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List of works by Lionel Trottet

Corrigendum to 'Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors' [Bioorg. Med. Chem. Lett. 29 (2019) 126675]

scientific article published on 16 December 2019

Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors

scientific article published on 07 September 2019

Development of a Series of Kynurenine 3-Monooxygenase Inhibitors Leading to a Clinical Candidate for the Treatment of Acute Pancreatitis.

scientific article

Discovery of Pyridones As Oral AMPK Direct Activators

scientific article

Effects of membrane type and liquid/liquid phase boundary on in vitro release of ketoprofen from gel formulations

scientific article

Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening

scientific article

Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2).

scientific article published on 18 November 2016

From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151.

scientific article

Ketoprofen: release from, permeation across and rheology of simple gel formulations that simulate increasing dryness

scientific article

Kynurenine-3-monooxygenase inhibition prevents multiple organ failure in rodent models of acute pancreatitis

scientific article

Myelination induction by a histamine H3 receptor antagonist in a mouse model of preterm white matter injury

scientific article published on 12 September 2018

Naphthyridines as novel BET family bromodomain inhibitors

scientific article

The discovery of I-BET726 (GSK1324726A), a potent tetrahydroquinoline ApoA1 up-regulator and selective BET bromodomain inhibitor

scientific article

The discovery of potent and selective kynurenine 3-monooxygenase inhibitors for the treatment of acute pancreatitis

scientific article published on 09 March 2017

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