List of works - Riccardo Baruchello

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

scientific article

A convenient synthesis of unsymmetrically substituted terphenyls of biologically active stilbenes via a double Suzuki cross-coupling protocol

A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach

scientific article published on June 2016

Antitumor effects of curcumin and structurally beta-diketone modified analogs on multidrug resistant cancer cells.

scientific article published on 13 November 2007

Arylamidonaphtalene sulfonate compounds as a novel class of heparanase inhibitors

scientific article published on 8 August 2017

Curcumin as a possible lead compound against hormone-independent, multidrug-resistant breast cancer.

scientific article

Design, synthesis and biological evaluation of novel stilbene-based antitumor agents.

scientific article

Design, synthesis, and biological evaluation of novel aminobisphosphonates possessing an in vivo antitumor activity through a gammadelta-T lymphocytes-mediated activation mechanism.

scientific article published on 21 October 2008

Development of hemiasterlin derivatives as potential anticancer agents that inhibit tubulin polymerization and synergize with a stilbene tubulin inhibitor.

scientific article published on 8 June 2011

Hemiasterlin derivative (R)(S)(S)-BF65 and Akt inhibitor MK-2206 synergistically inhibit SKOV3 ovarian cancer cell growth

scientific article published on 17 June 2016

Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines.

scientific article published on February 2005

Hydropathic analysis and biological evaluation of stilbene derivatives as colchicine site microtubule inhibitors with anti-leukemic activity

scientific article

Inhibition of activated STAT5 in Bcr/Abl expressing leukemia cells with new pimozide derivatives

scientific article published on August 2014

Inhibition of cell proliferation by a resveratrol analog in human pancreatic and breast cancer cells

scientific article published on March 2009

Lack of nucleophilic addition in the isoxazole and pyrazole diketone modified analogs of curcumin; implications for their antitumor and chemosensitizing activities

scientific article

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

scientific article published on November 23, 2011

Novel A-ring and B-ring modified combretastatin A-4 (CA-4) analogues endowed with interesting cytotoxic activity.

scientific article published on 11 September 2008

Novel combretastatin analogues endowed with antitumor activity

scientific article published on June 2006

Novel terphenyls and 3,5-diaryl isoxazole derivatives endowed with growth supporting and antiapoptotic properties.

scientific article

Pro-apoptotic activity of novel synthetic isoxazole derivatives exhibiting inhibitory activity against tumor cell growth in vitro

scientific article published on 24 August 2020

Stilbene-based anticancer agents: resveratrol analogues active toward HL60 leukemic cells with a non-specific phase mechanism

scientific article published on 31 March 2006

Studies on the apoptotic activity of natural and synthetic retinoids: discovery of a new class of synthetic terphenyls that potently support cell growth and inhibit apoptosis in neuronal and HL-60 cells.

scientific article published in June 2005

Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a.

scientific article published on 20 July 2011

Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents

scientific article published in July 2003

Synthesis and pharmacology of 6-substituted benztropines: discovery of novel dopamine uptake inhibitors possessing low binding affinity to the dopamine transporter

scientific article published in May 2005

Versatile synthesis of new cytotoxic agents structurally related to hemiasterlins

scientific article

List of works by Riccardo Baruchello

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

A convenient synthesis of unsymmetrically substituted terphenyls of biologically active stilbenes via a double Suzuki cross-coupling protocol

A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach

Antitumor effects of curcumin and structurally beta-diketone modified analogs on multidrug resistant cancer cells.

Arylamidonaphtalene sulfonate compounds as a novel class of heparanase inhibitors

Curcumin as a possible lead compound against hormone-independent, multidrug-resistant breast cancer.

Design, synthesis and biological evaluation of novel stilbene-based antitumor agents.

Design, synthesis, and biological evaluation of novel aminobisphosphonates possessing an in vivo antitumor activity through a gammadelta-T lymphocytes-mediated activation mechanism.

Development of hemiasterlin derivatives as potential anticancer agents that inhibit tubulin polymerization and synergize with a stilbene tubulin inhibitor.

Hemiasterlin derivative (R)(S)(S)-BF65 and Akt inhibitor MK-2206 synergistically inhibit SKOV3 ovarian cancer cell growth

Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines.

Hydropathic analysis and biological evaluation of stilbene derivatives as colchicine site microtubule inhibitors with anti-leukemic activity

Inhibition of activated STAT5 in Bcr/Abl expressing leukemia cells with new pimozide derivatives

Inhibition of cell proliferation by a resveratrol analog in human pancreatic and breast cancer cells

Lack of nucleophilic addition in the isoxazole and pyrazole diketone modified analogs of curcumin; implications for their antitumor and chemosensitizing activities

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

Novel A-ring and B-ring modified combretastatin A-4 (CA-4) analogues endowed with interesting cytotoxic activity.

Novel combretastatin analogues endowed with antitumor activity

Novel terphenyls and 3,5-diaryl isoxazole derivatives endowed with growth supporting and antiapoptotic properties.

Pro-apoptotic activity of novel synthetic isoxazole derivatives exhibiting inhibitory activity against tumor cell growth in vitro

Stilbene-based anticancer agents: resveratrol analogues active toward HL60 leukemic cells with a non-specific phase mechanism

Studies on the apoptotic activity of natural and synthetic retinoids: discovery of a new class of synthetic terphenyls that potently support cell growth and inhibit apoptosis in neuronal and HL-60 cells.

Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a.

Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents

Synthesis and pharmacology of 6-substituted benztropines: discovery of novel dopamine uptake inhibitors possessing low binding affinity to the dopamine transporter

Versatile synthesis of new cytotoxic agents structurally related to hemiasterlins