo-milling

scientific article published on 14 September 2007

Formation of drug nanocrystals under nanoconfinement afforded by liposomes

scholarly article in RSC Advances, vol. 6 no. 8, 2016

Formulation and characterization of self-nanoemulsifying drug delivery systems containing monoacyl phosphatidylcholine

Formulation of self-nanoemulsifying drug delivery systems containing monoacyl phosphatidylcholine and Kolliphor® RH40 using experimental design

scientific article published on 13 October 2017

Glass Forming Ability of Amorphous Drugs Investigated by Continuous Cooling and Isothermal Transformation

scientific article published on 26 August 2016

Glass-Transition Temperature of the β-Relaxation as the Major Predictive Parameter for Recrystallization of Neat Amorphous Drugs

scientific article published on 02 March 2018

High-Throughput Lipolysis in 96-Well Plates for Rapid Screening of Lipid-Based Drug Delivery Systems

scientific article published on 2 January 2017

High-shear granulation as a manufacturing method for cocrystal granules

scientific article published on 16 May 2013

Highly Elastic and Water Stable Zein Microfibers as a Potential Drug Delivery System for Wound Healing

scientific article published on 18 May 2020

Histidine residues in the peptide D-Lys(6)-GnRH: potential for copolymerization in polymeric nanoparticles

scientific article published in September 2009

Hot Melt Coating of Amorphous Carvedilol

scientific article published on 06 June 2020

Hot Melt Extrusion and Spray Drying of Co-amorphous Indomethacin-Arginine With Polymers

scientific article published on 3 November 2016

Hyaluronic acid-based nanogels improve in vivo compatibility of the anti-biofilm peptide DJK-5

scientific article published on 04 June 2019

Hydration of lipid films with an aqueous solution of Quil A: a simple method for the preparation of immune-stimulating complexes

scientific article published on 01 March 2000

Image Analytical Approach for Needle-Shaped Crystal Counting and Length Estimation

Imaging of dehydration in particulate matter using Raman line-focus microscopy

scientific article published on 17 May 2019

Immune responses induced by nano-self-assembled lipid adjuvants based on a monomycoloyl glycerol analogue after vaccination with the Chlamydia trachomatis major outer membrane protein

article

Immuno-stimulating complexes prepared by ethanol injection

scientific article published in June 2005

Immunogenicity of Liposomes Containing Lipid Core Peptides and the Adjuvant Quil A

scientific article published on 21 June 2006

Immunostimulatory biodegradable implants containing the adjuvant Quil-A—Part I: Physicochemical characterisation

scientific article published on 01 April 2008

Immunostimulatory biodegradable implants containing the adjuvant Quil-A—Part II:In vivoevaluation

scientific article published on 01 April 2008

Immunostimulatory colloidal delivery systems for cancer vaccines.

scientific article

Immunostimulatory lipid implants containing Quil-A and DC-cholesterol

scientific article published on 23 July 2008

Importance of in vitro dissolution conditions for the in vivo predictability of an amorphous solid dispersion containing a pH-sensitive carrier.

scientific article

Improvement of dissolution rate of indomethacin by inkjet printing

scientific article published on 25 March 2015

Improvement of the physicochemical properties of Co-amorphous naproxen-indomethacin by naproxen-sodium

scientific article

Improving co-amorphous drug formulations by the addition of the highly water soluble amino Acid, proline

scientific article published on 14 July 2014

In Situ Lipolysis and Synchrotron Small-Angle X-ray Scattering for the Direct Determination of the Precipitation and Solid-State Form of a Poorly Water-Soluble Drug During Digestion of a Lipid-Based Formulation

scientific article published on 11 September 2015

In Vitro, Ex Vivo and In Vivo Evaluation of Microcontainers for Oral Delivery of Insulin

scientific article published on 07 January 2020

In Vivo Precipitation of Poorly Soluble Drugs from Lipid-Based Drug Delivery Systems.

scientific article

In situ amorphisation of indomethacin with Eudragit® E during dissolution

scientific article published on 18 September 2013

In situ co-amorphisation in coated tablets - The combination of carvedilol with aspartic acid during immersion in an acidic medium

scientific article published on 12 January 2019

In situ co-amorphisation of arginine with indomethacin or furosemide during immersion in an acidic medium - a proof of concept study

scientific article published on 16 October 2018

In vitro and in vivo comparison between crystalline and co-amorphous salts of naproxen-arginine

scientific article published on 25 September 2018

In vitro and in vivo investigation of thermosensitive chitosan hydrogels containing silica nanoparticles for vaccine delivery

scientific article published on 13 July 2010

In vitro and in vivo performance of monoacyl phospholipid-based self-emulsifying drug delivery systems.

