Search filters

List of works by Arthur Christopoulos

3HN-methylscopolamine dissociation from muscarine receptors affected by low concentrations of allosteric modulators ⬇️

scientific article published on August 15, 1995

4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of the M1 Muscarinic Acetylcholine Receptor.

scientific article published in December 2015

A Hydrogen-Bonded Polar Network in the Core of the Glucagon-Like Peptide-1 Receptor Is a Fulcrum for Biased Agonism: Lessons from Class B Crystal Structures

scientific article

A Monod-Wyman-Changeux mechanism can explain G protein-coupled receptor (GPCR) allosteric modulation

scientific article published on 15 November 2011

A Positive Allosteric Modulator of the Adenosine A1 Receptor Selectively Inhibits Primary Afferent Synaptic Transmission in a Neuropathic Pain Model

scientific article published on 23 June 2015

A Structure-Activity Relationship Study of Bitopic N6-Substituted Adenosine Derivatives as Biased Adenosine A1 Receptor Agonists

scientific article published on 15 February 2018

A new mechanism of allostery in a G protein-coupled receptor dimer

scientific article (publication date: September 2014)

A simple method for quantifying functional selectivity and agonist bias

scientific article (publication date: 21 March 2012)

A simple method to generate stable cell lines for the analysis of transient protein-protein interactions.

scientific article published on April 2013

A structure-activity analysis of biased agonism at the dopamine D2 receptor

scientific article published on 8 November 2013

Accelerated structure-based design of chemically diverse allosteric modulators of a muscarinic G protein-coupled receptor

scientific article published on 06 September 2016

Activation and allosteric modulation of a muscarinic acetylcholine receptor

scientific article

Advances in G protein-coupled receptor allostery: from function to structure

scientific article

Allosteric Modulation as a Unifying Mechanism for Receptor Function and Regulation

scientific article

Allosteric interactions at muscarinic cholinoceptors ⬇️

scientific article published on March 1, 1998

Allosteric ligands of the glucagon-like peptide 1 receptor (GLP-1R) differentially modulate endogenous and exogenous peptide responses in a pathway-selective manner: implications for drug screening.

scientific article

Allosteric modulation as a unifying mechanism for receptor function and regulation

scientific article published in September 2017

Allosteric modulation of G protein-coupled receptors: a pharmacological perspective.

scientific article published on 15 July 2010

Allosteric modulation of M1 muscarinic acetylcholine receptor internalization and subcellular trafficking

scientific article

Allosteric modulation of a chemogenetically modified G protein-coupled receptor.

scientific article published on 29 November 2012

Allosteric modulation of endogenous metabolites as an avenue for drug discovery.

scientific article published on 10 May 2012

Allosteric modulation of seven transmembrane spanning receptors: theory, practice, and opportunities for central nervous system drug discovery

scientific article

Allosteric modulation of the cannabinoid CB1 receptor

scientific article

Allosteric modulators of G-protein-coupled receptors ⬇️

scientific article published on October 1, 2003

Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders

scientific article published on January 2009

Allosteric targeting of receptor tyrosine kinases.

scientific article published in November 2014

Allostery in GPCRs: 'MWC' revisited.

scientific article published on 14 September 2011

Analytical pharmacology: the impact of numbers on pharmacology

scientific article published on 10 March 2011

Application of an Allosteric Ternary Complex Model to the Technique of Pharmacological Resultant Analysis ⬇️

scientific article published on August 1, 1997

Assessment of the molecular mechanisms of action of novel 4-phenylpyridine-2-one and 6-phenylpyrimidin-4-one allosteric modulators at the M1 muscarinic acetylcholine receptors

scientific article published on 24 April 2018

Biased Agonism and Biased Allosteric Modulation at the CB1 Cannabinoid Receptor

scientific article published on 4 June 2015

Biased Agonism of Endogenous Opioid Peptides at the μ-Opioid Receptor.

scientific article published on 26 May 2015

Biased agonism at G protein-coupled receptors: the promise and the challenges--a medicinal chemistry perspective.

