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List of works by Paweł Kafarski

1,4-Phenylene-di(N-l-alanylaminomethylphosphonate) a new diaminophosphonate peptide receptor for lysine and arginine

3-D QSAR investigations of the inhibition of Leishmania major farnesyl pyrophosphate synthase by bisphosphonates.

scientific article published in November 2003

A Straightforward Synthesis of Six‐Membered‐Ring Heterocyclic α‐Aminophosphonic Acids from N ‐Acyliminium Ions

scientific article

A kinetic study on the isomerization of hop alpha-acids

scientific article published on 4 July 2008

A novel approach for obtaining α,β-diaminophosphonates bearing structurally diverse side chains and their interactions with transition metal ions studied by ITC

scientific article

A phosphonamidate containing aromatic N-terminal amino group as inhibitor of leucine aminopeptidase-design, synthesis and stability.

scientific article

A simple and green procedure for the microbial effective synthesis of 1-phenylethyl alcohol in both enantiomeric forms

scientific article published in April 2006

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases

scientific article published on 22 February 2007

Access to alpha-aminophosphonic acid derivatives and phosphonopeptides by [Rh(P-OP)]-catalyzed stereoselective hydrogenation

scientific article published on 11 June 2020

Accurate assay of enantiopurity of 1-hydroxy- and 2-hydroxyalkylphosphonate esters

Activity of bisphosphonates against Trypanosoma brucei rhodesiense

scientific article published in July 2002

Addition of H-phosphonates to quinine-derived carbonyl compounds. An unexpected C9 phosphonate-phosphate rearrangement and tandem intramolecular piperidine elimination

scientific article

Addition of thiols to the double bond of dipeptide C-terminal dehydroalanine as a source of new inhibitors of cathepsin C

scientific article published on 17 May 2017

Amidoalkylation of Phosphorus Trichloride with Acetamide and Alkyl Oxocycloalkanecarboxylates

scientific article

Amidoalkylation of Phosphorus Trichloride with Acetamide and Functionalized Cyclic Ketones-Evidence of Dominating Role of Side-Reactions

Amino polyphosphonates - chemical features and practical uses, environmental durability and biodegradation.

scientific article published on 30 July 2014

Aminobisphosphonates based on cyclohexane backbone as coordinating agents for metal ions. Thermodynamic, spectroscopic and biological studies

Aminophosphonic acids of potential medical importance

scientific article

An approach to the synthesis and assignment of the absolute configuration of all enantiomers of ethyl hydroxy(phenyl)methane(P-phenyl)phosphinate

Analysis of pD-dependent complexation of N-benzyloxycarbonylaminophosphonic acids by alpha-cyclodextrin. Enantiodifferentiation of phosphonic acid pKa values.

scientific article

Antibacterial activity of phosphono dipeptides based on 1-amino-1-methylethanephosphonic acid.

scientific article

Antibacterial activity of phosphono dipeptides related to alafosfalin

scientific article published on 01 November 1986

Antibacterial activity of phosphono peptides based on 4-amino-4-phosphonobutyric acid

scientific article published on 01 April 1993

Antifungal activity of the carrot seed oil and its major sesquiterpene compounds.

scientific article published in November 2004

Application of bacteria and fungi as biocatalysts for the preparation of optically active hydroxyphosphonates

Authentication of phacelia honeys (Phacelia tanacetifolia) based on a combination of HPLC and HPTLC analyses as well as spectrophotometric measurements

scientific article

BIOLOGICAL ACTIVITY OF AMINOPHOSPHONIC ACIDS

Biocatalytic resolution of enantiomeric mixtures of 1-aminoethanephosphonic acid

scientific article published on 14 July 2011

Biochemical bases for a widespread tolerance of cyanobacteria to the phosphonate herbicide glyphosate

scientific article published on 7 February 2008

Biodegradation of the aminopolyphosphonate DTPMP by the cyanobacterium Anabaena variabilis proceeds via a C-P lyase-independent pathway

