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List of works by Ulrike Holzgrabe

'Pro et contra' ionic liquid drugs - Challenges and opportunities for pharmaceutical translation

scientific article published on 10 June 2015

1,4-Substituted 4-(1H)-pyridylene-hydrazone-type inhibitors of AChE, BuChE, and amyloid-β aggregation crossing the blood-brain barrier

scientific article

11 The need for CE methods in pharmacopoeial monographs

11-Aminostrychnine and N-(Strychnine-11-yl)propionamide: Synthesis, Configuration, and Pharmacological Evaluation at Glycine Receptors

scientific article published on 06 August 2019

1H NMR analytical characterization of mineral oil hydrocarbons (PARAFFINS) for pharmaceutical use

scientific article published on 21 February 2019

1H NMR approach as an alternative to the classical p-anisidine value method

article published in 2012

1H NMR profiling as an approach to differentiate conventionally and organically grown tomatoes

scientific article published on 6 August 2014

1H and 13C nuclear magnetic resonance studies of the sites of protonation in itraconazole and fluconazole

scientific article

1H and 19F NMR relaxation studies of fleroxacin with Micrococcus luteus

scientific article published on 23 January 2007

1H and13C NMR studies of substituted isoquinolinium derivatives in different solvents

1H,19F and13C NMR spectral data of fifteen gyrase inhibitors and some metabolites

1H-NMR Spectroscopy as a New Tool in the Assessment of the Oxidative State in Edible Oils

35 Jahre Resistenzen gegen Antibiotika

4-[(2E)-2-(4-Chloro-benzyl-idene)hydrazinyl-idene]-1-methyl-1,4-dihydro-pyridine monohydrate

scientific article

5α‐Reduktase‐Inhibitoren – Benigne Prostatahyperplasie und vieles mehr. BPH, Alopezie und Co

scientific article published on 01 January 2008

A Fast and Efficient Track to Allosteric Modulators of Muscarinic Receptors: Microwave-Assisted Syntheses

A New Bioactive Compound From the Marine Sponge-Derived sp. SBT348 Inhibits Staphylococcal Growth and Biofilm Formation

scientific article published in 2018

A New Molecular Mechanism To Engineer Protean Agonism at a G Protein-Coupled Receptor

scientific article published on 6 February 2017

A Novel Mechanism of Inactivating Antibacterial Nitro Compounds in the Human Pathogen Staphylococcus aureus by Overexpression of a NADH-Dependent Flavin Nitroreductase

scientific article published on 13 November 2017

A Photoswitchable Dualsteric Ligand Controlling Receptor Efficacy.

scientific article published on 16 May 2017

A Sequence of Aldol Condensations and a Michael Addition Giving a Cyclohexenone Ring System

article

A Stable and Highly Potent Hexamethonium Derivative Which Modulates Muscarinic Receptors Allosterically in Guinea-pig Hearts

scientific article published on 01 February 1994

A Structural Biology Approach Enables the Development of Antimicrobials Targeting Bacterial Immunophilins

scientific article

A cell-permeable inhibitor to trap Gαq proteins in the empty pocket conformation

scientific article

A diversity oriented synthesis of natural product inspired molecular libraries

scientific article published on 19 October 2017

A long-time stability study of 50 drug substances representing common drug classes of pharmaceutical use

scientific article published on 02 May 2019

A miniaturized peptidyl-prolyl isomerase enzyme assay

scientific article published on 10 August 2017

A new in star in antibiotic heaven--daptomycin

scientific article

A new micellar electrokinetic capillary chromatography method for separation of the components of the aminoglycoside antibiotics

scientific article published in September 2003

A new synthetic route to compounds of the AFDX-type with affinity to muscarinic M2-receptor

article published in 2003

A novel class of allosteric modulators of the muscarinic M2 acetylcholine receptor: terphenyl derivatives

A riddle solved--why valerian-hops extract makes you drowsy

scientific article published in January 2004

A silver lining on the horizon: new antimycotics

scientific article published in January 2003

A small-molecule inhibitor of Nipah virus envelope protein-mediated membrane fusion

scientific article

A stability-study of expired ampoules manufactured more than 40 years ago.

scientific article published on 13 December 2017

A systematic review of the stability of finished pharmaceutical products and drug substances beyond their labeled expiry dates

scientific article published on 11 January 2019

A way out of a malaria-resistance?

scientific article published in January 2009

Absolute quantitative (1)h NMR spectroscopy for compound purity determination.

scientific article published on 7 November 2014

Acetylcholinesterase inhibitors with photoswitchable inhibition of β-amyloid aggregation

scientific article published on 14 March 2014

Agonists with supraphysiological efficacy at the muscarinic M2 ACh receptor.

