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List of works by Maurizio Pellecchia

A functional variant of lymphoid tyrosine phosphatase is associated with type I diabetes

scientific article (publication date: April 2004)

A novel small-molecule binds to the influenza A virus RNA promoter and inhibits viral replication

scientific article

Aryl-fluorosulfate-based Lysine Covalent Pan-Inhibitors of Apoptosis Protein (IAP) Antagonists with Cellular Efficacy

scientific article published on 08 October 2019

Control of vesicle fusion by a tyrosine phosphatase

scientific article

Covalent Inhibitors of Protein-Protein Interactions Targeting Lysine, Tyrosine, or Histidine Residues

scientific article published on 29 May 2019

Design of Potent pan-IAP and Lys-Covalent XIAP Selective Inhibitors Using a Thermodynamics Driven Approach

scientific article published on 09 July 2018

Discovery and binding studies on a series of novel Pin1 ligands

scientific article

Endoplasmic reticulum membrane reorganization is regulated by ionic homeostasis

scientific article

Enthalpy-Based Screening of Focused Combinatorial Libraries for the Identification of Potent and Selective Ligands.

scientific article published on 2 November 2017

Functional specialization in proline biosynthesis of melanoma

scientific journal article

Inhibition of Yersinia tyrosine phosphatase by furanyl salicylate compounds

scientific article

Multidentate Small-Molecule Inhibitors of Vaccinia H1-Related (VHR) Phosphatase Decrease Proliferation of Cervix Cancer Cells

scientific article

N-locking stabilization of covalent helical peptides: Application to Bfl-1 antagonists

scientific article published on 20 January 2020

NMR Studies of a Heterotypic Sam−Sam Domain Association: The Interaction between the Lipid Phosphatase Ship2 and the EphA2 Receptor † , ‡

scientific article

New crystal structures of HSC-70 ATP binding domain confirm the role of individual binding pockets and suggest a new method of inhibition

scientific article

Potential Therapeutic Targeting of Coronavirus Spike Glycoprotein Priming

scientific article published on 22 May 2020

Reduction of Circulating Cancer Cells and Metastases in Breast-Cancer Models by a Potent EphA2-Agonistic Peptide-Drug Conjugate.

scientific article published on 22 February 2018

Structural analysis of Siah1-Siah-interacting protein interactions and insights into the assembly of an E3 ligase multiprotein complex

scientific article

Structure-Based Design of Covalent Siah Inhibitors

scientific article

Structure-Based Design of Novel EphA2 Agonistic Agents with Nanomolar Affinity in Vitro and in Cell.

scientific article

Targeting Mcl-1 for the therapy of cancer

scientific article

Targeting Zinc Finger Domains with Small Molecules: Solution Structure and Binding Studies of the RanBP2-Type Zinc Finger of RBM5

scientific article

Targeting the Bcl-2 family for cancer therapy

scientific article

The FRB domain of mTOR: NMR solution structure and inhibitor design

scientific article

The PTB domain of tensin: NMR solution structure and phosphoinositides binding studies

scientific article

The Sam domain of the lipid phosphatase Ship2 adopts a common model to interact with Arap3-Sam and EphA2-Sam

scientific article

The solution structure of the bacterial HSP70 chaperone protein domain DnaK(393–507) in complex with the peptide NRLLLTG ⬇️

scientific article published on November 1, 2003

Therapeutic Targeting of MMP-12 for the Treatment of Chronic Obstructive Pulmonary Disease

scientific article published on 27 October 2020

Therapeutic Targeting of Pancreatic Cancer via EphA2 Dimeric Agonistic Agents

scientific article published on 10 May 2020

Therapy of prostate cancer using a novel cancer terminator virus and a small molecule BH-3 mimetic

scientific article

hBfl-1/hNOXA Interaction Studies Provide New Insights on the Role of Bfl-1 in Cancer Cell Resistance and for the Design of Novel Anticancer Agents.

scientific article published on 27 December 2016

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