scientific article

In vitro and in vivo performance of novel supersaturated self-nanoemulsifying drug delivery systems (super-SNEDDS)

article published in 2012

In vitro lipolysis data does not adequately predict the in vivo performance of lipid-based drug delivery systems containing fenofibrate

scientific article

In vivo activity of cationic immune stimulating complexes (PLUSCOMs).

scientific article published on 26 June 2008

In vivo evaluation of chitosan as an adjuvant in subcutaneous vaccine formulations

scientific article published on 9 August 2013

In-vitro release and oral bioactivity of insulin in diabetic rats using nanocapsules dispersed in biocompatible microemulsion.

scientific article

Incorporation of ovalbumin into ISCOMs and related colloidal particles prepared by the lipid film hydration method

scientific article

Induction of Cytotoxic T-Lymphocyte Responses Upon Subcutaneous Administration of a Subunit Vaccine Adjuvanted With an Emulsion Containing the Toll-Like Receptor 3 Ligand Poly(I:C).

scientific article

Influence of Copolymer Composition on In Vitro and In Vivo Performance of Celecoxib-PVP/VA Amorphous Solid Dispersions

scientific article published on 14 January 2016

Influence of Glass Forming Ability on the Physical Stability of Supersaturated Amorphous Solid Dispersions

scientific article published on 13 March 2019

Influence of Lipid Composition and Drug Load on the In Vitro Performance of Self-Nanoemulsifying Drug Delivery Systems

article

Influence of PVP molecular weight on the microwave assisted in situ amorphization of indomethacin

scientific article published on 3 October 2017

Influence of PVP/VA copolymer composition on drug-polymer solubility

scientific article

Influence of Polymer Molecular Weight on Drug-Polymer Solubility: A Comparison between Experimentally Determined Solubility in PVP and Prediction Derived from Solubility in Monomer

scientific article published on 3 March 2015

Influence of Polymorphic Form, Morphology, and Excipient Interactions on the Dissolution of Carbamazepine Compacts

scientific article published on 01 March 2007

Influence of Solvent Composition on the Performance of Spray-Dried Co-Amorphous Formulations

scientific article

Influence of Tableting on the Conformation and Thermal Stability of Trypsin as a Model Protein.

scientific article

Influence of drug load and physical form of cinnarizine in new SNEDDS dosing regimens: in vivo and in vitro evaluations

Influence of particle size and preparation methods on the physical and chemical stability of amorphous simvastatin

scientific article published on 24 July 2008

Influence of polymer molecular weight on in vitro dissolution behavior and in vivo performance of celecoxib:PVP amorphous solid dispersions.

scientific article published on 17 February 2016

Influence of postharvest processing and storage conditions on key antioxidants in pūhā (Sonchus oleraceusL.)

scientific article published on 12 February 2014

Influence of preparation pathway on the glass forming ability

scientific article published on 20 February 2017

Influence of preparation technique on co-amorphization of carvedilol with acidic amino acids

scientific article

Influence of sample characteristics on quantification of carbamazepine hydrate formation by X-ray powder diffraction and Raman spectroscopy

scientific article published on 13 December 2006

Influence of solvent evaporation rate and formulation factors on solid dispersion physical stability

scientific article published on 17 October 2011

Influence of the cooling rate and the blend ratio on the physical stability of co-amorphous naproxen/indomethacin

scientific article published on 13 October 2016

Influence of variation in molar ratio on co-amorphous drug-amino acid systems

scientific article published on 28 June 2016

Inhalable Antimicrobials for Treatment of Bacterial Biofilm-Associated Sinusitis in Cystic Fibrosis Patients: Challenges and Drug Delivery Approaches

scientific article

Inhalable co-amorphous budesonide-arginine dry powders prepared by spray drying

scientific article published on 15 April 2019

Inhibition of surface crystallisation of amorphous indomethacin particles in physical drug–polymer mixtures

scientific article published on 03 September 2013

Insights into the Early Dissolution Events of Amlodipine Using UV Imaging and Raman Spectroscopy

scientific article published on 20 June 2011

Insights into the Structure of Protein by Vibrational Spectroscopy

article

Interactions between fenoprofen sodium and poly (ethylene oxide) ⬇️

scientific article published on July 1, 1998

Interdependence of Dosage Form Microstructure and Performance.

