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List of works by Jesper Lau

Differential structural properties of GLP-1 and exendin-4 determine their relative affinity for the GLP-1 receptor N-terminal extracellular domain

scientific article

Discovery of the Once-Weekly Glucagon-Like Peptide-1 (GLP-1) Analogue Semaglutide

scientific article

Human glucagon receptor antagonists based on alkylidene hydrazides

scientific article published in February 2002

Human glucagon receptor antagonists with thiazole cores. A novel series with superior pharmacokinetic properties.

scientific article published in May 2009

New beta-alanine derivatives are orally available glucagon receptor antagonists

scientific article

Novel glucagon receptor antagonists with improved selectivity over the glucose-dependent insulinotropic polypeptide receptor.

scientific article

Optimization of alkylidene hydrazide based human glucagon receptor antagonists. Discovery of the highly potent and orally available 3-cyano-4-hydroxybenzoic acid [1-(2,3,5,6-tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide.

scientific article

Small molecule ago-allosteric modulators of the human glucagon-like peptide-1 (hGLP-1) receptor

article

Small-molecule agonists for the glucagon-like peptide 1 receptor

scholarly article

The Discovery and Development of Liraglutide and Semaglutide

article

Transmembrane α-Helix 2 and 7 Are Important for Small Molecule-Mediated Activation of the GLP-1 Receptor

scientific article published on 30 November 2011

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