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List of works by Erica C VanderPorten

Aminoisoxazoles as Potent Inhibitors of Tryptophan 2,3-Dioxygenase 2 (TDO2)

scientific article published on 02 April 2018

Design and evaluation of 1,7-naphthyridones as novel KDM5 inhibitors

scientific article

Design and synthesis of 2-amino-isoxazolopyridines as Polo-like kinase inhibitors

scientific article

Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors

scientific article

Differential effects of divalent manganese and magnesium on the kinase activity of leucine-rich repeat kinase 2 (LRRK2).

scientific article published in April 2010

Identification of 2-amino-5-aryl-pyrazines as inhibitors of human lactate dehydrogenase

scientific article

Identification of Small-Molecule Noncovalent Binders Utilizing SAMDI Technology

scientific article published on 05 June 2017

Identification of potent, selective KDM5 inhibitors

scientific article

Identification of substituted 2-thio-6-oxo-1,6-dihydropyrimidines as inhibitors of human lactate dehydrogenase

scientific article

Identification of substituted 3-hydroxy-2-mercaptocyclohex-2-enones as potent inhibitors of human lactate dehydrogenase

scientific article

Implementation of the CYP Index for the Design of Selective Tryptophan-2,3-dioxygenase Inhibitors

scientific article published on 04 March 2020

Label-free high-throughput assays to screen and characterize novel lactate dehydrogenase inhibitors

scientific article

Optimization of 5-(2,6-dichlorophenyl)-3-hydroxy-2-mercaptocyclohex-2-enones as potent inhibitors of human lactate dehydrogenase

scientific article

Quantitative Determination of Protein-Ligand Affinity by Size Exclusion Chromatography Directly Coupled to High-Resolution Native Mass Spectrometry

scientific article published on 12 December 2018

The Aurora kinase inhibitor SNS-314 shows broad therapeutic potential with chemotherapeutics and synergy with microtubule-targeted agents in a colon carcinoma model

scientific article published on April 2009