List of works - Basile Peres

6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein

scientific article published on 21 May 2012

ABCG2: recent discovery of potent and highly selective inhibitors

scientific article published on June 2013

Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations

scientific article published on 31 July 2020

Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens

scientific article published on 11 January 2019

Biomimetic synthesis of Tramadol

scientific article published in 2015

Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2

scientific article published on 05 July 2020

Design, synthesis and biological evaluation of novel ring-opened cromakalim analogues with relaxant effects on vascular and respiratory smooth muscles and as stimulators of elastin synthesis

scientific article

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands

scientific article

Ferrocene-embedded flavonoids targeting the Achilles heel of multidrug-resistant cancer cells through collateral sensitivity

scientific article published on March 2017

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

scientific article

Make azoles active again: chalcones as potent reversal agents of transporters-mediated resistance in Candida albicans

scientific article published on 25 July 2018

Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1

scientific article published on 06 May 2020

New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2.

scientific article published on 27 June 2016

Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2

scientific article published on 10 October 2019

Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models

scientific article published on 12 September 2018

Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2.

scientific article published on 13 December 2013

Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein

scientific article published on 06 January 2012

Synthesis and pharmacological evaluation of a series of the agomelatine analogues as melatonin MT1 /MT2 agonist and 5-HT2C antagonist

scientific article published on 12 September 2013

Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II).

scientific article published on 13 December 2014

Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands.

scientific article published on 27 August 2008

Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review ⬇️

scientific article published on 15 October 2017

Two independent ways of preparing hypercharged hydrolyzable polyaminorotaxane

scientific article published on 3 June 2008

List of works by Basile Peres

6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein

ABCG2: recent discovery of potent and highly selective inhibitors

Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations

Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens

Biomimetic synthesis of Tramadol

Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2

Design, synthesis and biological evaluation of novel ring-opened cromakalim analogues with relaxant effects on vascular and respiratory smooth muscles and as stimulators of elastin synthesis

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands

Ferrocene-embedded flavonoids targeting the Achilles heel of multidrug-resistant cancer cells through collateral sensitivity

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

Make azoles active again: chalcones as potent reversal agents of transporters-mediated resistance in Candida albicans

Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1

New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2.

Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2

Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models

Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2.

Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein

Synthesis and pharmacological evaluation of a series of the agomelatine analogues as melatonin MT1 /MT2 agonist and 5-HT2C antagonist

Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II).

Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands.

Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review ⬇️

Two independent ways of preparing hypercharged hydrolyzable polyaminorotaxane