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List of works by John Christopher Vederas

A carbonate-forming Baeyer-Villiger monooxygenase

scientific article published on 18 May 2014

A concise stereoselective synthesis of orthogonally protected lanthionine and β-methyllanthionine

scientific article published on 07 February 2007

A fungal ketoreductase domain that displays substrate-dependent stereospecificity

scientific article published on 11 March 2012

A mechanistic view of enzyme inhibition and peptide hydrolysis in the active site of the SARS-CoV 3C-like peptidase

scientific article

A pathway for the biosynthesis of fatty acid amides

scientific article published on 01 January 1999

Amidation of Salicyluric Acid and Gentisuric Acid: A Possible Role for Peptidylglycine α-Amidating Monooxygenase in the Metabolism of Aspirin

scientific article published on 01 November 2000

Amination of chiral enolates by dialkyl azodiformates. Synthesis of .alpha.-hydrazino acids and .alpha.-amino acids

article by Laird A. Trimble & John Christopher Vederas published October 1986 in Journal of the American Chemical Society

Amination with N-benzyloxycarbonyl-3-phenyloxaziridine as a route to sensitive chiral α-hydrazino acids: Synthesis of l-hydrazino serine

An acid metabolite of cyclosporine

scientific article published in 1985

An episulfide cation (thiiranium ring) trapped in the active site of HAV 3C proteinase inactivated by peptide-based ketone inhibitors

scientific article

Analogs of diaminopimelic acid as inhibitors of meso-diaminopimelate decarboxylase from Bacillus sphaericus and wheat germ.

scientific article published on October 1986

Analogs of diaminopimelic acid as inhibitors of meso-diaminopimelate dehydrogenase and LL-diaminopimelate epimerase

scientific article published in Journal of Biological Chemistry

Angiotensin-Converting Enzyme 2 Metabolizes and Partially Inactivates Pyr-Apelin-13 and Apelin-17: Physiological Effects in the Cardiovascular System

scientific article

Antimicrobial Leucocin Analogues with a Disulfide Bridge Replaced by a Carbocycle or by Noncovalent Interactions of Allyl Glycine Residues

scientific article published on 01 November 2006

Antimicrobial lipopeptide tridecaptin A1 selectively binds to Gram-negative lipid II

scientific article

Apelin directs endothelial cell differentiation and vascular repair following immune-mediated injury

scientific article published on 01 January 2020

Apelin protects against abdominal aortic aneurysm and the therapeutic role of neutral endopeptidase resistant apelin analogs

scientific article published on 12 June 2019

Application of stable isotope labelling methodology to the biosynthesis of the mycotoxin, terretonin, by aspergillus terreus: incorporation of 13C-labelled acetates and methionine, 2H- and 13C, 18O-labelled ethyl 3,5-dimethylorsellinate and oxygen-18

Approaches to the discovery of new antibacterial agents based on bacteriocins

scientific article published on April 2008

Aryl methylene ketones and fluorinated methylene ketones as reversible inhibitors for severe acute respiratory syndrome (SARS) 3C-like proteinase

scientific article published on 4 March 2008

Aspects of the biosynthesis of non-aromatic fungal polyketides by iterative polyketide synthases.

scientific article published in December 2000

Atypical genetic locus associated with constitutive production of enterocin B by Enterococcus faecium BFE 900.

scientific article

Author Correction: Feline coronavirus drug inhibits the main protease of SARS-CoV-2 and blocks virus replication

scientific article published on 20 October 2020

Bacillus amyloliquefaciens ssp. plantarum F11 isolated from Algerian salty lake as a source of biosurfactants and bioactive lipopeptides.

scientific article published on 23 November 2017

Bacterial diaminopimelate metabolism as a target for antibiotic design.

scientific article published in May 2000

Beta-lactones as a new class of cysteine proteinase inhibitors: inhibition of hepatitis A virus 3C proteinase by N-Cbz-serine beta-lactone.

scientific article

Biochemical and Structural Basis for Controlling Chemical Modularity in Fungal Polyketide Biosynthesis

scientific article

Biochemical, structural, and genetic characterization of tridecaptin A₁, an antagonist of Campylobacter jejuni.

scientific article

Biosyntheses of antibiotic A26771B by Penicillium turbatum and dehydrocurvularin by Alternaria cinerariae: comparison of stereochemistry of polyketide and fatty acid enoyl thiol ester reductases

article

Biosynthesis and full NMR assignment of fungichromin, a polyene antibiotic from Streptomyces cellulose

scientific article published in 1988

Biosynthesis of Cytochalasans. Part 4. The mode of incorporation of common naturally-occurring carboxylic acids into cytochalasin D

scientific article published on 01 November 1975

Biosynthesis of LL-D253? in Phoma pigmentivora. Incorporation of 13C, 2H, and 18O enriched precursors

Biosynthesis of ML-236C and the hypocholesterolemic agents compactin by Penicillium aurantiogriseum and lovastatin by Aspergillus terreus: determination of the origin of carbon, hydrogen and oxygen atoms by 13C NMR spectrometry and observation of unu

