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List of works by Satoshi Ōmura

2'-Amino-2'-deoxyadenosine produced by a strain of Actinomadura

scientific article

4'''-N-demethylspiramycin derivatives: synthesis and evaluation of effectiveness against drug-resistant bacteria

scientific article published in March 2008

6'-Hydroxy-3'-methoxy-mitorubrin, a new potentiator of antifungal miconazole activity, produced by Penicillium radicum FKI-3765-2. ⬇️

scientific article published in June 2010

A gamma-lactone form nafuredin, nafuredin-gamma, also inhibits helminth complex I.

scientific article published in January 2005

A gene cluster for biosynthesis of the sesquiterpenoid antibiotic pentalenolactone in Streptomyces avermitilis ⬇️

scientific article published on May 2006

A new alkaloid AM-2282 OF Streptomyces origin. Taxonomy, fermentation, isolation and preliminary characterization ⬇️

scientific article

A new anti-influenza virus antibiotic, 10-norparvulenone from Microsphaeropsis sp. FO-5050.

scientific article

A new antibiotic, OS-1804

scientific article published on April 1, 1977

A new antibiotic, antimycin Ag, produced by Streptomyces sp. K01-0031. ⬇️

scientific article published in January 2005

A new antibiotic, cypemycin. Taxonomy, fermentation, isolation and biological characteristics

scientific article

A new antibiotic, okicenone. I. Taxonomy, fermentation, isolation and biological characteristics ⬇️

scientific article published in August 1991

A new antibiotic, setomimycin, produced by a strain of Streptomyces

scientific article

A new antibiotic,, asukamycin, produced by Streptomyces ⬇️

scientific article published on September 1, 1976

A new antimicrobial antibiotic from Actinoplanes capillaceus sp. K95-5561T. ⬇️

scientific article

A new antitumor antibiotic, PO-357.

scientific article published in November 1976

A new species of Dinemasporium from sugar cane on Irabujima island, Japan

article by Yuichi Yamaguchi et al published December 2005 in Mycoscience

A simple screening system for anti-HIV drugs: syncytium formation assay using T-cell line tropic and macrophage tropic HIV env expressing cell lines--establishment and validation.

scientific article

A small-molecule inhibitor of the bacterial type III secretion system protects against in vivo infection with Citrobacter rodentium.

scientific article published on 8 December 2010

ACAT2 is localized to hepatocytes and is the major cholesterol-esterifying enzyme in human liver

scientific article

Absolute stereochemistry of fungal beauveriolide III and ACAT inhibitory activity of four stereoisomers

scientific article

Actinoallomurus radicium sp. nov., isolated from the roots of two plant species

scientific article

Actinohivin, a novel anti-HIV protein from an actinomycete that inhibits syncytium formation: isolation, characterization, and biological activities

scientific article

Actinohivin: specific amino acid residues essential for anti-HIV activity ⬇️

scientific article published on September 15, 2010

Actinoplanes capillaceus sp. nov., a new species of the genus Actinoplanes

scientific article

Acylated pregnane glycosides from Caralluma tuberculata and their antiparasitic activity

scientific article

Adecypenol, a unique adenosine deaminase inhibitor containing homopurine and cyclopentene rings. Taxonomy, production and enzyme inhibition

scientific article published in September 1986

Advances in drug discovery and biochemical studies

scientific article published on 23 March 2007

Alutenusin, a specific neutral sphingomyelinase inhibitor, produced by Penicillium sp. FO-7436. ⬇️

scientific article published in June 1999

Amphomycin inhibits phospho-N-acetylmuramyl-pentapeptide translocase in peptidoglycan synthesis of Bacillus ⬇️

scientific article published on February 14, 1979

An anthelmintic compound, nafuredin, shows selective inhibition of complex I in helminth mitochondria

scholarly article

Andrastins A-C, new protein farnesyltransferase inhibitors produced by Penicillium sp. FO-3929. I. Producing strain, fermentation, isolation, and biological activities. ⬇️

scientific article

Anti-atherosclerotic activity of triacsin C, an acyl-CoA synthetase inhibitor

scientific article published in May 2008

Anti-inflammatory effects of a novel non-antibiotic macrolide, EM900, on mucus secretion of airway epithelium.

scientific article published on 10 March 2015

Antiatherogenic activity of fungal beauveriolides, inhibitors of lipid droplet accumulation in macrophages

scholarly article

Antibiotics LL-Z1272 identified as novel inhibitors discriminating bacterial and mitochondrial quinol oxidases

scientific article

Antimalarial C-9 oxime derivatives from desmycosin, produced by click chemistry

scientific article published on 12 December 2012

Antimalarial tropones and their Plasmodium falciparum glyoxalase I (pfGLOI) inhibitory activity

scientific article published on 9 April 2014

Antiplasmodial and antitrypanosomal activity of plants from the Kingdom of Saudi Arabia

scientific article

Antitrypanosomal activity of some pregnane glycosides isolated from Caralluma species

scientific article published on 2 April 2009

Antitrypanosomal peptaibiotics, trichosporins B-VIIa and B-VIIb, produced by Trichoderma polysporum FKI-4452.

scientific article published on 30 April 2010

Antitumor activity of an antibiotic identical with or closely related to xanthomycin A ⬇️

scientific article published on July 1, 1981

Antitumor activity of prumycin

scientific article published on April 1, 1979

Antitumor activity of trienomycin A on murine tumors.