scientific article published on 05 May 2014

Biased allosteric agonism and modulation of metabotropic glutamate receptor 5: Implications for optimizing preclinical neuroscience drug discovery

scientific article published on 5 July 2016

Biased allosteric modulation at the CaS receptor engendered by structurally diverse calcimimetics

scientific article

Bitopic Binding Mode of an M1 Muscarinic Acetylcholine Receptor Agonist Associated with Adverse Clinical Trial Outcomes.

scientific article published on 25 April 2018

Bridging the gap: bitopic ligands of G-protein-coupled receptors.

scientific article

Calcium-sensing receptor-dependent activation of CREB phosphorylation in HEK293 cells and human parathyroid cells.

scientific article

Capadenoson, a clinically trialed partial adenosine A1 receptor agonist, can stimulate adenosine A2B receptor biased agonism.

scientific article published on 23 March 2017

Characterization of serotonin 5-HT2C receptor signaling to extracellular signal-regulated kinases 1 and 2.

scientific article published on June 2005

Characterization of signalling and regulation of common calcitonin receptor splice variants and polymorphisms

scientific article

Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M(2) and M(4) receptors

scientific article published on 7 May 2014

Complexing receptor pharmacology: modulation of family B G protein-coupled receptor function by RAMPs

scientific article

Consequences of splice variation on Secretin family G protein-coupled receptor function

scientific article

Correspondence: Reply to 'Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury'.

scientific article published on 7 February 2018

Crystal structure of the M5 muscarinic acetylcholine receptor

scientific article published on 26 November 2019

Crystal structures of the M1 and M4 muscarinic acetylcholine receptors

scientific article

Design and receptor interactions of obligate dimeric mutant of chemokine monocyte chemoattractant protein-1 (MCP-1).

scientific article published on 6 March 2012

Detection and quantification of allosteric modulation of endogenous m4 muscarinic acetylcholine receptor using impedance-based label-free technology in a neuronal cell line.

scientific article published on 22 December 2014

Development of M1 mAChR Allosteric and Bitopic Ligands: Prospective Therapeutics for the Treatment of Cognitive Deficits ⬇️

scientific article published on May 23, 2013

Development of a highly selective allosteric antagonist radioligand for the type 1 cholecystokinin receptor and elucidation of its molecular basis of binding

scientific article

Development of a photoactivatable allosteric ligand for the m1 muscarinic acetylcholine receptor

scientific article published on 9 September 2014

Development of a radioligand, [(3)H]LY2119620, to probe the human M(2) and M(4) muscarinic receptor allosteric binding sites

scientific article published on 7 May 2014

Differential activation and modulation of the glucagon-like peptide-1 receptor by small molecule ligands

scientific article published on 24 January 2013

Differential engagement of polar networks in the glucagon-like peptide 1 receptor by endogenous variants of the glucagon-like peptide 1

scientific article published on 25 August 2018

Differential impact of amino acid substitutions on critical residues of the human glucagon-like peptide-1 receptor involved in peptide activity and small-molecule allostery.

scientific article published on 28 January 2015

Discovery and Optimization of Potent and CNS Penetrant M5-Preferring Positive Allosteric Modulators Derived from a Novel, Chiral N-(Indanyl)piperidine Amide Scaffold

scientific article published on 26 April 2018

Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor Through Fragmentation of a Bitopic Ligand

scientific article published on 10 August 2015

Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor

scientific article

Divergent effects of strontium and calcium-sensing receptor positive allosteric modulators (calcimimetics) on human osteoclast activity.

scientific article published in May 2018

Drug-receptor kinetics and sigma-1 receptor affinity differentiate clinically evaluated histamine H receptor antagonists

article

Emerging paradigms in GPCR allostery: implications for drug discovery ⬇️

scientific article published on August 1, 2013

Endogenous allosteric modulators of G protein-coupled receptors

scientific article

Engendering biased signalling from the calcium-sensing receptor for the pharmacotherapy of diverse disorders

scientific article published on March 2014

Evidence for pleiotropic signaling at the mouse beta3-adrenoceptor revealed by SR59230A [3-(2-Ethylphenoxy)-1-[(1,S)-1,2,3,4-tetrahydronapth-1-ylamino]-2S-2-propanol oxalate].