scientific article published on 15 March 2017

Interlaboratory Validation of Small-Scale Solubility and Dissolution Measurements of Poorly Water-Soluble Drugs

scientific article

Investigating dehydration from compacts using terahertz pulsed, Raman, and near-infrared spectroscopy

scientific article

Investigating dissolution performance critical areas on coated tablets: A case study using terahertz pulsed imaging

scientific article published on 01 January 2010

Investigation of physical properties and stability of indomethacin-cimetidine and naproxen-cimetidine co-amorphous systems prepared by quench cooling, coprecipitation and ball milling

scientific article published on 14 December 2015

Investigation of properties and recrystallisation behaviour of amorphous indomethacin samples prepared by different methods

scientific article published on 21 December 2010

Investigation of the Formation Process of Two Piracetam Cocrystals during Grinding

scientific article published on 12 October 2011

Investigation of the Intra- and Interlaboratory Reproducibility of a Small Scale Standardized Supersaturation and Precipitation Method

scientific article

Investigation of the phase separation of PNIPAM using infrared spectroscopy together with multivariate data analysis

Investigations on the effect of different cooling rates on the stability of amorphous indomethacin

scientific article

Is there a correlation between the glass forming ability of a drug and its supersaturation propensity?

scientific article

Lipid based particulate formulations for the delivery of antigen.

scientific article

Lipid-Based Formulations Can Enable the Model Poorly Water-Soluble Weakly Basic Drug Cinnarizine To Precipitate in an Amorphous-Salt Form During In Vitro Digestion

scientific article published on 15 September 2016

Liposomal delivery of antigen to human dendritic cells

scientific article

Liposome-Based Adjuvants for Subunit Vaccines: Formulation Strategies for Subunit Antigens and Immunostimulators

scientific article

Liquid crystalline systems of phytantriol and glyceryl monooleate containing a hydrophilic protein: Characterisation, swelling and release kinetics

scientific article

Low-Frequency Raman Spectroscopic Study on Compression-Induced Destabilization in Melt-Quenched Amorphous Celecoxib

scientific article published on 10 July 2019

Lysozyme-magnesium aluminum silicate microparticles: Molecular interaction, bioactivity and release studies.

scientific article published on 17 July 2015

Mannosylated liposomes as antigen delivery vehicles for targeting to dendritic cells

scientific article published on 01 June 2006

Mannosylated saponins based on oleanolic and glycyrrhizic acids. Towards synthetic colloidal antigen delivery systems.

scientific article

Mechanical properties of excipients do not affect polymer matrix formation

scientific article published on 9 October 2009

Melt Extrusion and Spray Drying of Carbamazepine and Dipyridamole with Polyvinylpyrrolidone/Vinyl Acetate Copolymers

scientific article published on 01 January 2008

Melt Extrusion of High-Dose Co-Amorphous Drug-Drug Combinations : Theme: Formulation and Manufacturing of Solid Dosage Forms Guest Editors: Tony Zhou and Tonglei Li.

scientific article

Microcontainers as an oral delivery system for spray dried cubosomes containing ovalbumin

scientific article

Microcontainers for oral insulin delivery - In vitro studies of permeation enhancement

scientific article published on 16 August 2019

Microcontainers for protection of oral vaccines, in vitro and in vivo evaluation

scientific article published on 12 December 2018

Microemulsions containing lecithin and sugar-based surfactants: nanoparticle templates for delivery of proteins and peptides.

scientific article

Miscibility and interactions between 17beta-estradiol and Eudragit RS in solid dispersion.