Biosynthesis of aminovinyl-cysteine-containing peptides and its application in the production of potential drug candidates

scientific article

Biosynthesis of aspyrone and asperlactone, pentaketide metabolites of Aspergillus melleus. Incorporation studies with [1-13C, 18O2]acetate and 18O2 gas

Biosynthesis of averufin by Aspergillus parasiticus; detection of 18O-label by 13C-n.m.r. isotope shifts

Biosynthesis of cytochalasans. Part 6. The mode of incorporation of phenylalanine into cytochalasin D1.

scientific article

Biosynthesis of lovastatin and related metabolites formed by fungal iterative PKS enzymes

scientific article published on September 2010

Biosynthesis of macrolides. 5. Regiochemistry of the labeling of lasalocid A by [13C,18O]-labeled precursors

scientific article published in 1981

Biosynthesis of macrolides. 6. Mechanism of stereocontrol during the formation of lasalocid A

scientific article published in 1981

Biosynthesis of mevinolin. Spectral assignment by double-quantum coherence NMR after high carbon-13 incorporation

scientific article published in 1983

Biosynthesis of monocerin. Incorporation of 2H-, 13C-, and 18O-labelled acetates by Drechslera ravenelii

Biosynthesis of multicolosic acid, a polyketide metabolite from Penicillium multicolor: occurrence of large18O-induced β-isotope shifts in13C n.m.r. spectra

Biosynthesis of polyene antibiotics: intact incorporation of carbon-13 labeled octanoate into fungichromin by Streptomyces cellulosae

scientific article published in 1986

Biosynthesis of solanapyrone A, a phytotoxin of Alternaria solani

Biosynthesis of tajixanthone and shamixanthone by Aspergillus variecolor: incorporation of oxygen-18 gas

Biosynthesis of the Cytochalasans. Part III.13C-NMR. of cytochalasin B (phomin) and cytochalasin D. Incorporation of [1-13C]- and [2-13C]-sodium acetate

scientific article published on 01 January 1974

Biosynthesis of the aflatoxin precursor sterigmatocystin by Aspergillus versicolor; spin-echo resolution of 18O isotope shifts in 13C-n.m.r. spectroscopy

Biosynthesis of the hypocholesterolemic agent mevinolin by Aspergillus terreus. Determination of the origin of carbon, hydrogen, and oxygen atoms by carbon-13 NMR and mass spectrometry

article

Biosynthesis of the meroterpenoid austin, by Aspergillus ustus: synthesis and incorporation of 13C,18O-labelled ethyl 3,5-dimethylorsellinate

Biosynthesis of the meroterpenoid metabolite, andibenin B: incorporation of sodium [1-13C, 18O2]acetate and 18O2

Biosynthesis of the meroterpenoid metabolite, andilesin A, by Aspergillus variecolor: origins of the oxygen atoms

Biosynthesis of the meroterpenoid, austin, by Aspergillus ustus: incorporation of 18O2, sodium [1-13C, 18O2]acetate, and [Me-13C, 2H3]methionine

Biosynthetic incorporation of advanced precursors into dehydrocurvularin, a polyketide phytotoxin from Alternaria cinerariae

Biosynthetic incorporation of labeled tetraketide intermediates into dehydrocurvularin, a phytotoxin from Alternaria cinerariae, with assistance of .beta.-oxidation inhibitors

scientific article published in 1992

Catalytic mechanism and properties of pyridoxal 5'-phosphate independent racemases: how enzymes alter mismatched acidity and basicity

scientific article published on 01 December 2019

Characteristics and genetic determinant of a hydrophobic peptide bacteriocin, carnobacteriocin A, produced by Carnobacterium piscicola LV17A.

scientific article published in March 1994

Characterization of DcsC, a PLP-independent racemase involved in the biosynthesis of d-cycloserine

scientific article published on 06 February 2012

Characterization of a locus from Carnobacterium piscicola LV17B involved in bacteriocin production and immunity: evidence for global inducer-mediated transcriptional regulation

scientific article published on October 1997

Characterization of bacterial antimicrobial peptides active against Campylobacter jejuni

Characterization of leucocin A-UAL 187 and cloning of the bacteriocin gene from Leuconostoc gelidum

scientific article

Characterization of the genetic locus responsible for production and immunity of carnobacteriocin A: the immunity gene confers cross-protection to enterocin B.

scientific article published in March 2000

Characterization of the protein conferring immunity to the antimicrobial peptide carnobacteriocin B2 and expression of carnobacteriocins B2 and BM1

scientific article published on March 1995

Chemical and genetic characterization of bacteriocins produced by Carnobacterium piscicola LV17B.

scientific article published in April 1994

Chemical synthesis and biological activity of the neopetrosiamides and their analogues: revision of disulfide bond connectivity

scientific article

Chemical synthesis and biological evaluation of gallidermin-siderophore conjugates

scientific article published on 03 February 2011

Cloning and Characterization of the Gene Cluster Involved in the Production of the Circular Bacteriocin Carnocyclin A.