scientific article published on May 2013

Allosteric Modulators and Selective Agonists of Muscarinic Receptors

scientific article published on 01 January 2006

Allosteric Modulators of the Tertiary Alkanebisamino-Type. Variation of the Substitution of the Middle Chain Nitrogens

Allosteric effect on muscarinic M2-receptors of derivatives of the alkane-bis-ammonium compound W84. Comparison with bispyridinium-type allosteric modulators

Allosteric ligands for G protein-coupled receptors: a novel strategy with attractive therapeutic opportunities

scientific article published on May 2010

Allosteric modulators of ligand binding to muscarinic acetylcholine receptors

Allosteric site in M2 acetylcholine receptors: evidence for a major conformational change upon binding of an orthosteric agonist instead of an antagonist

scientific article published on 16 December 2005

Allosteric small molecules unveil a role of an extracellular E2/transmembrane helix 7 junction for G protein-coupled receptor activation

scientific article published on 21 September 2007

Alpha blockers and 5-alpha reductase inhibitors

scientific article published in January 2008

Alte Wege zu neuen Antibiotika – Platensimycin

scientific article published on 01 January 2006

Alternative Wege zu “Multidrug”-resistenten Bakterien via reaktiver Sauerstoffspezies

Alternatives to amino acid analysis for the purity control of pharmaceutical grade L-alanine

scientific article published in August 2010

Amadacyclin - a new tetracycline antibiotic in the pipeline

scientific article published in March 2010

Amino acid analysis for pharmacopoeial purposes

scientific article published on 22 March 2016

Amino acids: Aspects of impurity profiling by means of CE

scientific article published on 01 July 2007

An LC–MS/MS procedure for the quantification of naproxen in human plasma: Development, validation, comparison with other methods, and application to a pharmacokinetic study

article

An old drug as a carcinostatic. The new career of thalidomide

scientific article published in January 2007

Analysis of atropine, its degradation products and related substances of natural origin by means of reversed-phase high-performance liquid chromatography

scientific article published in August 2004

Analysis of the glucosinolate pattern ofArabidopsis thalianaseeds by capillary zone electrophoresis coupled to electrospray ionization-mass spectrometry

article

Analysis of the molecular size distribution of polyethylene glycols by CE-UV versus HPLC with evaporative light scattering detection

scientific article published in September 2008

Analytical challenges in drug counterfeiting and falsification-The NMR approach

scientific article published on 21 December 2010

Analytical characterisation of crude extracts from an African Ancistrocladus species using high-performance liquid chromatography and capillary electrophoresis coupled to ion trap mass spectrometry

scientific article published in January 2004

Anatoxin-a(s) — ein bakterielles Organophosphat

scientific article published on 01 September 1994

Anti-Schistosomal Activity of Cinnamic Acid Esters: Eugenyl and Thymyl Cinnamate Induce Cytoplasmic Vacuoles and Death in Schistosomula of Schistosoma mansoni

scientific article published on 12 June 2015

Anti-bacterial anacardic acid derivatives

scientific article published on 10 June 2020

Anti-trypanosomal activities and structural chemical properties of selected compound classes

scientific article

Anticancer effects of NSC‑631570 (Ukrain) in head and neck cancer cells: In vitro analysis of growth, invasion, angiogenesis and gene expression

scientific article published on 25 November 2019

Antileishmanial and cytotoxic compounds from Valeriana wallichii and identification of a novel nepetolactone derivative.

scientific article published on April 2015

Antileishmanial lead structures from nature: analysis of structure-activity relationships of a compound library derived from caffeic Acid bornyl ester.

scientific article published on 27 January 2014

Antitrypanosomal activity of quaternary naphthalimide derivatives

scientific article published on 04 January 2007

Artemisinin and successors

scientific article

Assessment of inhibitory potency of antibiotics by MRI: apparent T 2 as a marker of cell growth

Assignment of the major and minor components of gentamicin for evaluation of batches

