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List of works by Anders Hallberg

3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1

scholarly article by Benjamin Pelcman published in August 2015

A convenient synthesis of 1-(S)-[1′-(S)-(t-butyloxycarbonylamino)-2′-phenylethyl]oxirane. A useful building block in the synthesis of HIV protease inhibitors

article

A frame shifted disulfide bridged analogue of angiotensin II

scientific article published on 01 March 2003

A new class of HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold

scientific article published in December 2005

A new highly asymmetric chelation-controlled heck arylation

scientific article published in March 2003

A new regioselective Heck vinylation with enamides. Synthesis and investigation of fluorous-tagged bidentate ligands for fast separation

scientific article

A new structural theme in C2-symmetric HIV-1 protease inhibitors: ortho-substituted P1/P1' side chains

scientific article published on 18 April 2006

A one-pot isomerization-arylation of 2,3-epoxycyclohexanone under controlled microwave heating

scientific article published in June 2005

A selective AT2 receptor ligand with a gamma-turn-like mimetic replacing the amino acid residues 4-5 of angiotensin II.

scientific article

AT2-receptor stimulation enhances axonal plasticity after spinal cord injury by upregulating BDNF expression

scientific article published on 19 November 2012

AT2-selective angiotensin II analogues containing tyrosine-functionalized 5,5-bicyclic thiazabicycloalkane dipeptide mimetics.

scientific article

Acyl sulfonamides as potent protease inhibitors of the hepatitis C virus full-Length NS3 (protease-helicase/NTPase): a comparative study of different C-terminals

scientific article

Angiotensin AT2-receptor stimulation improves survival and neurological outcome after experimental stroke in mice

scientific article

Angiotensin II pseudopeptides containing 1,3,5-trisubstituted benzene scaffolds with high AT2 receptor affinity

scientific article published on October 2005

Angiotensin II type 2 receptor promotes adipocyte differentiation and restores adipocyte size in high-fat/high-fructose diet-induced insulin resistance in rats

scientific article published on 13 November 2012

Angiotensin II type 2 receptor stimulation improves fatty acid ovarian uptake and hyperandrogenemia in an obese rat model of polycystic ovary syndrome

scientific article published on 27 June 2014

Angiotensin II type 2 receptor stimulation: a novel option of therapeutic interference with the renin-angiotensin system in myocardial infarction?

scientific article

Angiotensin II, a neuropeptide at the frontier between endocrinology and neuroscience: is there a link between the angiotensin II type 2 receptor and Alzheimer’s disease? ⬇️

scientific article published on August 26, 2011

Angiotensin Peptides as AT2 Receptor Agonists

scientific article

Angiotensin type 2 receptor (AT2R) and receptor Mas: a complex liaison

scientific article

Angiotensin type 2 receptor stimulation ameliorates left ventricular fibrosis and dysfunction via regulation of tissue inhibitor of matrix metalloproteinase 1/matrix metalloproteinase 9 axis and transforming growth factor β1 in the rat heart

scientific article published on 30 December 2013

Aryl Radical Endo Cyclization of Enamidines. Selective Preparation of Trans and Cis Fused Octahydrobenzo[f]quinolines ⬇️

scientific article published on 01 January 1998

Aspartic protease inhibitors containing tertiary alcohol transition-state mimics

scientific article

Bicyclic Tripeptide Mimetics with Reverse Turn Inducing Properties

C2-symmetric inhibitors of Plasmodium falciparum plasmepsin II: synthesis and theoretical predictions

scientific article

Comparative functional properties of two structurally similar selective nonpeptide drug-like ligands for the angiotensin II type-2 (AT2) receptor. Effects on neurite outgrowth in NG108-15 cells ⬇️

scientific article published on December 2, 2012

Controlled Double-Bond Migration in Palladium-Catalyzed Intramolecular Arylation of Enamidines ⬇️

scientific article published on 01 October 1996

Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'.

scientific article published in February 2005

Design and synthesis of HIV-1 protease inhibitors. Novel tetrahydrofuran P2/P2'-groups interacting with Asp29/30 of the HIV-1 protease. Determination of binding from X-ray crystal structure of inhibitor protease complex

scientific article

Design and synthesis of P1-P3 macrocyclic tertiary-alcohol-comprising HIV-1 protease inhibitors

scientific article

Design and synthesis of dihydrofolate reductase inhibitors encompassing a bridging ester group. Evaluation in a mouse colitis model

scientific article published in July 2003

Design and synthesis of novel P2 substituents in diol-based HIV protease inhibitors

scientific article

Design and synthesis of plasmepsin I and plasmepsin II inhibitors with activity in Plasmodium falciparum-infected cultured human erythrocytes

scientific article published in February 2003

Design and synthesis of potent and selective BACE-1 inhibitors

scientific article

Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin II.

