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List of works by André Charette

3-Bromocamphor-8-sulfonic Acid

9-Silafluorenyl Dichlorides as Chemically Ligating Coupling Agents and Their Application in Peptide Synthesis

scientific article published on 4 October 2016

A Diels-Alder approach to the stereoselective synthesis of 2,3,5,6-tetra- and 2,3,4,5,6-pentasubstituted piperidines.

scientific article

A mild procedure for the Lewis acid-catalyzed ring-opening of activated cyclopropanes with amine nucleophiles

scientific article published on 4 June 2008

Access to Cyclopropyl-Fused Azacycles via a Palladium-Catalyzed Direct Alkenylation Strategy

scientific article published on 14 November 2016

An expedient and practical method for the synthesis of a diverse series of cyclopropane alpha-amino acids and amines

scientific article published in February 2004

Application of the chiral bis(phosphine) monoxide ligand to catalytic enantioselective addition of dialkylzinc reagents to beta-nitroalkenes

scientific article published on 01 January 2007

Asymmetric Rh(II)-catalyzed cyclopropanation of alkenes with diacceptor diazo compounds: p-methoxyphenyl ketone as a general stereoselectivity controlling group.

scientific article published on 18 May 2011

Asymmetric Synthesis of Bryostatin 2

scientific article published on 01 September 1998

Asymmetric Total Synthesis of (+)-Luciduline: Toward a General Approach to Related Lycopodium Alkaloids ⬇️

scientific article published on 01 June 2011

Asymmetric synthesis in a Norrish type II cleavage reaction induced by crystal chirality

scientific article published on 01 November 2003

Asymmetric, Catalytic Synthesis of α-Chiral Amines Using a Novel Bis(phosphine) Monoxide Chiral Ligand ⬇️

scientific article published on November 26, 2003

Borocyclopropanation of Styrenes Mediated by UV-light Under Continuous Flow Conditions

scientific article published on 12 September 2018

C-H functionalization of cyclopropanes: a practical approach employing a picolinamide auxiliary

scientific article published on 13 August 2013

Catalytic Asymmetric Synthesis of α,α-Difluoromethylated and α-Fluoromethylated Tertiary Alcohols

scientific article published on 09 September 2019

Catalytic Enantioselective Cyclopropanation of α-Fluoroacrylates: An Experimental and Theoretical Study

Catalytic Enantioselective Synthesis of Halocyclopropanes

scientific article published on 4 March 2016

Catalytic Enantioselective Synthesis of Highly Functionalized Difluoromethylated Cyclopropanes.

scientific article

Catalytic asymmetric addition of diorganozinc reagents to N-phosphinoylalkylimines

scholarly article

Catalytic asymmetric hydrogenation of N-iminopyridinium ylides: expedient approach to enantioenriched substituted piperidine derivatives.

scientific article published in June 2005

Catalytic asymmetric synthesis of alpha,alpha,alpha-trifluoromethylamines by the copper-catalyzed nucleophilic addition of diorganozinc reagents to imines

scientific article published on 01 June 2006

Catalytic enantioselective addition of dialkylzinc to N-diphenylphosphinoylimines. A practical synthesis of alpha-chiral amines

scientific article

Catalytic enantioselective addition of diorganozinc reagents to vinyl sulfones

scientific article published on 08 May 2008

Catalytic enantioselective reduction of beta,beta-disubstituted vinyl phenyl sulfones by using bisphosphine monoxide ligands

scientific article published on 01 January 2007

Chemoselective synthesis of ketones and ketimines by addition of organometallic reagents to secondary amides ⬇️

scientific article published on February 21, 2012

Complexation promoted additions to N-benzoyliminopyridinium ylides. A novel and highly regioselective approach to polysubstituted piperidines.