scientific article published in December 1987

Antiviral activities of pentalenolactones

scientific article published in August 1985

Aranorosin circumvents arbekacin-resistance in MRSA by inhibiting the bifunctional enzyme AAC(6')/APH(2″).

scientific article

Argifin; efficient solid phase total synthesis and evaluation of analogues of acyclic peptide

scientific article

Arisugacins A and B, novel and selective acetylcholinesterase inhibitors from Penicillium sp. FO-4259. I. Screening, taxonomy, fermentation, isolation and biological activity. ⬇️

scientific article published in August 1996

Arohynapenes A and B, new anticoccidial agents produced by Penicillium sp. Taxonomy, fermentation, and structure elucidation. ⬇️

scientific article published on January 1994

Atpenins, potent and specific inhibitors of mitochondrial complex II (succinate-ubiquinone oxidoreductase). ⬇️

scholarly article

Avermectins, New Family of Potent Anthelmintic Agents: Producing Organism and Fermentation ⬇️

scientific article published on March 1, 1979

Azithromycin inhibits the formation of flagellar filaments without suppressing flagellin synthesis in Salmonella enterica serovar typhimurium

scientific article

Beauveriolides, specific inhibitors of lipid droplet formation in mouse macrophages, produced by Beauveria sp. FO-6979. ⬇️

scientific article published in January 1999

Binding site for fungal beta-lactone hymeglusin on cytosolic 3-hydroxy-3-methylglutaryl coenzyme A synthase

scientific journal article

Biochemical and spectroscopic properties of cyanide-insensitive quinol oxidase from Gluconobacter oxydans.

scientific article published on 4 May 2009

Bioconversion and biosynthesis of 16-membered macrolide antibiotics. X. Final steps in the biosynthesis of spiramycin, using enzyme inhibitor: cerulenin ⬇️

scientific article published on January 1, 1979

Bioconversion and biosynthesis of 16-membered macrolide antibiotics. XIII. Regulation of spiramycin I 3-hydroxyl acylase formation by glucose, butyrate, and cerulenin

scientific article published on June 1, 1979

Biosynthesis of bioactive microbial metabolites and its application to the structural studies and production of hybrid compounds.

scientific article published on August 1996

Biosynthesis of kalafungin in Streptomyces tanashiensis

scientific article

Biosynthetic studies using carbon-13 enriched precursors on the 16-membered macrolide antibiotic leucomycin A3 ⬇️

scientific article published on October 29, 1975

Bottromycin derivatives: Efficient chemical modifications of the ester moiety and evaluation of anti-MRSA and anti-VRE activities ⬇️

scientific article published on August 18, 2010

Calpinactam, a new anti-mycobacterial agent, produced by Mortierella alpina FKI-4905.

scientific article published on 26 February 2010

Cerulenin resistance in a cerulenin-producing fungus. III. Studies on active-site peptides of fatty acid synthetase from Cephalosporium caerulens.

scientific article

Cerulenin resistance in a cerulenin-producing fungus. Isolation of cerulenin insensitive fatty acid synthetase

scientific article published on October 1, 1979

Cervinomycin A1 and A2, new antibiotics active against anaerobes, produced by Streptomyces cervinus sp. nov. ⬇️

scientific article published on June 1982

Chemical and biological studies on 16-membered macrolide antibiotics ⬇️

scientific article published on June 1, 1975

Chemical biology of natural indolocarbazole products: 30 years since the discovery of staurosporine

scientific article

Chemical modification of erythromycins. IV. Synthesis and biological properties of 6-O-methylerythromycin B.

scientific article published in May 1990

Chemical modification of erythromycins. V. Synthesis and antibacterial activity of 4''-O-methyl derivatives of erythromycin a 11,12-cyclic carbonate.

scientific article published in May 1990

Chemical modification of spiramycins. VI. Synthesis and antibacterial activities of 3,3''-di-O-acyl-4''-O-sulfonyl and 3,3''-di-O-acyl-4''-O-alkyl derivatives of spiramycin I.

scientific article

Chemical modification of tylosin. Thioether derivatives of tylosin and demycarosyltylosin.

scientific article

Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry

scientific article

Chlorogentisylquinone, a new neutral sphingomyelinase inhibitor, produced by a marine fungus.

scientific article published in November 2001

Chloropeptins I and II, novel inhibitors against gp120-CD4 binding from Streptomyces sp. ⬇️

scientific article published on October 1994

Chloropeptins, new anti-HIV antibiotics inhibiting gp120-CD4 binding from Streptomyces sp. I. Taxonomy, fermentation, isolation, and physico-chemical properties and biological activities. ⬇️

scientific article published on January 1997

Chlovalicin, a new cytocidal antibiotic produced by Sporothrix sp. FO-4649. I. Taxonomy, fermentation, isolation and biological activities. ⬇️

scientific article published in July 1996

Cholesterol synthesis inhibition elicits an integrated molecular response in human livers including decreased ACAT2

scientific article published on 13 March 2008

Citridones, new potentiators of antifungal miconazole activity, produced by Penicillium sp. FKI-1938. I. Taxonomy, fermentation, isolation and biological properties ⬇️

scientific article published in May 2005

Citridones, new potentiators of antifungal miconazole activity, produced by Penicillium sp. FKI-1938. II. Structure elucidation ⬇️

scientific article published in May 2005

Citrinamides, new potentiators of antifungal miconazole activity, produced by Penicillium sp. FKI-1938. ⬇️

scientific article

Cloning of the gene encoding avermectin B 5-O-methyltransferase in avermectin-producing Streptomyces avermitilis.