Atypical muscarinic allosteric modulation: cooperativity between modulators and their atypical binding topology in muscarinic M2 and M2/M5 chimeric receptors

scientific article

Azathioprine-induced reversible EBV-associated Hodgkin-like lymphoma after immunosuppressive therapy for autoimmune hepatitis

scientific article published in March 2018

Aziridine-2,3-dicarboxylate inhibitors targeting the major cysteine protease of Trypanosoma brucei as lead trypanocidal agents

scientific article published on 3 March 2006

Ball milling – a new concept for predicting degradation profiles in active pharmaceutical ingredients

scientific article published in 2021

Bemerkung zum DPhG-Statement: Wissenschaftliche Pharmazie und Homöopathie

scientific article published on 01 January 2006

Bioinspired Ion Pairs Transforming Papaverine into a Protic Ionic Liquid and Salts

scientific article published on 22 July 2020

Bioinspired co-crystals of Imatinib providing enhanced kinetic solubility

scientific article published on 04 May 2018

Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity

scientific article

Bisquaternary Ligands of the Common Allosteric Site of M2Acetylcholine Receptors: Search for the Minimum Essential Distances between the Pharmacophoric Elements

scientific article published on 01 March 1999

Bisquaternary dimers of strychnine and brucine. A new class of potent enhancers of antagonist binding to muscarinic M2 receptors

scientific article published in June 2003

Bistacrine derivatives as new potent antimalarials

scientific article

Bistacrines as potential antitrypanosomal agents.

scientific article

Bitopic muscarinic agonists and antagonists and uses thereof: a patent evaluation of US20160136145A1.

scientific article published on 14 December 2016

Bone penetration of amoxicillin and clavulanic acid evaluated by population pharmacokinetics and Monte Carlo simulation

scientific article published on 23 March 2009

CONTRIBUTION OF LATERAL SUBSTITUENTS IN HEPTANE-BISAMMONIUM DERIVATIVES TO THE ALLOSTERIC STABILIZATION OF ANTAGONIST BINDING TO M2-RECEPTORS

scientific article published on 01 January 1998

Capillary electrophoresis method for determination of related substances in glutathione reduced drug substance

Capillary electrophoresis separation of phenethylamine enantiomers using amino acid based ionic liquids

scientific article published on 17 October 2017

Capillary electrophoretic resolution of the enantiomers of 2,5-dimethyl-4-hydroxy-3(2H)-furanone, the key flavor compounds in strawberry fruit

Capillary zone electrophoresis as a tool for the quality control of goldenseal extracts

scientific article published in June 2005

Capillary zone electrophoresis for the determination of amodiaquine and three of its synthetic impurities in pharmaceutical formulations

scientific article published on 13 June 2018

Cer(IV) Oxidationen, 10. Mitt.: Oxidation von ω-Phenylalkyldicarbonyl- und dicarbonyl-analogen Verbindungen

Cer(IV)-Oxidationen von β-Aminoketonen. 3. Mitt.: Ein Syntheseweg zu 4-spirosubstituierten 1,2,3,4-Tetrahydroisochinolinen

Cer(IV)-Oxidationen von β-Aminoketonen. Teil IV: Synthese isomerer Phenanthridinone Cerium(IV)

Cer(IV)oxidationen von β-Aminoketonen, 6. Mitt.: Untersuchungen zum Reaktionsverlauf

Cer(IV)oxidationen von β-Aminoketonen, 8. Mitt.: Synthese von im Piperidinteil verschieden substituierten 1,2,3,4-Tetrahydroisochinolinen

Cer(IV)oxidationen von β–Aminoketonen. 7. Mitt.: Synthese von 4-Benzoylisochinolin und des davon abgeleiteten Lactams

Cer(IV)sulfat-Oxidationen: Intramolekulare Cyclisierung von N-Benzyl-β-aminoketonen zu 4-Benzoyl-1,2,3,4-tetrahydroisochinolinen

Cerium(IV)oxidations, Part IX: Cyclization of Diethyl 4-Phenylbutane-1, 1-dicarboxylate

scholarly article by Ulrike Holzgrabe et al published 1993 in Archiv der Pharmazie - Chemistry in Life Sciences

Cerulenin analogues as inhibitors of efflux pumps in drug-resistant Candida albicans

scientific article published in March 2009

Characterization of bacterial growth and the influence of antibiotics by means of UV resonance Raman spectroscopy.

scientific article published in July 2006

Characterization of complexes between phenethylamine enantiomers and β-cyclodextrin derivatives by capillary electrophoresis-Determination of binding constants and complex mobilities

scientific article published on 28 January 2017

Characterization of polydisperse macrogols and macrogol-based excipients via HPLC and charged aerosol detection

scientific article published on 27 July 2018

Charged aerosol detection in pharmaceutical analysis

scientific article published on 21 March 2012

Charged aerosol detector response modeling for fatty acids based on experimental settings and molecular features: a machine learning approach

scholarly article by Ruben Pawellek et al published 15 July 2021 in Journal of Cheminformatics