scientific article published in June 2005

Design and synthesis of potent inhibitors of the malaria aspartyl proteases plasmepsin I and II. Use of solid-phase synthesis to explore novel statine motifs

scientific article published in June 2004

Design, synthesis and SAR of potent statine-based BACE-1 inhibitors: exploration of P1 phenoxy and benzyloxy residues

scientific article

Design, synthesis, and biological evaluation of the first selective nonpeptide AT2 receptor agonist.

scientific article

Design, synthesis, and computational affinity prediction of ester soft drugs as inhibitors of dihydrofolate reductase from Pneumocystis carinii

scientific article published in May 2004

Design, synthesis, and incorporation of a beta-turn mimetic in angiotensin II forming novel pseudopeptides with affinity for AT1 and AT2 receptors

scientific article published in October 2006

Dimethylformamide as a carbon monoxide source in fast palladium-catalyzed aminocarbonylations of aryl bromides

scientific article

Direct angiotensin II type 2 receptor stimulation acts anti-inflammatory through epoxyeicosatrienoic acid and inhibition of nuclear factor kappaB.

scientific article

Direct angiotensin type 2 receptor (AT2R) stimulation attenuates T-cell and microglia activation and prevents demyelination in experimental autoimmune encephalomyelitis in mice

scientific article published in January 2015

Discovery of potent BACE-1 inhibitors containing a new hydroxyethylene (HE) scaffold: exploration of P1' alkoxy residues and an aminoethylene (AE) central core

scientific article

Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP).

scientific article published on 3 November 2010

Effect of 3-5 monocyclizations of angiotensin II and 4-aminoPhe6-Ang II on AT2 receptor affinity

scientific article

Evolution of Angiotensin Peptides and Peptidomimetics as Angiotensin II Receptor Type 2 (AT2) Receptor Agonists

scientific article published on 23 April 2020

Exploration of acyl sulfonamides as carboxylic acid replacements in protease inhibitors of the hepatitis C virus full-length NS3.

scientific article published on 5 October 2005

Fast synthesis of aryl triflates with controlled microwave heating

scientific article

First reported nonpeptide AT1 receptor agonist (L-162,313) acts as an AT2 receptor agonist in vivo

scientific article

Fmoc protected peptide mimetic based on a cyclohexane framework and incorporation into angiotensin II

Formamide as a combined ammonia synthon and carbon monoxide source in fast palladium-catalyzed aminocarbonylations of aryl halides

scientific article

From the first selective non-peptide AT(2) receptor agonist to structurally related antagonists

scientific article

HIV-1 Protease Inhibitors Based on Acyclic Carbohydrates

article

HIV-1 protease inhibitors with a transition-state mimic comprising a tertiary alcohol: improved antiviral activity in cells

scientific article

High-speed heck reactions in ionic liquid with controlled microwave heating

scientific article

High-speed synthesis of potent C2-symmetric HIV-1 protease inhibitors by in-situ aminocarbonylations

scientific article published in July 2005

In situ generation of carbon monoxide from solid molybdenum hexacarbonyl. A convenient and fast route to palladium-catalyzed carbonylation reactions

scientific article published on 01 March 2002

Inhibitor binding to the plasmepsin IV aspartic protease from Plasmodium falciparum

scientific article published in September 2006

Insulin-regulated aminopeptidase inhibitor-mediated increases in dendritic spine density are facilitated by glucose uptake

scientific article published on 26 September 2019

Intramolecular Enantioselective Palladium-Catalyzed Heck Arylation of Cyclic Enamides ⬇️

scientific article published on 01 February 1997

Macrocyclic inhibitors of the malarial aspartic proteases plasmepsin I, II, and IV.

scientific article published on 22 November 2005

Masked 3-aminoindan-1-ones by a palladium-catalyzed three-component annulation reaction

scientific article

Microwave-accelerated homogeneous catalysis in organic chemistry

scientific article

Microwave-accelerated synthesis of P1'-extended HIV-1 protease inhibitors encompassing a tertiary alcohol in the transition-state mimicking scaffold

scientific article published in March 2006

N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands

scientific article published on 07 November 2020

N-Aryl Isoleucine Derivatives as Angiotensin II AT2 Receptor Ligands

scientific article

N-Substituted pyrazole-3-carboxamides as inhibitors of human 15-lipoxygenase

scholarly article by Benjamin Pelcman published in August 2015

New inhibitors of the malaria aspartyl proteases plasmepsin I and II.

scientific article published in August 2003

New potent C2-symmetric malaria plasmepsin I and II inhibitors

scientific article published in April 2003

New selective AT2 receptor ligands encompassing a gamma-turn mimetic replacing the amino acid residues 4-5 of angiotensin II act as agonists.