scientific article

Cloning, sequencing and deduced functions of a cluster of Streptomyces genes probably encoding biosynthesis of the polyketide antibiotic frenolicin

scientific article published on May 1994

Comparative efficacies of different antibiotic treatments to eradicate nontypeable Haemophilus influenzae infection

scientific article

Computational analysis of the binding affinities of the natural-product cyclopentapeptides argifin and argadin to chitinase B from Serratia marcescens

scientific article published on 8 February 2008

Computer-aided rational molecular design of argifin-derivatives with increased inhibitory activity against chitinase B from Serratia marcescens.

scientific article published on 9 April 2009

Conexibacter arvalis sp. nov., isolated from a cultivated field soil sample

scientific article

Construction of a single component producer from the wild type avermectin producer Streptomyces avermitilis. ⬇️

scientific article published in June 1995

Control of Avermectin Biosynthesis in Streptomyces avermitilis for the Selective Production of a Useful Component ⬇️

scientific article published on July 1, 1995

Core structure in roselipins essential for eliciting inhibitory activity against diacylglycerol acyltransferase

scientific article published in January 2003

Crystal structure of the non-heme iron dioxygenase PtlH in pentalenolactone biosynthesis

scientific article

Culture conditions for screening of new antibiotics

scientific article published on February 1982

Cyslabdan, a new potentiator of imipenem activity against methicillin-resistant Staphylococcus aureus, produced by Streptomyces sp. K04-0144. I. Taxonomy, fermentation, isolation and structural elucidation

scientific article

Cyslabdan, a new potentiator of imipenem activity against methicillin-resistant Staphylococcus aureus, produced by Streptomyces sp. K04-0144. II. Biological activities ⬇️

scientific article

Cytochrome p450 complement (CYPome) of the avermectin-producer Streptomyces avermitilis and comparison to that of Streptomyces coelicolor A3(2).

scientific article published in August 2003

Deacetylravidomycin M, a new inhibitor of IL-4 signal transduction, produced by Streptomyces sp. WK-6326. I. Taxonomy, fermentation, isolation and biological activities. ⬇️

scientific article

Deacetylravidomycin M, a new inhibitor of IL-4 signal transduction, produced by Streptomyces sp. WK-6326. II. Structure elucidation

scientific article

Decursin and decursinol angelate selectively inhibit NADH-fumarate reductase of Ascaris suum

scientific article published on 18 October 2007

Demequina salsinemoris sp. nov., isolated on agar media supplemented with ascorbic acid or rutin

scientific article

Description of two novel species of the genus Kitasatospora Omura et al. 1982, Kitasatospora cineracea sp. nov. and Kitasatospora niigatensis sp. nov.

scientific article

Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity

scientific article

Design, synthesis, and biological activities of madindoline analogues

scientific article published on 14 February 2006

Design, synthesis, and biological evaluation of air-stable nafuredin-γ analogs as complex I inhibitors

scientific article published on 22 January 2015

Dinapinones, novel inhibitors of triacylglycerol synthesis in mammalian cells, produced by Penicillium pinophilum FKI-3864. ⬇️

scientific article published on 11 May 2011

Direct production of 5-oxo derivatives of avermectins by a recombinant strain of Streptomyces avermitilis. ⬇️

scientific article published in January 1995

Distribution and functional analysis of the phosphopantetheinyl transferase superfamily in Actinomycetales microorganisms.

scientific article published on 14 June 2018

EM, EM703 inhibit NF-kB activation induced by oxidative stress from diesel exhaust particle in human bronchial epithelial cells: importance in IL-8 transcription

scientific article

EM703 improves bleomycin-induced pulmonary fibrosis in mice by the inhibition of TGF-beta signaling in lung fibroblasts

scientific article published on 27 January 2006

EM703, a new derivative of erythromycin, inhibits transforming growth factor-beta signaling in human lung fibroblasts

scientific article

Effect of leucomycins and analogues on binding [14C ]erythromycin to Escherichia coli ribosomes

scientific article published on November 1974

Effects of a novel nonantibiotic macrolide, EM900, on cytokine and mucin gene expression in a human airway epithelial cell line

scientific article

Efficient total synthesis of novel bioactive microbial metabolites

scientific article published on 25 January 2008

Enantioselective total synthesis of atpenin A5.

scientific article published on 17 April 2009

Engineered Streptomyces avermitilis host for heterologous expression of biosynthetic gene cluster for secondary metabolites ⬇️

scientific article published on 17 January 2013

Enhancement of metabolites productivity of Penicillium pinophilum FKI-5653, by co-culture with Trichoderma harzianum FKI-5655. ⬇️

scientific article

Erythromycin derivatives inhibit HIV-1 replication in macrophages through modulation of MAPK activity to induce small isoforms of C/EBPbeta

scholarly article

Erythromycin suppresses nuclear factor-kappaB and activator protein-1 activation in human bronchial epithelial cells

scientific article

Euvesperins A and B, new circumventors of arbekacin resistance in MRSA, produced by Metarhizium sp. FKI-7236. ⬇️

scientific article

Expression of two human acyl-CoA:diacylglycerol acyltransferase isozymes in yeast and selectivity of microbial inhibitors toward the isozymes

scientific article published on 9 January 2009

F-244 (1233A), a specific inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A synthase: taxonomy of producing strain, fermentation, isolation and biological properties

scientific article published in February 1988

Ferroverdins, inhibitors of cholesteryl ester transfer protein produced by Streptomyces sp. WK-5344. I. Production, isolation and biological properties. ⬇️