scientific article published in December 2016

Bisphosphonic acids as effective inhibitors of Mycobacterium tuberculosis glutamine synthetase

scientific article published on 03 August 2015

Botanical Origin Authentication of Polish Phacelia Honey Using the Combination of Volatile Fraction Profiling by HS-SPME and Lipophilic Fraction Profiling by HPTLC

scientific article

Characterization of the Plasmodium falciparum M17 leucyl aminopeptidase. A protease involved in amino acid regulation with potential for antimalarial drug development

scientific article (publication date: 19 January 2007)

Chelating tendencies of bioactive aminophosphonates

scientific article published in January 1994

Chemical Profiling of Polyfloral Belgian Honey: Ellagic Acid and Pinocembrin as Antioxidants and Chemical Markers

scientific article

Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors

scientific article published on 5 May 2008

Chemometrics as a tool of origin determination of Polish monofloral and multifloral honeys

scientific article published on 18 March 2014

Chiral O-phosphorylated derivative of 2-hydroxy-2-phenylethylphosphonate as a valuable product of microbial biotransformation of diethyl 2-oxo-2-phenylethylphosphonate

Chiral discrimination of ethyl and phenyl N-benzyloxycarbonylaminophosphonates by cyclodextrins

Chromatographic fingerprint of the volatile fraction of rare Hedera helix honey and biomarkers identification

scientific article

Cinchona alkaloids as privileged chiral solvating agents for the enantiodiscrimination of N-protected aminoalkanephosphonates—a comparative NMR study

Combined effect of the DeltaPhe or DeltaAla residue and the p-nitroanilide group on a didehydropeptides conformation.

scientific article published in March 2008

Comparative study of fungal cell disruption--scope and limitations of the methods

scientific article

Comparison of adsorption mechanism on colloidal silver surface of alafosfalin and its analogs

Computer-Aided Analysis and Design of Phosphonic and Phosphinic Enzyme Inhibitors as Potential Drugs and Agrochemicals

Computer-aided analysis of the interactions of glutamine synthetase with its inhibitors

scientific article published on 28 February 2006

Computer-aided design and activity prediction of leucine aminopeptidase inhibitors

scientific article published on 01 August 2000

Computer-aided optimization of phosphinic inhibitors of bacterial ureases.

scientific article published on August 2010

Conformation of dehydropentapeptides containing four achiral amino acid residues - controlling the role of L-valine.

scientific article

Conformational investigations of bis(α-aminoalkyl)phosphinic acids and studies of the stability of their complexes with Cu(II)

Conformational isomers of the [(5-methyl-2-pyridinio)aminomethylene]diphosphonate dianion and [(5-methyl-2-pyridyl)aminomethylene]diphosphonate trianion in salts with 4-aminopyridine and ammonia.

scientific article published on 2 May 2009

Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate

Coordination abilities of difunctional, diaminophosphonic acid and its dipeptides towards Cu(II) ions

Coordination abilities of piperyd-1-yl-methane-1,1-diphosphonic acids towards zinc(II), magnesium(II) and calcium(II): potentiometric and NMR studies.

scientific article published on 23 February 2006

Coordination abilities of substituted β-aminophosphonates towards Cu2+ and Zn2+ ions

Copper(II) complexation by (pyridinyl)aminomethane-1,1-diphosphonic acid derivatives; spectroscopic and potentiometric studies

Copper(II) complexes of several monophosphono dipeptides: the role of phosphonic oxygen and thioether sulfur in complex stabilization

Correction to: New crystal structures of fluorinated α-aminophosphonic acid analogues of phenylglycine

scientific article

Crotonic acid as a bioactive factor in carrot seeds (Daucus carota L.).