scientific article published in June 2005

Non-peptide AT2-receptor agonists

scientific article published on 15 December 2010

Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: use of cyclopentane and cyclopentene P2-motifs

scientific article published on 22 August 2007

Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors

scientific article (publication date: April 2003)

P2'-truncated BACE-1 inhibitors with a novel hydroxethylene-like core.

scientific article published on 3 November 2009

Peptide-based inhibitors of hepatitis C virus full-length NS3 (protease-helicase/NTPase): model compounds towards small molecule inhibitors.

scientific article published in July 2003

Plasmepsins as potential targets for new antimalarial therapy

scientific article published in September 2006

Potent inhibitors of the Plasmodium falciparum enzymes plasmepsin I and II devoid of cathepsin D inhibitory activity

scientific article

Potent inhibitors of the hepatitis C virus NS3 protease: use of a novel P2 cyclopentane-derived template

scientific article published on 3 May 2006

Potent macrocyclic inhibitors of insulin-regulated aminopeptidase (IRAP) by olefin ring-closing metathesis.

scientific article published on 9 May 2011

Preparation of cis-5-methoxy-and-7-methoxy-1-acetoxy-1,2,3,4,4a,10a- hexahydro-9(10H)-phenanthrenone. An epoxide-arene reaction involving a selective 1,2-alkyl shift rearrangement

Presentation of a structurally diverse and commercially available drug data set for correlation and benchmarking studies

scientific article

Protected indanones by a Heck-aldol annulation reaction

scientific article

Rapid palladium-catalyzed synthesis of esters from aryl halides utilizing Mo(CO)(6) as a solid carbon monoxide source

scientific article

Regiochemical Control and Suppression of Double Bond Isomerization in the Heck Arylation of 1-(Methoxycarbonyl)-2,5-dihydropyrrole ⬇️

scientific article published on July 12, 1996

Relationships between structure and interaction kinetics for HIV-1 protease inhibitors

scientific article

Selective angiotensin II AT(2) receptor agonists with reduced CYP 450 inhibition

scientific article

Selective angiotensin II AT2 receptor agonists: Benzamide structure-activity relationships

scientific article

Selective terminal heck arylation of vinyl ethers with aryl chlorides: a combined experimental-computational approach including synthesis of betaxolol

scientific article published in May 2006

Short pseudopeptides containing turn scaffolds with high AT2 receptor affinity

scientific article published on 05 June 2006

Small-molecule AT2 receptor agonists

scientific article

Solid-phase library synthesis of reversed-statine type inhibitors of the malarial aspartyl proteases plasmepsin I and II.

scientific article

Stereoselective synthesis of 3-aminoindan-1-ones and subsequent incorporation into HIV-1 protease inhibitors

scientific article published in February 2006

Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

scientific article published on 25 April 2018

Structural determinants of subtype selectivity and functional activity of angiotensin II receptors

scientific article published on 29 October 2015

Structure-activity relationships for the selectivity of hepatitis C virus NS3 protease inhibitors.

scientific article published in April 2004

Symmetric fluoro-substituted diol-based HIV protease inhibitors. Ortho-fluorinated and meta-fluorinated P1/P1'-benzyloxy side groups significantly improve the antiviral activity and preserve binding efficacy

scientific article published in November 2004

Synthesis and Comparative Molecular Field Analysis (CoMFA) of Symmetric and Nonsymmetric Cyclic Sulfamide HIV-1 Protease Inhibitors

article

Synthesis of a new class of druglike angiotensin II C-terminal mimics with affinity for the AT2 receptor

scientific article

Synthesis of enantiomerically pure cis and trans 2-aminocyclopentanecarboxylic acids. Use of proline replacements in potential HIV-protease inhibitors

article

Synthesis of malarial plasmepsin inhibitors and prediction of binding modes by molecular dynamics simulations

scientific article published in September 2005

Synthesis of novel potent hepatitis C virus NS3 protease inhibitors: discovery of 4-hydroxy-cyclopent-2-ene-1,2-dicarboxylic acid as a N-acyl-L-hydroxyproline bioisostere

scientific article published on 25 October 2006

Synthesis of potent BACE-1 inhibitors incorporating a hydroxyethylene isostere as central core

scientific article

Synthesis ofC2Symmetric Potential Inhibitors of HIV-1 Protease From D-Mannitol

article

Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II.

scientific article published in September 2005

Tetrapeptides as potent protease inhibitors of Hepatitis C Virus full-length NS3 (protease-helicase/NTPase).

scientific article

Two-carbon-elongated HIV-1 protease inhibitors with a tertiary-alcohol-containing transition-state mimic

scientific article

Variations of the P2 group in HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold

scientific article published on 6 July 2006

Vinyl sulfide cyclized analogues of angiotensin II with high affinity and full agonist activity at the AT(1) receptor

scientific article published in April 2002

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