scientific article

Fourteen-member macrolides suppress interleukin-8 production but do not promote apoptosis of activated neutrophils

scientific article published on April 2002

Funalenone, a novel collagenase inhibitor produced by Aspergillus niger ⬇️

scientific article published in December 1999

Fungal citridone D having a novel phenylfuropyridine skeleton ⬇️

scientific article published in December 2006

Fungal phenalenones inhibit HIV-1 integrase ⬇️

scientific article published in January 2005

Fungerin, a fungal alkaloid, arrests the cell cycle in M phase by inhibition of microtubule polymerization

scientific article published on July 2004

Funicone-related compounds, potentiators of antifungal miconazole activity, produced by Talaromycesflavus FKI-0076. ⬇️

scientific article

Gastrointestinal motor-stimulating activity of macrolide antibiotics and the structure-activity relationship

scientific article published in November 1985

Generation of reactive oxygen species from conventional laboratory media

scientific article published on 30 March 2010

Generation of superoxide anions by a glycation reaction in conventional laboratory media

scientific article published on 31 May 2012

Genetic and biochemical features of spiramycin biosynthesis in Streptomyces ambofaciens--curing, protoplast regeneration and plasmid transfer. ⬇️

scientific article

Genetics of antibiotic-producing Streptomyces

scientific article published on December 1990

Genome-minimized Streptomyces host for the heterologous expression of secondary metabolism ⬇️

scientific article

Geosmin biosynthesis in Streptomyces avermitilis. Molecular cloning, expression, and mechanistic study of the germacradienol/geosmin synthase ⬇️

scientific article

Glisoprenins, new inhibitors of acyl-CoA: cholesterol acyltransferase produced by Gliocladium sp. FO-1513. I. Production, isolation and physico-chemical and biological properties

scientific article published in August 1992

Guadinomines, Type III secretion system inhibitors, produced by Streptomyces sp. K01-0509. I: taxonomy, fermentation, isolation and biological properties

scientific article

Guadinomines, Type III secretion system inhibitors, produced by Streptomyces sp. K01-0509. II: physico-chemical properties and structure elucidation ⬇️

scientific article published in April 2008

HIV-1 neutralization profile and plant-based recombinant expression of actinohivin, an Env glycan-specific lectin devoid of T-cell mitogenic activity

scientific article published in 2010

Herquline B, a new platelet aggregation inhibitor produced by Penicillium herquei Fg-372.

scientific article

High-resolution structures of a chitinase complexed with natural product cyclopentapeptide inhibitors: mimicry of carbohydrate substrate

scientific article

Hyper-inducible expression system for streptomycetes

scholarly article

Identification and functional analysis of genes controlling biosynthesis of 2-methylisoborneol

scholarly article

Identification of ACAT1- and ACAT2-specific inhibitors using a novel, cell-based fluorescence assay: individual ACAT uniqueness

scientific article published on 16 November 2003

Identification of new inhibitors for alternative NADH dehydrogenase (NDH-II).

scientific article

Identification of the active component that induces vancomycin resistance in MRSA.

scientific article published on 30 June 2010

Identification of the interaction site within acyl-CoA:cholesterol acyltransferase 2 for the isoform-specific inhibitor pyripyropene A

scientific article published on 19 February 2008

Improved catalytic and stereoselective glycosylation with glycosyl N-trichloroacetylcarbamate: application to various 1-hydroxy sugars

scientific article published on 4 February 2010

Improvement of macrolide antibiotic-producing streptomycete strains by the regeneration of protoplasts

scientific article

In vitro and in vivo activity of penicillinase inhibitor KA-107 against Staphylococcus aureus FS-1277

scientific article published on September 1973

In vitro and in vivo anti-Trypanosoma brucei activities of phenazinomycin and related compounds

scientific article published on 30 June 2010

In vitro and in vivo antimalarial activities of a carbohydrate antibiotic, prumycin, against drug-resistant strains of Plasmodia

scientific article

In vitro and in vivo antimalarial activity of puberulic acid and its new analogs, viticolins A–C, produced by Penicillium sp. FKI-4410 ⬇️

scientific article published on November 10, 2010

In vitro and in vivo antitrypanosomal activities of three peptide antibiotics: leucinostatin A and B, alamethicin I and tsushimycin

scientific article

In vitro and in vivo antitrypanosomal activitiy of two microbial metabolites, KS-505a and alazopeptin

scientific article

In vitro antimalarial activities of the microbial metabolites.

scientific article published in March 2003

In vitro antimalarial activity of biflavonoids from Wikstroemia indica

scientific article published on January 2004

In vitro antimalarial activity of prenylated flavonoids from Erythrina fusca

scientific article

In vitro antitrypanosomal activity of 12 low-molecular-weight antibiotics and observations of structure/activity relationships

scientific article published on 18 August 2010

In vitro antitrypanosomal activity of bis(bibenzyls)s and bibenzyls from liverworts against Trypanosoma brucei

scientific article

In vitro antitrypanosomal activity of five low-MW antibiotics

scientific article published on 14 December 2011

In vitro antitrypanosomal activity of plant terpenes against Trypanosoma brucei

scientific article

In vitro antitrypanosomal activity of some phenolic compounds from propolis and lactones from Fijian Kawa (Piper methysticum).

scientific article

In vitro antitrypanosomal activity of the cyclodepsipeptides, cardinalisamides A-C, from the insect pathogenic fungus Cordyceps cardinalis NBRC 103832.