scientific article

Modified thermoresponsive Poloxamer 407 and chitosan sol–gels as potential sustained-release vaccine delivery systems

scientific article published on 03 December 2014

Monitoring the Film Coating Unit Operation and Predicting Drug Dissolution Using Terahertz Pulsed Imaging

scientific article published on 01 December 2009

Monitoring the Isothermal Dehydration of Crystalline Hydrates Using Low-Frequency Raman Spectroscopy

scientific article published on 06 January 2021

Monitoring the intragastric distribution of a colloidal drug carrier model by magnetic resonance imaging460

scientific article published on 01 April 2001

Monoacyl phosphatidylcholine inhibits the formation of lipid multilamellar structures during in vitro lipolysis of self-emulsifying drug delivery systems

scientific article published on 23 November 2016

Multispectral UV Imaging for Determination of the Tablet Coating Thickness

scientific article

Multispectral UV imaging for fast and non-destructive quality control of chemical and physical tablet attributes

scientific article published on 3 December 2015

Multispectral UV imaging for surface analysis of MUPS tablets with special focus on the pellet distribution

scientific article published in October 2016

Multivariate Quantification of the Solid State Phase Composition of Co-Amorphous Naproxen-Indomethacin.

scientific article published on 27 October 2015

Nanomechanical Infrared Spectroscopy with Vibrating Filters for Pharmaceutical Analysis

scientific article

New perspectives on lipid and surfactant based drug delivery systems for oral delivery of poorly soluble drugs

scientific article

Nicotine-magnesium aluminum silicate microparticle surface modified with chitosan for mucosal delivery

scientific article published on 4 January 2013

Non-destructive quantification of pharmaceutical tablet coatings using terahertz pulsed imaging and optical coherence tomography

article

Noninvasive 3D characterization of layered samples using terahertz pulsed imaging and infrared optical coherence tomography

Nonlamellar liquid crystalline nanostructured particles: advances in materials and structure determination.

scientific article published on January 2009

Novel chitosan−magnesium aluminum silicate nanocomposite film coatings for modified-release tablets

scientific article published on 01 February 2011

On the role of salt formation and structural similarity of co-formers in co-amorphous drug delivery systems

scientific article published in November 2017

Optimization of Infrared Microscopy to Assess Secondary Structure of Insulin Molecules Within Individual Subvisible Particles in Aqueous Formulations

scientific article published on 26 October 2018

Oral insulin delivery using nanoparticles based on microemulsions with different structure-types: optimisation and in vivo evaluation

scientific article published on 9 January 2009

Organic acids as co-formers for co-amorphous systems - Influence of variation in molar ratio on the physicochemical properties of the co-amorphous systems

scientific article published on 21 July 2018

Performance comparison between crystalline and co-amorphous salts of indomethacin-lysine

scientific article published on 22 September 2017

Phosphatidyl choline-based colloidal systems for dermal and transdermal drug delivery

scientific article published in January 2009

Physical Characterization of Synthetic Phosphatidylinositol Dimannosides and Analogues in Binary Systems with Phosphatidylcholine

scientific article published on 30 January 2014

Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation

scientific article published on 3 July 2008

Physical stability and solubility of the thermotropic mesophase of fenoprofen calcium as pure drug and in a tablet formulation

scientific article published in October 2002

Physicochemical and biological characterization of synthetic phosphatidylinositol dimannosides and analogues

scientific article published on 25 March 2013

Poly(alkycyanoacrylate) nanoparticles for enhanced delivery of therapeutics – is there real potential?

scientific article published on 01 April 2009

Polymer incorporation method affects the physical stability of amorphous indomethacin in aqueous suspension

scientific article published on 16 June 2015

Polymeric microcontainers improve oral bioavailability of furosemide

Polymeric nanoparticles as an oral delivery system for biocontrol agents for the brushtail possum (Trichosurus vulpecula).

scientific article published in December 2009

Polymorphic form of piroxicam influences the performance of amorphous material prepared by ball-milling

scientific article published on 14 March 2012

Powder diffractometric assay of two polymorphic forms of ranitidine hydrochloride.

scientific article published in July 1999

Precipitation of a poorly soluble model drug during in vitro lipolysis: characterization and dissolution of the precipitate

scientific article published on December 2010

Predicting Crystallization of Amorphous Drugs with Terahertz Spectroscopy.

scientific article published in July 2015

Preparation and characterization of spray-dried co-amorphous drug-amino acid salts

scientific article published on 05 August 2015

Preparation and recrystallization behavior of spray-dried co-amorphous naproxen-indomethacin

scientific article

Preparation of an amorphous sodium furosemide salt improves solubility and dissolution rate and leads to a faster Tmax after oral dosing to rats

scientific article published on 27 September 2013

Preparation of biodegradable insulin nanocapsules from biocompatible microemulsions

scientific article published in June 2000

Preparation of glass solutions of three poorly water soluble drugs by spray drying, melt extrusion and ball milling

article

Preparation of phytantriol cubosomes by solvent precursor dilution for the delivery of protein vaccines

scientific article published on 13 January 2011

Probing Pharmaceutical Mixtures during Milling: The Potency of Low-Frequency Raman Spectroscopy in Identifying Disorder.