scientific article

Cyclodextrins as NMR probes in the study of the enantiomeric compositions of N-benzyloxycarbonylamino-phosphonic and phosphinic acids

article

Degradation of Amino-(3-methoxyphenyl)methanephosphonic Acid by Alternaria sp

Degradation of organophosphonates by Penicillium citrinum

Design, synthesis, and activity of analogues of phosphinothricin as inhibitors of glutamine synthetase

scientific article

Design, synthesis, and evaluation of novel organophosphorus inhibitors of bacterial ureases

scientific article

Determination of bisphosphonates anti-resorptive properties based on three forms of ceramic materials: Sorption and release process evaluation

Determination of optical purity of phosphonic acid analogues of aromatic amino acids by capillary electrophoresis with α-cyclodextrin

scientific article published on 01 October 2000

Development of a high performance thin layer chromatography method for the rapid qualification and quantification of phenolic compounds and abscisic acid in honeys

scientific article published on 19 April 2019

Diethyl boronobenzylphosphonates as substrates in Petasis reaction

Diethyl boronobenzylphosphonates as substrates in Suzuki–Miyaura reaction

scientific article

Dipeptides of -Substituted Dehydrocysteine as Artzyme Building Blocks: Synthesis, Complexing Abilities and Antiproliferative Properties

scientific article

Do differences in chemical composition of stem and cap of Amanita muscaria fruiting bodies correlate with topsoil type?

scientific article

Effect of an aliphatic spacer group on the adsorption mechanism of phosphonodipeptides containing N -terminal glycine on the colloidal silver surface

scientific article

Effect of an aliphatic spacer group on the adsorption mechanism on the colloidal silver surface of L-proline phosphonodipeptides

scientific article

Effectiveness and mode of action of phosphonate inhibitors of plant glutamine synthetase

scientific article published in January 2010

Electrochemical and spectroscopic investigations of selected N -heteroalkylaminomethylenebisphosphonic acids with Pb(II) ions

Enantiodifferentiation of N-benzyloxycarbonylaminophosphonic and phosphinic acids and their esters using cyclodextrins by means of capillary electrophoresis

scientific article published on 09 November 2006

Enantiodifferentiation of alpha-hydroxyalkanephosphonic acids in 31P NMR with application of alpha-cyclodextrin as chiral discriminating agent

scientific article published in January 2010

Enantiodifferentiation of aminophosphonic and aminophosphinic acids with α- and β-cyclodextrins

Enantioselective reduction of diethyl 2-oxoalkylphosphonates by baker's yeast

Enzymatic Resolution of Ethyl α-Hydroxyphosphinates in a Modified Reaction Environment

Enzymatic resolution of α-hydroxyphosphinates with two stereogenic centres and determination of absolute configuration of stereoisomers obtained

scientific article

First example of the chemical, oxidative cleavage of the C-P bond in aminophosphonate chemistry. The oxidation of 1-amino-1-(3,4-dihydroxyphenyl)methylphosphonic acid by NaIO4.

scientific article published on 8 April 2004

HPTLC Fingerprinting-Rapid Method for the Differentiation of Honeys of Different Botanical Origin Based on the Composition of the Lipophilic Fractions

scientific article published on 21 July 2018

Herbicidal Derivatives of Aminomethylenebisphosphonic Acid. Part III. Structure—Activity Relationship

Herbicidal Derivatives of Aminomethylenebisphosphonic Acid. Part IV. Hydroxyalkylidenebisphosphonates, Iminomethylenebisphosphonates and Ureidomethylenebisphosphonates

scientific article published on 01 December 1999

Herbicidal activity of phosphonic, phosphinic, and phosphonous acid analogues of phenylglycine and phenylalanine

Herbicidal pyridyl derivatives of aminomethylene-bisphosphonic acid inhibit plant glutamine synthetase

scientific article

High-performance liquid chromatographic enantiomer separation and determination of absolute configurations of phosphinic acid analogues of dipeptides and their α-aminophosphinic acid precursors

Hydrolysis of the Phosphonamidate Bond in Phosphono Dipeptide Analogues— the Influence of the Nature of the N-Terminal Functional Group