scientific article

Inhibition of acyl-CoA: cholesterol acyltransferase activity by cyclodepsipeptide antibiotics

scientific article published on October 1992

Inhibition of farnesyl-protein transferase by gliotoxin and acetylgliotoxin ⬇️

scientific article published on November 1, 1992

Inhibition of the biosynthesis of leucomycin, a macrolide antibiotic, by cerulenin

scientific article published in January 1974

Intracellular retention and degradation of tissue-nonspecific alkaline phosphatase with a Gly317-->Asp substitution associated with lethal hypophosphatasia

scientific article published in May 1998

Irumamycin, an antifungal 20-membered macrolide produced by a Streptomyces. Taxonomy, fermentation and biological properties ⬇️

scientific article published in December 1984

Isochromophilones I and II, Novel Inhibitors against gpl20-CD4 Binding Produced by Penicillium multicolor FO-2338. I. Screening, Taxonomy, Fermentation, Isolation and Biological Activity ⬇️

scientific article published on July 1, 1995

Isolation and characterization of elasnin, a new human granulocyte elastase inhibitor produced by a strain of Streptomyces ⬇️

scientific article published on November 1, 1978

Isolation and properties of spiramycin I 3-hydroxyl acylase from Streptomyces and ambofaciens ⬇️

scientific article published on December 1, 1979

Isolation and structure of a new antibiotic viridomycin F produced by Streptomyces sp. K96-0188. ⬇️

scientific article published in January 1999

Isolation and structure of an extracellular polysaccharide from streptomyces sp. FERM-P1185

scientific article published on July 1, 1976

Isolation of a new polyether antibiotic, lonomycin

scientific article published in January 1976

Isolation of a new sulfur-containing basic substance from a Thermo actinomyces species ⬇️

scientific article published in August 1975

Isolation of actinomycetes from the root of the plant, Ophiopogon japonicus, and proposal of two new species, Actinoallomurus liliacearum sp. nov. and Actinoallomurus vinaceus sp. nov.

scientific article

Isolation of isoflavonoids possessing antioxidant activity from the fermentation broth of Streptomyces sp. ⬇️

scientific article published on September 1989

Isolation of restriction-reduced mutants from Streptomyces

scientific article published on October 1, 1990

Ivermectin and malaria control.

scientific article

Ivermectin, 'wonder drug' from Japan: the human use perspective

scientific article

Izupeptins A and B, new glycopeptide antibiotics produced by an actinomycete.

scientific article

Jogyamycin, a new antiprotozoal aminocyclopentitol antibiotic, produced by Streptomyces sp. a-WM-JG-16.2.

scientific article published on 11 January 2012

Kitasatosporia, a new genus of the order Actinomycetales.

scientific article published on August 1982

Lanopylins A1, B1, A2 and B2, novel lanosterol synthase inhibitors from Streptomyces sp. K99-5041. ⬇️

scientific article

Louisianins A, B, C and D: non-steroidal growth inhibitors of testosterone-responsive SC 115 cells. I. Taxonomy, fermentation, isolation and biological characteristics. ⬇️

scientific article

Lys17 in the 'lasso' peptide lariatin A is responsible for anti-mycobacterial activity

scientific article

Macrolides with promotive activity of monocyte to macrophage differentiation

scientific article published in January 2005

Macrosphelide, a novel inhibitor of cell-cell adhesion molecule. I. Taxonomy, fermentation, isolation and biological activities

scientific article published on December 1995

Makomotindoline from Makomotake, Zizania latifolia infected with Ustilago esculenta

scientific article published on 17 May 2012

Mechanism of action of atpenin B on Raji cells.

scientific article published on September 1990

Molecular cloning of actinohivin, a novel anti-HIV protein from an actinomycete, and its expression in Escherichia coli

scientific article

Molecular insights into the biosynthesis of guadinomine: a type III secretion system inhibitor

scientific article

Molecular mechanisms of anti-inflammatory action of erythromycin in human bronchial epithelial cells: possible role in the signaling pathway that regulates nuclear factor-kappaB activation

scientific article published on May 2004

Molecular modeling of human acidic mammalian chitinase in complex with the natural-product cyclopentapeptide chitinase inhibitor argifin

scientific article published on 25 July 2009

Mycophenolic acid inhibits syncytium formation accompanied by reduction of gp120 expression

scientific article published on August 2005

NMR spectroscopy and computational analysis of interaction between Serratia marcescens chitinase B and a dipeptide derived from natural-product cyclopentapeptide chitinase inhibitor argifin ⬇️

scientific article published on August 15, 2010

New antibiotics miyakamides produced by a fungus

scientific article

New beauvericins, potentiators of antifungal miconazole activity, Produced by Beauveria sp. FKI-1366. I. Taxonomy, fermentation, isolation and biological properties ⬇️

scientific article published in February 2004

New beauvericins, potentiators of antifungal miconazole activity, Produced by Beauveria sp. FKI-1366. II. Structure elucidation

scientific article published in February 2004

New beauveriolides produced by amino acid-supplemented fermentation of Beauveria sp. FO-6979. ⬇️

scientific article published in January 2004

New brominated and halogen-less derivatives and structure-activity relationship of azaphilones inhibiting gp120-CD4 binding. ⬇️

scientific article published on November 1998

New inhibitors of melanogenesis, OH-3984 K1 and K2. I. Taxonomy, fermentation, isolation and biological characteristics

scientific article published in October 1993

New insecticidal antibiotics, hydroxyfungerins A and B, produced by Metarhizium sp. FKI-1079. ⬇️

scientific article published in December 2005

New isochaetochromin, an inhibitor of triacylglycerol synthesis in mammalian cells, produced by Penicillium sp. FKI-4942: I. Taxonomy, fermentation, isolation and biological properties

scientific article

New lycorine-type alkaloid from Lycoris traubii and evaluation of antitrypanosomal and antimalarial activities of lycorine derivatives

scientific article published on 30 October 2008

New monordens produced by amidepsine-producing fungus Humicola sp. FO-2942.