Chiral capillary electrophoresis: facts and fiction on the reproducibility of resolution with randomly substituted cyclodextrins

scientific article published in August 2004

Chiral discrimination of phenethylamines with β-cyclodextrin and heptakis(2,3-di-O-acetyl)β-cyclodextrin by capillary electrophoresis and NMR spectroscopy

scientific article published on 01 December 1994

Cinnamic Acid Bornyl Ester Derivatives from Valeriana wallichii Exhibit Antileishmanial In Vivo Activity in Leishmania major-Infected BALB/c Mice

scientific article

Comparable Bioavailability and Disposition of Pefloxacin in Patients with Cystic Fibrosis and Healthy Volunteers Assessed via Population Pharmacokinetics

scientific article published on 10 July 2019

Comparable population pharmacokinetics and pharmacodynamic breakpoints of cefpirome in cystic fibrosis patients and healthy volunteers

scientific article

Comparison of Conventional and Microwave Assisted Reactions Giving Aromatic Oxazolidines

Comparison of Cyclodextrin-Dipeptide Inclusion Complexes in the Absence and Presence of Urea by Means of Capillary Electrophoresis, Nuclear Magnetic Resonance and Molecular Modeling

Comparison of Pantoprazole Concentrations in Simultaneous Cerebrospinal Fluid and Serum Samples

scientific article

Comparison of chiral electrophoretic separation methods for phenethylamines and application on impurity analysis

scientific article published on 30 June 2010

Comparison of established and novel purity tests for the quality control of heparin by means of a set of 177 heparin samples

scientific article published on 08 September 2010

Comparison of extraction efficiency and selectivity between low-temperature pressurized microwave-assisted extraction and prolonged maceration

scientific article published on 31 August 2020

Comparison of pharmacological activities of three distinct kappa ligands (Salvinorin A, TRK-820 and 3FLB) on kappa opioid receptors in vitro and their antipruritic and antinociceptive activities in vivo

scientific article published on 21 September 2004

Comparison of structurally different allosteric modulators of muscarinic receptors by self-organizing neural networks

scientific article published in August 1996

Comparison of the pharmacokinetics and pharmacodynamic profile of carumonam in cystic fibrosis patients and healthy volunteers

scientific article published in October 2009

Comparison of the separation of aziridine isomers applying heptakis(2,3-di-O-methyl-6-sulfato)beta-CD and heptakis(2,3-di-O-acetyl-6-sulfato)beta-CD in aqueous and nonaqueous systems

scientific article published in October 2005

Competitive inhibition of renal tubular secretion of ciprofloxacin and metabolite by probenecid

scientific article

Competitive inhibition of renal tubular secretion of gemifloxacin by probenecid

scientific article published on 29 June 2009

Composition of OSCS-contaminated heparin occurring in 2008 in batches on the German market

scientific article

Contribution of lateral substituents in symmetrical and non-symmetrical heptane-bisammonio compounds to the allosteric stabilization of N-methylscopolamine binding to muscarinic M2 receptors

scientific article published in August 2003

Control of Cardiac Function in vivo with a Light-Regulated Drug

Control of impurities in L-aspartic acid and L-alanine by high-performance liquid chromatography coupled with a corona charged aerosol detector

scientific article published on 18 November 2009

Controlling Supramolecular Structures of Drugs by Light

scientific article published on 29 October 2020

Convergent, short synthesis of the muscarinic superagonist iperoxo

Cooperative interactions at M2 muscarinic acetylcholine receptors: structure/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators

scientific article published in April 2003

Corona Charged Aerosol Detector in studying retention and β-cyclodextrin complex stability using RP-HPLC

scientific article published on 22 October 2020

Critical aspects of analysis of Micrococcus luteus, Neisseria cinerea, and Pseudomonas fluorescens by means of capillary electrophoresis

scientific article published in October 2004

Crystal structure of (3S*,4R*)-4-fluoro-3-(4-meth-oxy-phen-yl)-1-oxo-2-phenyl-1,2,3,4-tetra-hydro-iso-quinoline-4-carb-oxy-lic acid

scientific article published on 23 May 2017

Crystal structure of 5,11-di-hydro-pyrido[2,3-b][1,4]benzodiazepin-6-one

scientific article published on 11 April 2015

Current role and future perspectives of multivariate (chemometric) methods in NMR spectroscopic analysis of pharmaceutical products

scientific article published on 27 May 2017

Cyclodextrin-Mediated Enantioseparation in Microemulsion Electrokinetic Chromatography

scientific article published on 01 January 2013

Cytochrome P450 1A2 phenotyping for student laboratories

Design, Synthesis and Evaluation of Novel 2-(Aminoalkyl)-isoindoline-1,3-dione Derivatives as Dual-Binding Site Acetylcholinesterase Inhibitors

scientific article published on 30 March 2012

Design, synthesis, and action of oxotremorine-related hybrid-type allosteric modulators of muscarinic acetylcholine receptors

scientific article published in January 2006

Designing Hybrids Targeting the Cholinergic System by Modulating the Muscarinic and Nicotinic Receptors: A Concept to Treat Alzheimer's Disease

scholarly article by Daniela Volpato & Ulrike Holzgrabe published 7 December 2018 in Molecules

