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List of works by Carole Pissot-Soldermann

Discovery and SAR of potent, orally available 2,8-diaryl-quinoxalines as a new class of JAK2 inhibitors

scientific article

Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing

scientific article published on 30 November 2020

Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors

scientific article

Modulation of Activation-Loop Phosphorylation by JAK Inhibitors Is Binding Mode Dependent

scientific article

Optimization of the In Vivo Potency of Pyrazolopyrimidine MALT1 Protease Inhibitors by Reducing Metabolism and Increasing Potency in Whole Blood

scientific article published on 20 November 2020

Paradoxical Increase of Permeability and Lipophilicity with the Increasing Topological Polar Surface Area within a Series of PRMT5 Inhibitors

scientific article published in 2022

Potent and selective inhibition of polycythemia by the quinoxaline JAK2 inhibitor NVP-BSK805

scientific article

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