List of works - Joachim Jose

1H and 13C NMR assignments of bioactive indeno[1,2-b]indole-10-one derivatives.

scientific article

A CE-based assay for human protein kinase CK2 activity measurement and inhibitor screening

scientific article published in January 2010

A FRET-based microplate assay for human protein kinase CK2, a target in neoplastic disease

scientific article published in April 2010

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds.

scientific article published on 3 April 2014

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.

scientific article published on 16 October 2014

Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery

scientific article

Identification of novel CK2 inhibitors with a benzofuran scaffold by novel non-radiometric in vitro assays

scientific article

Improved Surface Display of Human Hyal1 and Identification of Testosterone Propionate and Chicoric Acid as New Inhibitors

scientific article published on 26 March 2020

Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors.

scientific article

Indenoindoles and cyclopentacarbazoles as bioactive compounds: synthesis and biological applications.

scientific article published on 16 September 2013

Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion

scientific article published on 05 October 2020

Novel indeno[1,2-b]indoloquinones as inhibitors of the human protein kinase CK2 with antiproliferative activity towards a broad panel of cancer cell lines

scientific article published on 21 June 2012

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

scientific article published on 3 July 2015

Preparation and characterization of CK2 inhibitor-loaded cyclodextrin nanoparticles for drug delivery

scientific article published on 13 November 2012

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light

scientific article

Synthesis and biological evaluation of novel substituted pyrrolo[1,2-a]quinoxaline derivatives as inhibitors of the human protein kinase CK2.

scientific article published on 3 May 2013

Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2.

scientific article published on 8 June 2015

TF--a novel cell-permeable and selective inhibitor of human protein kinase CK2 induces apoptosis in the prostate cancer cell line LNCaP.

scientific article

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2

scientific article published on 12 November 2020

List of works by Joachim Jose

1H and 13C NMR assignments of bioactive indeno[1,2-b]indole-10-one derivatives.

A CE-based assay for human protein kinase CK2 activity measurement and inhibitor screening

A FRET-based microplate assay for human protein kinase CK2, a target in neoplastic disease

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds.

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.

Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery

Identification of novel CK2 inhibitors with a benzofuran scaffold by novel non-radiometric in vitro assays

Improved Surface Display of Human Hyal1 and Identification of Testosterone Propionate and Chicoric Acid as New Inhibitors

Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors.

Indenoindoles and cyclopentacarbazoles as bioactive compounds: synthesis and biological applications.

Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion

Novel indeno[1,2-b]indoloquinones as inhibitors of the human protein kinase CK2 with antiproliferative activity towards a broad panel of cancer cell lines

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Preparation and characterization of CK2 inhibitor-loaded cyclodextrin nanoparticles for drug delivery

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light

Synthesis and biological evaluation of novel substituted pyrrolo[1,2-a]quinoxaline derivatives as inhibitors of the human protein kinase CK2.

Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2.

TF--a novel cell-permeable and selective inhibitor of human protein kinase CK2 induces apoptosis in the prostate cancer cell line LNCaP.

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2