Determination of binding constants of cyclodextrin inclusion complexes with amino acids and dipeptides by potentiometric titration

scientific article published on 01 October 2004

Determination of clotrimazole in mice plasma by capillary electrophoresis

scientific article

Determination of erythromycin and related substances in commercial samples using liquid chromatography/ion trap mass spectrometry

scientific article published on 02 October 2006

Determination of free fatty acids in edible oils by1H NMR spectroscopy

Determination of free fatty acids in pharmaceutical lipids by 1H NMR and comparison with the classical acid value

scientific article published on 17 April 2013

Determination of protein binding of gyrase inhibitors by means of continuous ultrafiltration

scientific article published on 01 December 1998

Determination of the extent of protein binding of antibiotics by means of an automated continuous ultrafiltration method

scientific article published on 20 January 2006

Development and validation of a generic stability-indicating MEEKC method for five fluoroquinolone antibiotics

scientific article published on 12 May 2015

Development and validation of a separation method for the diastereomers and enantiomers of aziridine-type protease inhibitors

article

Development of a new type of allosteric modulator of muscarinic receptors: hybrids of the antagonist AF-DX 384 and the hexamethonio derivative W84.

scientific article

Development of a simple, rapid, and robust liquid chromatographic method for the simultaneous determination of sulfalene, sulfadoxine, and pyrimethamine in tablets.

scientific article published on 30 July 2016

Development of an enhanced separation of erythromycin and its related substances by liquid chromatography

article

Development of simplified HPLC methods for the detection of counterfeit antimalarials in resource-restraint environments

article

Development, synthesis and structure-activity-relationships of inhibitors of the macrophage infectivity potentiator (Mip) proteins of Legionella pneumophila and Burkholderia pseudomallei

scientific article

Die Entwicklung selektiver α2-Rezeptor-Agonisten

scientific article published on 01 November 2011

Die Fettsäuresynthese als Angriffspunkt

scientific article published on 01 January 2012

Die Natur als Apotheke gegen Tropenkrankheiten: Tirandamycin B gegen lymphatische Filariosen

scientific article published on 01 November 2011

Differentiation of Organically and Conventionally Grown Tomatoes by Chemometric Analysis of Combined Data from Proton Nuclear Magnetic Resonance and Mid-infrared Spectroscopy and Stable Isotope Analysis

scientific article

Diffusion ordered NMR spectroscopy measurements as screening method of potential reactions of API and excipients in drug formulations

scientific article published on 08 September 2018

Distinguishing paracetamol formulations: Comparison of potentiometric "Electronic Tongue" with established analytical techniques

scientific article published on 06 July 2020

Do we know the mechanism of chiral recognition between cyclodextrins and analytes?

scientific article published in January 2002

Do we need new drugs against human African trypanosomiasis?

scientific article

Drug Discovery: A Modern Decathlon

scientific article published on 06 March 2013

Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity

scientific article published on 8 October 2008

Dualsteric muscarinic antagonists--orthosteric binding pose controls allosteric subtype selectivity

scientific article published on 4 August 2014

Dynamic ligand binding dictates partial agonism at a G protein-coupled receptor.

scientific article

E-Z isomerism of anilinomethylenemalonic acid derivatives

Editorial: Pharmazie in unserer Zeit 1/2004

scholarly article by Ulrike Holzgrabe & Fritz Sörgel published January 2004 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 1/2012

scientific article published on 01 January 2012

Editorial: Pharmazie in unserer Zeit 2/2005

scholarly article by Ulrike Holzgrabe & Ulrich Jaehde published March 2005 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 2/2006

scholarly article by Ulrike Holzgrabe & Charlotte Kloft published March 2006 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 2/2008

scholarly article by Ulrike Holzgrabe & Matthias F. Melzig published March 2008 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 2/2009

scholarly article by Petra Högger & Ulrike Holzgrabe published March 2009 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 2/2011

scientific article published on 01 March 2011

Editorial: Pharmazie in unserer Zeit 3/2007

scholarly article by Ulrike Holzgrabe & Christa E. Müller published May 2007 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 5/2004

scholarly article by Ulrike Holzgrabe & Peter Christian Schmidt published September 2004 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 5/2006

scholarly article by Fritz Sörgel & Ulrike Holzgrabe published September 2006 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 6/2005

scientific article published on 01 January 2005

Editorial: Pharmazie in unserer Zeit 6/2007

scholarly article by Gerd Bendas et al published November 2007 in Pharmazie in unserer Zeit