scientific article published in June 2003

New rugulosins, anti-MRSA antibiotics, produced by Penicillium radicum FKI-3765-2.

scientific article published in April 2010

New sesquicillins, insecticidal antibiotics produced by Albophoma sp. FKI-1778. ⬇️

scientific article published in June 2005

New strategy for discovery of enzyme inhibitors: screening with intact mammalian cells or intact microorganisms having special functions

scientific article published on October 1990

Nosokomycins, new antibiotics discovered in an in vivo-mimic infection model using silkworm larvae. I: Fermentation, isolation and biological properties

scientific article published on 26 February 2010

Nosokomycins, new antibiotics discovered in an in vivo-mimic infection model using silkworm larvae. II: Structure elucidation ⬇️

scientific article published on 5 March 2010

Novel 12-membered non-antibiotic macrolides, EM900 series with anti-inflammatory and/or immunomodulatory activity; synthesis, structure-activity relationships and in vivo study

scientific article

Novel antibiotics, furaquinocins A and B. Taxonomy, fermentation, isolation and physico-chemical and biological characteristics

scientific article published in March 1990

Novel cytocidal antibiotics, glucopiericidinols A1 and A2. Taxonomy, fermentation, isolation, structure elucidation and biological characteristics

scientific article published in December 1989

Novel mitochondrial complex II isolated from Trypanosoma cruzi is composed of 12 peptides including a heterodimeric Ip subunit

scientific article published on 2 January 2009

OM-173, new nanaomycin-type antibiotics produced by a strain of Streptomyces. Taxonomy, production, isolation and biological properties ⬇️

scientific article published in October 1983

Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor

scientific article

Oral adjuvant activity for nasal influenza vaccines caused by combination of two trihydroxy fatty acid stereoisomers from the tuber of Pinellia ternata.

scientific article

Organization of the biosynthetic gene cluster for the polyketide anthelmintic macrolide avermectin in Streptomyces avermitilis

scientific article

Oxaline, a fungal alkaloid, arrests the cell cycle in M phase by inhibition of tubulin polymerization

scientific article

Oxetin, a new antimetabolite from an actinomycete. Fermentation, isolation, structure and biological activity

scientific article published on November 1984

Panowamycins A and B, new antitrypanosomal isochromans produced by Streptomyces sp. K07-0010. ⬇️

scientific article published on 25 January 2012

Penicillium viticola, a new species isolated from a grape in Japan

article

Pentacecilides, new inhibitors of lipid droplet formation in mouse macrophages produced by Penicillium cecidicola FKI-3765-1: II. Structure elucidation

scientific article published on 20 March 2009

Pentacecilides, new inhibitors of lipid droplet formation in mouse macrophages, produced by Penicillium cecidicola FKI-3765-1: I. Taxonomy, fermentation, isolation and biological properties ⬇️

scientific article published on 20 March 2009

Pentalenolactone biosynthesis. Molecular cloning and assignment of biochemical function to PtlH, a non-heme iron dioxygenase of Streptomyces avermitilis

scientific article

Pentalenolactone biosynthesis. Molecular cloning and assignment of biochemical function to PtlI, a cytochrome P450 of Streptomyces avermitilis

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Pentalenolactone biosynthesis: Molecular cloning and assignment of biochemical function to PtlF, a short-chain dehydrogenase from Streptomyces avermitilis, and identification of a new biosynthetic intermediate

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Phenatic acids A and B, new potentiators of antifungal miconazole activity produced by Streptomyces sp. K03-0132. ⬇️

scientific article published in April 2005

Phthoxazolin A, a specific inhibitor of cellulose biosynthesis from microbial origin. I. Discovery, taxonomy of producing microorganism, fermentation, and biological activity

scientific article published in August 1993

Phytohabitans flavus sp. nov., Phytohabitans rumicis sp. nov. and Phytohabitans houttuyneae sp. nov., isolated from plant roots, and emended description of the genus Phytohabitans

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Phytohabitans suffuscus gen. nov., sp. nov., an actinomycete of the family Micromonosporaceae isolated from plant roots

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Polymyxin B identified as an inhibitor of alternative NADH dehydrogenase and malate: quinone oxidoreductase from the Gram-positive bacterium Mycobacterium smegmatis

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Potent antimalarial activities of polyether antibiotic, X-206.

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Preparation of 13C- and 3H-labeled cerulenin and biosynthesis with 13C-NMR ⬇️

scientific article published on October 1, 1975

Production of 6,8a-seco-6,8a-deoxy derivatives of avermectins by a mutant strain of Streptomyces avermitilis.

scientific article published in January 1995

Production of 9-.BETA.-D-arabinofuranosyladenine by a new species of Streptomyces and its herbicidal activity ⬇️

scientific article published on October 1, 1979

Production of a new type of amidepsine with a sugar moiety by static fermentation of Humicola sp. FO-2942. ⬇️

scientific article published on 27 November 2009

Production of deoxyfrenolicin and a new antibiotic, frenolicin B by Streptomyces roseofulvus strain AM-3867.

