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List of works by Demetris P Papahatjis

(R)-N-(1-Methyl-2-hydroxyethyl)-13-(S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes

scientific article published on 21 September 2018

Addendum: Oil-In-Water Microemulsions as Hosts for Benzothiophene-Based Cytotoxic Compounds: An Effective Combination. 2018, , 13

scientific article published on 25 October 2018

C1'-cycloalkyl side chain pharmacophore in tetrahydrocannabinols

scientific article

Cannabilactones: a novel class of CB2 selective agonists with peripheral analgesic activity

scientific article

Combined 3D QSAR and molecular docking studies to reveal novel cannabinoid ligands with optimum binding activity

scientific article

DPS-2: A Novel Dual MEK/ERK and PI3K/AKT Pathway Inhibitor with Powerful Ex Vivo and In Vivo Anticancer Properties

Design and synthesis of (13S)-methyl-substituted arachidonic acid analogues: templates for novel endocannabinoids

scientific article published on April 2010

Mapping the melatonin receptor. 7. Subtype selective ligands based on beta-substituted N-acyl-5-methoxytryptamines and beta-substituted N-acyl-5-methoxy-1-methyltryptamines

scientific article published on June 2006

Novel 1',1'-chain substituted Delta(8)-tetrahydrocannabinols

scientific article

Novel 1',1'-chain substituted hexahydrocannabinols: 9β-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist.

scientific article

Oil-In-Water Microemulsions as Hosts for Benzothiophene-Based Cytotoxic Compounds: An Effective Combination

scientific article published on 16 June 2018

Pharmacophoric requirements for the cannabinoid side chain. Probing the cannabinoid receptor subsite at C1'.

scientific article

Structural modifications of the cannabinoid side chain towards C3-aryl and 1',1'-cycloalkyl-1'-cyano cannabinoids

scientific article published on 4 January 2006

The application of 3D-QSAR studies for novel cannabinoid ligands substituted at the C1' position of the alkyl side chain on the structural requirements for binding to cannabinoid receptors CB1 and CB2.

scientific article

The cannabinoid CB1 receptor biphasically modulates motor activity and regulates dopamine and glutamate release region dependently

scientific article published on March 6, 2012

The role of halogen substitution in classical cannabinoids: a CB1 pharmacophore model

scientific article published on 19 October 2004