Editorial: Pharmazie in unserer Zeit 6/2009

scientific article published in January 2009

Editorial: Pharmazie in unserer Zeit 6/2010

scientific article published on 01 November 2010

Editorial: Pharmazie in unserer Zeit 6/2011

scientific article published on 01 November 2011

Effect of various cyclodextrin derivatives on the resolution of fencamfamine isomers with capillary electrophoresis and nuclear magnetic resonance

article published in 1998

Effect of β-cyclodextrin acetylation on the resolution of phenethylamines with capillary electrophoresis and nuclear magnetic resonance spectroscopy

Effects of fluoroquinolones on HERG channels and on pancreatic beta-cell ATP-sensitive K+ channels

scientific article published on 8 September 2006

Elevation of ligand binding to muscarinic M(2) acetylcholine receptors by bis(ammonio)alkane-type allosteric modulators

scientific article published in August 2002

Emergency admission of peramivir in the U.S.A

scientific article published in January 2010

Enantioseparation by Capillary Electrophoresis Using Cyclodextrins in an Amino Acid-Based Ionic Liquid Running Buffer

scientific article published on 01 January 2019

Enantioseparation of chiral tropa alkaloids by means of cyclodextrin-modified microemulsion electrokinetic chromatography

scientific article published on 01 August 2007

Enantioseparation of dihydropyridine derivatives by means of neutral and negatively charged beta-cyclodextrin derivatives using capillary electrophoresis

scientific article published on 01 November 2000

Enantioseparation of dopa and related compounds by cyclodextrin-modified microemulsion electrokinetic chromatography

scientific article published on 24 May 2008

Enantioseparation of linear and cyclic chiral bis(phenethyl)amines by means of cyclodextrin-modified capillary electrophoresis

scientific article published on 01 September 2001

Enantioseparation of tropa alkaloids by means of anionic cyclodextrin-modified capillary electrophoresis

scientific article published on 01 June 1999

Engineered Context-Sensitive Agonism: Tissue-Selective Drug Signaling through a G Protein-Coupled Receptor

scientific article published on 15 November 2016

Erratum to: Comparison of established and novel purity tests for the quality control of heparin by means of a set of 177 heparin samples

scholarly article published in Analytical and Bioanalytical Chemistry

Evaluation by monte carlo simulation of the pharmacokinetics of two doses of meropenem administered intermittently or as a continuous infusion in healthy volunteers.

scientific article

Evaluation of amino sugar, low molecular peptide and amino acid impurities of biotechnologically produced amino acids by means of CE.

scientific article

Evaluation of enantiomeric purity of magnesium-L-aspartate dihydrate

scientific article

Evaluation of the extent of protein binding by means of NMR diffusion and relaxation experiments, and automated continuous ultrafiltration.

scientific article published on 22 January 2009

Evaluation of the impurity profile of alcuronium by means of capillary electrophoresis

scientific article published in June 2002

Evaluation of the impurity profile of amino acids by means of CE.

scientific article

Evaluation of the stability of gentamicin in different antibiotic carriers using a validated MEKC method

scientific article published on 18 June 2008

Evidence for a multiple binding mode of bispyridinium-type allosteric modulators of muscarinic receptors

article

FRET Studies of Quinolone-Based Bitopic Ligands and Their Structural Analogues at the Muscarinic M1 Receptor

scientific article published on 24 January 2017

FRET zur Bestimmung der minimalen Hemmkonzentration von Antibiotika

scientific article published on 01 January 2012

Fatty acid composition analysis in polysorbate 80 with high performance liquid chromatography coupled to charged aerosol detection

article

Fenton's oxidation: a tool for the investigation of potential drug metabolites

scientific article

Ficts and facts of epinephrine and norepinephrine stability in injectable solutions

scientific article published on 18 May 2012

FimH-Inhibitoren - eine neue Möglichkeit chronische Harnwegsinfektionen zu behandeln und zu verhindern

scientific article published on 01 March 2012

First population pharmacokinetic analysis showing increased quinolone metabolite formation and clearance in patients with cystic fibrosis compared to healthy volunteers

scholarly article by Yuanyuan Jiao et al published 15 October 2018 in European Journal of Pharmaceutical Sciences

Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties

scientific article published on 19 March 2019

Fluorine walk: The impact of fluorine in quinolone amides on their activity against African sleeping sickness

scientific article published on 30 April 2018

Focus on PAINS: false friends in the quest for selective anti-protozoal lead structures from Nature?

