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List of works by Guillermina Estiu

A molecular mechanism of artemisinin resistance in Plasmodium falciparum malaria

scientific article (publication date: 30 April 2015)

Computational studies of the cholesterol transport between NPC2 and the N-terminal domain of NPC1 (NPC1(NTD))

scientific article published on 19 September 2013

Design and synthesis of a crosslinker for studying intracellular steroid trafficking pathways

scientific article published on 27 March 2015

Discovery of selective small-molecule HDAC6 inhibitor for overcoming proteasome inhibitor resistance in multiple myeloma

scientific article

Identifying Ligand Binding Conformations of the β2-Adrenergic Receptor by Using Its Agonists as Computational Probes

scientific article published on December 31, 2012

On the inhibition of histone deacetylase 8

scientific article published on 3 April 2010

Residues in the 11 A channel of histone deacetylase 1 promote catalytic activity: implications for designing isoform-selective histone deacetylase inhibitors

scientific article published on 27 August 2008

Structural origin of selectivity in class II-selective histone deacetylase inhibitors

scientific article published on 16 April 2008

Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs

scientific article published on 18 June 2013

Synthesis and conformation-activity relationships of the peptide isosteres of FK228 and largazole

scientific article

Synthesis and modeling of new benzofuranone histone deacetylase inhibitors that stimulate tumor suppressor gene expression

scientific article published in May 2009

The cytoplasmic prolyl-tRNA synthetase of the malaria parasite is a dual-stage target of febrifugine and its analogs

scientific article