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List of works by Maria Preobrazhenskaya

1-Benzyl-indole-3-carbinol is a novel indole-3-carbinol derivative with significantly enhanced potency of anti-proliferative and anti-estrogenic properties in human breast cancer cells

scientific article

3-Aminomethyl derivatives of 4,11-dihydroxynaphtho[2,3-f]indole-5,10-dione for circumvention of anticancer drug resistance.

scientific article published on March 2005

A novel acyclic oligomycin A derivative formed via retro-aldol rearrangement of oligomycin A.

scientific article published on 23 May 2012

Altered transcription and replication are the mechanisms of cytotoxicity of antitumor antibiotic olivomycin A

scientific article published on 01 November 2010

An analogue of the antibiotic teicoplanin prevents flavivirus entry in vitro

scientific article

Anthracycline antibiotics and their derivatives--inhibitors of topoisomerase I

scientific article published in May 2008

Antiretroviral activity of semisynthetic derivatives of glycopeptide antibiotics

scientific article published on June 2003

Antitumor antibiotic streptonigrin and its derivatives as inhibitors of nitric oxide-dependent activation of soluble guanylyl cyclase

scientific article

Bacterial eukaryotic type serine-threonine protein kinases: from structural biology to targeted anti-infective drug design

scientific article

Characterization of HERG potassium channel inhibition using CoMSiA 3D QSAR and homology modeling approaches

scientific article published on May 2003

Chemical modification and biological evaluation of new semisynthetic derivatives of 28,29-Didehydronystatin A1 (S44HP), a genetically engineered antifungal polyene macrolide antibiotic

scientific article published in January 2009

Correction to The Carboxyl Terminus of Eremomycin Facilitates Binding to the Non-d-Ala-d-Ala Segment of the Peptidoglycan Pentapeptide Stem

scientific article published on 06 July 2016

Erratum: Modification of the antibiotic olivomycin I at the 2′-keto group of the side chain. Novel derivatives, antitumor and topoisomerase I-poisoning activity

scholarly article published in The Journal of Antibiotics

Glycopeptide antibiotic analogs efficient against vancomycin-resistant bacteria: a patent evaluation (WO2013022763).

scientific article

Inhibition of feline (FIPV) and human (SARS) coronavirus by semisynthetic derivatives of glycopeptide antibiotics

scientific article published on 6 April 2006

Inhibition of hepatitis C virus replication by semi-synthetic derivatives of glycopeptide antibiotics

scientific article published on 24 March 2011

Modification of olivomycin A at the side chain of the aglycon yields the derivative with perspective antitumor characteristics

scientific article

Modification of the antibiotic olivomycin I at the 2'-keto group of the side chain. Novel derivatives, antitumor and topoisomerase I-poisoning activity

scientific article

N-Alkoxy derivatization of indole-3-carbinol increases the efficacy of the G1 cell cycle arrest and of I3C-specific regulation of cell cycle gene transcription and activity in human breast cancer cells ⬇️

scientific article

Naphtho[2,3-f]indole-5,10-dione aminoalkyl derivatives: a new class of topoisomerase I inhibitors

scientific article published in March 2008

Naphthoindole-based analogues of tryptophan and tryptamine: synthesis and cytotoxic properties.

scientific article published on 23 January 2007

Novel semisynthetic derivative of antibiotic Eremomycin active against drug-resistant gram-positive pathogens including Bacillus anthracis.

scientific article published on 3 July 2007

N′-(α-Aminoacyl)- and N′-α-(N-Alkylamino)acyl Derivatives of Vancomycin and Eremomycin

scientific article published on 01 April 2007

N′-(α-Aminoacyl)- and N′-α-(Nα-Alkylamino)acyl Derivatives of Vancomycin and Eremomycin

scientific article published on 01 April 2007

O-glycosides of N-hydroxyindoles

scientific article published in October 2001

Partial circumvention of P-glycoprotein-mediated multidrug resistance by doxorubicin-14-O-hemiadipate

scientific article

Patents on glycopeptides of the vancomycin family and their derivatives as antimicrobials: January 1999 ? June 2003

Polycyclic peptide and glycopeptide antibiotics and their derivatives as inhibitors of HIV entry.

scientific article published on 6 May 2006

REDOR constraints on the peptidoglycan lattice architecture of Staphylococcus aureus and its FemA mutant

scientific article

Reaction of the antitumor antibiotic olivomycin I with aryl diazonium salts. Synthesis, cytotoxic and antiretroviral potency of 5-aryldiazenyl-6-O-deglycosyl derivatives of olivomycin I.