scientific article published in December 2010

Comparison of 10,11-Dehydrocurvularin Polyketide Synthases from Alternaria cinerariae and Aspergillus terreus Highlights Key Structural Motifs

scientific article

Comparison of fatty acid and polyketide biosynthesis: stereochemistry of cladosporin and oleic acid formation in Cladosporium cladosporioides

scientific article published in 1989

Comparison of stereochemistry of fatty acid and cladosporin biosynthesis in Cladosporium cladosporioides using deuterium-decoupled proton, carbon-13 NMR shift correlation

scientific article published in 1988

Complete reconstitution of a highly reducing iterative polyketide synthase

scientific article published on October 2009

Conjugate addition of radicals generated from diacyloxyiodobenzenes to dehydroamino acid derivatives; a synthesis of diaminopimelic acid analogues

scientific article

Conversion of cyclic nonaketides to lovastatin and compactin by a lovC deficient mutant of Aspergillus terreus.

scientific article published in June 2001

Conversion of serine .beta.-lactones to chiral .alpha.-amino acids by copper-containing organolithium and organomagnesium reagents

scientific article published in 1987

Conversion of serine to stereochemically pure .beta.-substituted .alpha.-amino acids via .beta.-lactones

scientific article published in 1985

Crystal structure and biochemical studies of the trans-acting polyketide enoyl reductase LovC from lovastatin biosynthesis

scientific article

Crystal structure of LL-diaminopimelate aminotransferase from Arabidopsis thaliana: a recently discovered enzyme in the biosynthesis of L-lysine by plants and Chlamydia

scientific article

Crystal structure of diaminopimelate epimerase from Arabidopsis thaliana, an amino acid racemase critical for L-lysine biosynthesis

scientific article

Design, synthesis, and evaluation of inhibitors for severe acute respiratory syndrome 3C-like protease based on phthalhydrazide ketones or heteroaromatic esters

scientific article published on 24 March 2007

Dess-Martin periodinane oxidative rearrangement for preparation of α-keto thioesters.

scientific article published on 3 January 2018

Development of Class IIa Bacteriocins as Therapeutic Agents

scientific article

Diacylglycerol Acyltransferase 1 Is Regulated by Its N-Terminal Domain in Response to Allosteric Effectors.

scientific article published on 21 August 2017

Differential Hydrogen Exchange During Biosynthesis of Cytochalasins B and D

Differential response of orthologous L,L-diaminopimelate aminotransferases (DapL) to enzyme inhibitory antibiotic lead compounds.

scientific article published on 9 November 2013

Dissecting the Binding Interactions of Teixobactin with the Bacterial Cell-Wall Precursor Lipid II

scientific article published on 12 November 2019

Double Oxidation of the Cyclic Nonaketide Dihydromonacolin L to Monacolin J by a Single Cytochrome P450 Monooxygenase, LovA

scientific article published on 15 April 2011

Draft Genome Sequence of Bacillus paralicheniformis F47, Isolated from an Algerian Salty Lake.

scientific article published on 29 March 2018

Draft Genome Sequence of Enterococcus canintestini 49, a Potential Probiotic That Produces Multiple Bacteriocins

scientific article published on 5 October 2017

Draft Genome Sequence of the Bacteriocin-Producing Strain Enterococcus faecium M3K31, Isolated from Griffon Vultures (Gyps fulvus subsp. fulvus).

scientific article

Draft Genome Sequence of the Thermophilic Bacterium Bacillus licheniformis SMIA-2, an Antimicrobial- and Thermostable Enzyme-Producing Isolate from Brazilian Soil

scientific article published on 23 April 2020

Draft Genome Sequences of Bacillus cereus E41 and Bacillus anthracis F34 Isolated from Algerian Salt Lakes

scientific article

Draft Genome Sequences of Paenibacillus polymyxa NRRL B-30509 and Paenibacillus terrae NRRL B-30644, Strains from a Poultry Environment That Produce Tridecaptin A and Paenicidins

scientific article

Drug discovery and natural products: end of an era or an endless frontier?

scientific article

Dual modes of modification of hepatitis A virus 3C protease by a serine-derived beta-lactone: selective crystallization and formation of a functional catalytic triad in the active site

scientific article

Dynamic relationships among type IIa bacteriocins: temperature effects on antimicrobial activity and on structure of the C-terminal amphipathic alpha helix as a receptor-binding region

scientific article published in July 2004

Dynamics of catalysis revealed from the crystal structures of mutants of diaminopimelate epimerase

scientific article

Effect of amino acid substitutions on the activity of carnobacteriocin B2. Overproduction of the antimicrobial peptide, its engineered variants, and its precursor in Escherichia coli.

