Search filters

List of works by Pierre Germain

9-cis-retinoic acid analogues with bulky hydrophobic rings: new RXR-selective agonists

scientific article published in December 2004

A unique secondary-structure switch controls constitutive gene repression by retinoic acid receptor

scientific article

An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor β (RARβ, NR1B2) Selective Agonist.

scientific article published on May 2015

C3 halogen and c8'' substituents on stilbene arotinoids modulate retinoic Acid receptor subtype function

scientific article published in October 2009

Characterization of the interaction between retinoic acid receptor/retinoid X receptor (RAR/RXR) heterodimers and transcriptional coactivators through structural and fluorescence anisotropy studies

scientific article published on 4 November 2004

Co-regulator recruitment and the mechanism of retinoic acid receptor synergy

scientific article published in January 2002

Differential action on coregulator interaction defines inverse retinoid agonists and neutral antagonists

scientific article

Insights into the mechanism of the site-selective sequential palladium-catalyzed cross-coupling reactions of dibromothiophenes/dibromothiazoles and arylboronic acids. Synthesis of PPARβ/δ agonists

scientific article published on 13 November 2006

International Union of Pharmacology. LX. Retinoic acid receptors

scientific article

International Union of Pharmacology. LXIII. Retinoid X receptors

scientific article

Modulating retinoid X receptor with a series of (E)-3-[4-hydroxy-3-(3-alkoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)phenyl]acrylic acids and their 4-alkoxy isomers

scientific article

Modulators of the structural dynamics of the retinoid X receptor to reveal receptor function

scientific article

Monitoring ligand-mediated nuclear receptor-coregulator interactions by noncovalent mass spectrometry

scientific article published in December 2004

Neofunctionalization in vertebrates: the example of retinoic acid receptors

scientific article

New retinoid chemotypes: 9-cis-retinoic acid analogs with hydrophobic rings derived from terpenes as selective RAR agonists

scientific article

Nuclear receptor superfamily: Principles of signaling

RARbeta ligand-binding domain bound to an SRC-1 co-activator peptide: purification, crystallization and preliminary X-ray diffraction analysis

scientific article published on 20 October 2004

Rational design of RAR-selective ligands revealed by RARbeta crystal structure

scientific article

Retinoid receptor subtype-selective modulators through synthetic modifications of RARgamma agonists.

scientific article published on 18 May 2009

Retinoids: potential in cancer prevention and therapy.

scientific article

Silicon analogues of the retinoid agonists TTNPB and 3-methyl-TTNPB, disila-TTNPB and disila-3-methyl-TTNPB: chemistry and biology

scientific article published on September 2007

Structure, function and modulation of retinoic acid receptor beta, a tumor suppressor

scientific article published on 22 February 2007

Synthesis of the PPARbeta/delta-selective agonist GW501516 and C4-thiazole-substituted analogs

scientific article published on 18 October 2005