List of works - Heinz Heimgartner

(S)-N-[(4-{(S)-1-[2-(4-Meth-oxy-benz-amido)-2-methyl-propano-yl]pyrrolidine-2-carboxamido}-3,4,5,6-tetra-hydro-2H-pyran-4-yl)carbon-yl]proline dimethyl sulfoxide monosolvate (4-MeBz-Aib-Pro-Thp-Pro-OH).

scientific article published on 20 February 2013

1,3-Dipolar Cycloadditions ofα-Diazo Ketones Derived fromN-Protected (S)-Proline with Aromatic and Cycloaliphatic Thioketones

scientific article published in February 2015

1,3-Dipolar cycloadditions of fluorinated nitrones with thioketones

scientific article published in September 2014

1,3-thiazolidine derivatives from regioselective [2+3]-cycloadditions of azomethine ylides with thioketones.

scientific article published on 18 April 2003

2-Unsubstituted Imidazole N-Oxides as Novel Precursors of Chiral 3-Alkoxyimidazol-2-ylidenes Derived from trans-1,2-Diaminocyclohexane and Other Chiral Amino Compounds

scientific article published on 02 December 2019

3-(2,6-dimethylphenyl)-2-selenoxo-1,3-thiazolidin-4-one suppresses hydrogen peroxide-induced cytotoxicity on PC12 cells via activation of MAPK.

scientific article published on 29 September 2011

A novel 2H-azirin-3-amine as a synthon for a sulfur-containing dipeptide segment

scientific article published on 20 March 2013

A novel application of 2-silylated 1,3-dithiolanes for the synthesis of aryl/hetaryl-substituted ethenes and dibenzofulvenes.

scientific article published on 8 September 2017

Attempts toward the synthesis of the peptaibol antiamoebin by using the 'azirine/oxazolone method'.

scientific article published in May 2013

Bis(1-chloro-2,2,4,4-tetramethyl-3-oxocyclobutan-1-yl)pentasulfane: an occupancy modulated structure.

scientific article published on 19 July 2004

Chemoselective trifluoromethylation of the C N group of α-iminoketones derived from arylglyoxals

scientific article published in December 2014

Coexistence of hydrogen-bonded loop and extended tetrapeptide conformations

scientific article published on 01 January 2007

Crystal structure of (E)-1,2-diferrocenyl-1,2-bis(furan-2-yl)ethene.

scientific article published on 6 April 2018

Di- and tripeptide segments of zervamicin II-2: Z-Thr(OBn)-Aib-N(Me)Ph and Z-Val-Aib-Hyp(OBn)-OMe

scientific article published on 13 April 2006

Dialkyl dicyanofumarates and dicyanomaleates as versatile building blocks for synthetic organic chemistry and mechanistic studies.

scientific article published on 24 October 2017

Dimerization reactions of aryl selenophen-2-yl-substituted thiocarbonyl S-methanides as diradical processes: a computational study.

scientific article published on 03 March 2017

Diradical reaction mechanisms in [3 + 2]-cycloadditions of hetaryl thioketones with alkyl- or trimethylsilyl-substituted diazomethanes

scientific article published on 14 April 2016

Efficient synthesis of ferrocifens and other ferrocenyl-substituted ethylenes via a 'sulfur approach'

scientific article published on 01 June 2018

Exploration of Fluoral Hydrazones Derived from Carbohydrazides for the Synthesis of Trifluoromethylated Heterocycles

scientific article published in 2014

First thia-Diels-Alder reactions of thiochalcones with 1,4-quinones

scientific article published on 19 July 2018

Hetero-Diels-Alder reactions of hetaryl and aryl thioketones with acetylenic dienophiles.

scientific article published on 28 April 2015

Highly Constrained Linear Oligopeptides Containing Heterocyclicα-Amino Carboxylic Acids

scientific article published in September 2013

Intra- and intermolecular Se···X (X = Se, O) interactions in selenium-containing heterocycles: 3-benzoylimino-5-(morpholin-4-yl)-1,2,4-diselenazole

scientific article published on 18 April 2014

New 21- and 24-atom Aib-containing cyclopeptides

scientific article published on 01 September 2008

New Optically Active Bis-Heterocycles Derived from (S)-Proline

scientific article published in September 2012

New Selenosemicarbazides Derived from Imidazole-Based Carbohydrazides

scientific article published in March 2013

Nucleophilic trifluoromethylation of aziridinyl ketones: A convenient access to fluorinated aziridinyl alcohols

scientific article published in December 2013

Reaction of Thioketones with (R)-2-Vinyloxirane: Regio- and Stereoselective Formation of (S)-4-Vinyl-1,3-oxathiolanes

Reactions of Acid Chlorides/Ketenes with 2-Substituted 4,5-Dihydro-4,4-dimethyl-1,3-thiazoles: Formation of Penam Derivatives

scientific article published in August 2013

Regio- and Stereoselectivity in theLewis Acid- and NaH-Induced Reactions of Thiocamphor with (R)-2-Vinyloxirane