scientific article

Effect of analogues of diaminopimelic acid on the meso -diaminopimelate-adding enzyme from Escherichia coli

scientific article published on 01 August 1996

Enzymatic synthesis of resorcylic acid lactones by cooperation of fungal iterative polyketide synthases involved in hypothemycin biosynthesis

scientific article published on April 2010

Enzymatic synthesis of valerena-4,7(11)-diene by a unique sesquiterpene synthase from the valerian plant (Valeriana officinalis). ⬇️

scientific article

Exploration of inhibitors for diaminopimelate aminotransferase

scientific article published on 06 February 2010

Explorations of fungal biosynthesis of reduced polyketides - a personal viewpoint

scientific article

Feline coronavirus drug inhibits the main protease of SARS-CoV-2 and blocks virus replication

scientific article published on 05 May 2020

Feline coronavirus drug inhibits the main protease of SARS-CoV-2 and blocks virus replication

scientific article published on 27 August 2020

For the record: The three-dimensional structure of the ternary complex ofCorynebacterium glutamicumdiaminopimelate dehydrogenase-NADPH-L-2-amino-6-methylene-pimelate

scientific article

Formation of peptide amides by peptidylglycine .alpha.-amidating monooxygenase: a new assay and stereochemistry of hydrogen loss

scientific article published in 1988

Fracturing rings to understand lantibiotics

scientific article

Functional characterization of recombinant hyoscyamine 6β-hydroxylase from Atropa belladonna

scientific article published on 26 May 2012

Fundamental functionality: recent developments in understanding the structure-activity relationships of lantibiotic peptides

scientific article

Fungal xanthone biosynthesis. Distribution of acetate-derived oxygens in ravenelin

scientific article published in 1982

Further studies on the biosynthesis of granaticin ⬇️

scientific article published on 01 January 1986

Genes of the sbo-alb locus of Bacillus subtilis are required for production of the antilisterial bacteriocin subtilosin

scientific article

Genetic characterization and heterologous expression of brochocin-C, an antibotulinal, two-peptide bacteriocin produced by Brochothrix campestris ATCC 43754

scientific article

Genetic determinants of reutericyclin biosynthesis in Lactobacillus reuteri

scientific article published on 9 January 2015

Heteroaromatic ester inhibitors of hepatitis A virus 3C proteinase: Evaluation of mode of action

scientific article

Highly selective but multifunctional oxygenases in secondary metabolism

scientific article published on 24 September 2014

Hydrophobic Interactions as Substitutes for a Conserved Disulfide Linkage in the Type IIa Bacteriocins, Leucocin A and Pediocin PA-1

scientific article published on 01 August 2008

Identification and Heterologous Expression of the sec-Dependent Bacteriocin Faerocin MK from Enterococcus faecium M3K31.

scientific article published on 6 January 2018

Identification and comparison of natural rubber from two Lactuca species.

scientific article

Identification and three-dimensional structure of carnobacteriocin XY, a class IIb bacteriocin produced by Carnobacteria.

scientific article published on 9 April 2017

Identification of Active Site Cysteine Residues that Function as General Bases: Diaminopimelate Epimerase

article

Identification of an N-terminal formylated, two-peptide bacteriocin from Enterococcus faecalis 710C.

scientific article

Identification of didecyldimethylammonium salts and salicylic acid as antimicrobial compounds in commercial fermented radish kimchi

scientific article published on 17 March 2015

Identification of sterigmatocystin as a metabolite of Monocillium nordinii ⬇️

scientific article published on August 1, 1981

In vitro and ex vivo inhibition of hepatitis A virus 3C proteinase by a peptidyl monofluoromethyl ketone.

scientific article published on May 1997

Incorporation of deuterium-labelled analogs of isopentenyl diphosphate for the elucidation of the stereochemistry of rubber biosynthesis

scientific article published on 23 January 2006

Inhibition of cytoplasmic aspartate aminotransferase from porcine heart by R and S isomers of aminooxysuccinate and hydrazinosuccinate

scientific article published in Journal of Biological Chemistry

Inhibitors of 3C cysteine proteinases from Picornaviridae

scientific article published in January 2004

Insights into radicicol biosynthesis via heterologous synthesis of intermediates and analogs

scientific article

Insights into the Mechanism of Action of the Two-Peptide Lantibiotic Lacticin 3147.

scientific article published on 22 November 2017

Insights into the draft genome sequence of bioactives-producing DNG9 isolated from Algerian soil-oil slough

scientific article published on 11 October 2018

Intact incorporation of acetate-derived di- and tetraketides during biosynthesis of dehydrocurvularin, a macrolide phytotoxin from Alternaria cinerariae

scientific article published in 1990

Investigation of fungal iterative polyketide synthase functions using partially assembled intermediates

scientific article published on 28 January 2013

Investigation of the ring-closing metathesis of peptides in water

scientific article published on 04 December 2012

Isolation and characterization of carnocyclin a, a novel circular bacteriocin produced by Carnobacterium maltaromaticum UAL307.

scientific article

Isolation of a variant of subtilosin A with hemolytic activity

scientific article published on 24 July 2009

Isolation, expression and biochemical characterization of recombinant hyoscyamine-6β-hydroxylase from Brugmansia sanguinea - tuning the scopolamine production

scientific article published on 02 May 2018

Isolation, structural characterization, and properties of mattacin (polymyxin M), a cyclic peptide antibiotic produced by Paenibacillus kobensis M.

