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List of works by Michel Detheux

A natural ligand for the orphan receptor GPR15 modulates lymphocyte recruitment to epithelia

scientific article published on 12 September 2017

Adaptation of aequorin functional assay to high throughput screening

scientific article published in February 2002

Aequorin-Based Functional Assays for G-Protein-Coupled Receptors, Ion Channels, and Tyrosine Kinase Receptors ⬇️

scientific article published on January 1, 2002

Analysis of C-terminally substituted tachykinin-like peptide agonists by means of aequorin-based luminescent assays for human and insect neurokinin receptors

scientific article

Design and in vitro characterization of PAC1/VPAC1-selective agonists with potent neuroprotective effects

scientific article

Design, Synthesis, and Structure−Activity Relationships of Novel Bicyclic Azole-amines as Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5 ⬇️

scientific article published on October 14, 2010

Distinct recognition of OX1 and OX2 receptors by orexin peptides.

scientific article

Functional analysis of synthetic insectatachykinin analogs on recombinant neurokinin receptor expressing cell lines

scientific article published on November 2002

Functional characterization of human receptors for short chain fatty acids and their role in polymorphonuclear cell activation

scientific article (publication date: 11 July 2003)

Identification and characterization of an endogenous chemotactic ligand specific for FPRL2

scientific article

Identification of a binding domain of the endothelin-B receptor using a selective IRL-1620-derived photoprobe

scientific article published in September 2004

Identification of natural ligands for the orphan G protein-coupled receptors GPR7 and GPR8

scientific article

Oxysterols direct immune cell migration via EBI2 ⬇️

scientific article published on July 27, 2011

PTHrP fragments 1-16 and 1-23 do not bind to either the ETA or the ETB endothelin receptors

scientific article published on 20 April 2005

Pharmacological characterization of human NPFF(1) and NPFF(2) receptors expressed in CHO cells by using NPY Y(1) receptor antagonists

scientific article (publication date: 20 September 2002)

Preclinical assessment of a novel small molecule inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1).

scientific article published on 6 November 2014

Preclinical assessment of a novel small molecule inhibitor of tryptophan 2,3-dioxygenase 2 (TDO2)

Recombinant aequorin as a reporter for receptor-mediated changes of intracellular Ca2+ -levels in Drosophila S2 cells

scientific article published on November 2001

Serotonin 5-HT(2B) receptor loss of function mutation in a patient with fenfluramine-associated primary pulmonary hypertension.

scientific article

Significance of N-terminal proteolysis of CCL14a to activity on the chemokine receptors CCR1 and CCR5 and the human cytomegalovirus-encoded chemokine receptor US28.

scientific article

Specific recruitment of antigen-presenting cells by chemerin, a novel processed ligand from human inflammatory fluids

scientific article

Substitution of conserved glycine residue by alanine in natural and synthetic neuropeptide ligands causes partial agonism at the stomoxytachykinin receptor.

scientific article published on July 2004

Transmembrane domain V of the endothelin-A receptor is a binding domain of ETA-selective TTA-386-derived photoprobes

scientific article published in May 2005

Vasopressin-like peptide and its receptor function in an indirect diuretic signaling pathway in the red flour beetle

scientific article published on 10 May 2008

iTeos Therapeutics.

scientific article published on 6 June 2017

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