List of works - Maria Camilla Cerlesi

A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism

scientific article

A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.

scientific article published on 13 May 2014

Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo).

scientific article

Correction for "Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines".

scientific article published on 9 May 2016

Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues

scientific article

In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations.

scientific article published on 22 October 2016

Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist

scientific article published on 02 August 2016

Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues.

scientific article published on 13 March 2014

Pharmacological characterization of tachykinin tetrabranched derivatives

scientific article

Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt1]N/OFQ(1-13).

scientific article

Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic

scientific article

Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity.

scientific article published in June 2015

Structure activity studies of nociceptin/orphanin FQ(1-13)-NH2 derivatives modified in position 5.

scientific article

Structure- and conformation-activity studies of nociceptin/orphanin FQ receptor dimeric ligands

scientific article published on 06 April 2017

Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids

scientific article published on 3 August 2017

Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration

scientific article published on 12 December 2015

Synthesis of mixed opioid affinity cyclic endomorphin-2 analogues with fluorinated phenylalanines

scientific article published on 3 April 2015

Synthesis, biological evaluation and structural analysis of novel peripherally active morphiceptin analogs

scientific article published on 26 February 2016

List of works by Maria Camilla Cerlesi

A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism

A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.

Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo).

Correction for "Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines".

Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues

In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations.

Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist

Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues.

Pharmacological characterization of tachykinin tetrabranched derivatives

Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt1]N/OFQ(1-13).

Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic

Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity.

Structure activity studies of nociceptin/orphanin FQ(1-13)-NH2 derivatives modified in position 5.

Structure- and conformation-activity studies of nociceptin/orphanin FQ receptor dimeric ligands

Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids

Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration

Synthesis of mixed opioid affinity cyclic endomorphin-2 analogues with fluorinated phenylalanines

Synthesis, biological evaluation and structural analysis of novel peripherally active morphiceptin analogs

Synthesis, enantiomeric separation and docking studies of spiropiperidine analogues as ligands of the nociceptin/orphanin FQ receptor