List of works - Masayuki Inoue

Biological Effects of a Simplified Synthetic Analogue of Ion-Channel-Forming Polytheonamide B on Plasma Membrane and Lysosomes

scientific article published on 25 October 2019

Comprehensive Structure-Activity Relationship Studies of Macrocyclic Natural Products Enabled by Their Total Syntheses

scientific article published on 04 April 2019

Conformational equilibrium shift underlies altered K+ channel gating as revealed by NMR

scientific article published on 14 October 2020

Construction of a 6/5/9-membered tricyclic structure of cladiellins via radical-polar crossover reaction

scientific article published on 25 February 2019

Construction of the septahydroxylated ABC-ring system of dihydro-β-agarofurans: application of 6-exo-dig radical cyclization

scientific article published on 27 March 2017

Convergent Assembly of Highly Oxygenated Natural Products Enabled by Intermolecular Radical Reactions

scientific article published on 06 January 2021

Convergent Synthesis of Taxol Skeleton via Decarbonylative Radical Coupling Reaction

scientific article published on 19 November 2018

Convergent Total Synthesis of Asimicin via Decarbonylative Radical Dimerization

scientific article published on 20 November 2018

Development of a high-throughput strategy for discovery of potent analogues of antibiotic lysocin E

scientific article published on 05 July 2019

Discovery of gramicidin A analogues with altered activities by multidimensional screening of a one-bead-one-compound library

scientific article published on 01 October 2020

Evolution of Radical-Based Convergent Strategies for Total Syntheses of Densely Oxygenated Natural Products.

scientific article

Full solid-phase total synthesis of macrocyclic natural peptides using four-dimensionally orthogonal protective groups

scientific article published on 24 June 2019

In honor of Professor Samuel J. Danishefsky

scientific article published on 27 May 2019

Solid-Phase Total Synthesis and Dual Mechanism of Action of the Channel-Forming 48-mer Peptide Polytheonamide B

scientific article published on 07 August 2018

Solid-Phase Total Synthesis of Yaku'amide B Enabled by Traceless Staudinger Ligation

scientific article published on 03 February 2020

Synthesis of the Tetracyclic Structure of Batrachotoxin Enabled by Bridgehead Radical Coupling and Pd/Ni-Promoted Ullmann Reaction

scientific article published on 12 December 2017

Target Identification of Yaku'amide B and Its Two Distinct Activities against Mitochondrial FoF1-ATP Synthase

scientific article published on 12 September 2018

The liver-brain-gut neural arc maintains the Treg cell niche in the gut

scientific article published on 11 June 2020

Total Synthesis and Biological Mode of Action of WAP-8294A2: A Menaquinone-Targeting Antibiotic.

scientific article

Total Synthesis of (-)-Morphine

scientific article published on 4 April 2017

Total Synthesis of 1-Hydroxytaxinine

scientific article published on 25 July 2019

Total Synthesis of 5-epi-Eudesm-4(15)-ene-1β,6β-diol via Decarbonylative Radical Coupling Reaction

scientific article published on 09 September 2019

Total Synthesis of Diospyrodin and Its Three Diastereomers

scientific article published on 06 August 2020

Total Synthesis of Resiniferatoxin Enabled by Radical-Mediated Three-Component Coupling and 7-endo Cyclization

scientific article

Total Synthesis of Talatisamine

scientific article published on 19 November 2019

Total Synthesis of Zaragozic Acid C: Implementation of Photochemical C(sp3)-H Acylation

scientific article published on 16 January 2017

Total synthesis and biological evaluation of 19-hydroxysarmentogenin-3-O-a-L-rhamnoside, trewianin, and their aglycons

scientific article published on 25 October 2018

Unified Total Synthesis of Five Bufadienolides

scientific article published on 26 October 2020

Unified Total Synthesis of Polyoxins J, L, and Fluorinated Analogues on the Basis of Decarbonylative Radical Coupling Reactions.

scientific article published on 20 July 2017

List of works by Masayuki Inoue

Biological Effects of a Simplified Synthetic Analogue of Ion-Channel-Forming Polytheonamide B on Plasma Membrane and Lysosomes

Comprehensive Structure-Activity Relationship Studies of Macrocyclic Natural Products Enabled by Their Total Syntheses

Conformational equilibrium shift underlies altered K+ channel gating as revealed by NMR

Construction of a 6/5/9-membered tricyclic structure of cladiellins via radical-polar crossover reaction

Construction of the septahydroxylated ABC-ring system of dihydro-β-agarofurans: application of 6-exo-dig radical cyclization

Convergent Assembly of Highly Oxygenated Natural Products Enabled by Intermolecular Radical Reactions

Convergent Synthesis of Taxol Skeleton via Decarbonylative Radical Coupling Reaction

Convergent Total Synthesis of Asimicin via Decarbonylative Radical Dimerization

Development of a high-throughput strategy for discovery of potent analogues of antibiotic lysocin E

Discovery of gramicidin A analogues with altered activities by multidimensional screening of a one-bead-one-compound library

Evolution of Radical-Based Convergent Strategies for Total Syntheses of Densely Oxygenated Natural Products.

Full solid-phase total synthesis of macrocyclic natural peptides using four-dimensionally orthogonal protective groups

In honor of Professor Samuel J. Danishefsky

Solid-Phase Total Synthesis and Dual Mechanism of Action of the Channel-Forming 48-mer Peptide Polytheonamide B

Solid-Phase Total Synthesis of Yaku'amide B Enabled by Traceless Staudinger Ligation

Synthesis of the Tetracyclic Structure of Batrachotoxin Enabled by Bridgehead Radical Coupling and Pd/Ni-Promoted Ullmann Reaction

Target Identification of Yaku'amide B and Its Two Distinct Activities against Mitochondrial FoF1-ATP Synthase

The liver-brain-gut neural arc maintains the Treg cell niche in the gut

Total Synthesis and Biological Mode of Action of WAP-8294A2: A Menaquinone-Targeting Antibiotic.

Total Synthesis of (-)-Morphine

Total Synthesis of 1-Hydroxytaxinine

Total Synthesis of 5-epi-Eudesm-4(15)-ene-1β,6β-diol via Decarbonylative Radical Coupling Reaction

Total Synthesis of Diospyrodin and Its Three Diastereomers

Total Synthesis of Resiniferatoxin Enabled by Radical-Mediated Three-Component Coupling and 7-endo Cyclization

Total Synthesis of Talatisamine

Total Synthesis of Zaragozic Acid C: Implementation of Photochemical C(sp3)-H Acylation

Total synthesis and biological evaluation of 19-hydroxysarmentogenin-3-O-a-L-rhamnoside, trewianin, and their aglycons

Unified Total Synthesis of Five Bufadienolides

Unified Total Synthesis of Polyoxins J, L, and Fluorinated Analogues on the Basis of Decarbonylative Radical Coupling Reactions.