Hydrophosphonylation of nanoparticle Schiff bases as a mean for preparation of aminophosphonate-functionalized nanoparticles

scientific article published on 18 July 2013

Hypervalent-iodine mediated one-pot synthesis of isoxazolines and isoxazoles bearing a difluoromethyl phosphonate moiety

scientific article

Identification of phosphinate dipeptide analog inhibitors directed against the Plasmodium falciparum M17 leucine aminopeptidase as lead antimalarial compounds.

scientific article published on 26 October 2007

Improvement of Large Animal Model for Studying Osteoporosis

Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.

scientific article published on 2 February 2008

Influence of aliphatic spacer group on adsorption mechanisms of phosphonate derivatives of l-phenylalanine: Surface-enhanced Raman, Raman, and infrared studies

Influence of solvents on conformation of dehydropeptides

Inhibition of aminopeptidases by aminophosphonates

scientific article

Inhibition of aminopeptidases by phosphonic acid and phosphinic acid analogues of aspartic and glutamic acids

scientific article published on 01 January 1993

Insight into the mechanism of three component condensation leading to aminomethylenebisphosphonates

Interaction of mushroom tyrosinase with aromatic amines, o-diamines and o-aminophenols

scientific article

Interactions of N-heteroalkylaminomethylenebisphosphonic acids with Cd(II) ions: Electrochemical and spectroscopic investigations

Interactions of zinc(II), magnesium(II) and calcium(II) with aminomethane-1,1-diphosphonic acids in aqueous solutions

scientific article

Interactions of zinc(II), magnesium(II) and calcium(II) with iminodimethylenediphosphonic acids in aqueous solutions †

scientific article

Investigation of molecular structures and adsorption mechanisms of phosphonodipeptides by surface-enhanced Raman, Raman, and infrared spectroscopies

Kinetic resolution of (±)-diethyl- and dibenzyl hydroxy(phenyl)methanephosphonates and their acyl derivatives with lipases

Kinetics of photochemical isomerization of TFA-Gly-ZΔPhe into TFA-Gly-EΔPhe

scientific article

Leucine aminopeptidase as a target for inhibitor design

scientific article

Long range phosphorus–phosphorus coupling constants in bis(phosphorylhydroxymethyl)benzene derivatives

Mannitol in Amanita muscaria--an osmotic blood-brain barrier disruptor enhancing its hallucinogenic action?

scientific article published on 8 August 2013

Mass spectrometric and PM5 study of N-(2-pyridyl)-aminomethyldiphoshonic acids and their complexes with alkali cations

Mass spectrometric and PM5 study of some piperidine-N-methyldiphosphonic acids and their complexes with alkali cations

Metabolism of the phosphonate herbicide glyphosate by a non-nitrate-utilizing strain of Penicillium chrysogenum

scientific article published in September 2001

Metallo-aminopeptidase inhibitors

scientific article published on 10 May 2010

Michael additions to double bonds of esters of N-protected (s)-phenylalanyldehydroalanine (X-(s)-Phe-ΔAla-OMe) and its phosphonic acid counterpart (X-(s)-Phe-ΔAla-PO(OEt)2)

scientific article

Mode of Action of Herbicidal Derivatives of Aminomethylenebisphosphonic Acid. Part II. Reversal of Herbicidal Action by Aromatic Amino Acids

Mode of biosorption of chromium(III) by Spirulina species cells from aqueous solutions

scientific article published on 01 July 2006

N,N′-Ethylenediaminobis(benzylphosphonic acids) as a potent class of chelators for metal ions

N-(Phosphonoacetyl)amino phosphonates. Phosphonate analogues of N-(phosphonoacetyl)-L-aspartic acid (PALA).

scientific article published in November 1985

N-Arylaminomethylenebisphosphonates Bearing Fluorine Atoms: Synthesis and Antiosteoporotic Activity