scientific article

Isotope shifts in13C-n.m.r. spectra of18O-labelled acetals; multiple labelling effects at β-carbons

Key Residues in Octyl-Tridecaptin A1Analogues Linked to Stable Secondary Structures in the Membrane

scientific article published on 09 May 2014

Lipopeptides from Bacillus and Paenibacillus spp.: A Gold Mine of Antibiotic Candidates

scientific article

Loss of Apelin exacerbates myocardial infarction adverse remodeling and ischemia-reperfusion injury: therapeutic potential of synthetic Apelin analogues.

scientific article published on July 2013

LovG: the thioesterase required for dihydromonacolin L release and lovastatin nonaketide synthase turnover in lovastatin biosynthesis

scientific article published on 07 May 2013

Lovastatin Nonaketide Synthase Catalyzes an Intramolecular Diels−Alder Reaction of a Substrate Analogue

article

Magnitudes of 18O isotope shifts in 13C nuclear magnetic resonance spectra of ketones and alcohols

Mechanism of substrate recognition and PLP-induced conformational changes in LL-diaminopimelate aminotransferase from Arabidopsis thaliana

scientific article

Membrane permeabilization, orientation, and antimicrobial mechanism of subtilosin A.

scientific article published in October 2005

Modification of the Swern Oxidation: Use of Stoichiometric Amounts of an Easily Separable, Recyclable, and Odorless Sulfoxide That Can Be Polymer-Bound

scientific article published on 01 November 1996

Modification of the Swern Oxidation: Use of a Soluble Polymer-Bound, Recyclable, and Odorless Sulfoxide

article by Joanna M. Harris et al published April 1998 in Journal of Organic Chemistry

Modulation of Polyketide Synthase Activity by Accessory Proteins During Lovastatin Biosynthesis

scientific article published in Science

Molecular cloning and characterization of drimenol synthase from valerian plant (Valeriana officinalis)

article

Molecular docking identifies the binding of 3-chloropyridine moieties specifically to the S1 pocket of SARS-CoV Mpro

scientific article published on 22 September 2007

Monacolin N, a compound resulting from derailment of type I iterative polyketide synthase function en route to lovastatin

scientific article published in July 2003

Multiple On-Resin Olefin Metathesis to Form Ring-Expanded Analogues of the Lantibiotic Peptide, Lacticin 3147 A2

scientific article published on 01 February 2007

N-Acylglycine Amidation: Implications for the Biosynthesis of Fatty Acid Primary Amides†

scientific article published on 01 March 1999

N-phthalimidoaziridines by diastereoselective Addition to α,β-unsaturated amides: a route to chiral β-substituted α-hydrazino acid derivatives

article

NMR Solution Structure of ImB2, a Protein Conferring Immunity to Antimicrobial Activity of the Type IIa Bacteriocin, Carnobacteriocin B2†,‡

scientific article published on 01 September 2004

NMR method to detect stereospecific deuterium labeling at diastereotopic methylene hydrogens: selective proton, carbon-13 heteronuclear shift correlation

scientific article published in 1985

NMR solution structure of the precursor for carnobacteriocin B2, an antimicrobial peptide from Carnobacterium piscicola

scientific article published in May 2004

New insights into natural rubber biosynthesis from rubber‐deficient lettuce mutants expressing goldenrod or guayule <i>cis</i>‐prenyltransferase

scientific article published in 2023

Nitrogen-15- and carbon-13-labeled media from Anabaena sp. for universal isotopic labeling of bacteriocins: NMR resonance assignments of leucocin A from Leuconostoc gelidum and nisin A from Lactococcus lactis

scientific article published on 01 January 1993

Novel pyrano and vinylphenol adducts of deoxyanthocyanidins in sorghum sourdough

scientific article published on 13 November 2014

Nuclear Magnetic Resonance Solution Structures of Lacticin Q and Aureocin A53 Reveal a Structural Motif Conserved among Leaderless Bacteriocins with Broad-Spectrum Activity

scientific article

Nuclear magnetic resonance solution structure of PisI, a group B immunity protein that provides protection against the type IIa bacteriocin piscicolin 126, PisA

scientific article

Nucleosides and nucleotides part 24 Investigation of ribo- and deoxyribonucleosides and -nucleotides by fast- atom-bombardment mass spectrometry

One-Step Transformation of Coenzyme A into Analogues by Transamidation

scientific article published on 10 April 2017

Optimizing PEG-Extended Apelin Analogues as Cardioprotective Drug Leads: Importance of the KFRR Motif and Aromatic Head Group for Improved Physiological Activity

scientific article published on 01 October 2020

PLP-independent racemization: mechanistic and mutational studies of O-ureidoserine racemase (DcsC).