scientific article published in November 2017

Process Optimization and Upscaling of Spray-Dried Drug-Amino acid Co-Amorphous Formulations

scientific article published on 09 January 2019

Properties of the Sodium Naproxen-Lactose-Tetrahydrate Co-Crystal upon Processing and Storage.

scientific article published on 19 April 2016

Protein delivery using nanoparticles based on microemulsions with different structure-types.

scientific article

Pseudo-ternary phase diagrams of aqueous mixtures of Quil A, cholesterol and phospholipid prepared by the lipid-film hydration method

scientific article

Quality of generic medicines in South Africa: perceptions versus reality - a qualitative study

scientific article

Quantification of binary polymorphic mixtures of ranitidine hydrochloride using NIR spectroscopy

Quantification of microwave-induced amorphization of celecoxib in PVP tablets using transmission Raman spectroscopy.

scientific article published on 8 February 2018

Quantification of the types of water in Eudragit RLPO polymer and the kinetics of water loss using FTIR

scientific article published on 19 October 2013

Quantifying ternary mixtures of different solid-state forms of indomethacin by Raman and near-infrared spectroscopy.

scientific article published on 17 July 2007

Quantitative analysis of polymorphic mixtures of ranitidine hydrochloride by Raman spectroscopy and principal components analysis

scientific article

Quantitative solid-state analysis of three solid forms of ranitidine hydrochloride in ternary mixtures using Raman spectroscopy and X-ray powder diffraction

scientific article

Quil A-lipid powder formulations releasing ISCOMs and related colloidal structures upon hydration

scientific article published on 25 January 2005

Raman spectroscopy for quantitative analysis of pharmaceutical solids.

scientific article published on February 2007

Ranitidine hydrochloride X-ray assay using a neural network.

scientific article published in July 2000

Rapid Assessment of Tablet Film Coating Quality by Multispectral UV Imaging

scientific article published on 13 October 2015

Rapid and specific high-performance liquid chromatography for the in vitro quantification of D-Lys6-GnRH in a microemulsion-type formulation in the presence of peptide oxidation products

scientific article published in February 2010

Recent advances and potential applications of modulated differential scanning calorimetry (mDSC) in drug development

scientific article published on 22 December 2015

Recent advances in co-amorphous drug formulations

scientific article

Refining stability and dissolution rate of amorphous drug formulations

scientific article published on 23 April 2014

Relaxation and Crystallization of Amorphous Carbamazepine Studied by Terahertz Pulsed Spectroscopy

scientific article published on 01 October 2007

Release and bioactivity of PACA nanoparticles containing D-Lys6-GnRH for brushtail possum fertility control

scientific article published on 31 October 2010

Screening for differences in the amorphous state of indomethacin using multivariate visualization

scientific article published on 11 November 2006

Selection of excipients for melt extrusion with two poorly water-soluble drugs by solubility parameter calculation and thermal analysis.

scientific article

Self-assembled geometric liquid-crystalline nanoparticles imaged in three dimensions: hexosomes are not necessarily flat hexagonal prisms

scientific article

Self-microemulsifying drug delivery system and nanoemulsion for enhancing aqueous miscibility of Alpinia galanga oil.

scientific article

Silica nanoparticles to control the lipase-mediated digestion of lipid-based oral delivery systems

scientific article published in April 2010

Silica-lipid hybrid (SLH) microcapsules: a novel oral delivery system for poorly soluble drugs

scientific article published on 30 October 2008

Simple measurements for prediction of drug release from polymer matrices – Solubility parameters and intrinsic viscosity

scientific article published on 07 February 2015

Solid Lipid Nanoparticles

article from 2006

Solid State Characterization of Ciprofloxacin Liposome Nanocrystals

scientific article published on 29 November 2018

Solid state properties and drug release behavior of co-amorphous indomethacin-arginine tablets coated with Kollicoat® Protect

scientific article published on 8 June 2017

Solid-State Transition Mechanism in Carbamazepine Polymorphs by Time-Resolved Terahertz Spectroscopy

scientific article published on 01 September 2007

Solid-state properties and dissolution behaviour of tablets containing co-amorphous indomethacin–arginine

scientific article published on 18 July 2015

Solvent change co-precipitation with hydroxypropyl methylcellulose phthalate to improve dissolution characteristics of a poorly water-soluble drug

scientific article published on 01 August 2002

Solvent-mediated amorphous-to-crystalline transformation of nitrendipine in amorphous particle suspensions containing polymers

scientific article published on 29 March 2012

Spatial confinement can lead to increased stability of amorphous indomethacin

scientific article

Spray dried cubosomes with ovalbumin and Quil-A as a nanoparticulate dry powder vaccine formulation