Future Information Technology Tools for Fighting Substandard and Falsified Medicines in Low- and Middle-Income Countries

scholarly article by Huma Rasheed et al published 2018 in Frontiers in Pharmacology

Geometrical and Structural Dynamics of Imatinib within Biorelevant Colloids

article

Glufosfamid – ein neues Lost-Derivat: PerfektesDrug-Targeting

scientific article published on 01 January 2006

H1-Antihistaminika der ersten Generation. Problemlos in der Empfehlung?

scientific article published on 01 January 2007

Helfen Sie uns, unseren wissenschaftlichen Nachwuchs zu fördern!

scientific article published on 01 January 2008

High-performance liquid chromatography evaluation of the enantiomeric purity of amino acids by means of automated precolumn derivatization with ortho-phthalaldehyde and chiral thiols.

scientific article

How safe was oseltamivir care in the flu pandemic?

scientific article

Ibuprofen for Alzheimer's?

scientific article published in January 2002

Identification and characterization of diarylimidazoles as hybrid inhibitors of butyrylcholinesterase and amyloid beta fibril formation

scientific article

Identification and control of impurities in streptomycin sulfate by high-performance liquid chromatography coupled with mass detection and corona charged-aerosol detection

scientific article

Identification and quantitation of the ingredients in a counterfeit Vietnamese herbal medicine against rheumatic diseases

scientific article published on 19 April 2014

Improving anti-trypanosomal activity of alkamides isolated from Achillea fragrantissima

scientific article published on 3 November 2017

Impurity profile of amino acids?

scientific article published on 01 August 2005

Impurity profiling of N,N'-ethylenebis-l-cysteine diethyl ester (Bicisate).

scientific article published on 5 December 2017

Impurity profiling of atropine sulfate by microemulsion electrokinetic chromatography

scientific article

Impurity profiling of carbocisteine by HPLC-CAD, qNMR and UV/vis spectroscopy

scientific article published on 25 February 2014

Impurity profiling of ibandronate sodium by HPLC–CAD

scientific article published on 06 June 2015

Impurity profiling of l -asparagine monohydrate by ion pair chromatography applying low wavelength UV detection

scientific article published on 30 August 2016

Impurity profiling of l-aspartic acid and glycine using high-performance liquid chromatography coupled with charged aerosol and ultraviolet detection

scientific article published on 05 February 2020

Impurity profiling of l-methionine by HPLC on a mixed mode column

scientific article published on 02 February 2016

In search of novel agents for therapy of tropical diseases and human immunodeficiency virus

scientific article published on 27 December 2007

Indirect Enantioseparation of Amino Acids by CE Using Automated In-Capillary Derivatization with ortho-Phthalaldehyde and N-Acetyl-l-Cysteine

article published in 2016

Influence of charged aerosol detector instrument settings on the ultra-high-performance liquid chromatography analysis of fatty acids in polysorbate 80

scientific article published on 18 September 2018

Influence of the capillary diameter on the separation efficiency and sensitivity: a systematic approach

scientific article

Inhibition of cytochrome P450 3A4 by extracts and kavalactones of Piper methysticum (Kava-Kava).

scientific article

Inhibition of flucloxacillin tubular renal secretion by piperacillin

scientific article

Inhibition of hypusine biosynthesis in plasmodium: a possible, new strategy in prevention and therapy of malaria

scientific article published on November 2006

Inhibition von Virulenzfaktoren: Ein neuer Ansatz zur Entwicklung von Antibiotika

scientific article published on 01 January 2006

Inhibitoren der New‐Delhi‐Metallolactamase

scientific article published on 01 July 2012

Inhibitors of macrophage infectivity potentiator-like PPIases affect neisserial and chlamydial pathogenicity

scientific article published on August 2016

Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases

scientific article published on 15 January 2010

Interlaboratory Comparison Test as an Evaluation of Applicability of an Alternative Edible Oil Analysis by (1)H NMR Spectroscopy

scientific article

Interlaboratory study of a NACE method for the determination ofR-timolol content inS-timolol maleate: Assessment of uncertainty

scientific article published on 01 June 2006

Investigation of Multi-Component Drugs by NMR Spectroscopy

Investigation of tryptophan-related yellowing in parenteral amino acid solution: Development of a stability-indicating method and assessment of degradation products in pharmaceutical formulations

scientific article published on 27 August 2019

Ionic Liquids in Capillary Electrophoresis

scientific article published on 01 January 2016

Ionic liquid versus prodrug strategy to address formulation challenges

scientific article published on 23 December 2014

Isolation and Characterization of Galloylglucoses Effective against Multidrug-Resistant Strains of Escherichia coli and Klebsiella pneumoniae