scientific article

Paenibacillus polymyxa PKB1 produces variants of polymyxin B-type antibiotics

scientific article

Peptide aldehyde inhibitors of hepatitis A virus 3C proteinase

scientific article

Peptide amidation in an invertebrate: purification, characterization, and inhibition of peptidylglycine alpha-hydroxylating monooxygenase from the heads of honeybees (Apis mellifera).

scientific article published in January 1994

Peptidomimetic α-Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV-2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and <i>in Vitro</i> Biological Stability

scientific article published on 09 July 2021

Photolysis of Diacyl Peroxides:  A Radical-Based Approach for the Synthesis of Functionalized Amino Acids

scientific article published on 01 August 2003

Plasma kallikrein cleaves and inactivates apelin-17: Palmitoyl- and PEG-extended apelin-17 analogs as metabolically stable blood pressure-lowering agents

scientific article published on 18 January 2019

Polymer-supported alkyl azodicarboxylates for Mitsunobu reactions

scientific article published in 1989

Preparation and use of cysteine orthoesters for solid-supported synthesis of peptides

scientific article published in May 2010

Production of New Cladosporin Analogues by Reconstitution of the Polyketide Synthases Responsible for the Biosynthesis of this Antimalarial Agent

scientific article

Production of piscicolin 126 by Carnobacterium maltaromaticum UAL26 is controlled by temperature and induction peptide concentration

scientific article published on 23 August 2006

Protein farnesyltransferase inhibitors interfere with farnesyl diphosphate binding by rubber transferase

scientific article published in October 2003

Pseudoxazolones, a new class of inhibitors for cysteine proteinases: inhibition of hepatitis A virus and human rhinovirus 3C proteinases

Purification and characterization of antimicrobial peptides from fish isolate Carnobacterium maltaromaticum C2: Carnobacteriocin X and carnolysins A1 and A2.

scientific article

Purification and characterization of brochocin A and brochocin B(10-43), a functional fragment generated by heterologous expression in Carnobacterium piscicola

scientific article

Putative Diels-Alder-Catalyzed Cyclization during the Biosynthesis of Lovastatin.

scientific article

Reaction of .beta.-hydroxy .alpha.-amino acid derivatives with (diethylamino)sulfur trifluoride (DAST). Synthesis of .beta.-fluoro .alpha.-amino acids

Response of methicillin-resistant Staphylococcus aureus to amicoumacin A

scientific article

Retention of Configuration in Photolytic Decarboxylation of Peresters to Form Chiral Acetals and Ethers

scientific article published on 01 February 2009

Revision of the biosynthetic origin of oxygens in mevinolin (lovastatin), a hypocholesterolemic drug from Aspergillus terreus MF 4845

scientific article published in 1994

Ribosomally synthesized and post-translationally modified peptide natural products: overview and recommendations for a universal nomenclature

scientific article

Selection of entomopathogenic fungus Beauveria bassiana (Deuteromycotina: Hyphomycetes) for the biocontrol of Dendroctonus ponderosae (Coleoptera: Curculionidae, Scolytinae) in Western Canada

scientific article published on 18 February 2021

Serine and threonine beta-lactones: a new class of hepatitis A virus 3C cysteine proteinase inhibitors

scientific article published in March 2002

Solid Supported Chemical Syntheses of Both Components of the Lantibiotic Lacticin 3147

scientific article published on 17 August 2011

Solid-supported synthesis and biological evaluation of the lantibiotic peptide bis(desmethyl) lacticin 3147 A2.

scientific article

Solution Structure of Enterocin HF, an Antilisterial Bacteriocin Produced by Enterococcus faecium M3K31

scientific article

Solution Structures of Phenol-Soluble Modulins α1, α3, and β2, Virulence Factors from Staphylococcus aureus

scientific article

Solution structure of acidocin B, a circular bacteriocin produced by Lactobacillus acidophilus M46.

scientific article published on 13 February 2015

Solution structures of the linear leaderless bacteriocins enterocin 7A and 7B resemble carnocyclin A, a circular antimicrobial peptide

scientific article

Spermicidal bacteriocins: lacticin 3147 and subtilosin A.

scientific article published on 17 November 2007

Stereochemical features of enoyl thiol ester reductase in averufin and fatty acid biosynthesis in Aspergillus parasiticus

scientific article published in 1988

Stereochemistry and mechanism of reactions catalyzed by tryptophanase Escherichia coli

scientific article

Stereochemistry of lysine formation by meso-diaminopimelate decarboxylase from wheat germ: use of proton-carbon-13 NMR shift correlation to detect stereospecific deuterium labeling

scientific article published on 01 June 1985

Stereoselective Syntheses of 4-Oxa Diaminopimelic Acid and Its Protected Derivatives via Aziridine Ring Opening

scientific article published on 12 September 2007

Stereospecific Synthesis of Phosphonate Analogs of Diaminopimelic Acid (DAP), Their Interaction with DAP Enzymes, and Antibacterial Activity of Peptide Derivatives

Stereospecificity of sodium borohydride reduction of tyrosine decarboxylase from Streptococcus faecalis ⬇️

scientific article (publication date: 25 June 1979)

