List of works - Jacek Stawiński

31P NMR Studies on Oxidative Transformations of Aryl Nucleoside H-Phosphonate Diesters

31P NMR and Computational Studies on Stereochemistry of Conversion of Phosphoramidate Diesters into the Corresponding Phosphotriesters

scientific article published on 01 July 2011

9-Fluorenemethyl H-phosphonoselenoate--a versatile reagent for transferring an H-phosphonoselenoate group

scientific article published in May 2003

A New Reagent System for Efficient Silylation of Alcohols: Silyl Chloride-N-Methylimidazole-Iodine

A cautionary note on the use of the 31P NMR spectroscopy in stereochemical correlation analysis

scientific article

A convenient stereochemical notation for p-chiral nucleotide analogs

scientific article published on 01 March 2007

A new approach to stereospecific synthesis of P-chiral phosphorothioates. Preparation of diastereomeric dithymidyl-(3′-5′) phosphorothioates

scientific article published on 19 December 2003

A new method for the synthesis of nucleoside 2′,3′-O,O-cyclic phosphorodithioates via aryl cyclic phosphites as intermediates

article published in 2001

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 2. Dinucleoside monophosphate analogues

scientific article published in January 2006

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 4. A relationship between the Dp/Lp notation and stereochemistry of reactions

scientific article

A proposal for a convenient notation forP-chiral nucleotide analogues. Part 3. Compounds with one nucleoside residue and nonnucleosidic derivatives

scientific article published on 01 January 2006

A proposal for a new stereochemical notation for P-chiral nucleotide analogues and related compounds

scientific article published in January 2005

ARYL NUCLEOSIDE H-PHOSPHONATES AS A TOOL FOR INVESTIGATION OF STEREOSPECIFICITY DURING COUPLING

scientific article published on 01 January 2005

Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2',3'-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity

scientific article published on 4 June 2015

Aryl H-phosphonates 17: (N-aryl)phosphoramidates of pyrimidine nucleoside analogues and their synthesis, selected properties, and anti-HIV activity

scientific article published on 9 September 2011

Aryl H-phosphonates. 19. New anti-HIV pronucleotide phosphoramidate diesters containing amino- and hydroxypyridine auxiliaries

scientific article published on 17 December 2018

Aryl H-phosphonates. Part IV. A new method for internucleotide bond formation based on transesterification of aryl nucleoside H-phosphonate diesters

article published in 1996

Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 5'-alpha-hydroxyphosphonates

scientific article published on 14 November 2005

Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters

scientific article published on 23 February 2009

ArylH-Phosphonates. 14. Synthesis of New Nucleotide Analogues with Phosphonate−Phosphate Internucleosidic Linkage

scientific article published on 01 October 2003

ArylH-Phosphonates. 6. Synthetic Studies on the Preparation of NucleosideN-Alkyl-H-phosphonamidates

Chemical and Stereochemical Aspects of Oxidative Coupling of HPhosphonate and H-Phosphonothioate Diesters. Reactions with N,N-, N,Oand O,O-Binucleophiles

Chemoselectivity in oxidative coupling of bifunctional nucleophiles with dinucleoside H-phosphonate and dinucleoside H-phosphonothioate diesters

scientific article published on 01 May 2003

Computational Study of the Mechanism and Selectivity of Palladium-Catalyzed Propargylic Substitution with Phosphorus Nucleophiles

scientific article published on 13 August 2012

Controlling stereochemistry during oxidative coupling. Preparation of Rp or Sp phosphoramidates from one P-chiral precursor

scientific article published on 29 September 2004

DEVELOPING SYNTHETIC METHODS FOR BIOACTIVE PHOSPHORUS COMPOUNDS USING H-PHOSPHONATE CHEMISTRY: A PROGRESS REPORT

scientific article published on 01 January 2005

Design, synthesis and QSAR studies of dispiroindole derivatives as new antiproliferative agents.

scientific article published on 11 August 2013

Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report

scientific article published on 01 May 2003

Di- and oligonucleotide synthesis using H-phosphonate chemistry

scientific article published on 01 January 2005

Efficient synthesis of mono- and diarylphosphinic acids: a microwave-assisted palladium-catalyzed cross-coupling of aryl halides with phosphinate

Exploring Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents

H-Phosphonate Chemistry in the Synthesis of Electrically Neutral and Charged Antiviral and Anticancer Pronucleotides

scientific article

H-Phosphonates: Versatile synthetic precursors to biologically active phosphorus compounds

