Search filters

List of works by Michael J Romanowski

2-Aminobenzimidazoles as potent Aurora kinase inhibitors.

scientific article

Design and synthesis of 2-amino-isoxazolopyridines as Polo-like kinase inhibitors

scientific article

Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors

scientific article

Discovery of a potent and selective aurora kinase inhibitor

scientific article

Fragment-based discovery of nonpeptidic BACE-1 inhibitors using tethering

scientific article

SNS-314, a pan-Aurora kinase inhibitor, shows potent anti-tumor activity and dosing flexibility in vivo

scientific article published in August 2009

Structural analysis of caspase-1 inhibitors derived from Tethering.

scientific article published on 9 April 2005

Structure of theBrachydanio rerioPolo-like kinase 1 (Plk1) catalytic domain in complex with an extended inhibitor targeting the adaptive pocket of the enzyme

scientific article

Structures of the wild-type and activated catalytic domains of Brachydanio rerio Polo-like kinase 1 (Plk1): changes in the active-site conformation and interactions with ligands

scientific article

Tethering identifies fragment that yields potent inhibitors of human caspase-1

scientific article published on 04 November 2005

Water-soluble prodrugs of an Aurora kinase inhibitor

scientific article published on 19 January 2009

Paulina is supported by:

About Paulina

Help