N-Benzyl Residues as the P1' Substituents in Phosphorus-Containing Extended Transition State Analog Inhibitors of Metalloaminopeptidases

scientific article published on 22 September 2020

N-Pyridyl-aminomethylene-bisphosphonic Acids Inhibit the First Enzyme in the Shikimate Pathway, 3-Deoxy-D-arabino- heptulosonate-7-phosphate Synthase

scientific article published in 1996

N-substituted aminomethanephosphonic and aminomethane-P-methylphosphinic acids as inhibitors of ureases.

scientific article

NMR and theoretical study on the structure of O,O-dimethyl-1,4-oxoazetin-2-ylphosphonate

scientific article

New crystal structures of fluorinated α-aminophosphonic acid analogues of phenylglycine

scientific article

Novel, automated, semi-industrial modular photobioreactor system for cultivation of demanding microalgae that produce fine chemicals—The next story of H. pluvialis and astaxanthin

scientific article

Organophosphonate utilization by the thermophile Geobacillus caldoxylosilyticus T20

scientific article

Organophosphonate utilization by the wild-type strain of Pseudomonas fluorescens ⬇️

scientific article published on September 1, 1992

Organophosphonate utilization by the wild‐type strain ofcladosporium resinae

Organophosphorus Supramolecular Chemistry Part 1. Receptors for Organophosphorus Compounds

Organophosphorus Supramolecular Chemistry. Part 2. Organophosphorus Receptors

Palladium-Catalyzed Hydrophosphonylation of Alkenes with Dialkyl H-Phosphonates

Pentapeptides containing two dehydrophenylalanine residues--synthesis, structural studies and evaluation of their activity towards cathepsin C.

scientific article published in October 2008

Peptide and Pseudopeptide Bond Synthesis in Phosphorus Dipeptide Analogs

scientific article published on 01 January 2020

Peptide p-nitrophenylanilides containing (E)-dehydrophenylalanine—synthesis, structural studies and evaluation of their activity towards cathepsin C

Phenolic compounds and abscisic acid as potential markers for the floral origin of two Polish unifloral honeys

Phosphinothricin analogues as inhibitors of plant glutamine synthetases

scientific article published in February 2006

Phosphonate degradation by Spirulina strains: cyanobacterial biofilters for the removal of anticorrosive polyphosphonates from wastewater

scientific article

Phosphonic Acid Analogs of Fluorophenylalanines as Inhibitors of Human and Porcine Aminopeptidases N: Validation of the Importance of the Substitution of the Aromatic Ring

scientific article published on 09 April 2020

Phosphonic Acid Analogues of Phenylglycine as Inhibitors of Aminopeptidases: Comparison of Porcine Aminopeptidase N, Bovine Leucine Aminopeptidase, Tomato Acidic Leucine Aminopeptidase and Aminopeptidase from Barley Seeds

scientific article published on 17 September 2019

Phosphonic Analogues of Phenylglycine as Inhibitors of Aminopeptidases: Comparison of Porcine Aminopeptidase N, Bovine Leucine Aminopeptidase and Aminopeptidase from Barley Seeds

scientific article

Phosphonic acid analogue of forfenicine ? synthesis, antibacterial activity and degradation byPseudomonas fluorescens

Phosphonic analogues of tyrosine and 3,4-dihydroxyphenylalanine (dopa) influence mushroom tyrosinase activity

scientific article

Phosphonic and phosphinic acid analogues of tyrosine and 3,4-dihydroxyphenylalanine (dopa) as potential antimelanotic agents

scientific article published on 01 November 1990

Phosphonopeptides containing free phosphonic groups: recent advances

scientific article

Phosphorus NMR as a tool to study mineralization of organophosphonates—The ability of Spirulina spp. to degrade glyphosate

article published in 2007

Phosphorus Profile of Basidiomycetes

Phosphorylation as a method of tuning the enantiodiscrimination potency of quinine-An NMR study

scientific article published on 17 February 2012

Physiologic Activity of Bisphosphonates – Recent Advances

Phytotoxicity of aminobisphosphonates targeting both δ1 -pyrroline-5-carboxylate reductase and glutamine synthetase.

