List of works - Kathy Andrews

A novel in vitro image-based assay identifies new drug leads for giardiasis.

scientific article published on 27 January 2017

Acaricidal activity of eugenol based compounds against scabies mites

scientific article

Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites

scientific article published on 26 March 2018

Adaptation of the [3H]Hypoxanthine Uptake Assay for In Vitro-Cultured Plasmodium knowlesi Malaria Parasites.

scientific article published on 25 April 2016

Adherence of Plasmodium falciparum infected erythrocytes to CHO-745 cells and inhibition of binding by protein A in the presence of human serum

scientific article published on September 2005

An ELISA method to assess HDAC inhibitor-induced alterations to P. falciparum histone lysine acetylation

scientific article published on 02 November 2020

Anti-malarial effect of histone deacetylation inhibitors and mammalian tumour cytodifferentiating agents

scientific article published in May 2000

Antimalarial Isocyano and Isothiocyanato Sesquiterpenes with Tri- and Bicyclic Skeletons from the Nudibranch Phyllidia ocellata

scientific article published on 09 June 2015

Antimalarial activity of azadipeptide nitriles

scientific article

Antimalarial activity of compounds comprising a primary benzene sulfonamide fragment.

scientific article published on 14 September 2013

Antimalarial activity of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors

scientific article published on 21 July 2008

Antimalarial activity of pyrroloiminoquinones from the Australian marine sponge Zyzzya sp. ⬇️

scientific article

Antimalarial activity of sera from subjects taking HIV protease inhibitors.

scientific article published on March 2007

Antimalarial activity of the anticancer histone deacetylase inhibitor SB939.

scientific article

Antimalarial asexual stage-specific and gametocytocidal activities of HIV protease inhibitors

scientific article published on 22 December 2009

Antimalarial histone deacetylase inhibitors containing cinnamate or NSAID components

scientific article published on 22 September 2010

Antiparasitic activity of alkaloids from plant species of Papua New Guinea and Australia.

scientific article published on 26 June 2010

Antiretrovirals as antimalarial agents.

scientific article published on 3 November 2004

Apparent bias for P. falciparum parasites carrying the wild-type pfcrt allele in the placenta

scientific article published on 11 February 2010

Carrageenans inhibit the in vitro growth of Plasmodium falciparum and cytoadhesion to CD36.

scientific article published on 13 July 2005

Catalyst-Controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile-1.

scientific article published on 10 November 2017

Chemical investigation of an antimalarial Chinese medicinal herb Picrorhiza scrophulariiflora.

scientific article published on 27 August 2013

Comparative gene expression profiling of P. falciparum malaria parasites exposed to three different histone deacetylase inhibitors

scientific article

Comparison of different PCR protocols for the detection and diagnosis of Plasmodium falciparum

scientific article published on 7 September 2005

Correction to Catalyst-Controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile-1

scientific article published on 31 July 2018

Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone

scientific article published on 03 May 2019

Defining the targets of antiparasitic compounds.

scientific article

Design and synthesis of screening libraries based on the muurolane natural product scaffold.

scientific article

Direct activation of human endothelial cells by Plasmodium falciparum-infected erythrocytes

scientific article published on June 2005

Discovery of HDAC inhibitors with potent activity against multiple malaria parasite life cycle stages

scientific article

Drug repurposing and human parasitic protozoan diseases

scientific article

Effect of cytokine treatment on the in vitro expression of the P. falciparum adhesion receptor chondroitin-4-sulphate on the surface of human choriocarcinoma (BeWo) cells

scientific article published on 16 February 2007

Effect of sequence variation in Plasmodium falciparum histidine- rich protein 2 on binding of specific monoclonal antibodies: Implications for rapid diagnostic tests for malaria

scientific article

Entonalactams A-C: Isoindolinone derivatives from an Australian rainforest fungus belonging to the genus Entonaema.

scientific article published on 3 June 2015

Erratum to "Profiling the anti-protozoal activity of anti-cancer HDAC inhibitors against Plasmodium and Trypanosoma parasites" [Int. J. Parasitol. Drugs Drug Res. 5 (2015) 117-126].

