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List of works by Jean-Christophe Harmange

Design and evaluation of 1,7-naphthyridones as novel KDM5 inhibitors

scientific article

Design, synthesis, and evaluation of orally active benzimidazoles and benzoxazoles as vascular endothelial growth factor-2 receptor tyrosine kinase inhibitors

scientific article

Discovery and optimization of a potent and selective triazolopyridinone series of c-Met inhibitors

scientific article

Discovery and optimization of potent and selective triazolopyridazine series of c-Met inhibitors

scientific article

Discovery and optimization of triazolopyridazines as potent and selective inhibitors of the c-Met kinase

scientific article

Discovery of (R)-6-(1-(8-Fluoro-6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl)-3-(2-methoxyethoxy)-1,6-naphthyridin-5(6H)-one (AMG 337), a Potent and Selective Inhibitor of MET...

scientific article

Discovery of 2,4-bis-arylamino-1,3-pyrimidines as insulin-like growth factor-1 receptor (IGF-1R) inhibitors ⬇️

scientific article published on February 23, 2011

Discovery of potent and selective 8-fluorotriazolopyridine c-Met inhibitors

scientific article

Discovery of triazine-benzimidazoles as selective inhibitors of mTOR

scientific article

Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors

scientific article

Evaluation of a series of naphthamides as potent, orally active vascular endothelial growth factor receptor-2 tyrosine kinase inhibitors

scientific article

Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials

scientific article

Identification of potent, selective KDM5 inhibitors

scientific article

Novel 2,3-dihydro-1,4-benzoxazines as potent and orally bioavailable inhibitors of tumor-driven angiogenesis

scientific article

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