List of works - Anna Di Fiore

2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity

scientific article

Anticancer steroid sulfatase inhibitors: synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography

scientific article

Benzoxaborole as a new chemotype for carbonic anhydrase inhibition

scientific article

Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of N-substituted benzenesulfonamides to human isoform II

scientific article

Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties

scientific article

Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV

scientific article

Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors

scientific article

Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide

scientific article

Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide

scientific article

Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX

scientific article

Crystal structure of the most catalytically effective carbonic anhydrase enzyme known, SazCA from the thermophilic bacterium Sulfurihydrogenibium azorense

scientific article

Hydroxamate represents a versatile zinc binding group for the development of new carbonic anhydrase inhibitors

scientific article

Structural analysis of BldR from Sulfolobus solfataricus provides insights into the molecular basis of transcriptional activation in Archaea by MarR family proteins

scientific article

Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents

scientific article

The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies

scientific article

The unswapped chain of bovine seminal ribonuclease: Crystal structure of the free and liganded monomeric derivative

scientific article

Thermostable Carbonic Anhydrases in Biotechnological Applications

scientific article

X-ray structure of the first `extremo-α-carbonic anhydrase', a dimeric enzyme from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1

scientific article

List of works by Anna Di Fiore

2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity

Anticancer steroid sulfatase inhibitors: synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography

Benzoxaborole as a new chemotype for carbonic anhydrase inhibition

Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of N-substituted benzenesulfonamides to human isoform II

Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties

Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV

Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors

Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide

Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide

Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX

Crystal structure of the most catalytically effective carbonic anhydrase enzyme known, SazCA from the thermophilic bacterium Sulfurihydrogenibium azorense

Hydroxamate represents a versatile zinc binding group for the development of new carbonic anhydrase inhibitors

Structural analysis of BldR from Sulfolobus solfataricus provides insights into the molecular basis of transcriptional activation in Archaea by MarR family proteins

Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents

The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies

The unswapped chain of bovine seminal ribonuclease: Crystal structure of the free and liganded monomeric derivative

Thermostable Carbonic Anhydrases in Biotechnological Applications

X-ray structure of the first `extremo-α-carbonic anhydrase', a dimeric enzyme from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1