scientific article published on 30 May 2016

Evaluation of the role of the endocytic receptor L-SIGN for cytoadhesion of Plasmodium falciparum-infected erythrocytes

scientific article published on 4 May 2005

Evidence for trafficking of PfEMP1 to the surface of P. falciparum-infected erythrocytes via a complex membrane network

scientific article published in June 2003

Ex vivo activity of histone deacetylase inhibitors against multidrug-resistant clinical isolates of Plasmodium falciparum and P. vivax

scientific article

FgoI, a Type II restriction endonuclease from the thermoanaerobeFervidobacterium gondwanenseAB39T

scientific article published on 01 October 1998

HDAC inhibitors in parasitic diseases ⬇️

scientific article published on November 29, 2011

HIV and malaria co-infection: interactions and consequences of chemotherapy.

scientific article published on 02 May 2008

Histone deacetylase inhibitor AR-42 and achiral analogues kill malaria parasites in vitro and in mice

scientific article published in December 2021

Identification of novel quinazoline derivatives as potent antiplasmodial agents

scientific article published on 17 October 2018

Inhibition of Plasmodium falciparum growth in vitro and adhesion to chondroitin-4-sulfate by the heparan sulfate mimetic PI-88 and other sulfated oligosaccharides.

scientific article

Inhibition of chondroitin-4-sulfate-specific adhesion of Plasmodium falciparum-infected erythrocytes by sulfated polysaccharides

scientific article

Intrapulmonary pharmacokinetics of antibiotics used to treat nosocomial pneumonia caused by Gram-negative bacilli: A systematic review

scientific article published on 23 November 2018

Lysine acetylation in sexual stage malaria parasites is a target for antimalarial small molecules.

scientific article

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond

scientific article (publication date: July 2016)

Pestalactams A-C: novel caprolactams from the endophytic fungus Pestalotiopsis sp. ⬇️

scientific article

Plagiarism

scientific article published in August 2009

Plasmodium falciparum: new molecular targets with potential for antimalarial drug development

scientific article

Plasmodium gametocyte inhibition identified from a natural-product-based fragment library

scientific article

Potencies of human immunodeficiency virus protease inhibitors in vitro against Plasmodium falciparum and in vivo against murine malaria

scientific article

Potent antimalarial activity of histone deacetylase inhibitor analogues.

scientific article published on 22 January 2008

Profiling the anti-protozoal activity of anti-cancer HDAC inhibitors against Plasmodium and Trypanosoma parasites

scientific article published on 20 June 2015

Proteomic analysis of Plasmodium falciparum histone deacetylase 1 complex proteins

Psammaplysin H, a new antimalarial bromotyrosine alkaloid from a marine sponge of the genus Pseudoceratina.

scientific article published on 21 November 2010

Psammaplysin derivatives from the Balinese marine sponge Aplysinella strongylata

scientific article

Recovery of adhesion to chondroitin-4-sulphate in Plasmodium falciparum varCSA disruption mutants by antigenically similar PfEMP1 variants

scientific article

Reevaluating the classification of Halobacteroides and Haloanaerobacter species based on sequence comparisons of the 16S ribosomal RNA gene

scientific article published in December 1995

Regioselectively modified sulfated cellulose as prospective drug for treatment of malaria tropica

scientific article published on January 2007

Stronger activity of human immunodeficiency virus type 1 protease inhibitors against clinical isolates of Plasmodium vivax than against those of P. falciparum.

scientific article published on 28 April 2008

Structural basis for binding of Plasmodium falciparum erythrocyte membrane protein 1 to chondroitin sulfate and placental tissue and the influence of protein polymorphisms on binding specificity

scientific article published on 11 June 2007

Structure-Activity and Structure-Toxicity Relationships of Peptoid-Based Histone Deacetylase Inhibitors with Dual-Stage Antiplasmodial Activity

scientific article published on 19 February 2019

Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum

scientific article published on 11 December 2014

Synergistic interactions of the antiretroviral protease inhibitors saquinavir and ritonavir with chloroquine and mefloquine against Plasmodium falciparum in vitro.

scientific article published on 6 November 2006

Synthesis and Antiplasmodial Evaluation of Analogues Based on the Tricyclic Core of Thiaplakortones A-D.