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Production of ‘hybrid’ antibiotics by genetic engineering

scientific article published in Nature

Promising lead compounds for novel antiprotozoals

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Purpactins, new inhibitors of acyl-CoA:cholesterol acyltransferase produced by Penicillium purpurogenum. I. Production, isolation and physico-chemical and biological properties ⬇️

scientific article published on February 1, 1991

Purpactins, new inhibitors of acyl-CoA:cholesterol acyltransferase produced by Penicillium purpurogenum. III. Chemical modification of purpactin A.

scientific article published on February 1991

Recent development of two chitinase inhibitors, Argifin and Argadin, produced by soil microorganisms

scientific article

Relationship between the structures of fatty acid amide derivatives and their antimicrobial activities

scientific article published on August 1974

Remarkable influence of the aromatic substructure in 9-methoxystrobilurin derivatives on their antifungal activity

scientific article published on October 2002

Research and development of clarithromycin

scientific article published on September 1, 1992

Screening and isolation of penicillinase inhibitor, KA-107.

scientific article published on September 1973

Screening for new antitrichomonal substances of microbial origin and antitrichomonal activity of trichostatin A.

scientific article published in April 1988

Search for protein farnesyltransferase inhibitors of microbial origin: our strategy and results as well as the results obtained by other groups

scientific article published on January 2007

Selective and potent in vitro antitrypanosomal activities of ten microbial metabolites

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Selective inhibition of bleomycin-induced G2 cell cycle checkpoint by simaomicin alpha

scientific article published on May 2004

Selective production of fungal beauveriolide I or III by fermentation in amino acid-supplemented media

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Selective production of specific components of avermectins in Streptomyces avermitilis.

scientific article published in May 1991

Selectivity of microbial acyl-CoA: cholesterol acyltransferase inhibitors toward isozymes.

scientific article published in January 2007

Selectivity of pyripyropene derivatives in inhibition toward acyl-CoA:cholesterol acyltransferase 2 isozyme.

scientific article published in August 2008

Siccanin rediscovered as a species-selective succinate dehydrogenase inhibitor

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Simaomicin alpha: effects on the cell cycle of synchronized, cultured Plasmodium falciparum

scientific article published in April 2008

Sinefungin VA and dehydrosinefungin V, new antitrypanosomal antibiotics produced by Streptomyces sp. K05-0178 ⬇️

scientific article published on September 22, 2010

Solid-phase total synthesis of the chitinase inhibitor Argadin using a supported acetal resin.

scientific article published on 3 July 2009

Spoxazomicins A-C, novel antitrypanosomal alkaloids produced by an endophytic actinomycete, Streptosporangium oxazolinicum K07-0460(T). ⬇️

scientific article published on 9 March 2011

Spylidone, a novel inhibitor of lipid droplet accumulation in mouse macrophages produced by Phoma sp. FKI-1840. ⬇️

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Staurosporine, a Potentially Important Gift from a Microorganism ⬇️

scientific article published on July 1, 1995

Stemphones, novel potentiators of imipenem activity against methicillin-resistant staphylococcus aureus, produced by Aspergillus sp. FKI-2136. ⬇️

scientific article published in November 2005

Stereostructure of luminamicin, an anaerobic antibiotic, via molecular dynamics, NMR spectroscopy, and the modified Mosher method

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Stimulation of leucomycin production by magnesium phosphate and its relevance to nitrogen catabolite regulation

scientific article published on November 1980

Streptosporangium oxazolinicum sp. nov., a novel endophytic actinomycete producing new antitrypanosomal antibiotics, spoxazomicins

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Structural analysis of the gene coding for hepatitis B virus surface antigen and its product

scientific article published in January 1985

Structural and computational analysis of the quinone-binding site of complex II (succinate-ubiquinone oxidoreductase): a mechanism of electron transfer and proton conduction during ubiquinone reduction

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Structural study of isoflavonoids possessing antioxidant activity isolated from the fermentation broth of Streptomyces sp. ⬇️

scientific article published on September 1989

Structure and total synthesis of fungal calpinactam, a new antimycobacterial agent

scientific article published in February 2010

Structure determination and total synthesis of (+)-16-hydroxy-16,22-dihydroapparicine

scientific article published on 20 June 2013

Structure determination and total synthesis of bottromycin A2: a potent antibiotic against MRSA and VRE.

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Structure of a new antimicrobial unsaturated fatty acid from Sm. kitasatoenis NU-23-1 ⬇️

scientific article published on December 1, 1976

Structure of nanaomycin E, a new nanaomycin ⬇️

scientific article published on May 1, 1979

Structure of the spiramycins (foromacidines) and their relationship with the leucomycins and carbomycins (magnamycins) ⬇️

scientific article

Structure-activity Relationships of Pyripyropenes Fungal Acyl-CoA: Cholesterol Acyltransferase Inhibitors ⬇️

scientific article published on July 1, 1995

Structure-activity relationships of stemphones, potentiators of imipenem activity against methicillin-resistant Staphylococcus aureus ⬇️

scientific article

Structures and Biological Properties of Kinamycin A, B, C, and D ⬇️

scientific article published on May 1, 1973

Studies on a novel antitumor antibiotic, phenazinomycin: taxonomy, fermentation, isolation, and physicochemical and biological characteristics ⬇️