scientific article published on December 2004

Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy.

scientific article published on 28 September 2016

Extracellular loops 2 and 3 of the calcitonin receptor selectively modify agonist binding and efficacy.

scientific article published on 15 February 2018

Functional Selectivity and Classical Concepts of Quantitative Pharmacology

scientific article

Functional and structural perspectives on allosteric modulation of GPCRs.

scientific article published on 22 December 2013

G-protein-coupled receptor Mas is a physiological antagonist of the angiotensin II type 1 receptor

scientific article

Glucagon-like peptide-1 receptor dimerization differentially regulates agonist signaling but does not affect small molecule allostery.

scientific article

Glucagon-like peptide-1 receptor internalisation controls spatiotemporal signalling mediated by biased agonists

scientific article published on 07 September 2018

H2 relaxin is a biased ligand relative to H3 relaxin at the relaxin family peptide receptor 3 (RXFP3).

scientific article

High throughput, quantitative analysis of human osteoclast differentiation and activity

scientific article published on 14 December 2016

Identification of global and ligand-specific calcium sensing receptor activation mechanisms

scientific article published on 10 April 2018

Identification of molecular phenotypes and biased signaling induced by naturally occurring mutations of the human calcium-sensing receptor.

scientific article

Impact of chronic congestive heart failure on pharmacokinetics and vasomotor effects of infused nitrite ⬇️

scientific article published on June 1, 2013

Impact of clinically relevant mutations on the pharmacoregulation and signaling bias of the calcium-sensing receptor by positive and negative allosteric modulators

scientific article published on 31 January 2013

Impact of species variability and 'probe-dependence' on the detection and in vivo validation of allosteric modulation at the M4 muscarinic acetylcholine receptor.

scientific article

Improving virtual screening of G protein-coupled receptors via ligand-directed modeling.

scientific article published on 13 November 2017

Inhibition of tumor angiogenesis and growth by a small-molecule multi-FGF receptor blocker with allosteric properties

scientific article

Insurmountable AT1 receptor antagonism: message in a model? ⬇️

scientific article published on 01 November 2001

Interaction studies of multiple binding sites on m4 muscarinic acetylcholine receptors

scientific article published on 18 May 2006

International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands.

scientific article

International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology

scientific article (publication date: December 2003)

Investigation of the Interaction of a Putative Allosteric Modulator,N-(2,3-Diphenyl-1,2,4-thiadiazole-5-(2H)-ylidene) Methanamine Hydrobromide (SCH-202676), with M1Muscarinic Acetylcholine Receptors ⬇️

scientific article published on November 14, 2003

Involvement of the sigma1 (sigma1) receptor in the anti-amnesic, but not antidepressant-like, effects of the aminotetrahydrofuran derivative ANAVEX1-41.

scientific article

Isoform-Specific Biased Agonism of Histamine H3 Receptor Agonists

scientific article published on 18 November 2016

Key interactions by conserved polar amino acids located at the transmembrane helical boundaries in Class B GPCRs modulate activation, effector specificity and biased signalling in the glucagon-like peptide-1 receptor

scientific article

Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists

scientific article published on 4 August 2015

Ligand-Dependent Modulation of G Protein Conformation Alters Drug Efficacy

scientific article published on 6 October 2016

Ligand-Independent Adenosine A2B Receptor Constitutive Activity as a Promoter of Prostate Cancer Cell Proliferation

scientific article published on 20 January 2016

M1 muscarinic allosteric modulators slow prion neurodegeneration and restore memory loss

scientific article

Measurements of ligand bias and functional affinity

scientific article

Mechanisms of ERK1/2 regulation by seven-transmembrane-domain receptors.