Solid-state conformations of linear depsipeptide amides with an alternating sequence of α,α-disubstituted α-amino acid and α-hydroxy acid

scientific article published on 06 December 2019

Solution-phase synthesis of Aib-containing cyclic hexapeptides

scientific article published on 01 November 2004

Studies on the Reaction of Aryl Glyoxals withl-Prolinol: Unexpected Formation of Morpholin-2-one Derivatives and Stereoselective Trifluoromethylation of the Bicyclic System

scientific article published on 12 June 2015

Studies on the synthesis and some reactions of (S)-proline hydrazides

scientific article published in May 2012

Synthesis and selected transformations of 2-unsubstituted 1-(adamantyloxy)imidazole 3-oxides: straightforward access to non-symmetric 1,3-dialkoxyimidazolium salts

scientific article published on 19 February 2019

Synthesis of 1,3,5-Triazineselones from Imidoyl Isoselenocyanates and Amidines

scientific article published in 2012

Synthesis of Aib- and Phe(2Me)-Containing Cyclopentapeptides

scientific article published in February 2015

Synthesis of Aib-Pro Oligopeptides by Repeated Azirine Coupling with the Aib-Pro Synthon

scientific article published in August 2012

Synthesis of Cyclopentapeptides with Three to Five Aib Units

scientific article published in February 2015

Synthesis of Z-Protected Aib- and Phe(2Me)-Containing Pentapeptides and Their Crystal Structures

scientific article published in May 2014

Synthesis of ferrocenyl-substituted 1,3-dithiolanes via [3 + 2]-cycloadditions of ferrocenyl hetaryl thioketones with thiocarbonyl S-methanides

scientific article published on 08 July 2016

Synthesis of the protected 6-16 segment of zervamicin 11-2, an application of the azirine/oxazolone method.

scientific article published in November 2003

The 'azirine/oxazolone method' in peptaibol synthesis: preparation of a derivative of trichotoxin A-50 (G)

scientific article published on 01 June 2007

The [4+2]-Cycloaddition of α-Nitrosoalkenes with Thiochalcones as a Prototype of Periselective Hetero-Diels-Alder Reactions-Experimental and Computational Studies

scientific article published on 22 November 2019

The first total synthesis of the peptaibol hypomurocin A1 and its conformation analysis: an application of the 'azirine/oxazolone method'

scientific article published on 01 September 2005

Thermal [2+2]-Cycloadditions of Diphenylketene with Aryl- and Hetaryl-Substituted Thioketones

scientific article published in 2015

Thio- and Dithioesters as Dipolarophiles in Reactions with Thiocarbonyl Ylides

Total synthesis of the peptaibols hypomurocin A3 and hypomurocin A5, and their conformation analysis

scientific article published on 01 November 2012

Unexpected Course of the Reaction of 2-Unsubstituted 1H-Imidazole 3-Oxides with Ethyl Acrylate

scientific article published in April 2012

Unexpected Reaction Course of 3-Amino-5-aryl-1H-pyrazoles with Dialkyl Dicyanofumarates

scientific article published in April 2013

[2 + 3]-Cycloadditions of PhosphonodithioformateS-Methanides with CS, NN, and CC Dipolarophiles

cis-(6RS,13RS)-3,3,10,10-Tetramethyl-6,13-diphenyl-1,8-dioxa-4,11-diazacyclotetradecane-2,5,9,12-tetraone and two of its precursors

scientific article published on 24 May 2006

List of works by Heinz Heimgartner

(S)-N-[(4-{(S)-1-[2-(4-Meth-oxy-benz-amido)-2-methyl-propano-yl]pyrrolidine-2-carboxamido}-3,4,5,6-tetra-hydro-2H-pyran-4-yl)carbon-yl]proline dimethyl sulfoxide monosolvate (4-MeBz-Aib-Pro-Thp-Pro-OH).

1,3-Dipolar Cycloadditions ofα-Diazo Ketones Derived fromN-Protected (S)-Proline with Aromatic and Cycloaliphatic Thioketones

1,3-Dipolar cycloadditions of fluorinated nitrones with thioketones

1,3-thiazolidine derivatives from regioselective [2+3]-cycloadditions of azomethine ylides with thioketones.

2-Unsubstituted Imidazole N-Oxides as Novel Precursors of Chiral 3-Alkoxyimidazol-2-ylidenes Derived from trans-1,2-Diaminocyclohexane and Other Chiral Amino Compounds

3-(2,6-dimethylphenyl)-2-selenoxo-1,3-thiazolidin-4-one suppresses hydrogen peroxide-induced cytotoxicity on PC12 cells via activation of MAPK.

A novel 2H-azirin-3-amine as a synthon for a sulfur-containing dipeptide segment

A novel application of 2-silylated 1,3-dithiolanes for the synthesis of aryl/hetaryl-substituted ethenes and dibenzofulvenes.

Attempts toward the synthesis of the peptaibol antiamoebin by using the 'azirine/oxazolone method'.

Bis(1-chloro-2,2,4,4-tetramethyl-3-oxocyclobutan-1-yl)pentasulfane: an occupancy modulated structure.

