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List of works by Isabella Pugliesi

3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one, a novel adenosine receptor antagonist with A(2A)-mediated neuroprotective effects

scientific article

3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists

scientific article published on 7 February 2012

A3 receptor ligands: past, present and future trends

scientific article published on January 2010

Allosteric modulators of human A2B adenosine receptor

scientific article published on 19 December 2013

Arylthioamides as H2S Donors: l-Cysteine-Activated Releasing Properties and Vascular Effects in Vitro and in Vivo

scientific article

Derivatives of Benzimidazol-2-ylquinoline and Benzimidazol-2-ylisoquinoline as Selective A1 Adenosine Receptor Antagonists with Stimulant Activity on Human Colon Motility

scientific article published on 27 July 2011

Evaluation of novel N1-methyl-2-phenylindol-3-ylglyoxylamides as a new chemotype of 18 kDa translocator protein-selective ligand suitable for the development of positron emission tomography radioligands

scientific article

Identification of novel molecular scaffolds for the design of MMP-13 inhibitors: A first round of lead optimization

article

Medicinal chemistry of indolylglyoxylamide TSPO high affinity ligands with anxiolytic-like effects.

scientific article published on January 2012

Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives

scientific article published on 8 September 2013

Novel irreversible fluorescent probes targeting the 18 kDa translocator protein: synthesis and biological characterization.

scientific article

Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors

scientific article published on 16 September 2013

Structural requirements to obtain highly potent and selective 18 kDa Translocator Protein (TSPO) Ligands.

scientific article published on January 2011

Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein

scientific article

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