scientific article

Mechanistic insights into allosteric structure-function relationships at the M1 muscarinic acetylcholine receptor.

scientific article

Microglial activation and progressive brain changes in schizophrenia

scientific article published on 12 October 2015

Minireview: Signal bias, allosterism, and polymorphic variation at the GLP-1R: implications for drug discovery

scientific article published on 17 July 2013

Modulating receptor function through RAMPs: can they represent drug targets in themselves?

scientific article published on 16 January 2009

Molecular Mechanism of Action of Triazolobenzodiazepinone Agonists of the Type 1 Cholecystokinin Receptor. Possible Cooperativity across the Receptor Homodimeric Complex.

scientific article published on 10 December 2015

Molecular Mechanisms of Action of M5 Muscarinic Acetylcholine Receptor Allosteric Modulators

scientific article published on 26 July 2016

Molecular basis for benzodiazepine agonist action at the type 1 cholecystokinin receptor.

scientific article published on 10 June 2013

Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor.

scientific article published on 17 January 2014

Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptor

scientific article

Murine GPRC6A Mediates Cellular Responses to L-Amino Acids, but Not Osteocalcin Variants

scientific article published on 19 January 2016

Muscarinic M5 receptors modulate ethanol seeking in rats

scientific article published on 5 February 2018

Muscarinic acetylcholine receptors: novel opportunities for drug development

scientific article

Novel Allosteric Modulators of G Protein-coupled Receptors

scientific article

Novel Fused Arylpyrimidinone Based Allosteric Modulators of the M1 Muscarinic Acetylcholine Receptor.

scientific article published on 18 February 2016

Novel GPCR paradigms at the μ-opioid receptor

scientific article

Novel Irreversible Agonists Acting at the A1 Adenosine Receptor

scientific article

Novel persistent activation of muscarinic M1 receptors by xanomeline ⬇️

scientific article published on September 3, 1997

On the mechanism of interaction of potent surmountable and insurmountable antagonists with the prostaglandin D2 receptor CRTH2

scientific article

Orthosteric and allosteric modes of interaction of novel selective agonists of the M1 muscarinic acetylcholine receptor

scientific article published on 22 April 2010

Overview of Receptor Allosterism

scientific article published on 01 December 2010

Pharmacological analysis of the mode of interaction of McN-A-343 at atrial muscarinic M2 receptors ⬇️

scientific article published on November 27, 1997

Pharmacological discrimination of calcitonin receptor: receptor activity-modifying protein complexes

scientific article published on 3 February 2005

Phase-plate cryo-EM structure of a biased agonist-bound human GLP-1 receptor-Gs complex

scientific article published on 21 February 2018

Phase-plate cryo-EM structure of a class B GPCR-G-protein complex

scientific article published on 24 April 2017

Polar transmembrane interactions drive formation of ligand-specific and signal pathway-biased family B G protein-coupled receptor conformations ⬇️

scientific article published on March 11, 2013

Polymorphism and ligand dependent changes in human glucagon-like peptide-1 receptor (GLP-1R) function: allosteric rescue of loss of function mutation.

scientific article

Positive Allosteric Modulation of the Muscarinic M1 Receptor Improves Efficacy of Antipsychotics in Mouse Glutamatergic Deficit Models of Behavior

scientific article published on 14 September 2016

Positive allosteric mechanisms of adenosine A<sub>1</sub> receptor-mediated analgesia

scientific article published on 08 September 2021

Positive and negative allosteric modulators promote biased signaling at the calcium-sensing receptor.

