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List of works by Alastair R Hawkins

A prodrug approach for improving antituberculosis activity of potent Mycobacterium tuberculosis type II dehydroquinase inhibitors

scientific article

Chemical Modification of a Dehydratase Enzyme Involved in Bacterial Virulence by an Ammonium Derivative: Evidence of its Active Site Covalent Adduct

scientific article

Competitive inhibitors of Helicobacter pylori type II dehydroquinase: synthesis, biological evaluation, and NMR studies.

scientific article

Determination of the bound conformation of a competitive nanomolar inhibitor of mycobacterium tuberculosis type II dehydroquinase by NMR spectroscopy

scientific article published on 01 September 2006

Exploring the water-binding pocket of the type II dehydroquinase enzyme in the structure-based design of inhibitors

scientific article

Mechanistic basis of the inhibition of type II dehydroquinase by (2S)- and (2R)-2-benzyl-3-dehydroquinic acids

scientific article

Mycobacterium tuberculosis shikimate kinase inhibitors: design and simulation studies of the catalytic turnover

scientific article

Synthesis and biological evaluation of new nanomolar competitive inhibitors of Helicobacter pylori type II dehydroquinase. Structural details of the role of the aromatic moieties with essential residues

scientific article

Tetrahydrobenzothiophene derivatives: conformationally restricted inhibitors of type II dehydroquinase

scientific article

Understanding the key factors that control the inhibition of type II dehydroquinase by (2R)-2-benzyl-3-dehydroquinic acids

scientific article

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