Spray-drying of inhalable, multifunctional formulations for the treatment of biofilms formed in cystic fibrosis

scientific article published on 22 October 2019

Stabilisation of amorphous furosemide increases the oral drug bioavailability in rats

Statistical Analysis of a Method to Predict Drug-Polymer Miscibility

scientific article published on 5 November 2015

Structural Elucidation of Rapid Solution-Mediated Phase Transitions in Pharmaceutical Solids Using in Situ Synchrotron SAXS/WAXS

scientific article published on 14 August 2012

Structural investigations on nanoemulsions, solid lipid nanoparticles and nanostructured lipid carriers by cryo-field emission scanning electron microscopy and Raman spectroscopy

scientific article published on 30 March 2006

Studies on the lipase-induced degradation of lipid-based drug delivery systems. Part II - Investigations on the mechanisms leading to collapse of the lipid structure.

scientific article

Studying the Propensity of Compounds to Supersaturate: A Practical and Broadly Applicable Approach

scientific article published on 31 July 2016

Supersaturated self-nanoemulsifying drug delivery systems (Super-SNEDDS) enhance the bioavailability of the poorly water-soluble drug simvastatin in dogs

scientific article

Supersaturating drug delivery systems: The potential of co-amorphous drug formulations.

scientific article

Supersaturation of zafirlukast in fasted and fed state intestinal media with and without precipitation inhibitors.

scientific article published on 31 May 2016

Swelling lecithin: cholesterol implants for the controlled release of proteins.

scientific article

Synthesis, Formulation, and Adjuvanticity of Monodesmosidic Saponins with Olenanolic Acid, Hederagenin and Gypsogenin Aglycones, and some C-28 Ester Derivatives

scientific article published on 30 September 2015

Systematic Investigation of the Role of Surfactant Composition and Choice of oil: Design of a Nanoemulsion-Based Adjuvant Inducing Concomitant Humoral and CD4+ T-Cell Responses.

scientific article published on 17 May 2017

Temperature dependent terahertz pulsed spectroscopy of carbamazepine

Temperature-Modulated Micromechanical Thermal Analysis with Microstring Resonators Detects Multiple Coherent Features of Small Molecule Glass Transition

scientific article published on 13 February 2020

Terahertz pulsed imaging as an advanced characterisation tool for film coatings--a review.

scientific article published on 06 April 2013

Terahertz pulsed imaging as an analytical tool for sustained-release tablet film coating

scientific article published on 04 July 2008

Terahertz pulsed spectroscopy and imaging in the pharmaceutical setting--a review

scientific article published on February 2007

The Effect of Digestion and Drug Load on Halofantrine Absorption from Self-nanoemulsifying Drug Delivery System (SNEDDS).

scientific article published on 20 October 2015

The Influence of Milling on the Dissolution Performance of Simvastatin.

scientific article published on 17 December 2010

The Influence of Polymers on the Supersaturation Potential of Poor and Good Glass Formers

scientific article published on 21 September 2018

The Precipitation Behavior of Poorly Water-Soluble Drugs with an Emphasis on the Digestion of Lipid Based Formulations.

scientific article

The Role of Configurational Entropy in Amorphous Systems.