scientific article

Continuous Flow Synthesis and Purification of Aryldiazomethanes through Hydrazone Fragmentation

scientific article published on 9 December 2016

Controlled and Chemoselective Reduction of Secondary Amides ⬇️

scientific article published on September 22, 2010

Convenient one-pot synthesis of (E)-beta-aryl vinyl halides from benzyl bromides and dihalomethanes

scientific article published on 01 December 2008

Copper-catalyzed direct alkenylation of N-iminopyridinium ylides

scientific article published in February 2010

Corrigendum: Safe and Facile Access to Nonstabilized Diazoalkanes Using Continuous Flow Technology

scientific article published on 01 February 2020

Cycloadditions of aromatic azomethine imines with 1,1-cyclopropane diesters

scientific article published on 08 February 2008

Cyclopropanation of protected chiral, acyclic allylic alcohols: expedient access to the anti-cyclopropylcarbinol derivatives

scientific article published on 01 October 2002

Defying ring strain: new approaches to cyclopropanes.

scientific article published in January 2010

Diastereoselective Borocyclopropanation of Allylic Ethers Using a Boromethylzinc Carbenoid.

scientific article published on 18 January 2017

Diastereoselective Fluorocyclopropanation of Chiral Allylic Alcohols Using an α-Fluoroiodomethylzinc Carbenoid

scientific article published on 26 August 2015

Diastereoselective zinco-cyclopropanation of chiral allylic alcohols with gem-dizinc carbenoids.

scientific article published in September 2005

Difluorocarbene Addition to Alkenes and Alkynes in Continuous Flow

scientific article published on 27 April 2016

Direct Functionalization Processes: A Journey from Palladium to Copper to Iron to Nickel to Metal-Free Coupling Reactions ⬇️

scientific article published on October 26, 2012

Directed functionalization of 1,2-dihydropyridines: stereoselective synthesis of 2,6-disubstituted piperidines

scientific article published in July 2014

Doubly activated cyclopropanes as synthetic precursors for the preparation of 4-nitro- and 4-cyano-dihydropyrroles and pyrroles

scientific article published on 01 June 2005

Dual role of silanol groups in cyclopropanation and Hiyama-Denmark cross-coupling reactions

scientific article published in March 2010

Electrophilic activation of lactams with Tf2O and pyridine: expedient synthesis of (+/-)-tetraponerine T4

scientific article published on 01 November 2005

Enantio- and diastereoselective iodocyclopropanation of allylic alcohols by using a substituted zinc carbenoid

scientific article published in November 2009

Enantioselective synthesis of 1,2,3-trisubstituted cyclopropanes using gem-dizinc reagents

scientific article published in November 2009

Engineered, highly reactive substrates of microbial transglutaminase enable protein labeling within various secondary structure elements

scientific article published on 31 August 2017

Evidence for the structure of the enantioactive ligand in the phosphine-copper-catalyzed addition of diorganozinc reagents to imines

scientific article published on 01 December 2004

Expedient stereoselective synthesis of coronafacic acid through intramolecular Diels-Alder cyclization

scientific article published on 26 January 2007

Expedient synthesis of cyclopropane alpha-amino acids by the catalytic asymmetric cyclopropanation of alkenes using iodonium ylides derived from methyl nitroacetate.

scientific article published in December 2005

Experimental evidence for the all-up reactive conformation of chiral rhodium(II) carboxylate catalysts: enantioselective synthesis of cis-cyclopropane alpha-amino acids

scientific article published in November 2009

First evidence for the formation of a geminal dizinc carbenoid: a highly stereoselective synthesis of 1,2,3-substituted cyclopropanes

scientific article published in January 2002

Formal synthesis of belactosin A and hormaomycin via a diastereoselective intramolecular cyclopropanation of an alpha-nitro diazoester

scientific article published in February 2010

General C-H Arylation Strategy for the Synthesis of Tunable Visible Light-Emitting Benzo[a]imidazo[2,1,5-c,d]indolizine Fluorophores.

scientific article published on 25 April 2017

General Catalytic Enantioselective Access to Monohalomethyl and Trifluoromethyl Cyclopropanes

scientific article published on 25 June 2018

General method for the expedient synthesis of salt-free diorganozinc reagents using zinc methoxide

scientific article published on 12 February 2008

General method for the synthesis of phenyliodonium ylides from malonate esters: easy access to 1,1-cyclopropane diesters.

