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List of works by Milan Kožíšek

Anomalous adsorptive properties of HIV protease: Indication of two-dimensional crystallization?

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Crystal structures of the effector-binding domain of repressor Central glycolytic gene Regulator fromBacillus subtilisreveal ligand-induced structural changes upon binding of several glycolytic intermediates

scientific article

Design of HIV protease inhibitors based on inorganic polyhedral metallacarboranes

scientific article

Dispersion Interactions Govern the Strong Thermal Stability of a Protein

scientific article published on 01 January 2007

Enzymatic and structural analysis of the I47A mutation contributing to the reduced susceptibility to HIV protease inhibitor lopinavir

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Fine tuning of the catalytic activity of colicin E7 nuclease domain by systematic N-terminal mutations.

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Functional and Structural Characterization of Novel Type of Linker Connecting Capsid and Nucleocapsid Protein Domains in Murine Leukemia Virus.

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GS-8374, a Prototype Phosphonate-Containing Inhibitor of HIV-1 Protease, Effectively Inhibits Protease Mutants with Amino Acid Insertions

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Human DNA-Damage-Inducible 2 Protein Is Structurally and Functionally Distinct from Its Yeast Ortholog.

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Kinetic, Thermodynamic, and Structural Analysis of Drug Resistance Mutations in Neuraminidase from the 2009 Pandemic Influenza Virus

scientific article published on 21 June 2018

Kinetic, thermodynamic and structural analysis of tamiphosphor binding to neuraminidase of H1N1 (2009) pandemic influenza

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Molecular Characterization of Clinical Isolates of Human Immunodeficiency Virus Resistant to the Protease Inhibitor Darunavir

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Molecular analysis of the HIV-1 resistance development: enzymatic activities, crystal structures, and thermodynamics of nelfinavir-resistant HIV protease mutants

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Mutations in HIV-1 gag and pol Compensate for the Loss of Viral Fitness Caused by a Highly Mutated Protease

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Ninety-Nine Is Not Enough: Molecular Characterization of Inhibitor-Resistant Human Immunodeficiency Virus Type 1 Protease Mutants with Insertions in the Flap Region

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Potent inhibition of drug-resistant HIV protease variants by monoclonal antibodies

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Preorganization of the catalytic Zn(2+)-binding site in the HNH nuclease motif--A solution study

scientific article published on 09 April 2015

Re-evaluation of binding properties of recombinant lymphocyte receptors NKR-P1A and CD69 to chemically synthesized glycans and peptides

scientific article published on 17 January 2014

Specific Inhibitors of HIV Capsid Assembly Binding to the C-Terminal Domain of the Capsid Protein: Evaluation of 2-Arylquinazolines as Potential Antiviral Compounds.

scientific article published on 21 December 2015

Stabilization of antibody structure upon association to a human carbonic anhydrase IX epitope studied by X-ray crystallography, microcalorimetry, and molecular dynamics simulations

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Structural studies of the yeast DNA damage-inducible protein Ddi1 reveal domain architecture of this eukaryotic protein family.

scientific article published on 20 September 2016

Structure-aided design of novel inhibitors of HIV protease based on a benzodiazepine scaffold.

scientific article

Substrate binding activates the designed triple mutant of the colicin E7 metallonuclease

scientific article published on 26 August 2014

Synthesis and evaluation of 2-pyridinylpyrimidines as inhibitors of HIV-1 structural protein assembly

scientific article published on 16 June 2016

Tetraphenylporphyrin-cobalt(III) Bis(1,2-dicarbollide) Conjugates: From the Solution Characteristics to Inhibition of HIV Protease

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Thermodynamic and structural analysis of HIV protease resistance to darunavir - analysis of heavily mutated patient-derived HIV-1 proteases

scientific article

Urea and Guanidinium Induced Denaturation of a Trp-Cage Miniprotein

scientific article published on 02 June 2011