How to get the most out of two phosphorus chemistries. Studies on H-phosphonates

scientific article

Iodine-promoted silylation of alcohols with silyl chlorides. Synthetic and mechanistic studies

Microwave-Assisted Palladium-Catalyzed Cross-Coupling of Aryl and Vinyl Halides with H-Phosphonate Diesters

scientific article published on 23 September 2008

Minimal length of the lactose operator sequence for the specific recognition by the lactose repressor

scientific article

New 3'-O-aromatic acyl-5-fluoro-2'-deoxyuridine derivatives as potential anticancer agents

scientific article published on 04 March 2016

New antiglioma zwitterionic pronucleotides with an FdUMP framework

scientific article published on 21 December 2017

Novel reactivity of Fhit proteins: catalysts for fluorolysis of nucleoside 5'-phosphoramidates and nucleoside 5'-phosphosulfates to generate nucleoside 5'-phosphorofluoridates

scientific article published on 01 June 2015

Novel, Stereoselective and Stereospecific Synthesis of Allenylphosphonates and Related Compounds via Palladium-Catalyzed Propargylic Substitution

Nucleoside 3′,5′-Cyclic H-Phosphonates, New Useful Precursors for the Synthesis of Nucleoside 3′,5′-Cyclic Phosphates and Their Analogues

scientific article published on 01 August 2013

Nucleoside Di- and Triphosphates as a New Generation of Anti-HIV Pronucleotides. Chemical and Biological Aspects

scientific article

Nucleoside H-Phosphonates XX. Efficient Method for the Preparation of Nucleoside H-Phosphonoselenoate Monoesters

Nucleoside H-Phosphonates. 17. Synthetic and (31)P NMR Studies on the Preparation of Dinucleoside H-Phosphonothioates

scientific article published on 01 September 1996

Nucleoside H-phosphonates. III. Chemical synthesis of oligodeoxyribonucleotides by the hydrogenphosphonate approach

scientific article (publication date: 1986)

Nucleoside Phosphonates. Development of Synthetic Methods and Reagents

NucleosideH-Phosphonates. 18. Synthesis of Unprotected Nucleoside 5‘-H-Phosphonates and Nucleoside 5‘-H-Phosphonothioates and Their Conversion into the 5‘-Phosphorothioate and 5‘-Phosphorodithioate Monoesters

O-Silylated C3-halohydrins as a novel class of protected building blocks for total, regio- and stereocontrolled synthesis of glycerolipid frameworks

scientific article published on 26 November 2009

On the Sulfurization ofH-Phosphonate Diesters and Phosphite Triesters Using Elemental Sulfur

Oxidative transformations of nucleoside fluorenemethyl H-phosphonoselenoate diesters

scientific article

Oxyonium phosphobetaines – unusually stable nucleophilic catalyst–phosphate complexes formed from H-phosphonates and N-oxides

scholarly article in RSC Advances, vol. 6 no. 18, 2016

Palladium-Catalyzed C−P Bond Formation: Mechanistic Studies on the Ligand Substitution and the Reductive Elimination. An Intramolecular Catalysis by the Acetate Group in PdIIComplexes

Palladium-catalyzed propargylic substitution with phosphorus nucleophiles: efficient, stereoselective synthesis of allenylphosphonates and related compounds

scientific article published on 01 October 2010

Pd(0)-Catalyzed Phosphorus−Carbon Bond Formation. Mechanistic and Synthetic Studies on the Role of the Palladium Sources and Anionic Additives

Preparation of Arylphosphonates by Palladium(0)-Catalyzed Cross-Coupling in the Presence of Acetate Additives: Synthetic and Mechanistic Studies

Preparation of benzylphosphonates via a palladium(0)-catalyzed cross-coupling of H-phosphonate diesters with benzyl halides. Synthetic and mechanistic studies

Preparation of nucleoside H-phosphonoselenoate monoesters via the phosphinate approach

scientific article published in January 2005

Reaction of Boranephosphonate Diesters with Pyridines or Tertiary Amines in the Presence of Iodine: Synthetic and Mechanistic Studies

scientific article published on 26 February 2020

Reaction of boranephosphonate diesters with amines in the presence of iodine: the case for the intermediacy of H-phosphonate derivatives.

scientific article published on 23 April 2018

Recent Advances in H-Phosphonate Chemistry. Part 2. Synthesis of C-Phosphonate Derivatives

scientific article published on 01 January 2015

Recent advances in H-phosphonate chemistry. Part 1. H-phosphonate esters: synthesis and basic reactions

scientific article

Regioselective and stereospecific acylation across oxirane- and silyloxy systems as a novel strategy to the synthesis of enantiomerically pure mono-, di- and triglycerides

scientific article published on 11 October 2007

Regioselective and stereospecific cleavage of a terminal oxirane system: a novel synthetic approach to lipid mediator congeners--1,2(2,3)-diacyl-3(1)-halo-sn-glycerols.