scientific article published on 25 May 2010

The Role of Glass Transition Temperatures in Coamorphous Drug–Amino Acid Formulations

scientific article published on 30 July 2018

The ability of two in vitro lipolysis models reflecting the human and rat gastro-intestinal conditions to predict the in vivo performance of SNEDDS dosing regimens

scientific article published on 27 December 2017

The administration route is decisive for the ability of the vaccine adjuvant CAF09 to induce antigen-specific CD8(+) T-cell responses: The immunological consequences of the biodistribution profile

scientific article published on 26 August 2016

The application of MALDI TOF MS in biopharmaceutical research ⬇️

scientific article published on December 13, 2010

The effect of surfactants on the dissolution behavior of amorphous formulations

scientific article published on 05 March 2016

The impact of surface- and nano-crystallisation on the detected amorphous content and the dissolution behaviour of amorphous indomethacin

scientific article published on 06 June 2012

The influence of co-formers on the dissolution rates of co-amorphous sulfamerazine/excipient systems

scientific article published on 16 March 2016

The influence of pressure on the intrinsic dissolution rate of amorphous indomethacin

scientific article published on 20 August 2014

The influence of thermal and mechanical preparative techniques on the amorphous state of four poorly soluble compounds

scientific article published in September 2005

The influence of various excipients on the conversion kinetics of carbamazepine polymorphs in aqueous suspension

article

The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion

scientific article

The significance of the amorphous potential energy landscape for dictating glassy dynamics and driving solid-state crystallisation

scientific article published on 2 November 2017

The use of molecular descriptors in the development of co-amorphous formulations

scientific article published on 9 April 2018

Themed issue: Improve dissolution, solubility and bioavailability of poorly soluble drugs

scientific article published on 01 November 2010

Thermal degradation of amorphous glibenclamide

scientific article

Thermotropic liquid crystalline drugs.

scientific article

Towards characterization and identification of solid state pharmaceutical mixtures through second harmonic generation

scientific article published in April 2006

Transcutaneous immunization using microneedles and cubosomes: Mechanistic investigations using Optical Coherence Tomography and Two-Photon Microscopy

scientific article published on 23 August 2013

Transdermal delivery of hydrophobic and hydrophilic local anesthetics from o/w and w/o Brij 97-based microemulsions.

scientific article published in January 2007

Transformations between Co-Amorphous and Co-Crystal Systems and Their Influence on the Formation and Physical Stability of Co-Amorphous Systems

scientific article published on 25 January 2019

UV imaging of Multiple Unit Pellet System (MUPS) tablets: A case study of acetylsalicylic acid stability.

scientific article published on 02 August 2017

Ultrasensitive Microstring Resonators for Solid State Thermomechanical Analysis of Small and Large Molecules

scientific article published on 05 December 2018

Understanding the influence of polymorphism on phonon spectra: lattice dynamics calculations and terahertz spectroscopy of carbamazepine.

scientific article published in January 2006

Understanding the solid-state forms of fenofibrate--a spectroscopic and computational study

scientific article published on 12 June 2008

Undesired co-amorphisation of indomethacin and arginine during combined storage at high humidity conditions

scientific article published on 15 April 2018

Unintended and in situ amorphisation of pharmaceuticals.

scientific article published on 23 December 2015

Unravelling the relationship between degree of disorder and the dissolution behavior of milled glibenclamide

scientific article published on 17 December 2013

Using Potentiometric Free Drug Sensors to Determine the Free Concentration of Ionizable Drugs in Colloidal Systems

scientific article published on 23 May 2017

Using different structure types of microemulsions for the preparation of poly(alkylcyanoacrylate) nanoparticles by interfacial polymerization.

scientific article published in August 2005

Using in vitro lipolysis and SPECT/CT in vivo imaging to understand oral absorption of fenofibrate from lipid-based drug delivery systems

scientific article published on 23 November 2019

Using terahertz pulsed spectroscopy to quantify pharmaceutical polymorphism and crystallinity

scientific article published in April 2005

Using terahertz pulsed spectroscopy to study crystallinity of pharmaceutical materials

Utilizing nanoparticles for improving anti-biofilm effects of azithromycin: A head-to-head comparison of modified hyaluronic acid nanogels and coated poly (lactic-co-glycolic acid) nanoparticles

scientific article published on 03 August 2019

Visualizing solvent mediated phase transformation behavior of carbamazepine polymorphs by principal component analysis

scientific article published on 21 February 2008

Visualizing the conversion of carbamazepine in aqueous suspension with and without the presence of excipients: A single crystal study using SEM and Raman microscopy

scientific article published on 03 June 2006

W/O microemulsions for ocular delivery: evaluation of ocular irritation and precorneal retention.

scientific article published on 19 January 2006

Whey proteins as stabilizers in amorphous solid dispersions

scientific article published on 04 December 2018

pH-triggered drug release from biodegradable microwells for oral drug delivery

scientific article published on June 2015

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