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List of works by Bruce Fahr

A diaminocyclohexyl analog of SNS-032 with improved permeability and bioavailability properties

scientific article

Allosteric inhibition of protein tyrosine phosphatase 1B.

scientific article published on 18 July 2004

Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors

scientific article

Fragment-based discovery of nonpeptidic BACE-1 inhibitors using tethering

scientific article

Identification of potent and novel small-molecule inhibitors of caspase-3

scientific article published on 01 November 2003

Identification of potent and selective small-molecule inhibitors of caspase-3 through the use of extended tethering and structure-based drug design

scientific article published in November 2002

Methyl-substitution of an iminohydantoin spiropiperidine β-secretase (BACE-1) inhibitor has a profound effect on its potency

scientific article

Modifications of the isonipecotic acid fragment of SNS-032: analogs with improved permeability and lower efflux ratio

scientific article published on 2 October 2008

Structural analysis of caspase-1 inhibitors derived from Tethering.

scientific article published on 9 April 2005

Tethering identifies fragment that yields potent inhibitors of human caspase-1

scientific article published on 04 November 2005

Total Synthesis of Aeruginosin 98B ⬇️

scientific article published on November 12, 2012

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