Stereospecificity of thymidylate synthetase

Structural characterization of lacticin 3147, a two-peptide lantibiotic with synergistic activity.

scientific article published in March 2004

Structural characterization of the highly cyclized lantibiotic paenicidin A via a partial desulfurization/reduction strategy

scientific article

Structural characterization of thioether-bridged bacteriocins

scientific article published on 11 September 2013

Structural features of many circular and leaderless bacteriocins are similar to those in saposins and saposin-like peptides

scientific article published on 11 January 2017

Structural insights into stereochemical inversion by diaminopimelate epimerase: an antibacterial drug target

scholarly article

Structural variations in keto-glutamines for improved inhibition against hepatitis A virus 3C proteinase

scientific article

Structure and biosynthesis of carnolysin, a homologue of enterococcal cytolysin with D-amino acids.

scientific article

Structure and genetics of circular bacteriocins

scientific article published on 12 June 2011

Structure function relationship of inducer peptide pheromones involved in bacteriocin production in Carnobacterium maltaromaticum and Enterococcus faecium

scientific article published on 01 November 2007

Structure of subtilosin A, a cyclic antimicrobial peptide from Bacillus subtilis with unusual sulfur to alpha-carbon cross-links: formation and reduction of alpha-thio-alpha-amino acid derivatives

scientific article

Structure of subtilosin A, an antimicrobial peptide from Bacillus subtilis with unusual posttranslational modifications linking cysteine sulfurs to alpha-carbons of phenylalanine and threonine

scientific article

Studies on the biosynthesis of the mycotoxin austin, a meroterpenoid metabolite of Aspergillus ustus

Studies on tridecaptin B(1), a lipopeptide with activity against multidrug resistant Gram-negative bacteria

scientific article published on June 2015

Substitution of a conserved disulfide in the type IIa bacteriocin, leucocin A, with L-leucine and L-serine residues: effects on activity and three-dimensional structure

scientific article

Substrate and inhibitor binding sites in Corynebacterium glutamicum diaminopimelate dehydrogenase

scientific article

Syntheses of Conjugated Pyrones for the Enzymatic Assay of Lovastatin Nonaketide Synthase, an Iterative Polyketide Synthase

scientific article published on 01 January 2007

Synthesis and Biological Activity of Oxa-Lacticin A2, a Lantibiotic Analogue with Sulfur Replaced by Oxygen

scientific article published on 01 December 2009

Synthesis and Structure–Activity Relationship Studies of N-Terminal Analogues of the Antimicrobial Peptide Tridecaptin A1

scientific article published on 30 January 2014

Synthesis and acylation of salts of L-threonine .beta.-lactone: a route to .beta.-lactone antibiotics

Synthesis and biological activity of isopentenyl diphosphate analogues

scientific article published in February 2004

Synthesis and biological evaluation of nucleoside dicarboxylates as potential mimics of nucleoside diphosphates

scientific article published on 18 January 2007

Synthesis and biological studies of neopetrosiamides as inhibitors of cancer cell invasion

scientific article published on March 2013

Synthesis and evaluation of keto-glutamine analogues as inhibitors of hepatitis A virus 3C proteinase

scientific article published in May 2002

Synthesis and evaluation of keto-glutamine analogues as potent inhibitors of severe acute respiratory syndrome 3CLpro

scientific article published in December 2004

Synthesis and reactivity of .beta.-lactones derived from L-threonine and related amino acids

Synthesis and structure-activity relationships of o-sulfonamido-arylhydrazides as inhibitors of LL-diaminopimelate aminotransferase (LL-DAP-AT).

scientific article

Synthesis and testing of azaglutamine derivatives as inhibitors of hepatitis A virus (HAV) 3C proteinase

scientific article

Synthesis of (+)-obafluorin, a .beta.-lactone antibiotic

Synthesis of 3-fluorodiaminopimelic acid isomers as inhibitors of diaminopimelate epimerase: stereocontrolled enzymatic elimination of hydrogen fluoride

article published in 1990

Synthesis of Biologically Active Dicarba Analogues of the Peptide Hormone Oxytocin Using Ring-Closing Metathesis

scientific article published on 01 January 2003

Synthesis of Chiral Spin-Labeled Amino Acids

scientific article published on 10 December 2019

Synthesis of Protein Farnesyltransferase and Protein Geranylgeranyltransferase Inhibitors: Rapid Access to Chaetomellic Acid A and Its Analogues

scientific article published on 01 September 1996

Synthesis of Tridecaptin-Antibiotic Conjugates with in Vivo Activity against Gram-Negative Bacteria

scientific article

Synthesis of a C-phosphonate disaccharide as a potential inhibitor of peptidoglycan polymerization by transglycosylase

Synthesis of mono- and disaccharide analogs of moenomycin and lipid II for inhibition of transglycosylase activity of penicillin-binding protein 1b.

