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List of works by Yesim A Tahirovic

An NMDAR positive and negative allosteric modulator series share a binding site and are interconverted by methyl groups.

scientific article published on 24 May 2018

CCR5 receptor antagonists in preclinical to phase II clinical development for treatment of HIV.

scientific article published on 28 October 2016

Context-dependent GluN2B-selective inhibitors of NMDA receptor function are neuroprotective with minimal side effects

scientific article

Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties

scientific article published on 15 August 2018

Discovery of N-Alkyl Piperazine Side Chain Based CXCR4 Antagonists with Improved Drug-like Properties

scientific article published on 09 April 2018

Discovery of Tetrahydroisoquinoline-Containing CXCR4 Antagonists with Improved in Vitro ADMET Properties.

scientific article

Enantiomeric propanolamines as selective N-methyl-D-aspartate 2B receptor antagonists.

scientific article

Small molecule and peptide-based CXCR4 modulators as therapeutic agents. A patent review for the period from 2010 to 2018

scientific article published on 07 January 2020

Structural elements of a pH-sensitive inhibitor binding site in NMDA receptors

scientific article published in Nature Communications

Synthesis and SAR of 1,2,3,4-Tetrahydroisoquinoline-Based CXCR4 Antagonists

scientific article published on 8 December 2017

Synthesis of Novel Tetrahydroisoquinoline CXCR4 Antagonists with Rigidified Side-Chains.

scientific article published on 20 December 2017

Synthesis, structural activity-relationships, and biological evaluation of novel amide-based allosteric binding site antagonists in NR1A/NR2B N-methyl-D-aspartate receptors

scientific article

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