scientific article

Reinvestigation of the 31P NMR evidence for the formation of diorganyl phosphoropyridinium intermediates

article

Searching for anti-glioma activity. Ribonucleoside analogues with modifications in nucleobase and sugar moieties

scientific article published on 10 November 2016

Silylation-Mediated Transesterification ofO-Phenyl H-Phosphonothioates − A New Entry to Nucleoside H-Phosphonothioate Monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 1. Synthesis and 31P NMR analysis of 16 diribonulceoside (3'-5')-H-phosphonates and the corresponding phosphorothioates

scientific article

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 5. The role of Brønsted and H-bonding base catalysis in ribonucleoside H-phosphonate condensation-chemical and stereochemical consequences

scientific article published on August 2010

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 7. Stereoselective formation of ribonucleoside (RP)- and (SP)-3′-H-phosphonothioate monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 3: Investigations on a mechanism of asymmetric induction

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 6: Optimization of the reaction conditions towards highest stereoselectivity

Stereospecific and regioselective opening of an oxirane system. A new efficient entry to 1- or 3-monoacyl- and 1- or 3-monoalkyl-sn-glycerols

Studies on Oxidative Transformations of Dinucleoside H-Phosphonoselenoates

Studies on aryl H-phosphonates. 3. Mechanistic investigations related to the disproportionation of diphenyl H-phosphonate under anhydrous basic conditions

Studies on aryl H-phosphonates. I. An efficient method for the preparation of deoxyribo- and ribonucleoside 3′-H-phosphonate monoesters by transesterification of diphenyl H-phosphonate

Studies on reactions of nucleoside H-phosphonate diesters with bifunctional reagents. Part 4. Chemoselectivity during oxidative coupling of nucleoside H-phosphonate diesters with amino alcohols controlled by protonation of the amino function

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 1. Reaction with amino alcohols

article published in 1993

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 2. Stability of nucleoside H-phosphonate diesters in the presence of amino alcohols

Studies on the decomposition pathways of diastereoisomeric mixtures of aryl nucleoside α-hydroxyphosphonates under hydrolytic conditions. Synthesis of α-hydroxyphosphonate monoesters

Studies towards synthesis of dinucleoside arylphosphonates with metal complexing properties

scientific article published in May 2003

Synthesis and QSAR study of novel cytotoxic spiro[3H-indole-3,2'(1'H)-pyrrolo[3,4-c]pyrrole]-2,3',5'(1H,2'aH,4'H)-triones.

scientific article

Synthesis of Nucleotide Analogues with Pyridylphosphonate and Pyridylphosphono thio ate Internucleotide Linkages

Synthesis of nucleoside phosphorothio-, phosphorodithio- and phosphoroselenoate diesters via oxidative esterification of the corresponding H-phosphonate analogues

scientific article published on 01 January 2008

Synthesis of oligodeoxyribo- and oligoribonucleotides according to the H-phosphonate method

scientific article published on 01 December 2004

The Case for the Intermediacy of Monomeric Metaphosphate Analogues during Oxidation ofH-Phosphonothioate,H-Phosphonodithioate, andH-Phosphonoselenoate Monoesters: Mechanistic and Synthetic Studies

scientific article published on 29 May 2008

The case of triethylammonium cation loss during purification of certain nucleotide analogues: a cautionary note

scientific article

The influences of a nitrogen atom position in dinucleoside 2-,3-,4-pyridylphosphonates on fragmentation patterns in electrospray ionization multistage tandem mass spectra

scientific article published on 01 January 2006

List of works by Jacek Stawiński

31P NMR Studies on Oxidative Transformations of Aryl Nucleoside H-Phosphonate Diesters

31P NMR and Computational Studies on Stereochemistry of Conversion of Phosphoramidate Diesters into the Corresponding Phosphotriesters

9-Fluorenemethyl H-phosphonoselenoate--a versatile reagent for transferring an H-phosphonoselenoate group

A New Reagent System for Efficient Silylation of Alcohols: Silyl Chloride-N-Methylimidazole-Iodine

A cautionary note on the use of the 31P NMR spectroscopy in stereochemical correlation analysis

A convenient stereochemical notation for p-chiral nucleotide analogs

A new approach to stereospecific synthesis of P-chiral phosphorothioates. Preparation of diastereomeric dithymidyl-(3′-5′) phosphorothioates

