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List of works by Stephan Kopp

A subset of highly effective propafenone-type multidrug resistance modulators lacks effects on cardiac action potential and mechanical twitch parameters of rat papillary muscles

scientific article published on 9 September 2003

A three-dimensional model for the substrate binding domain of the multidrug ATP binding cassette transporter LmrA.

scientific article published on 10 August 2004

Identification of ligand-binding regions of P-glycoprotein by activated-pharmacophore photoaffinity labeling and matrix-assisted laser desorption/ionization-time-of-flight mass spectrometry.

scientific article

In silico screening with benzofurane- and benzopyrane-type MDR-modulators

scientific article published on March 2003

Intramolecular distribution of hydrophobicity influences pharmacological activity of propafenone-type MDR modulators

scientific article published on June 2004

Multispecificity of drug transporters: probing inhibitor selectivity for the human drug efflux transporters ABCB1 and ABCG2.

scientific article published on December 2007

P-glycoprotein substrate binding domains are located at the transmembrane domain/transmembrane domain interfaces: a combined photoaffinity labeling-protein homology modeling approach

scientific article published on 27 October 2004

Role of transmembrane domain/transmembrane domain interfaces of P-glycoprotein (ABCB1) in solute transport. Convergent information from photoaffinity labeling, site directed mutagenesis and in silico importance prediction

scientific article published on January 2006

Self-organizing maps for identification of new inhibitors of P-glycoprotein

scientific article

Similarity based SAR (SIBAR) as tool for early ADME profiling

scientific article