scientific article published in January 2009

Grob Fragmentation of 2-Azabicyclo[2.2.2]oct-7-ene: Tool for the Stereoselective Synthesis of Polysubstituted Piperidines ⬇️

scientific article published on June 15, 2012

Highly Enantioselective Synthesis of 1,2,3‐Substituted Cyclopropanes by Using α‐Iodo‐ and α‐Chloromethylzinc Carbenoids ⬇️

scientific article published on September 25, 2012

Highly chemoselective metal-free reduction of tertiary amides

scientific article published on 13 December 2007

Highly efficient synthesis of O-(2,4-dinitrophenyl)hydroxylamine. Application to the synthesis of substituted N-benzoyliminopyridinium ylides.

scientific article published in September 2003

Highly efficient two-step synthesis of C-sp3-centered geminal diiodides

scientific article published on 01 December 2004

Highly enantioselective Simmons-Smith fluorocyclopropanation of allylic alcohols via the halogen scrambling strategy of zinc carbenoids

scientific article

Highly regioselective intermolecular arylation of 1,2,3,4-tetrahydropyridines

scientific article published on 01 October 2008

Hypervalent iodine(III) reagents as safe alternatives to alpha-nitro-alpha-diazocarbonyls

scientific article published on 01 June 2003

Improved procedure for the synthesis of gem-diiodoalkanes by the alkylation of diiodomethane. scope and limitations

scientific article

Improved zinc-catalyzed Simmons-Smith reaction: access to various 1,2,3-trisubstituted cyclopropanes

scientific article published on 20 February 2014

In situ generation of zinc carbenoids from diazo compounds and zinc salts: asymmetric synthesis of 1,2,3-substituted cyclopropanes

scientific article published on 01 November 2009

Intramolecular Simmons-Smith cyclopropanation. Studies into the reactivity of alkyl-substituted zinc carbenoids, effect of directing groups and synthesis of bicyclo[n.1.0]alkanes

scientific article published on 01 February 2010

Intramolecular pyridine activation-dearomatization reaction: highly stereoselective synthesis of polysubstituted indolizidines and quinolizidines

scientific article published on 01 August 2009

Intramolecular sp(3) Functionalization of Cyclopropyl α-Amino Acid-Derived Benzamides.

scientific article published in December 2015

Iodomethylzinc phosphates: powerful reagents for the cyclopropanation of alkenes

scientific article

Iron-catalyzed direct arylation through an aryl radical transfer pathway

scientific article published in February 2010

Iron-catalyzed synthesis of cyclopropanes by in situ generation and decomposition of electronically diversified diazo compounds

scientific article published on 01 November 2018

Lithium Iodide

scientific article (publication date: 15 April 2006)

Mechanism-Driven Elaboration of an Enantioselective Bromocyclopropanation Reaction of Allylic Alcohols

scientific article published on 30 September 2015

Mild method for the conversion of amides to thioamides

scientific article published on 01 July 2003

Multicomponent one-pot procedure for the synthesis of free alpha-chiral amines from aldehydes

scientific article published on 01 December 2005

New Family of Cyclopropanating Reagents: Synthesis, Reactivity, and Stability Studies of Iodomethylzinc Phenoxides This work was supported by the E.W.R. Steacie Fund, the National Science and Engineering Research Council (NSERC) of Canada, Merck Fro

scientific article

New methodology toward chiral, non-racemic 2,5-cis-substituted piperidines via Suzuki cross-coupling

scientific article published on 01 August 2006

Nickel(0)/NaHMDS adduct-mediated intramolecular alkylation of unactivated arenes via a homolytic aromatic substitution mechanism

scientific article published on 12 July 2012

Non-stabilized diazoalkane synthesis the oxidation of free hydrazones by iodosylbenzene and application in MIRC cyclopropanation