scientific article

Plant P5C reductase as a new target for aminomethylenebisphosphonates.

scientific article published on 3 May 2007

Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials

scientific article published on 30 September 2009

Possible fungistatic implications of betulin presence in betulaceae plants and their hymenochaetaceae parasitic fungi.

scientific article

Potentiometric and spectroscopic studies of the cobalt(II), nickel(II) and manganese(II) complexes with some aminodiphosphonic acids in aqueous solution

scientific article

Potentiometric and spectroscopic studies of the copper(II) complexes with some aminodiphosphonic acids in aqueous solution

scientific article

Preliminary pharmacological evaluation of newly synthesized derivatives of phosphonoamino acids

scientific article published on September 1986

Preliminary pharmacological investigation on 38 aminophosphonic acids and their derivatives

scientific article published on September 1985

Preliminary studies on the mechanisms of action of phosphonic analogues of morphactins on plants and bacteria

scientific article published in 1990

Preparation of 1-aminoalkylphosphonic acids and 2-aminoalkylphosphonic acids by reductive amination of oxoalkylphosphonates

Preparation of the library of fluorescent aromatic aminophosphonate phenyl and benzyl esters

Preparation, crystal and molecular structure, and evaluation of plant growth regulating activity of guanidinoalkanephosphinates and phosphonates

Prospects of in vivo 31P NMR method in glyphosate degradation studies in whole cell system

scientific article

Proteases as anti-cancer targets--molecular and biological basis for development of inhibitor-like drugs against cancer

scientific article published on September 2009

Quantitative structure-activity relationships for gammadelta T cell activation by bisphosphonates

scientific article published on January 2004

Quantum chemical analysis of the interactions of transition state analogs with leucine aminopeptidase

Quinazoline Antifolate Thymidylate Synthase Inhibitors: Replacement of Glutamic Acid by Aminophosphonic Acids

Quinine as chiral discriminator for determination of enantiomeric excess of diethyl 1,2-dihydroxyalkanephosphonates

Rapid determination of ibotenic acid and muscimol in human urine

scientific article published on 20 July 2014

Reaction of N-(Benzyloxycarbonyl)aminobenzyl-phosphonous Acid with Ethyl Orthoformate

Reaction of benzolactams with triethyl phosphite prompted by phosphoryl chloride affords benzoannulated monophosphonates instead of expected bisphoshonates

Reactions of Piperazin-2-one, Morpholin-3-one, and Thiomorpholin-3-one with Triethyl Phosphite Prompted by Phosphoryl Chloride: Scope and Limitations

scientific article published on 22 May 2019

Recent advances in design of new urease inhibitors: A review

article

Redox reaction between amino-(3,4-dihydroxyphenyl)methyl phosphonic acid and dopaquinone is responsible for the apparent inhibitory effect on tyrosinase

scientific article published in August 2002

Reductive biotransformation of diethyl β-, γ- and δ-oxoalkylphosphonates by cells of baker’s yeast

scientific article published on 01 February 2000

Regio- and stereoselective synthesis of 2-amino-1-hydroxy-2-aryl ethylphosphonic esters

Remarkable potential of the α-aminophosphonate/phosphinate structural motif in medicinal chemistry

scientific article published on 05 August 2011

Selective synthesis of α-fluoro-β-keto- and α-fluoro-β-aminophosphonates via electrophilic fluorination by selectfluor

scientific article published on 18 January 2011

Separation of amino acid enantiomers using supported liquid membrane extraction with chiral phosphates and phosphonates

Separation of aminoalkanephosphonic acid enantiomers by indirect UV detection capillary electrophoresis with application of cyclodextrins

scientific article published on 01 August 2003

Separation of aromatic aminophosphonic acid enantiomers by capillary electrophoresis with the application of cyclodextrins

scientific article published on 01 December 2002

Simple and effective method for the deracemization of ethyl 1-hydroxyphosphinate using biocatalysts with lipolytic activity