A new method for the synthesis of nucleoside 2′,3′-O,O-cyclic phosphorodithioates via aryl cyclic phosphites as intermediates

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 2. Dinucleoside monophosphate analogues

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 4. A relationship between the Dp/Lp notation and stereochemistry of reactions

A proposal for a convenient notation forP-chiral nucleotide analogues. Part 3. Compounds with one nucleoside residue and nonnucleosidic derivatives

A proposal for a new stereochemical notation for P-chiral nucleotide analogues and related compounds

ARYL NUCLEOSIDE H-PHOSPHONATES AS A TOOL FOR INVESTIGATION OF STEREOSPECIFICITY DURING COUPLING

Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2',3'-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity

Aryl H-phosphonates 17: (N-aryl)phosphoramidates of pyrimidine nucleoside analogues and their synthesis, selected properties, and anti-HIV activity

Aryl H-phosphonates. 19. New anti-HIV pronucleotide phosphoramidate diesters containing amino- and hydroxypyridine auxiliaries

Aryl H-phosphonates. Part IV. A new method for internucleotide bond formation based on transesterification of aryl nucleoside H-phosphonate diesters

Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 5'-alpha-hydroxyphosphonates

Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters

ArylH-Phosphonates. 14. Synthesis of New Nucleotide Analogues with Phosphonate−Phosphate Internucleosidic Linkage

ArylH-Phosphonates. 6. Synthetic Studies on the Preparation of NucleosideN-Alkyl-H-phosphonamidates

Chemical and Stereochemical Aspects of Oxidative Coupling of HPhosphonate and H-Phosphonothioate Diesters. Reactions with N,N-, N,Oand O,O-Binucleophiles

Chemoselectivity in oxidative coupling of bifunctional nucleophiles with dinucleoside H-phosphonate and dinucleoside H-phosphonothioate diesters

Computational Study of the Mechanism and Selectivity of Palladium-Catalyzed Propargylic Substitution with Phosphorus Nucleophiles

Controlling stereochemistry during oxidative coupling. Preparation of Rp or Sp phosphoramidates from one P-chiral precursor

DEVELOPING SYNTHETIC METHODS FOR BIOACTIVE PHOSPHORUS COMPOUNDS USING H-PHOSPHONATE CHEMISTRY: A PROGRESS REPORT

Design, synthesis and QSAR studies of dispiroindole derivatives as new antiproliferative agents.

Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report

Di- and oligonucleotide synthesis using H-phosphonate chemistry

Efficient synthesis of mono- and diarylphosphinic acids: a microwave-assisted palladium-catalyzed cross-coupling of aryl halides with phosphinate

Exploring Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents

H-Phosphonate Chemistry in the Synthesis of Electrically Neutral and Charged Antiviral and Anticancer Pronucleotides

H-Phosphonates: Versatile synthetic precursors to biologically active phosphorus compounds

How to get the most out of two phosphorus chemistries. Studies on H-phosphonates

Iodine-promoted silylation of alcohols with silyl chlorides. Synthetic and mechanistic studies

Microwave-Assisted Palladium-Catalyzed Cross-Coupling of Aryl and Vinyl Halides with H-Phosphonate Diesters

Minimal length of the lactose operator sequence for the specific recognition by the lactose repressor

New 3'-O-aromatic acyl-5-fluoro-2'-deoxyuridine derivatives as potential anticancer agents

New antiglioma zwitterionic pronucleotides with an FdUMP framework

Novel reactivity of Fhit proteins: catalysts for fluorolysis of nucleoside 5'-phosphoramidates and nucleoside 5'-phosphosulfates to generate nucleoside 5'-phosphorofluoridates

Novel, Stereoselective and Stereospecific Synthesis of Allenylphosphonates and Related Compounds via Palladium-Catalyzed Propargylic Substitution

Nucleoside 3′,5′-Cyclic H-Phosphonates, New Useful Precursors for the Synthesis of Nucleoside 3′,5′-Cyclic Phosphates and Their Analogues

Nucleoside Di- and Triphosphates as a New Generation of Anti-HIV Pronucleotides. Chemical and Biological Aspects

Nucleoside H-Phosphonates XX. Efficient Method for the Preparation of Nucleoside H-Phosphonoselenoate Monoesters

Nucleoside H-Phosphonates. 17. Synthetic and (31)P NMR Studies on the Preparation of Dinucleoside H-Phosphonothioates

