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List of works by Lars Richter

A residue close to α1 loop F disrupts modulation of GABAA receptors by benzodiazepines while their binding is maintained

scientific article published on 11 November 2010

An updated unified pharmacophore model of the benzodiazepine binding site on gamma-aminobutyric acid(a) receptors: correlation with comparative models

scientific article

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands

scientific article

Exploiting open data: a new era in pharmacoinformatics

scientific article

Kinetics for Drug Discovery: an industry-driven effort to target drug residence time

scientific article

Ligand Desolvation Steers On-Rate and Impacts Drug Residence Time of Heat Shock Protein 90 (Hsp90) Inhibitors

scientific article published on 10 May 2018

Medicinal chemistry in the era of big data

scientific article published on 14 July 2015

Molecular analysis of the site for 2-arachidonylglycerol (2-AG) on the β₂ subunit of GABA(A) receptors

scientific article

SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2– Benzodiazepine Site

scientific article published on 08 August 2018

Structure based classification for bile salt export pump (BSEP) inhibitors using comparative structural modeling of human BSEP.

scientific article published on 19 May 2017

The application of the open pharmacological concepts triple store (Open PHACTS) to support drug discovery research

scientific article published in 2014

Topliss Batchwise Schemes Reviewed in the Era of Open Data Reveal Significant Differences between Enzymes and Membrane Receptors

scientific article published on 21 September 2017

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