scientific article

Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity

scientific article published on 7 September 2012

Role of the acyl groups in carbohydrate chains in cytotoxic properties of olivomycin A.

scientific article published on 22 May 2013

Role of the glycopeptide framework in the antibacterial activity of hydrophobic derivatives of glycopeptide antibiotics

scientific article published in March 2003

Search for inhibitors of bacterial and human protein kinases among derivatives of diazepines[1,4] annelated with maleimide and indole cycles

scientific article published in December 2008

Staphylococcus aureus peptidoglycan stem packing by rotational-echo double resonance NMR spectroscopy

scientific article published on 14 May 2013

Structure-activity relationship studies of a series of antiviral and antibacterial aglycon derivatives of the glycopeptide antibiotics vancomycin, eremomycin, and dechloroeremomycin

scientific article

Structure-antifungal activity relationships of polyene antibiotics of the amphotericin B group

scientific article

Structures of Staphylococcus aureus cell-wall complexes with vancomycin, eremomycin, and chloroeremomycin derivatives by 13C{19F} and 15N{19F} rotational-echo double resonance

scientific article published on April 2006

Studies of complex formation of olivomycin A and its derivatives with DNA

scientific article published on 01 November 2010

Study of 1-deoxy-1-(indol-3-yl)-L-sorbose, 1-deoxy-1-(indol-3-yl)-L-tagatose, and their analogs

scientific article published in January 2003

Study on retroaldol degradation products of antibiotic oligomycin A.

scientific article published on 2 October 2013

Synthesis and antibacterial activity of alkyl derivatives of the glycopeptide antibiotic A40926 and their amides.

scientific article published in August 2005

Synthesis and antitumor activity of new D-galactose-containing derivatives of doxorubicin

scientific article published on June 2003

Synthesis and cytotoxic potency of novel tris(1-alkylindol-3-yl)methylium salts: role of N-alkyl substituents.

scientific article published on 23 July 2010

Synthesis and cytotoxic properties of 4,11-bis[(aminoethyl)amino]anthra[2,3-b]thiophene-5,10-diones, novel analogues of antitumor anthracene-9,10-diones

scientific article

Synthesis and cytotoxicity of oligomycin A derivatives modified in the side chain

scientific article published on 6 April 2013

Synthesis and mode of action of hydrophobic derivatives of the glycopeptide antibiotic eremomycin and des-(N-methyl-D-leucyl)eremomycin against glycopeptide-sensitive and -resistant bacteria

scientific article published in March 2002

Synthesis and properties of a novel brominated oligomycin A derivative

scientific article published on 08 February 2012

Synthesis and structure-activity relationship studies of 4,11-diaminonaphtho[2,3-f]indole-5,10-diones

scientific article published on 2 May 2006

Synthesis and study of the antifungal activity of new mono- and disubstituted derivatives of a genetically engineered polyene antibiotic 28,29-didehydronystatin A1 (S44HP).

scientific article published on 4 December 2009

Synthesis of 1-(omega-aminoalkyl)naphthoindolediones with antiproliferative properties

scientific article published on July 2004

Synthesis of 6H-pyrrolo[3',4':2,3][1,4]diazepino[6,7,1-hi]indole-8,10(7H,9H)-diones using 3-bromo-4-(indol-1-yl)maleimide scaffold

scientific article published in March 2003

Target protein interactions of indole-3-carbinol and the highly potent derivative 1-benzyl-I3C with the C-terminal domain of human elastase uncouples cell cycle arrest from apoptotic signaling

scientific article

The Carboxyl Terminus of Eremomycin Facilitates Binding to the Non-d-Ala-d-Ala Segment of the Peptidoglycan Pentapeptide Stem

scientific article published on 31 May 2016

The Influence of 1′-Methyl- and 1′-Ethylascorbigen on Metabolism of Arachidonic Acid in Murine Spleen Cells

scientific article published on 01 February 1993

The first examples of chemical modification of oligomycin A.

scientific article published on 13 November 2009

The first series of 4,11-bis[(2-aminoethyl)amino]anthra[2,3-b]furan-5,10-diones: Synthesis and anti-proliferative characteristics

scientific article published on 19 November 2010

The formation of 2-hydroxy-4-hydroxymethyl-3-(indol-3-yl)-cyclopent-2-enone derivatives from ascorbigens

scientific article

The interaction of per-O-acetylated acyclic 1-(1-butylindol-3-yl)-1-deoxy-ketoses with silylated uracil

scientific article published in January 2004

Thienoquinolines as novel disruptors of the PKCε/RACK2 protein-protein interaction

scientific article published on 08 April 2014

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