Nucleophilic addition of phenol derivatives to methyl 1-nitrocyclopropanecarboxylates

scientific article published in August 2008

Nucleophilic addition to 3-substituted pyridinium salts: expedient syntheses of (-)-L-733,061 and (-)-CP-99,994

scientific article published on 01 September 2004

One-Pot Synthesis of 1-Iodoalkynes and Trisubstituted Alkenes from Benzylic and Allylic Bromides ⬇️

scientific article published on October 17, 2012

One-pot synthesis of 3,4,5-trisubstituted 1,2,4-triazoles via the addition of hydrazides to activated secondary amides

scientific article published on 20 February 2015

Organic chemistry: Short cuts to complexity

scientific article published on 01 November 2008

Orthoacylimines: A New Class of Chiral Auxiliaries for Nucleophilic Addition of Organolithium Reagents to Imines ⬇️

scientific article published on April 18, 2003

Palladium-Catalyzed Suzuki-Type Cross-Couplings of Iodocyclopropanes with Boronic Acids: Synthesis of trans-1,2-Dicyclopropyl Alkenes ⬇️

scientific article published on December 13, 1996

Palladium-catalyzed benzylic C-H insertion of 2-substituted N-iminopyridinium ylides

scientific article published on 22 March 2008

Palladium-catalyzed direct C-h arylation of N-iminopyridinium ylides: application to the synthesis of (+/-)-anabasine

scientific article published on 8 December 2007

Palladium-catalyzed synthesis of functionalized tetraarylphosphonium salts

scientific article published on 23 December 2007

Photoinduced alkyl group exchange of ethylzinc alkoxides: X-ray crystal structure of an iodomethylzinc methoxide

scientific article published on 01 March 2002

Potassium tert-butoxide promoted intramolecular arylation via a radical pathway

article published in 2011

Preparation of a storable zinc carbenoid species and its application in cyclopropanation, chain extension, and [2,3]-sigmatropic rearrangement reactions

scientific article published on 01 February 2010

Probing the importance of the hemilabile site of bis(phosphine) monoxide ligands in the copper-catalyzed addition of diethylzinc to N-phosphinoylimines: discovery of new effective chiral ligands

scientific article published on 19 July 2008

Rapid Access to 3-Aminoindazoles from Tertiary Amides

scientific article published on 8 July 2015

Recent Progress Toward the Synthesis of Trifluoromethyl- and Difluoromethyl-Substituted Cyclopropanes

scientific article published on 3 November 2016

Removal, recovery, and recycling of triarylphosphonium-supported tin reagents for various organic transformations

scientific article published on 02 August 2007

Rhodium catalysed enantioselective synthesis of mono-(halo)-methyl-cyclopropanes

scientific article published on 01 January 2019

Rhodium-catalyzed cyclopropanation of fluorinated olefins: a straightforward route to highly functionalized fluorocyclopropanes

scientific article published on 13 March 2015

Safe and Facile Access to Nonstabilized Diazoalkanes Using Continuous Flow Technology

scientific article published on 19 April 2018

Samarium(II) Iodide

scientific article by Gary A. Molander and André Charette

Silver ion-induced Grob fragmentation of gamma-amino iodides: highly stereoselective synthesis of polysubstituted piperidines

scientific article published on 01 December 2008

Silver-promoted, palladium-catalyzed direct arylation of cyclopropanes: facile access to spiro 3,3'-cyclopropyl oxindoles.

scientific article published in March 2013

Simmons-Smith Cyclopropanation Reaction

scientific article (publication date: 18 July 2001)

Spectroscopic characterization of (diiodomethyl)zinc iodide: application to the stereoselective synthesis and functionalization of iodocyclopropanes

scientific article

Stereoselective Rh2(S-IBAZ)4-catalyzed cyclopropanation of alkenes, alkynes, and allenes: asymmetric synthesis of diacceptor cyclopropylphosphonates and alkylidenecyclopropanes

scientific article published on 15 January 2013

Stereoselective Synthesis of 2,3,6-Trisubstituted Tetrahydropyridines via Tf2O-Mediated Grob Fragmentation: Access to Indolizidines (−)-209I and (−)-223J ⬇️

scientific article published on November 5, 2010

Stereoselective cyclopropanation reactions

scientific article (publication date: April 2003)

