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List of works by Roberto Pellicciari

Asymmetric synthesis of the four diastereoisomers of a novel non-steroidal farnesoid X receptor (FXR) agonist: role of the chirality on the biological activity

scientific article

Chiral ligand-exchange separation and resolution of extremely rigid glutamate analogs: 1-aminospiro[2.2]pentyl-1,4-dicarboxylic acids

scientific article published on 22 May 2010

Evaluation of the enantiomeric selectivity in the chiral ligand-exchange chromatography of amino acids by a computational model

scientific article published on 01 April 2004

Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5.

scientific article published on 13 August 2008

Novel potent and selective bile acid derivatives as TGR5 agonists: biological screening, structure-activity relationships, and molecular modeling studies

scientific article

Preparative resolution of 1-aminoindan-1,5-dicarboxylic acid (AIDA) by chiral ligand-exchange chromatography.

scientific article published in May 2004

Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists

scientific article published on 20 April 2012

Synthesis and chromatographic resolution of conformationally constrained analogues of homotaurine

article by Maria Carmela Fulco et al published October 2009 in Tetrahedron

TGR5 activation inhibits atherosclerosis by reducing macrophage inflammation and lipid loading

scientific article

TGR5-mediated bile acid sensing controls glucose homeostasis

scientific article

Targeting bile-acid signalling for metabolic diseases

scientific article published on August 2008