scientific article

Synthesis and antimalarial evaluation of amide and urea derivatives based on the thiaplakortone A natural product scaffold

scientific article

Synthesis and antimalarial evaluation of novel benzopyrano[4,3-b]benzopyran derivatives

scientific article published on 23 July 2011

Synthesis and evaluation of antimalarial properties of novel 4-aminoquinoline hybrid compounds

scientific article published on 3 June 2014

Synthesis, antimalarial properties, and SAR studies of alkoxyurea-based HDAC inhibitors.

scientific article published on 4 February 2014

Synthesis, biological characterisation and structure activity relationships of aromatic bisamidines active against Plasmodium falciparum

scientific article published on 23 December 2016

The Key Glycolytic Enzyme Phosphofructokinase Is Involved in Resistance to Antiplasmodial Glycosides.

scientific article published on 8 December 2020

The activity of protease inhibitors against Giardia duodenalis and metronidazole-resistant Trichomonas vaginalis.

scientific article

The histone H4 gene of Plasmodium falciparum is developmentally transcribed in asexual parasites

scientific article published on 9 May 2003

Total synthesis of thiaplakortone a: derivatives as metabolically stable leads for the treatment of malaria

scientific article

List of works by Kathy Andrews

A novel in vitro image-based assay identifies new drug leads for giardiasis.

Acaricidal activity of eugenol based compounds against scabies mites

Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites

Adaptation of the [3H]Hypoxanthine Uptake Assay for In Vitro-Cultured Plasmodium knowlesi Malaria Parasites.

Adherence of Plasmodium falciparum infected erythrocytes to CHO-745 cells and inhibition of binding by protein A in the presence of human serum

An ELISA method to assess HDAC inhibitor-induced alterations to P. falciparum histone lysine acetylation

Anti-malarial effect of histone deacetylation inhibitors and mammalian tumour cytodifferentiating agents

Antimalarial Isocyano and Isothiocyanato Sesquiterpenes with Tri- and Bicyclic Skeletons from the Nudibranch Phyllidia ocellata

Antimalarial activity of azadipeptide nitriles

Antimalarial activity of compounds comprising a primary benzene sulfonamide fragment.

Antimalarial activity of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors

Antimalarial activity of pyrroloiminoquinones from the Australian marine sponge Zyzzya sp. ⬇️

Antimalarial activity of sera from subjects taking HIV protease inhibitors.

Antimalarial activity of the anticancer histone deacetylase inhibitor SB939.

Antimalarial asexual stage-specific and gametocytocidal activities of HIV protease inhibitors

Antimalarial histone deacetylase inhibitors containing cinnamate or NSAID components

Antiparasitic activity of alkaloids from plant species of Papua New Guinea and Australia.

Antiretrovirals as antimalarial agents.

Apparent bias for P. falciparum parasites carrying the wild-type pfcrt allele in the placenta

Carrageenans inhibit the in vitro growth of Plasmodium falciparum and cytoadhesion to CD36.

Catalyst-Controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile-1.

Chemical investigation of an antimalarial Chinese medicinal herb Picrorhiza scrophulariiflora.

Comparative gene expression profiling of P. falciparum malaria parasites exposed to three different histone deacetylase inhibitors

Comparison of different PCR protocols for the detection and diagnosis of Plasmodium falciparum

Correction to Catalyst-Controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile-1

Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone

Defining the targets of antiparasitic compounds.

Design and synthesis of screening libraries based on the muurolane natural product scaffold.

Direct activation of human endothelial cells by Plasmodium falciparum-infected erythrocytes

Discovery of HDAC inhibitors with potent activity against multiple malaria parasite life cycle stages

Drug repurposing and human parasitic protozoan diseases

Effect of cytokine treatment on the in vitro expression of the P. falciparum adhesion receptor chondroitin-4-sulphate on the surface of human choriocarcinoma (BeWo) cells

Effect of sequence variation in Plasmodium falciparum histidine- rich protein 2 on binding of specific monoclonal antibodies: Implications for rapid diagnostic tests for malaria

Entonalactams A-C: Isoindolinone derivatives from an Australian rainforest fungus belonging to the genus Entonaema.

Erratum to "Profiling the anti-protozoal activity of anti-cancer HDAC inhibitors against Plasmodium and Trypanosoma parasites" [Int. J. Parasitol. Drugs Drug Res. 5 (2015) 117-126].

