Search filters

List of works by Pravin S Shirude

1,4-azaindole, a potential drug candidate for treatment of tuberculosis

scientific article

Alkylidene Oxapenem β-Lactamase Inhibitors Revisited: Potent Broad Spectrum Activity but New Stability Challenges

scientific article published on 20 June 2014

Aminopyrazinamides: Novel and Specific GyrB Inhibitors that Kill Replicating and Nonreplicating Mycobacterium tuberculosis ⬇️

scientific article published on December 31, 2012

Azaindoles: noncovalent DprE1 inhibitors from scaffold morphing efforts, kill Mycobacterium tuberculosis and are efficacious in vivo.

scientific article published on 21 November 2013

Challenges and opportunities in tuberculosis drug discovery: an industry perspective

scientific article published in April 2013

Diarylethynyl amides that recognize the parallel conformation of genomic promoter DNA G-quadruplexes

scientific article published on November 2008

Discovery of pyrazolopyridones as a novel class of noncovalent DprE1 inhibitor with potent anti-mycobacterial activity

scientific article published on 22 May 2014

Ensemble and single molecule FRET analysis of the structure and unfolding kinetics of the c-kit promoter quadruplexes

scientific article

G-quadruplex DNA bound by a synthetic ligand is highly dynamic

scientific article published on September 2009

G-quadruplex recognition by bis-indole carboxamides

scientific article published on 5 June 2008

Impact of CO2-solvent separators on the degradation of benzyl-2,3-dihydroxypiperidine-1-carboxylate during preparative supercritical fluid chromatographic (SFC) purification

scientific article published on 14 November 2017

Lead optimization of 1,4-azaindoles as antimycobacterial agents

scientific article published on 20 June 2014

Macrocyclic and helical oligoamides as a new class of G-quadruplex ligands

scientific article

Methyl-thiazoles: a novel mode of inhibition with the potential to develop novel inhibitors targeting InhA in Mycobacterium tuberculosis

scientific article

Oxazole-based peptide macrocycles: a new class of G-quadruplex binding ligands

scientific article published on October 2006

Quinolinyl Pyrimidines: Potent Inhibitors of NDH-2 as a Novel Class of Anti-TB Agents

scientific article

Rigid cyanine dye nucleic acid labels

scientific article published on 26 March 2008

Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity

scientific article published on 23 September 2019

Single molecule conformational analysis of DNA G-quadruplexes

scientific article published on 06 February 2008

Single molecule conformational analysis of the biologically relevant DNA G-quadruplex in the promoter of the proto-oncogene c-MYC.

scientific article published on 20 March 2008

Single-molecule conformational analysis of G-quadruplex formation in the promoter DNA duplex of the proto-oncogene c-kit.

scientific article

Synthesis of aqueous Au core-Ag shell nanoparticles using tyrosine as a pH-dependent reducing agent and assembling phase-transferred silver nanoparticles at the air-water interface.

scientific article

Synthesis of bis-indole carboxamides as G-quadruplex stabilizing and inducing ligands.

scientific article

Triarylpyridines: a versatile small molecule scaffold for G-quadruplex recognition

scientific article published on 29 January 2008

Trisubstituted isoalloxazines as a new class of G-quadruplex binding ligands: small molecule regulation of c-kit oncogene expression

scientific article published on 5 October 2007

Paulina is supported by:

About Paulina

Help