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Isolation of a novel compound (MIMO2) from the methanolic extract of Moringa oleifera leaves: protective effects against vanadium-induced cytotoxity

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Kappa-receptor selective binding of opioid ligands with a heterocyclic bicyclo[3.3.1]nonan-9-one structure

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Keto-Enol-Tautomerism and Configurational Isomerism of 2,6-Disubstituted 4-Piperidone-3,5-dicarboxylates

Ketolide und Oxazolidinone in der Pipeline: Und die Reise geht weiter…

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Lactivicin – ein Antibiotikum gegen Penicillin-resistente Pneumokokken

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Large-scale attack against Plasmodium

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Ligand Binding Ensembles Determine Graded Agonist Efficacies at a G Protein-coupled Receptor

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Ligand-Specific Allosteric Coupling Controls G-Protein-Coupled Receptor Signaling

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Mechanism of action of the diazabicyclononanone-type kappa-agonists

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Mechanochemical Oxidative Degradation of Thienopyridine Containing Drugs: Toward a Simple Tool for the Prediction of Drug Stability

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Microwave-enhanced hydrogenations at medium pressure using a newly constructed reactor

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Muscarinic Allosteric Modulators: Atypical Structure-Activity-Relationships in Bispyridinium-type Compounds

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NMR Spectroscopic and Molecular Modelling Studies on Cyclodextrin-Dipeptide Inclusion Complexes

NMR spectroscopy in pharmaceutical and biomedical analysis

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NMR spectroscopy in pharmacy

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Neue Antiepileptika im Überblick

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Neue Hoffnung für Krebspatienten?

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Neuroprotective Effects of Isosteviol Sodium in Murine Brain Capillary Cerebellar Endothelial Cells (cerebEND) After Hypoxia

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Novel Population Pharmacokinetic Approach to Explain the Differences between Cystic Fibrosis Patients and Healthy Volunteers via Protein Binding

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Preface

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Syntheses and Biological Activities of NewN1-Aryl Substituted Quinolone Antibacterials

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Synthesis and evaluation of antitrypanosomal activity of some thiosemicarbazide derivatives of 1-butyl-6-fluoro-7-morpholino-4-oxo-1,4-dihydroquinoline-3-carboxylic acid

Synthesis and opioid receptor affinity of a series of 2, 4-diaryl-substituted 3,7-diazabicylononanones

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Synthesis and structure-activity relationships of new quinolone-type molecules against Trypanosoma brucei

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Synthesis, bioactivity and molecular modeling studies on potential anti-Alzheimer piperidinehydrazide-hydrazones

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Synthesis, biological activity, and docking studies of new acetylcholinesterase inhibitors of the bispyridinium type

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Systematic comparison of the population pharmacokinetics and pharmacodynamics of piperacillin in cystic fibrosis patients and healthy volunteers

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Systematic development of high affinity bis(ammonio)alkane-type allosteric enhancers of muscarinic ligand binding

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Tacrine-xanomeline and tacrine-iperoxo hybrid ligands: Synthesis and biological evaluation at acetylcholinesterase and M1 muscarinic acetylcholine receptors

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Tamper-proof tablets for distinction between counterfeit and originator drugs through PEG coding

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Targeting acetylcholinesterase to treat neurodegeneration

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Targeting protein folding; a novel approach for the treatment of pathogenic bacteria

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Tautomerism of 4-hydroxy-2,5-dimethyl-3(2H)-furanone: evidence for its enantioselective biosynthesis

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The Influence of Fluoroquinolone Drugs on the Bacterial Growth ofS. epidermidisUtilizing the Unique Potential of Vibrational Spectroscopy

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The Role of Orthosteric Building Blocks of Bitopic Ligands for Muscarinic M1 Receptors

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The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling

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The contamination of valsartan and other sartans, Part 2: Untargeted screening reveals contamination with amides additionally to known nitrosamine impurities

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Valeriana wallichii root extracts and fractions with activity against Leishmania spp

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Vibrational spectroscopic characterization of fluoroquinolones

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Zwei Fliegen mit einer Klappe – Platencin, ein neues Antibiotikum

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Zwitterionic-hydrophilic interaction liquid chromatography for l-ascorbic acid 2-phosphate magnesium, a raw material in cell therapy

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qNMR Spectroscopy in Drug Analysis – A General View

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