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List of works by Charlotte Gauthier

6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein

scientific article published on 21 May 2012

A Synthetic Chalcone as a Potent Inducer of Glutathione Biosynthesis

scientific article published on January 30, 2012

ABCG2 is not able to catalyze glutathione efflux and does not contribute to GSH-dependent collateral sensitivity

scientific article

ABCG2: recent discovery of potent and highly selective inhibitors

scientific article published on June 2013

Investigation of chalcones as selective inhibitors of the breast cancer resistance protein: critical role of methoxylation in both inhibition potency and cytotoxicity

scientific article published on 02 April 2012

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

scientific article

Methoxy stilbenes as potent, specific, untransported, and noncytotoxic inhibitors of breast cancer resistance protein

scientific article published on 11 November 2011

New structure-activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity

scientific article published on 30 September 2013

Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position

scientific article

Structure-activity relationships of chromone derivatives toward the mechanism of interaction with and inhibition of breast cancer resistance protein ABCG2.

scientific article published on 13 December 2013

Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein

scientific article published on 06 January 2012

Symmetric bis-chalcones as a new type of breast cancer resistance protein inhibitors with a mechanism different from that of chromones

scientific article published on 24 March 2014