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List of works by Jean-Robert Ioset

A Sample-Centric and Knowledge-Driven Computational Framework for Natural Products Drug Discovery ⬇️

Absolute configuration of a tetrahydrophenanthrene from Heliotropium ovalifolium by LC-NMR of its Mosher esters.

scientific article published in January 2003

Addressing the Most Neglected Diseases through an Open Research Model: the Discovery of Fenarimols as Novel Drug Candidates for Eumycetoma

Addressing the most neglected diseases through an open research model: The discovery of fenarimols as novel drug candidates for eumycetoma.

scientific article published on 26 April 2018

An LC/DAD-UV/MS method for the rapid detection of aristolochic acid in plant preparations

scientific article published in September 2002

Antileishmanial activities associated with plants used in the Malian traditional medicine

scientific article published on 06 October 2006

Antileishmanial and antifungal acridone derivatives from the roots of Thamnosma rhodesica

scientific article published in April 2004

Antiprotozoal Activity Profiling of Approved Drugs: A Starting Point toward Drug Repositioning

scientific article

Assessing anti-T. cruzi candidates in vitro for sterile cidality

scientific article published on 26 August 2016

Bio-guided isolation of cholinesterase inhibitors from the bulbs of Crinum x powellii

scientific article published in November 2005

Catechol pyrazolinones as trypanocidals: fragment-based design, synthesis, and pharmacological evaluation of nanomolar inhibitors of trypanosomal phosphodiesterase B1

article

Complete LC/MS analysis of a Tinnevelli senna pod extract and subsequent isolation and identification of two new benzophenone glucosides

scientific article published in April 2002

Correction: Identification of Compounds with Anti-Proliferative Activity against Strain 427 by a Whole Cell Viability Based HTS Campaign

Development and Validation of a Novel Leishmania donovani Screening Cascade for High-Throughput Screening Using a Novel Axenic Assay with High Predictivity of Leishmanicidal Intracellular Activity.

scientific article

Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation

scientific article published on 24 August 2015

Drug discovery and development for neglected diseases: the DNDi model

scientific article

Drugs for Neglected Diseases initiative model of drug development for neglected diseases: current status and future challenges

scientific article published on September 2011

Ellagic acid derivatives from Syzygium cumini stem bark: investigation of their antiplasmodial activity.

scientific article

Evaluation of Parameters Impacting Drug Susceptibility in Intracellular Trypanosoma cruzi Assay Protocols

scientific article published on 13 October 2016

Flavonoid profiling among wild type and related GM wheat varieties

article

Four new sesquiterpenoid derivatives from the heartwood of Mansonia gagei

scientific article published in September 2002

Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign

scientific article

Identification of two isomeric meroterpenoid naphthoquinones fromCordia linnaei by liquid chromatography-mass spectrometry and liquid chromatography-nuclear magnetic resonance spectroscopy

article

Limonoid orthoacetates and antiprotozoal compounds from the roots of Pseudocedrela kotschyi

scientific article published on January 2007

Novel 3-nitro-1H-1,2,4-triazole-based amides and sulfonamides as potential antitrypanosomal agents

scientific article published on 23 May 2012

Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents

scientific article published on 20 August 2013

Novel 3-nitrotriazole-based amides and carbinols as bifunctional antichagasic agents

scientific article

Novel benzoxaborole, nitroimidazole and aminopyrazoles with activity against experimental cutaneous leishmaniasis

scientific article published on 26 February 2019

On-line characterisation of apple polyphenols by liquid chromatography coupled with mass spectrometry and ultraviolet absorbance detection

scientific article

Phenotypic screening approaches for Chagas disease drug discovery

scientific article published on 13 December 2017

Qualitative and quantitative determination of yohimbine in authentic yohimbe bark and in commercial aphrodisiacs by HPLC-UV-API/ MS methods

scientific article

Repurposing of the Open Access Malaria Box for Kinetoplastid Diseases Identifies Novel Active Scaffolds against Trypanosomatids

scientific article

Screening strategies to identify new chemical diversity for drug development to treat kinetoplastid infections

scientific article

Selection and optimization of hits from a high-throughput phenotypic screen against Trypanosoma cruzi.

scientific article published on October 2013

Simple field assays to check quality of current artemisinin-based antimalarial combination formulations

scientific article

Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals

scientific article

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