Slow Inversion of Stereoisomers of 4-Amino-1-benzylpiperid-4-yl Phosphonic Acids and Their Esters

Solid state and solution behaviour of N-(2-pyridyl)- and N-(4-methyl-2-pyridyl)aminomethane-1,1-diphosphonic acids

Solid-state molecular organization and solution behavior of methane-1,1-diphosphonic acid derivatives of heterocyclic amines: the role of the topochemical ring modification and the intramolecular hydrogen bonds in monosubstituted [...]

scientific article

Solution conformations of 2-amino-1-hydroxy-2-aryl ethylphosphonic acids and their diethyl esters

Specificity of the zinc(II), magnesium(II) and calcium(II) complexation by (pyridin-2-yl)aminomethane-1,1-diphosphonic acids and related 1,3-(thiazol-2-yl) and 1,3-(benzothiazol-2-yl) derivatives.

scientific article published on 19 November 2009

Stereochemical control of biocatalytic asymmetric reduction of diethyl 2-oxopropylphosphonate employing yeasts

Stereoselective separations of chiral phosphinic acid pseudodipeptides by CEC using silica monoliths modified with an anion-exchange-type chiral selector

scientific article published on 01 November 2006

Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.

scientific article published in January 2003

Stereoselective synthesis, solution structure and metal complexes of (1S,2S)-2-amino-1-hydroxyalkylphosphonic acids

Structural Analogues of Selfotel

scientific article

Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase

scientific article

Structural properties of L-X-L-Met-L-Ala phosphonate tripeptides: a combined FT-IR, FT-RS, and SERS spectroscopy studies and DFT calculations

scientific article

Structure of the Plasmodium falciparum M17 aminopeptidase and significance for the design of drugs targeting the neutral exopeptidases

scientific article

Sublethal detergent concentrations increase metabolization of recalcitrant polyphosphonates by the cyanobacterium Spirulina platensis

scientific article

Substituted phosphonic analogues of phenylglycine as inhibitors of phenylalanine ammonia lyase from potatoes

scientific article published on 15 June 2018

Supported liquid membrane separation of amine and amino acid derivatives with chiral esters of phosphoric acids as carriers

Synthesis and Inhibitory Studies of Phosphonic Acid Analogues of Homophenylalanine and Phenylalanine towards Alanyl Aminopeptidases

scientific article published on 14 September 2020

Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin C.

scientific article

Synthesis and evaluation of effective inhibitors of plant δ1-pyrroline-5-carboxylate reductase

scientific article

Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides

scientific article

Synthesis of Hybrid Tripeptide Peptidomimetics Containing Dehydroamino Acid and Aminophosphonic Acid in the Chain and Evaluation of Their Activity toward Cathepsin C

scientific article published in 2022

Synthesis of Triethyl N-Formyl-N-phosphonomethylglycinate and Diethyl N-Formyl-N-phosphonomethylglycine and Studies of Their Rotational Conformers by Dynamic NMR

Synthesis of cyclooctapeptides: constraints analogues of the peptidic neurotoxin, ω-agatoxine IVB—an experimental point of view

Synthesis of dehydrodipeptide esters and their evaluation as inhibitors of cathepsin C.

scientific article published on 16 April 2015

Synthesis of fluorescent (benzyloxycarbonylamino)(aryl)methylphosphonates

scientific article

Synthesis of phosphonate derivatives of 2,3-dihydroindene

Synthesis of tetrapeptide p-nitrophenylanilides containing dehydroalanine and dehydrophenylalanine and their influence on cathepsin C activity

scientific article published in March 2001

Synthetic Procedures Leading towards Aminobisphosphonates

scientific article

Tailoring the structure of aminobisphosphonates to target plant P5C reductase

scientific article published on 10 April 2008

Tetra-2-methoxyethyl phenylene-1,4-di(benzyloaminomethanephosphonate) a new ligand for metal ions and amino acids. Electrospray ionization mass spectrometric and NMR studies