scientific article

Prediction of Loops in G Protein-Coupled Receptor Homology Models: Effect of Imprecise Surroundings and Constraints

scientific article published on 15 March 2016

Probe dependence in the allosteric modulation of a G protein-coupled receptor: implications for detection and validation of allosteric ligand effects

scientific article published on 11 October 2011

Probing structural requirements of positive allosteric modulators of the M4 muscarinic receptor

scientific article

Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonist

scientific article

Prolonged calcitonin receptor signaling by salmon, but not human calcitonin, reveals ligand bias

scientific article

Proof of concept study for designed multiple ligands targeting the dopamine D2, serotonin 5-HT2A, and muscarinic M1 acetylcholine receptors

scientific article published on 30 January 2015

Proposed Mode of Binding and Action of Positive Allosteric Modulators at Opioid Receptors

scientific article published on 03 February 2016

Quantification of adenosine A(1) receptor biased agonism: Implications for drug discovery

scientific article published on 12 November 2015

Quantification of allosteric interactions at G protein-coupled receptors using radioligand binding assays

scientific article published on 01 March 2011

Quantification of functional selectivity at the human α(1A)-adrenoceptor.

scientific article published on 26 October 2010

Quantification of ligand bias for clinically relevant β2-adrenergic receptor ligands: implications for drug taxonomy.

scientific article published on 23 December 2013

RAMPs as Drug Targets ⬇️

scientific article published on January 1, 2012

Recent advances in understanding GLP-1R (glucagon-like peptide-1 receptor) function.

scientific article published on February 2013

Receptor expression modulates calcium-sensing receptor mediated intracellular Ca2+ mobilization

scientific article published on 21 January 2015

Relative affinity of angiotensin peptides and novel ligands at AT1 and AT2 receptors.

scientific article published on October 2011

Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M₁ muscarinic acetylcholine receptor.

scientific article

Reversible and specific extracellular antagonism of receptor-histidine kinase signaling

scientific article published on 03 December 2001

Role of the Second Extracellular Loop of the Adenosine A1 Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity.

scientific article published on 28 September 2016

Roles of intraloops-2 and -3 and the proximal C-terminus in signalling pathway selection from the human calcium-sensing receptor

scientific article published on 28 July 2014

Second extracellular loop of human glucagon-like peptide-1 receptor (GLP-1R) differentially regulates orthosteric but not allosteric agonist binding and function.

scientific article published on 6 December 2011

Second extracellular loop of human glucagon-like peptide-1 receptor (GLP-1R) has a critical role in GLP-1 peptide binding and receptor activation

scientific article published on 6 December 2011

Separation of on-target efficacy from adverse effects through rational design of a bitopic adenosine receptor agonist

scientific article published on 11 March 2014

Signalling bias in new drug discovery: detection, quantification and therapeutic impact.

scientific article published on 15 February 2012

Small molecule allosteric modulation of the glucagon-like Peptide-1 receptor enhances the insulinotropic effect of oxyntomodulin.

scientific article published on 28 August 2012

Small-molecule-biased formyl peptide receptor agonist compound 17b protects against myocardial ischaemia-reperfusion injury in mice.

scientific article published on 07 February 2017

Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor

scientific article

Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs.

scientific article published on 13 October 2013

Structural basis of receptor sulfotyrosine recognition by a CC chemokine: the N-terminal region of CCR3 bound to CCL11/eotaxin-1

scientific article

Structural features embedded in G protein-coupled receptor co-crystal structures are key to their success in virtual screening

scientific article

Structure of the Adenosine A1 Receptor Reveals the Basis for Subtype Selectivity

scientific article published in February 2017

Structure of the adenosine-bound human adenosine A1 receptor–Gi complex

scientific article published in Nature

Structure-Activity Relationships of Pan-Gα Coupled Muscarinic Acetylcholine Receptor Positive Allosteric Modulators

Structure-activity relationships of privileged structures lead to the discovery of novel biased ligands at the dopamine D₂ receptor.

scientific article published on 30 May 2014

Structure-activity study of N-((trans)-4-(2-(7-cyano-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)cyclohexyl)-1H-indole-2-carboxamide (SB269652), a bitopic ligand that acts as a negative allosteric modulator of the dopamine D2 receptor.