Nucleoside H-phosphonates. III. Chemical synthesis of oligodeoxyribonucleotides by the hydrogenphosphonate approach

Nucleoside Phosphonates. Development of Synthetic Methods and Reagents

NucleosideH-Phosphonates. 18. Synthesis of Unprotected Nucleoside 5‘-H-Phosphonates and Nucleoside 5‘-H-Phosphonothioates and Their Conversion into the 5‘-Phosphorothioate and 5‘-Phosphorodithioate Monoesters

O-Silylated C3-halohydrins as a novel class of protected building blocks for total, regio- and stereocontrolled synthesis of glycerolipid frameworks

On the Sulfurization ofH-Phosphonate Diesters and Phosphite Triesters Using Elemental Sulfur

Oxidative transformations of nucleoside fluorenemethyl H-phosphonoselenoate diesters

Oxyonium phosphobetaines – unusually stable nucleophilic catalyst–phosphate complexes formed from H-phosphonates and N-oxides

Palladium-Catalyzed C−P Bond Formation: Mechanistic Studies on the Ligand Substitution and the Reductive Elimination. An Intramolecular Catalysis by the Acetate Group in PdIIComplexes

Palladium-catalyzed propargylic substitution with phosphorus nucleophiles: efficient, stereoselective synthesis of allenylphosphonates and related compounds

Pd(0)-Catalyzed Phosphorus−Carbon Bond Formation. Mechanistic and Synthetic Studies on the Role of the Palladium Sources and Anionic Additives

Preparation of Arylphosphonates by Palladium(0)-Catalyzed Cross-Coupling in the Presence of Acetate Additives: Synthetic and Mechanistic Studies

Preparation of benzylphosphonates via a palladium(0)-catalyzed cross-coupling of H-phosphonate diesters with benzyl halides. Synthetic and mechanistic studies

Preparation of nucleoside H-phosphonoselenoate monoesters via the phosphinate approach

Reaction of Boranephosphonate Diesters with Pyridines or Tertiary Amines in the Presence of Iodine: Synthetic and Mechanistic Studies

Reaction of boranephosphonate diesters with amines in the presence of iodine: the case for the intermediacy of H-phosphonate derivatives.

Recent Advances in H-Phosphonate Chemistry. Part 2. Synthesis of C-Phosphonate Derivatives

Recent advances in H-phosphonate chemistry. Part 1. H-phosphonate esters: synthesis and basic reactions

Regioselective and stereospecific acylation across oxirane- and silyloxy systems as a novel strategy to the synthesis of enantiomerically pure mono-, di- and triglycerides

Regioselective and stereospecific cleavage of a terminal oxirane system: a novel synthetic approach to lipid mediator congeners--1,2(2,3)-diacyl-3(1)-halo-sn-glycerols.

Reinvestigation of the 31P NMR evidence for the formation of diorganyl phosphoropyridinium intermediates

Searching for anti-glioma activity. Ribonucleoside analogues with modifications in nucleobase and sugar moieties

Silylation-Mediated Transesterification ofO-Phenyl H-Phosphonothioates − A New Entry to Nucleoside H-Phosphonothioate Monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 1. Synthesis and 31P NMR analysis of 16 diribonulceoside (3'-5')-H-phosphonates and the corresponding phosphorothioates

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 5. The role of Brønsted and H-bonding base catalysis in ribonucleoside H-phosphonate condensation-chemical and stereochemical consequences

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 7. Stereoselective formation of ribonucleoside (RP)- and (SP)-3′-H-phosphonothioate monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 3: Investigations on a mechanism of asymmetric induction

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 6: Optimization of the reaction conditions towards highest stereoselectivity

Stereospecific and regioselective opening of an oxirane system. A new efficient entry to 1- or 3-monoacyl- and 1- or 3-monoalkyl-sn-glycerols

Studies on Oxidative Transformations of Dinucleoside H-Phosphonoselenoates

Studies on aryl H-phosphonates. 3. Mechanistic investigations related to the disproportionation of diphenyl H-phosphonate under anhydrous basic conditions

Studies on aryl H-phosphonates. I. An efficient method for the preparation of deoxyribo- and ribonucleoside 3′-H-phosphonate monoesters by transesterification of diphenyl H-phosphonate

Studies on reactions of nucleoside H-phosphonate diesters with bifunctional reagents. Part 4. Chemoselectivity during oxidative coupling of nucleoside H-phosphonate diesters with amino alcohols controlled by protonation of the amino function

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 1. Reaction with amino alcohols

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 2. Stability of nucleoside H-phosphonate diesters in the presence of amino alcohols