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List of works by Janina Karolak-Wojciechowska

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

scientific article published on 10 August 2015

A structure-activity relationship study of the affinity of selected imidazo[1,2-a]pyridine derivatives, congeners of zolpidem, for the omega 1-subtype of the benzodiazepine receptor

scientific article published in January 2001

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

scientific article

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 5. Synthesis of some triazolo[4,3-b]pyridazine and pyridazino[6,1-c]triazine derivatives as potential benzodiazepine receptor ligands

scientific article published on 01 November 1996

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 6. Aromatization of some tetrahydrotriazolo[4,3-b]pyridazine derivatives with potential activity as benzodiazepine receptor ligands

scientific article published on 01 July 1997

Bicyclic [b]-heteroannulated pyridazine derivatives--II. Structure-activity relationships in the 6-aryltriazolo-[4,3-b]pyridazine ligands of the benzodiazepine receptor

scientific article published in August 1994

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

scientific article published on 2 December 2015

Conformational investigation of alpha, beta-dehydropeptides. Part VI. Molecular and crystal structure of benzyloxycarbonylglycyl-(Z)-dehydrophenylalanine

scientific article published on 01 October 1994

Convenient way of synthesis and crystal structure of 1-[(5-chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine, a histamine H4 receptor antagonist

Crystal and Molecular Structure of 4-[ω-(Benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a Different Pharmacological Activity

Crystallographic and spectroscopic studies of 5-arylidene-2-amino-imidazol-4-ones

scientific article published in July 2009

Crystallographic studies of (Z) and (E) isomers of 2-amino-5-(2-chlorobenzylidene)-1-methyl-1H-imidazol-4(5H)-one

scientific article published in March 2010

Design, synthesis, and anticonvulsant activity of new N-Mannich bases derived from spirosuccinimides and spirohydantoins.

scientific article published on 30 June 2010

Desulfurization of 2-thiouracil nucleosides: conformational studies of 4-pyrimidinone nucleosides

scientific article published on 01 April 2011

Efficient synthesis of 2'-deoxyzebularine and its α-anomer by the silyl method of N-glycosylation. Crystal structures and conformational study in solution.

scientific article published on 28 March 2014

Five-membered heterocycles. Part III. Aromaticity of 1,3-imidazole in 5+n hetero-bicyclic molecules

article

Four- and five-coordinate copper(II) complexes with N-(4,4-diphenyl-5-oxo-4,5-dihydro-1H-imidazol-2-yl)glycine

scientific article published on 12 January 2008

From crystallographic data to the creation of a binding model with a receptor

scientific article

Fused 2-thiohydantoin derivatives: evaluation as potential antioxidants

scientific article published on 01 April 1997

Glycine derivatives of imidazolones as potential ligands of glycine binding site of NMDA receptors. Part 1

scientific article published on 01 September 1998

Imidazo-thiazine, -diazinone and -diazepinone derivatives. Synthesis, structure and benzodiazepine receptor binding

scientific article published in May 2001

Imidazo[2,1-b]thiazepines: synthesis, structure and evaluation of benzodiazepine receptor binding.

scientific article published in March 2004

Impact of the aryl substituent kind and distance from pyrimido[2,1-f]purindiones on the adenosine receptor selectivity and antagonistic properties.

scientific article published in April 2003

Inhibition of cryptosporidium parvum in vitro by 9-(alkylthio)acridine derivatives

scientific article

N9-benzyl-substituted 1,3-dimethyl- and 1,3-dipropyl-pyrimido[2,1-f]purinediones: synthesis and structure-activity relationships at adenosine A1 and A2A receptors

scientific article published on 19 April 2007

Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: Structure–activity relationships as adenosine A1 and A2A receptor ligands

scientific article published on 22 August 2007

Quantitative analysis of structure-activity relationship in the acridine serie. Part 1: Antiparasitic 9-thioaryl-acridine derivatives

scientific article published on 01 September 2000

Quantitative analysis of structure-activity relationship in the acridine series. Part 2: Antitumor 9-thiadiazolo-acridine derivatives

scientific article published on 01 November 2000

Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors.

scientific article

Structural and electronic conditions for anticonvulsant activity of bicyclic hydantoin derivatives

scientific article published on 01 February 1995

Structure and activity studies on glycine receptor ligands. Part 5. Diphenyl imidazolin-4-one glycinamides

scientific article published on 01 September 1998

Structure of an anticonvulsant N-methyl-m-bromophenylsuccinimide ⬇️

scientific article published on January 15, 1992

Structure-activity relationship investigations of the modulating effect of core substituents on the affinity of pyrazoloquinolinone congeners for the benzodiazepine receptor

scientific article

Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

scientific article published on 01 November 1999

Structures of three N-pyridyl-2-phenylsuccinimides and structural evidence for substituent effects on anticonvulsant properties

scientific article published on 01 January 1990

Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α₁-adrenoceptor antagonistic properties

scientific article published on 05 June 2012

Synthesis and anticonvulsant activity of new fluorinated N-phenyl- and N-benzyl-2-azaspiro[4.4]nonane- and [4.5]decane-1,3-dione derivatives: Part III

scientific article published in March 2006

Synthesis and anticonvulsant properties of new N-Mannich bases derived from 3,3-diphenyl- and 3-ethyl-3-methyl-pyrrolidine-2,5-diones. Part III.

scientific article published on 25 November 2012

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

scientific article

Synthesis and biological activity of tricyclic aryloimidazo-, pyrimido-, and diazepinopurinediones

scientific article published on 17 July 2006

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

scientific article

Synthesis and effects on chloroquine susceptibility in Plasmodium falciparum of a series of new dihydroanthracene derivatives

scientific article published on July 2002

Synthesis, biological activity and molecular modelling studies of tricyclic alkylimidazo-, pyrimido- and diazepinopurinediones

scientific article published on 02 April 2013

Synthesis, physicochemical and anticonvulsant properties of N-benzyl and N-aminophenyl derivatives of 2-azaspiro[4.4]nonane and [4.5]decane-1,3-dione. Part I.

scientific article published in June 2005

Synthesis, physicochemical and anticonvulsant properties of new N-pyridyl derivatives of 3-phenyl- and 3,3-diphenyl-succinimides

scientific article published on 01 July 1999

Tricyclic oxazolo[2,3-f]purinediones: potency as adenosine receptor ligands and anticonvulsants.

scientific article published in September 2004

Use of molecular electrostatic potentials for analysis of anticonvulsant activities of phenylsuccinimides

scientific article published on 01 January 1993

tert-Butyl N-[(S)-3-isobutyl-2-oxooxetan-3-yl]carbamate

scientific article published on 6 December 2007

tert-Butyl N-[(S)-3-isopropyl-2-oxo-oxetan-3-yl]carbamate

scientific article published on 6 February 2008

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