Evaluation of the role of the endocytic receptor L-SIGN for cytoadhesion of Plasmodium falciparum-infected erythrocytes

Evidence for trafficking of PfEMP1 to the surface of P. falciparum-infected erythrocytes via a complex membrane network

Ex vivo activity of histone deacetylase inhibitors against multidrug-resistant clinical isolates of Plasmodium falciparum and P. vivax

FgoI, a Type II restriction endonuclease from the thermoanaerobeFervidobacterium gondwanenseAB39T

HDAC inhibitors in parasitic diseases ⬇️

HIV and malaria co-infection: interactions and consequences of chemotherapy.

Histone deacetylase inhibitor AR-42 and achiral analogues kill malaria parasites in vitro and in mice

Identification of novel quinazoline derivatives as potent antiplasmodial agents

Inhibition of Plasmodium falciparum growth in vitro and adhesion to chondroitin-4-sulfate by the heparan sulfate mimetic PI-88 and other sulfated oligosaccharides.

Inhibition of chondroitin-4-sulfate-specific adhesion of Plasmodium falciparum-infected erythrocytes by sulfated polysaccharides

Intrapulmonary pharmacokinetics of antibiotics used to treat nosocomial pneumonia caused by Gram-negative bacilli: A systematic review

Lysine acetylation in sexual stage malaria parasites is a target for antimalarial small molecules.

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond

Pestalactams A-C: novel caprolactams from the endophytic fungus Pestalotiopsis sp. ⬇️

Plagiarism

Plasmodium falciparum: new molecular targets with potential for antimalarial drug development

Plasmodium gametocyte inhibition identified from a natural-product-based fragment library

Potencies of human immunodeficiency virus protease inhibitors in vitro against Plasmodium falciparum and in vivo against murine malaria

Potent antimalarial activity of histone deacetylase inhibitor analogues.

Profiling the anti-protozoal activity of anti-cancer HDAC inhibitors against Plasmodium and Trypanosoma parasites

Proteomic analysis of Plasmodium falciparum histone deacetylase 1 complex proteins

Psammaplysin H, a new antimalarial bromotyrosine alkaloid from a marine sponge of the genus Pseudoceratina.

Psammaplysin derivatives from the Balinese marine sponge Aplysinella strongylata

Recovery of adhesion to chondroitin-4-sulphate in Plasmodium falciparum varCSA disruption mutants by antigenically similar PfEMP1 variants

Reevaluating the classification of Halobacteroides and Haloanaerobacter species based on sequence comparisons of the 16S ribosomal RNA gene

Regioselectively modified sulfated cellulose as prospective drug for treatment of malaria tropica

Stronger activity of human immunodeficiency virus type 1 protease inhibitors against clinical isolates of Plasmodium vivax than against those of P. falciparum.

Structural basis for binding of Plasmodium falciparum erythrocyte membrane protein 1 to chondroitin sulfate and placental tissue and the influence of protein polymorphisms on binding specificity

Structure-Activity and Structure-Toxicity Relationships of Peptoid-Based Histone Deacetylase Inhibitors with Dual-Stage Antiplasmodial Activity

Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum

Synergistic interactions of the antiretroviral protease inhibitors saquinavir and ritonavir with chloroquine and mefloquine against Plasmodium falciparum in vitro.

Synthesis and Antiplasmodial Evaluation of Analogues Based on the Tricyclic Core of Thiaplakortones A-D.

Synthesis and antimalarial evaluation of amide and urea derivatives based on the thiaplakortone A natural product scaffold

Synthesis and antimalarial evaluation of novel benzopyrano[4,3-b]benzopyran derivatives

Synthesis and evaluation of antimalarial properties of novel 4-aminoquinoline hybrid compounds

Synthesis, antimalarial properties, and SAR studies of alkoxyurea-based HDAC inhibitors.

Synthesis, biological characterisation and structure activity relationships of aromatic bisamidines active against Plasmodium falciparum

The Key Glycolytic Enzyme Phosphofructokinase Is Involved in Resistance to Antiplasmodial Glycosides.

The activity of protease inhibitors against Giardia duodenalis and metronidazole-resistant Trichomonas vaginalis.

The histone H4 gene of Plasmodium falciparum is developmentally transcribed in asexual parasites

Total synthesis of thiaplakortone a: derivatives as metabolically stable leads for the treatment of malaria