scientific article published in July 1989

Studies on bacterial cell wall inhibitors. VII. Azureomycins A and B, new antibiotics produced by Pseudonocardia azurea nov. sp. Taxonomy of the producing organism, isolation, characterization and biological properties

scientific article published on October 1, 1979

Studies on bacterial cell wall inhibitors. VIII. Mode of action of a new antibiotic, azureomycin B, in Bacillus cereus T

scientific article published on October 1, 1979

Studies on cerulenin, 3. Isolation and physico-chemical properties of cerulenin

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Studies on cerulenin. V. Structure of cerulenin

scientific article published in November 1967

Studies on penicillinase inhibitors produced by microorganisms

scientific article published on August 1, 1972

Studies on the ionophorous antibiotics. XVII. The structures of lonomycins B and C

scientific article published on September 1, 1978

Superoxide dismutase produced by soil bacteria increases bacterial colony growth from soil samples ⬇️

scientific article published on August 1, 2003

Suppression of bone resorption by madindoline A, a novel nonpeptide antagonist to gp130.

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Synthesis and anti-platelet aggregation activity of water-soluble staurosporine derivatives

scientific article published in October 1996

Synthesis and biological activities of novel 4″-alkylidene avermectin derivatives ⬇️

scientific article published on November 17, 2003

Synthesis and biological activity of analogues of diazaquinomycin A, a new thymidylate synthase inhibitor

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Synthesis and biological evaluation of a beauveriolide analogue library

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Synthesis and biological evaluation of a focused library of beauveriolides

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Synthesis and biological evaluation of novel 4"-alkoxy avermectin derivatives.

scientific article published in August 2004

Synthesis and inhibitory activities of isochromophilone analogues against gp120-CD4 binding

scientific article published on July 1996

Synthesis and nematocidal activities of jietacin A and its analogs

scientific article published in July 1991

Synthesis and stereochemical determination of an antiparasitic pseudo-aminal type monoterpene indole alkaloid

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Takanawaenes, novel antifungal antibiotics produced by Streptomyces sp. K99-5278. I. Taxonomy, fermentation, isolation and biological properties ⬇️

scientific article published in May 2003

Tensidols, new potentiators of antifungal miconazole activity, produced by Aspergillus niger FKI-2342. ⬇️

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Tensyuic acids, new antibiotics produced by Aspergillus niger FKI-2342. ⬇️

scientific article published in September 2007

Terpendoles, novel ACAT inhibitors produced by Albophoma yamanashiensis. I. Production, isolation and biological properties. ⬇️

scientific article published on January 1995

The antibiotic cerulenin, a novel tool for biochemistry as an inhibitor of fatty acid synthesis

scientific article published on September 1976

The chemistry of leucomycins. IV. Structure of leucomycin A.

scientific article published in March 1968

The effects of macrolides (EM900, clarithromycin and azithromycin) on IL-17-induced IL-8 production by airway epithelial cells

scientific article published on March 2009

The first total synthesis of (+/-)-arisugacin A, a potent, orally bioavailable inhibitor of acetylcholinesterase

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The high mannose-type glycan binding lectin actinohivin: dimerization greatly improves anti-HIV activity

scientific article published on 22 June 2011

The non-osteogenic mouse pluripotent cell line, C3H10T1/2, is induced to differentiate into osteoblastic cells by recombinant human bone morphogenetic protein-2 ⬇️

scientific article published on October 15, 1990

The selectivity of beauveriolide derivatives in inhibition toward the two isozymes of acyl-CoA: cholesterol acyltransferase.

scientific article published in April 2009

The site of inhibition of cell wall synthesis by 3-amino-3-deoxy-D-glucose in Staphylococcus aureus ⬇️

scientific article published on 01 July 1979

Thiotetromycin, a new antibiotic. Taxonomy, production, isolation, and physicochemical and biological properties. ⬇️

scientific article published in February 1983

Three new Pochonia taxa (Clavicipitaceae) from soils in Japan

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Three-dimensional solution structure of bottromycin A2: a potent antibiotic active against methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococci

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Total synthesis and determination of the absolute configuration of guadinomines B and C2.

scientific article published in January 2008

Verticilide, a new ryanodine-binding inhibitor, produced by Verticillium sp. FKI-1033.

scientific article published on 8 January 2010

Virantmycin, a potent antiviral antibiotic produced by a strain of Streptomyces ⬇️

scientific article published in November 1980

X-ray crystallography of protylonolide and absolute configuration of tylosin

scientific article published on August 1980

Xanthoradone C, a new potentiator of imipenem activity against methicillin-resistant Staphylococcus aureus, produced by Penicillium radicum FKI-3765-2.

scientific article published on 30 April 2010

Xanthoradones, new potentiators of imipenem activity against methicillin-resistant Staphylococcus aureus, produced by Penicillium radicum FKI-3765-2 II. Structure elucidation.

scientific article published on 17 July 2009

Xanthoradones, new potentiators of imipenem activity against methicillin-resistant Staphylococcus aureus, produced by Penicillium radicum FKI-3765-2: I. Taxonomy, fermentation, isolation and biological properties ⬇️

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Yaequinolones J1 and J2, novel insecticidal antibiotics from Penicillium sp. FKI-2140.

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Yaequinolones, new insecticidal antibiotics produced by Penicillium sp. FKI-2140. I. Taxonomy, fermentation, isolation and biological activity ⬇️

scientific article published in October 2006

Yaequinolones, new insecticidal antibiotics produced by Penicillium sp. FKI-2140. II. Structural elucidation.

scientific article published in October 2006

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