scientific article published on 24 June 2015

Structure-function studies of allosteric agonism at M2 muscarinic acetylcholine receptors

scientific article published on 24 May 2007

Structures of the human cholecystokinin 1 (CCK1) receptor bound to Gs and Gq mimetic proteins provide insight into mechanisms of G protein selectivity

scientific article published on 04 June 2021

Structure–Function Studies of Muscarinic Acetylcholine Receptors ⬇️

scientific article published on January 1, 2012

Synthesis and Pharmacological Evaluation of Heterocyclic Carboxamides: Positive Allosteric Modulators of the M1 Muscarinic Acetylcholine Receptor with Weak Agonist Activity and Diverse Modulatory Profiles

scientific article published on 23 March 2018

Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT2C agonists ⬇️

scientific article published on February 9, 2012

Synthesis and characterization of novel 2-amino-3-benzoylthiophene derivatives as biased allosteric agonists and modulators of the adenosine A(1) receptor.

scientific article published on 17 February 2012

Synthesis and pharmacological evaluation of M4 muscarinic receptor positive allosteric modulators derived from VU10004.

scientific article published on 17 April 2015

Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M ₁ muscarinic acetylcholine receptor.

scientific article published on 5 June 2014

Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptor.

scientific article published on 17 June 2013

Systematic analysis of factors influencing observations of biased agonism at the mu-opioid receptor.

scientific article

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview

scientific article published on December 2017

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein-coupled receptors

scientific article published on 01 December 2019

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Introduction and Other Protein Targets

scientific article published on 01 December 2019

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors ⬇️

journal article from 'British Journal of Pharmacology' published in 2021

The Extracellular Surface of the GLP-1 Receptor Is a Molecular Trigger for Biased Agonism

scientific article

The action of a negative allosteric modulator at the dopamine D2 receptor is dependent upon sodium ions

scientific article published on 19 January 2018

The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.

scientific article published in March 2001

The complexity of signalling mediated by the glucagon-like peptide-1 receptor.

scientific article published on April 2016

The effect of social isolation on rat brain expression of genes associated with endocannabinoid signaling.

scientific article published on 27 April 2010

The hybrid molecule, VCP746, is a potent adenosine A2B receptor agonist that stimulates anti-fibrotic signalling

scientific article published on 9 August 2016

The role of kinetic context in apparent biased agonism at GPCRs

scientific article published on 24 February 2016

The role of transmembrane domain 3 in the actions of orthosteric, allosteric, and atypical agonists of the M4 muscarinic acetylcholine receptor.

scientific article published on 7 February 2011

The structural determinants of the bitopic binding mode of a negative allosteric modulator of the dopamine D2 receptor

scientific article published on 8 January 2018

The synthesis and biological evaluation of 2-amino-4,5,6,7,8,9-hexahydrocycloocta[b]thiophenes as allosteric modulators of the A1 adenosine receptor.

scientific article published on 4 May 2011

Towards a structural understanding of allosteric drugs at the human calcium-sensing receptor

scientific article published on 22 March 2016

Towards tissue-specific pharmacology: insights from the calcium-sensing receptor as a paradigm for GPCR (patho)physiological bias

scientific article published on 09 March 2015

Two distinct domains of the glucagon-like peptide-1 receptor control peptide-mediated biased agonism.

scientific article published in May 2018

Tyrosine sulfation of chemokine receptor CCR2 enhances interactions with both monomeric and dimeric forms of the chemokine monocyte chemoattractant protein-1 (MCP-1)

scientific article published on 13 February 2013

Use of Cysteine Trapping to Map Spatial Approximations between Residues Contributing to the Helix N-capping Motif of Secretin and Distinct Residues within Each of the Extracellular Loops of Its Receptor

scientific article published on 6 January 2016

Use of a spreadsheet to quantitate the equilibrium binding of an allosteric modulator ⬇️

scientific article published on August 14, 1998

VCP746, a novel A1 adenosine receptor biased agonist, reduces hypertrophy in a rat neonatal cardiac myocyte model.

scientific article published on 5 July 2016

Paulina is supported by:

About Paulina

Help