Stereoselective formation of amines by nucleophilic addition to azomethine derivatives

scientific article published on 01 January 2014

Stereoselective syntheses of L-pipecolic acid and (2S,3S)-3-hydroxypipecolic acid from a chiral N-imino-2-phenyl-1,2-dihydropyridine intermediate

scientific article published in March 2010

Stereoselective synthesis of 2,6-disubstituted 3-piperidinols: application to the expedient synthesis of (+)-julifloridine

scientific article published on 01 June 2005

Stereoselective synthesis of pyridinones: application to the synthesis of (-)-barrenazines

scientific article published on 01 July 2006

Structure and reactivity of "unusual" N-heterocyclic carbene (NHC) palladium complexes synthesized from imidazolium salts

article published in 2004

Structure and reactivity of a new anionic N-heterocyclic carbene silver(I) complex

scientific article published on 01 July 2005

Synthesis of 2- and 2,3-substituted pyrazolo[1,5-a]pyridines: scope and mechanistic considerations of a domino direct alkynylation and cyclization of N-iminopyridinium ylides using alkenyl bromides, alkenyl iodides, and alkynes

scientific article published on 30 September 2011

Synthesis of 2-substituted pyrazolo[1,5-a]pyridines through cascade direct alkenylation/cyclization reactions

scientific article published on 01 February 2010

Synthesis of 3-Aminoimidazo[1,2-a]pyridines from α-Aminopyridinyl Amides

scientific article published on 26 July 2016

Synthesis of Fluoro, Monofluoromethyl, Difluoromethyl and Trifluoromethyl-Substituted Three Membered Rings

scientific article published on 17 September 2020

Synthesis of N-diphenylphosphinoylimines using the Kresze reaction

scientific article published in December 2005

Synthesis of enantioenriched allenes from 1,1-cyclopropanediesters

scientific article published in February 2010

Synthesis of enantiopure substituted piperidines via an aziridinium ring expansion

scientific article published on June 28, 2011

Synthesis of pyridine and dihydropyridine derivatives by regio- and stereoselective addition to N-activated pyridines

scientific article published on 21 February 2012

Tetraarylphosphonium salts as solubility-control groups: phosphonium-supported triphenylphosphine and azodicarboxylate reagents

scientific article published in February 2006

Tetraarylphosphonium salts as soluble supports for oxidative catalysts and reagents

scientific article published in November 2009

Tetraarylphosphonium salts as soluble supports for the synthesis of small molecules

scientific article published on 01 January 2007

Tetraarylphosphonium-supported carbodiimide reagents: synthesis, structure optimization and applications

scientific article published on 4 March 2008

TfNH2 as achiral hydrogen-bond donor additive to enhance the selectivity of a transition metal catalyzed reaction. Highly enantio- and diastereoselective rhodium-catalyzed cyclopropanation of alkenes using alpha-cyano diazoacetamide.

scientific article published in May 2009

Total Synthesis of (+)-Cystothiazole A ⬇️

scientific article published on October 30, 2003

Total Synthesis of Bryostatin 2

article by David A. Evans et al published August 1999 in Journal of the American Chemical Society

Total synthesis of (+)-lepadin B: stereoselective synthesis of nonracemic polysubstituted hydroquinolines using an RC-ROM process

scientific article published on 27 September 2008

Transition metal-catalyzed cyclopropanation of alkenes in water: catalyst efficiency and in situ generation of the diazo reagent

scientific article published on 01 December 2002

Triflic anhydride mediated synthesis of imidazo[1,5-a]azines

scientific article published on 24 April 2013

Umpolung Direct Arylation Reactions: Facile Process Requiring Only Catalytic Palladium and Substoichiometric Amount of Silver Salts ⬇️

scientific article published on October 20, 2010

Use of achiral additives to increase the stereoselectivity in Rh(II)-catalyzed cyclopropanations

scientific article published on 07 January 2010

Utilization of BozPhos as an Effective Ligand in Enantioselective C-H Functionalization of Cyclopropanes: Synthesis of Dihydroisoquinolones and Dihydroquinolones

scientific article published on 29 March 2019

[4+2] Cycloaddition of 2-substituted 1,2-dihydropyridines with nitrosobenzene: asymmetric synthesis of trans-2-substituted 3-amino-1,2,3,6-tetrahydropyridines

scientific article

trans-Directing ability of amide groups in cyclopropanation: application to the asymmetric cyclopropanation of alkenes with diazo reagents bearing two carboxy groups

scientific article published in January 2008

trans-Directing ability of the amide group: enabling the enantiocontrol in the synthesis of 1,1-dicarboxy cyclopropanes. Reaction development, scope, and synthetic applications.

scientific article published in December 2009

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