scientific article

Synthesis of optically pure .alpha.-amino acids via salts of .alpha.-amino-.beta.-propiolactone

article by Lee D. Arnold et al published March 1988 in Journal of the American Chemical Society

Synthesis of oxytocin analogues with replacement of sulfur by carbon gives potent antagonists with increased stability

scientific article published in September 2005

Synthesis of pseudoxazolones and their inhibition of the 3C cysteine proteinases from hepatitis A virus and human rhinovirus-14

Synthesis of sterically encumbered 11β-aminoprogesterone derivatives and evaluation as 11β-hydroxysteroid dehydrogenase inhibitors and mineralocorticoid receptor antagonists

scientific article published on 07 September 2013

Synthesis of the lantibiotic lactocin S using peptide cyclizations on solid phase

scientific article published in January 2010

Synthesis of β-Cyclopropylalanines by Photolysis of Diacyl Peroxides

scientific article published on 01 November 2003

Synthesis, Stability, and Antimicrobial Activity of (+)-Obafluorin and Related .beta.-Lactone Antibiotics

Synthetic Modification within the "RPRL" Region of Apelin Peptides: Impact on Cardiovascular Activity and Stability to Neprilysin and Plasma Degradation.

scientific article

Targeting the apelin pathway as a novel therapeutic approach for cardiovascular diseases

scientific article published on 04 November 2016

The 3D solution structure of thurincin H, a bacteriocin with four sulfur to α-carbon crosslinks

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The 3D structure of thuricin CD, a two-component bacteriocin with cysteine sulfur to α-carbon cross-links

scientific article

The ABC Transporter CclEFGH Facilitates the Production of the Circular Bacteriocin Carnocyclin A

article

The Enzymatic Formation of Novel Bile Acid Primary Amides

scientific article published on 01 February 2000

The Metalloprotease Neprilysin Degrades and Inactivates Apelin Peptides.

scientific article published on 5 July 2016

The Synthesis of Active and Stable Diaminopimelate Analogues of the Lantibiotic Peptide Lactocin S

scientific article published on 24 January 2012

The Three-dimensional Structure of Carnocyclin A Reveals That Many Circular Bacteriocins Share a Common Structural Motif ⬇️

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The activity of bacteriocins from Carnobacterium maltaromaticum UAL307 against gram-negative bacteria in combination with EDTA treatment

scientific article published on 7 February 2011

The circular bacteriocin, carnocyclin A, forms anion-selective channels in lipid bilayers

scientific article

The distribution of acetate-derived oxygens in the tetronic acids of Penicillium multicolor

The expanding structural variety among bacteriocins from Gram-positive bacteria

scientific article published on 01 November 2018

The first isolation of an alkoxy-N,N-dialkylaminodifluorosulfane from the reaction of an alcohol and DAST: an efficient synthesis of (2S,3R,6S)-3-fluoro-2,6-diaminopimelic acid

The first stereospecific synthesis of l-tetrahydrodipicolinic acid†; a key intermediate of diaminopimelate metabolism

The stereoselective synthesis of aziridine analogues of diaminopimelic acid (DAP) and their interaction with dap epimerase

scientific article published on 15 November 2005

The structure of LL-diaminopimelate aminotransferase from Chlamydia trachomatis: implications for its broad substrate specificity

scientific article

The use of stable isotopes in biosynthetic studies

scientific article published on June 1987

Three-Dimensional Structure of Leucocin A in Trifluoroethanol and Dodecylphosphocholine Micelles: Spatial Location of Residues Critical for Biological Activity in Type IIa Bacteriocins from Lactic Acid Bacteria, ⬇️

scientific article published on December 9, 1997

Thuricin CD, a posttranslationally modified bacteriocin with a narrow spectrum of activity against Clostridium difficile.

scientific article published on 30 April 2010

Total Synthesis and Stereochemical Assignment of the Antimicrobial Lipopeptide Cerexin A1

scientific article published on 14 October 2015

Transformations of cyclic nonaketides by Aspergillus terreus mutants blocked for lovastatin biosynthesis at the lovA and lovC genes

scientific article published in January 2003

Two-peptide bacteriocins produced by lactic acid bacteria

scientific article

Unacylated tridecaptin A₁ acts as an effective sensitiser of Gram-negative bacteria to other antibiotics

scientific article published on 27 September 2014

Understanding Programming of Fungal Iterative Polyketide Synthases: The Biochemical Basis for Regioselectivity by the Methyltransferase Domain in the Lovastatin Megasynthase.

scientific article published on 2 December 2015

Unsaturated α-aminopimelic acids as potent inhibitors of meso-diaminopimelic acid (DAP) D-dehydrogenase

Use of a copper-chelated lipid speeds up NMR measurements from membrane proteins

scientific article published on May 2010

Vinylogous Amide Analogues of Diaminopimelic Acid (DAP) as Inhibitors of Enzymes Involved in Bacterial Lysine Biosynthesis

scientific article published on 01 November 2000

[Drug discovery and natural products: end of era or an endless frontier?]

scientific article published on 01 March 2011

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