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List of works by Johan D Oslob

2-Aminobenzimidazoles as potent Aurora kinase inhibitors.

scientific article

A small-molecule inhibitor of sarcomere contractility suppresses hypertrophic cardiomyopathy in mice.

scientific article published on February 2016

Binding of small molecules to an adaptive protein-protein interface

scientific article

Discovery and Development of Potent LFA-1/ICAM-1 Antagonist SAR 1118 as an Ophthalmic Solution for Treating Dry Eye.

scientific article

Discovery of a potent and selective aurora kinase inhibitor

scientific article

Discovery of a potent small molecule IL-2 inhibitor through fragment assembly

scientific article published in April 2003

Discovery of tetrahydroisoquinoline (THIQ) derivatives as potent and orally bioavailable LFA-1/ICAM-1 antagonists

scientific article published on 23 July 2010

Identification of nonpeptidic small-molecule inhibitors of interleukin-2.

scientific article

Imidazopyridine-Based Fatty Acid Synthase Inhibitors That Show Anti-HCV Activity and in Vivo Target Modulation

scientific article

Integrating fragment assembly and biophysical methods in the chemical advancement of small-molecule antagonists of IL-2: an approach for inhibiting protein-protein interactions

scientific article

Small-molecule inhibition of TNF-alpha

scientific article

Structure–activity relationship (SAR) of the α-amino acid residue of potent tetrahydroisoquinoline (THIQ)-derived LFA-1/ICAM-1 antagonists

scientific article published on 05 November 2010

Water-soluble prodrugs of an Aurora kinase inhibitor

scientific article published on 19 January 2009