The Computer-Aided Design, Synthesis, and Activity Prediction of New Leucine Aminopeptidase Inhibitors

The Herbicidally Active Compound N-2-(6-Methyl-Pyridyl)-Aminomethylene Bisphosphonic Acid Inhibits In Vivo Aromatic Biosynthesis

scientific article published on 01 October 1999

The M18 aspartyl aminopeptidase of the human malaria parasite Plasmodium falciparum.

scientific article published on 20 August 2007

The ability of soil-borne fungi to degrade organophosphonate carbon-to-phosphorus bonds

scientific article published in October 1997

The application of organophosphorus flame-retardants in epoxy resin

scientific article

The chemical composition of the floral extract of Epipogium aphyllum sw. (Orchidaceae): A clue for their pollination biology

article

The experimental osteoporosis in sheep--clinical approach

scientific article published in September 2015

The influence of α-aminophosphonic acids on the activity of aminopeptidase from barley seeds—an approach to determine the enzyme specificity

The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity

scientific article

The overproduction of 2,4-DTBP accompanying to the lack of available form of phosphorus during the biodegradative utilization of aminophosphonates by Aspergillus terreus.

scientific article

The role of hydrogen bonding in conformational stabilization of 3,5,6- and 3,5-substituted (pyridin-2-yl)aminomethane-1,1-diphosphonic acids and related (pyrimidin-2-yl) derivative

The use of molecular modelling for comparison of three possible modes of action of herbicidally active derivatives of aminomethylenebisphosphonic acid

scientific article published in 2002

Theoretical study of spin-spin coupling across the hydrogen (O-H...N) bond in adenosine derivatives

scientific article published on 24 February 2009

Three-Component Reaction of Benzylamines, Diethyl Phosphite and Triethyl Orthoformate: Dependence of the Reaction Course on the Structural Features of the Substrates and Reaction Conditions.

scientific article published on 11 March 2017

Three-Component Reaction of Diamines with Triethyl Orthoformate and Diethyl Phosphite and Anti-Proliferative and Antiosteoporotic Activities of the Products

scientific article published on 20 March 2020

Toward very potent, non-covalent organophosphonate inhibitors of cathepsin C and related enzymes by 2-amino-1-hydroxy-alkanephosphonates dipeptides

scientific article published on 24 May 2013

Transesterification of monophenyl phosphonamidates—chemical modelling of serine protease inhibition

Unexpected formation of hydroxyborazaphosphonic acid in the reaction of (N-benzyl)benzylideneimine-2-boronic acid with diethyl phosphite

Vibrational characterization of L -valine phosphonate dipeptides: FT-IR, FT-RS, and SERS spectroscopy studies and DFT calculations

Vibrational characterization of L-leucine phosphonate analogues: FT-IR, FT-Raman, and SERS spectroscopy studies and DFT calculations

scientific article published on 19 September 2011

Whole-cell Proteus mirabilis urease inhibition by aminophosphinates for the control of struvite formation.

scientific article

Z/E Isomerism in (Pyridinyl)aminomethane-1,1-diphosphonic Acids Derived from 2-, 3-, and 4-Aminopyridines

[(5-Bromopyridinium-2-ylamino)(phosphono)methyl]phosphonate.

scientific article published on 11 February 2006

alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases

scientific article published on 20 April 2005

Δ1-pyrroline-5-carboxylate reductase as a new target for therapeutics: inhibition of the enzyme from Streptococcus pyogenes and effects in vivo

scientific article published on 09 July 2011

“Twin” phosphorous atoms of tetraethyl 2-methyl-piperyd-1-ylmethylenebisphosphonates

article by Piotr Młynarz et al published 2007 in Heteroatom Chemistry

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