Chemoselective trifluoromethylation of the C N group of α-iminoketones derived from arylglyoxals

Coexistence of hydrogen-bonded loop and extended tetrapeptide conformations

Crystal structure of (E)-1,2-diferrocenyl-1,2-bis(furan-2-yl)ethene.

Di- and tripeptide segments of zervamicin II-2: Z-Thr(OBn)-Aib-N(Me)Ph and Z-Val-Aib-Hyp(OBn)-OMe

Dialkyl dicyanofumarates and dicyanomaleates as versatile building blocks for synthetic organic chemistry and mechanistic studies.

Dimerization reactions of aryl selenophen-2-yl-substituted thiocarbonyl S-methanides as diradical processes: a computational study.

Diradical reaction mechanisms in [3 + 2]-cycloadditions of hetaryl thioketones with alkyl- or trimethylsilyl-substituted diazomethanes

Efficient synthesis of ferrocifens and other ferrocenyl-substituted ethylenes via a 'sulfur approach'

Exploration of Fluoral Hydrazones Derived from Carbohydrazides for the Synthesis of Trifluoromethylated Heterocycles

First thia-Diels-Alder reactions of thiochalcones with 1,4-quinones

Hetero-Diels-Alder reactions of hetaryl and aryl thioketones with acetylenic dienophiles.

Highly Constrained Linear Oligopeptides Containing Heterocyclicα-Amino Carboxylic Acids

Intra- and intermolecular Se···X (X = Se, O) interactions in selenium-containing heterocycles: 3-benzoylimino-5-(morpholin-4-yl)-1,2,4-diselenazole

New 21- and 24-atom Aib-containing cyclopeptides

New Optically Active Bis-Heterocycles Derived from (S)-Proline

New Selenosemicarbazides Derived from Imidazole-Based Carbohydrazides

Nucleophilic trifluoromethylation of aziridinyl ketones: A convenient access to fluorinated aziridinyl alcohols

Reaction of Thioketones with (R)-2-Vinyloxirane: Regio- and Stereoselective Formation of (S)-4-Vinyl-1,3-oxathiolanes

Reactions of Acid Chlorides/Ketenes with 2-Substituted 4,5-Dihydro-4,4-dimethyl-1,3-thiazoles: Formation of Penam Derivatives

Regio- and Stereoselectivity in theLewis Acid- and NaH-Induced Reactions of Thiocamphor with (R)-2-Vinyloxirane

Solid-state conformations of linear depsipeptide amides with an alternating sequence of α,α-disubstituted α-amino acid and α-hydroxy acid

Solution-phase synthesis of Aib-containing cyclic hexapeptides

Studies on the Reaction of Aryl Glyoxals withl-Prolinol: Unexpected Formation of Morpholin-2-one Derivatives and Stereoselective Trifluoromethylation of the Bicyclic System

Studies on the synthesis and some reactions of (S)-proline hydrazides

Synthesis and selected transformations of 2-unsubstituted 1-(adamantyloxy)imidazole 3-oxides: straightforward access to non-symmetric 1,3-dialkoxyimidazolium salts

Synthesis of 1,3,5-Triazineselones from Imidoyl Isoselenocyanates and Amidines

Synthesis of Aib- and Phe(2Me)-Containing Cyclopentapeptides

Synthesis of Aib-Pro Oligopeptides by Repeated Azirine Coupling with the Aib-Pro Synthon

Synthesis of Cyclopentapeptides with Three to Five Aib Units

Synthesis of Z-Protected Aib- and Phe(2Me)-Containing Pentapeptides and Their Crystal Structures

Synthesis of ferrocenyl-substituted 1,3-dithiolanes via [3 + 2]-cycloadditions of ferrocenyl hetaryl thioketones with thiocarbonyl S-methanides

Synthesis of the protected 6-16 segment of zervamicin 11-2, an application of the azirine/oxazolone method.

The 'azirine/oxazolone method' in peptaibol synthesis: preparation of a derivative of trichotoxin A-50 (G)

The [4+2]-Cycloaddition of α-Nitrosoalkenes with Thiochalcones as a Prototype of Periselective Hetero-Diels-Alder Reactions-Experimental and Computational Studies

The first total synthesis of the peptaibol hypomurocin A1 and its conformation analysis: an application of the 'azirine/oxazolone method'

Thermal [2+2]-Cycloadditions of Diphenylketene with Aryl- and Hetaryl-Substituted Thioketones

Thio- and Dithioesters as Dipolarophiles in Reactions with Thiocarbonyl Ylides

Total synthesis of the peptaibols hypomurocin A3 and hypomurocin A5, and their conformation analysis

Unexpected Course of the Reaction of 2-Unsubstituted 1H-Imidazole 3-Oxides with Ethyl Acrylate

Unexpected Reaction Course of 3-Amino-5-aryl-1H-pyrazoles with Dialkyl Dicyanofumarates

[2 + 3]-Cycloadditions of PhosphonodithioformateS-Methanides with CS, NN, and CC Dipolarophiles

cis-(6RS,13RS)-3,3,10,10-Tetramethyl-6,13-diphenyl-1,8-dioxa-4,11-diazacyclotetradecane-2,5,9,12-tetraone and two of its precursors